Allopregnanolone Regenerative Therapeutic for Mild Alzheimer's Disease

NCT ID: NCT04838301

Last Updated: 2025-05-11

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

RECRUITING

Clinical Phase

PHASE2

Total Enrollment

200 participants

Study Classification

INTERVENTIONAL

Study Start Date

2023-08-15

Study Completion Date

2026-04-30

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

A phase 2, double-blind, randomized, placebo-controlled clinical trial to evaluate the safety and efficacy of Allopregnanolone as a regenerative therapeutic for Alzheimer's disease.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

This is a proof-of-concept phase 2 clinical trial to investigate the long-term safety and efficacy of Allo to function as a regenerative therapeutic to restore structural integrity and cognitive function of the brain in participants with mild Alzheimer's disease (AD) dementia. Study participants will be male and female, APOE ε4 positive diagnosed with probable AD, Mini-Mental State Exam (MMSE) 20 to 26, ages 55 to 80 years old.

After a 2-4-week screening period, participants will be randomized to 4 mg Allo (administered intravenously over 30 minutes, once per week, in clinic) or matching placebo, 1:1 allocation, for a period of 12 months. After 12 months, all participants in the placebo group will be crossed-over to receive Allo for the remainder of the study (6 month open-label phase). Brain imaging to evaluate the primary endpoint will be conducted at baseline, 6 and 12 months.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Alzheimer Dementia Late Onset Alzheimer Disease Neurodegenerative Diseases

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Participants are assigned to the active intervention or placebo in parallel for 12 months. After 12 months, all participants in the placebo group will be crossed-over to receive Allo for the remainder of the study (6 month open-label phase).
Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors
After 12 months participants and study personnel will be aware of the open label phase, but initial randomization will remain blind during the entire length of the study (placebo-controlled and open-label periods); that is, all participants and study personnel are blinded to each participant's randomization to initial treatment group.

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Allo group

Allopregnanolone 4mg IV 30-minute infusion once per week for 12 months.

Group Type EXPERIMENTAL

Allopregnanolone

Intervention Type DRUG

Allopregnanolone 4mg IV via 30-minute infusion, once per week.

Control group

Placebo (normal saline) IV 30-minute infusion once per week for 12 months.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type OTHER

Normal saline solution IV via 30-minute infusion, once per week

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

Allopregnanolone

Allopregnanolone 4mg IV via 30-minute infusion, once per week.

Intervention Type DRUG

Placebo

Normal saline solution IV via 30-minute infusion, once per week

Intervention Type OTHER

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

Allo

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Men and postmenopausal women
* Age 55 to 80 years old
* Meets NIA-AA criteria for probable AD dementia
* MMSE of 20-26
* APOE ε4 positive
* Geriatric Depression Scale short form (GDS-S) score of ≤ 6
* No medical contraindications to participation
* Capacity to provide informed consent at screening

Exclusion Criteria

* Dementia other than probable AD
* Use of benzodiazepines, anticonvulsants, antipsychotics, or other drugs that might interact with the GABA-A receptor complex
* History of stroke with a modified Hachinski Ischemic Scale score \>4
* History of seizure disorder, focal brain lesion, traumatic brain injury
* History within the last 5 years of a primary or recurrent malignant disease
* Unstable or clinically significant cardiovascular, kidney or liver disease
* MRI indicative of any other significant abnormality, including but not limited to one or more significant ARIA-E or macro-hemorrhage findings, or multiple microhemorrhages (\>8), or Fazekas score of 3; encephalomalacia, aneurysms, vascular malformations, subdural hematoma, or space occupying lesions
* Any conditions that would contraindicate MRI studies.
Minimum Eligible Age

55 Years

Maximum Eligible Age

80 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

National Institute on Aging (NIA)

NIH

Sponsor Role collaborator

Syneos Health

OTHER

Sponsor Role collaborator

University of Southern California

OTHER

Sponsor Role collaborator

ADM Diagnostics

UNKNOWN

Sponsor Role collaborator

University of Arizona

OTHER

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Roberta Brinton

Director, Center for Innovation in Brain Science; Professor, Departments of Pharmacology and Neurology

Responsibility Role PRINCIPAL_INVESTIGATOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Roberta D Brinton, PhD

