Dose Ranging Study Of Bococizumab (PF-04950615; RN316) In Hypercholesterolemic Japanese Subjects

NCT ID: NCT02055976

Last Updated: 2019-02-08

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

218 participants

Study Classification

INTERVENTIONAL

Study Start Date

2014-03-31

Study Completion Date

2015-01-31

Brief Summary

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The purpose of this study is to evaluate the low density lipoprotein cholesterol (LDL-C) lowering effect of Bococizumab (PF-04950615;RN316) administered subcutaneously at every two weeks (Q14D) in hypercholesterolemic Japanese subjects whose LDL-C is not controlled by a stable dose of atorvastatin, or who are naïve to a treatment by lipid lowering drug and whose LDL-C is not controlled.

Detailed Description

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Conditions

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Hypercholesterolemia

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Investigators Outcome Assessors

Study Groups

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Population A

A total of 9 groups in two population. Population A comprises hypercholesterolemic Japanese subjects whose LDL-C is not controlled by a stable dose of atorvastatin. A subject who is receiving a stable dose of atorvastatin will be randomized into one out of 5 dose groups.

Group Type EXPERIMENTAL

Bococizumab (PF-04950615;RN316)

Intervention Type DRUG

Atorvastatin plus PF-04950615 50 mg subcutaneous administration at every two weeks (Q14D SC) for 16 week

Bococizumab (PF-04950615;RN316)

Intervention Type DRUG

Atorvastatin plus PF-04950615 100 mg Q14D SC for 16 week

Bococizumab (PF-04950615;RN316)

Intervention Type DRUG

Atorvastatin plus PF-04950615 150 mg Q14D SC for 16 week

Placebo

Intervention Type DRUG

Atorvastatin plus PF-04950615 Placebo Q14D SC for 16 week

Ezetimibe

Intervention Type DRUG

Atorvastatin plus Ezetimibe 10 mg oral administration once daily for 16 week (open)

Population B

A total of 9 groups in two population. Population B comprises hypercholesterolemic Japanese subjects who are naïve for a treatment by lipid lowering drug and whose fasting LDL-cholesterol is not controlled. A subject who is treatment naïve will be randomized into one out of 4 dose groups.

Group Type EXPERIMENTAL

Bococizumab (PF-04950615;RN316)

Intervention Type DRUG

50 mg Q14D SC for 16 week

Bococizumab (PF-04950615;RN316)

Intervention Type DRUG

100 mg Q14D SC for 16 week

Bococizumab (PF-04950615;RN316)

Intervention Type DRUG

150 mg Q14D SC for 16 week

Placebo

Intervention Type DRUG

Placebo Q14D SC for 16 week

Interventions

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Bococizumab (PF-04950615;RN316)

Atorvastatin plus PF-04950615 50 mg subcutaneous administration at every two weeks (Q14D SC) for 16 week

Intervention Type DRUG

Bococizumab (PF-04950615;RN316)

Atorvastatin plus PF-04950615 100 mg Q14D SC for 16 week

Intervention Type DRUG

Bococizumab (PF-04950615;RN316)

Atorvastatin plus PF-04950615 150 mg Q14D SC for 16 week

Intervention Type DRUG

Placebo

Atorvastatin plus PF-04950615 Placebo Q14D SC for 16 week

Intervention Type DRUG

Ezetimibe

Atorvastatin plus Ezetimibe 10 mg oral administration once daily for 16 week (open)

Intervention Type DRUG

Bococizumab (PF-04950615;RN316)

50 mg Q14D SC for 16 week

Intervention Type DRUG

Bococizumab (PF-04950615;RN316)

100 mg Q14D SC for 16 week

Intervention Type DRUG

Bococizumab (PF-04950615;RN316)

150 mg Q14D SC for 16 week

Intervention Type DRUG

Placebo

Placebo Q14D SC for 16 week

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Subjects whose LDL-C is not controlled by a stable dose of atorvastatin (Population A).
* Subjects who are naïve to a treatment by lipid lowering drug and whose LDL-C is not controlled (Population B).

Exclusion Criteria

* Severe acute or chronic medical or psychiatric condition or laboratory abnormality.
* Pregnant females; breastfeeding females; males and females of childbearing potential; males and females of childbearing potential who are unwilling or unable to use a highly effective method of contraception.
* Subjects who were administered or prior exposed to PF-04950615 and/or anti-body targeting PCSK9.
Minimum Eligible Age

20 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Maebashi Hirosegawa Clinic

Maebashi, Gunma, Japan

Site Status

Yokohama Minoru Clinic

Yokohama, Kanagawa, Japan

Site Status

Heishinkai Medical Group Incorporated OCROM Clinic

Suita, Osaka, Japan

Site Status

Meiwa Hospital

Chiyoda-ku, Tokyo, Japan

Site Status

Tokyo-Eki Center-building Clinic

Chuo-ku, Tokyo, Japan

Site Status

Heishinkai Medical Group Incorporated ToCROM Clinic

Shinjuku-ku, Tokyo, Japan

Site Status

Clinical Research Hospital Tokyo

Shinjuku-ku, Tokyo, Japan

Site Status

Oda Clinic

Shinjuku-ku, Tokyo, Japan

Site Status

Sekino Hospital

Toshima-ku, Tokyo, Japan

Site Status

Countries

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Japan

References

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Wang EQ, Kaila N, Plowchalk D, Gibiansky L, Yunis C, Sweeney K. Population PK/PD modeling of low-density lipoprotein cholesterol response in hypercholesterolemic participants following administration of bococizumab, a potent anti-PCSK9 monoclonal antibody. CPT Pharmacometrics Syst Pharmacol. 2023 Dec;12(12):2013-2026. doi: 10.1002/psp4.13050. Epub 2023 Nov 22.

Reference Type DERIVED
PMID: 37994400 (View on PubMed)

Yokote K, Suzuki A, Li Y, Matsuoka N, Teramoto T. Pharmacokinetics and exploratory efficacy biomarkers of bococizumab, an anti-PCSK9 monoclonal antibody, in hypercholesterolemic Japanese subjects . Int J Clin Pharmacol Ther. 2019 Dec;57(12):575-589. doi: 10.5414/CP203418.

Reference Type DERIVED
PMID: 31549625 (View on PubMed)

Yokote K, Kanada S, Matsuoka O, Sekino H, Imai K, Tabira J, Matsuoka N, Chaudhuri S, Teramoto T. Efficacy and Safety of Bococizumab (RN316/PF-04950615), a Monoclonal Antibody Against Proprotein Convertase Subtilisin/Kexin Type 9, in Hypercholesterolemic Japanese Subjects Receiving a Stable Dose of Atorvastatin or Treatment-Naive - Results From a Randomized, Placebo-Controlled, Dose-Ranging Study. Circ J. 2017 Sep 25;81(10):1496-1505. doi: 10.1253/circj.CJ-16-1310. Epub 2017 May 23.

Reference Type DERIVED
PMID: 28539539 (View on PubMed)

Related Links

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Other Identifiers

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B1481036

Identifier Type: -

Identifier Source: org_study_id

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