Role: PRINCIPAL_INVESTIGATOR

University of Arizona

Lon Schneider, MD

Role: PRINCIPAL_INVESTIGATOR

University of Southern California

Gerson D Hernandez, MD, MPH

Role: STUDY_DIRECTOR

University of Arizona

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Perseverance Research Center

Scottsdale, Arizona, United States

Site Status RECRUITING

ATP Clinical Research

Costa Mesa, California, United States

Site Status RECRUITING

Syrentis Clinical Research

Santa Ana, California, United States

Site Status RECRUITING

Optimus U Corporation

Miami, Florida, United States

Site Status RECRUITING

Miami Jewish Health

Miami, Florida, United States

Site Status RECRUITING

Combined Research

Orlando, Florida, United States

Site Status RECRUITING

Conquest Research

Winter Park, Florida, United States

Site Status RECRUITING

MedVadis Research

Waltham, Massachusetts, United States

Site Status RECRUITING

Countries

Review the countries where the study has at least one active or historical site.

United States

Central Contacts

Reach out to these primary contacts for questions about participation or study logistics.

Claudia M Lopez, BS

Role: CONTACT

520-626-6276

Facility Contacts

Find local site contact details for specific facilities participating in the trial.

Nicole Hank, PhD

Role: primary

4804716132

Bobby Shih

Role: primary

714-277-4472

Caitlyn Villanueva

Role: backup

714-277-4472

Emily Watson

Role: primary

714-542-3008 ext. 314

Rebecca Bonar

Role: backup

714-542-3008

Yaneicy Gonazalez Rojas, MD

Role: primary

Mariolga Aymat

Role: primary

305-751-8626 ext. 64103

Alexander Gomez

Role: backup

305-751-8626 ext. 64199

Adrian Delgado

Role: primary

407-440-4493

Yenilady Estevez

Role: backup

407-440-4493

Melissa O'Neill

Role: primary

407-916-0060

Rathod Meera

Role: backup

407-916-0060

Donald Counihan

Role: primary

781-373-2940

Jessica O'Brien

Role: backup

781-373-2940

References

Explore related publications, articles, or registry entries linked to this study.

Raikes AC, Hernandez GD, Matthews DC, Lukic AS, Law M, Shi Y, Schneider LS, Brinton RD. Exploratory imaging outcomes of a phase 1b/2a clinical trial of allopregnanolone as a regenerative therapeutic for Alzheimer's disease: Structural effects and functional connectivity outcomes. Alzheimers Dement (N Y). 2022 Mar 14;8(1):e12258. doi: 10.1002/trc2.12258. eCollection 2022.

Reference Type BACKGROUND
PMID: 35310526 (View on PubMed)

Hernandez GD, Solinsky CM, Mack WJ, Kono N, Rodgers KE, Wu CY, Mollo AR, Lopez CM, Pawluczyk S, Bauer G, Matthews D, Shi Y, Law M, Rogawski MA, Schneider LS, Brinton RD. Safety, tolerability, and pharmacokinetics of allopregnanolone as a regenerative therapeutic for Alzheimer's disease: A single and multiple ascending dose phase 1b/2a clinical trial. Alzheimers Dement (N Y). 2020 Dec 16;6(1):e12107. doi: 10.1002/trc2.12107. eCollection 2020.

Reference Type BACKGROUND
PMID: 33344752 (View on PubMed)

Brinton RD. Neurosteroids as regenerative agents in the brain: therapeutic implications. Nat Rev Endocrinol. 2013 Apr;9(4):241-50. doi: 10.1038/nrendo.2013.31. Epub 2013 Feb 26.

Reference Type BACKGROUND
PMID: 23438839 (View on PubMed)

Brinton RD, Wang JM. Therapeutic potential of neurogenesis for prevention and recovery from Alzheimer's disease: allopregnanolone as a proof of concept neurogenic agent. Curr Alzheimer Res. 2006 Jul;3(3):185-90. doi: 10.2174/156720506777632817.

Reference Type BACKGROUND
PMID: 16842093 (View on PubMed)

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

R01AG063826

Identifier Type: NIH

Identifier Source: secondary_id

View Link

Allo-20-001

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.