A Pharmacokinetic and Pharmacodynamic Study of PF-04950615 (RN316) in Subjects With Hypercholesterolemia

NCT ID: NCT01435382

Last Updated: 2018-07-23

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

49 participants

Study Classification

INTERVENTIONAL

Study Start Date

2011-10-31

Study Completion Date

2012-04-30

Brief Summary

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This Phase 1 study has been designed to evaluate the absolute bioavailability of PF-04950615 (RN316) in subjects with hypercholesterolemia who are not currently on lipid-lowering therapy.

Detailed Description

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Conditions

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Hypercholesterolemia Dyslipidemias Hyperlipidemias Lipid Metabolism Disorders Metabolic Diseases

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

NONE

Study Groups

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Group A

Group Type EXPERIMENTAL

PF-04950615 (RN316)

Intervention Type BIOLOGICAL

Dose A - single-dose intravenous infusion

Group B

Group Type EXPERIMENTAL

PF-04950615 (RN316)

Intervention Type BIOLOGICAL

Dose B - single-dose subcutaneous injection

Group C

Group Type EXPERIMENTAL

PF-04950615 (RN316)

Intervention Type BIOLOGICAL

Dose C - single-dose subcutaneous injection

Group D

Group Type EXPERIMENTAL

PF-04950615 (RN316)

Intervention Type BIOLOGICAL

Dose D - single-dose subcutaneous injection

Interventions

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PF-04950615 (RN316)

Dose A - single-dose intravenous infusion

Intervention Type BIOLOGICAL

PF-04950615 (RN316)

Dose B - single-dose subcutaneous injection

Intervention Type BIOLOGICAL

PF-04950615 (RN316)

Dose C - single-dose subcutaneous injection

Intervention Type BIOLOGICAL

PF-04950615 (RN316)

Dose D - single-dose subcutaneous injection

Intervention Type BIOLOGICAL

Eligibility Criteria

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Inclusion Criteria

* Fasting LDL-C greater than or equal to 130 mg/dL at two qualifying screening visits.
* Total body weight greater than or equal to 50 kg (110 lbs) and less than or equal to 150 kg (330 lbs)

Exclusion Criteria

* Lipid-lowering prescription medications, homeopaths, herbal medicines, or nutritional supplements.
* Poorly controlled type 1 or type 2 diabetes.
* History of a cardiovascular or cerebrovascular event or related procedure during the past year.
* Poorly controlled hypertension.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Profil Institute for Clinical Research, Inc.

Chula Vista, California, United States

Site Status

Elite Research Institute

Miami, Florida, United States

Site Status

Vince and Associates Clinical Research

Overland Park, Kansas, United States

Site Status

PAREXEL International - Baltimore Early Phase Clinical Unit

Baltimore, Maryland, United States

Site Status

Jasper Clinic, Inc.

Kalamazoo, Michigan, United States

Site Status

Prism Research

Saint Paul, Minnesota, United States

Site Status

Medpace Clinical Pharmacology Unit

Cincinnati, Ohio, United States

Site Status

Countries

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United States

References

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Wang EQ, Kaila N, Plowchalk D, Gibiansky L, Yunis C, Sweeney K. Population PK/PD modeling of low-density lipoprotein cholesterol response in hypercholesterolemic participants following administration of bococizumab, a potent anti-PCSK9 monoclonal antibody. CPT Pharmacometrics Syst Pharmacol. 2023 Dec;12(12):2013-2026. doi: 10.1002/psp4.13050. Epub 2023 Nov 22.

Reference Type DERIVED
PMID: 37994400 (View on PubMed)

Udata C, Garzone PD, Gumbiner B, Joh T, Liang H, Liao KH, Williams JH, Meng X. A Mechanism-Based Pharmacokinetic/Pharmacodynamic Model for Bococizumab, a Humanized Monoclonal Antibody Against Proprotein Convertase Subtilisin/Kexin Type 9, and Its Application in Early Clinical Development. J Clin Pharmacol. 2017 Jul;57(7):855-864. doi: 10.1002/jcph.867. Epub 2017 Feb 9.

Reference Type DERIVED
PMID: 28181260 (View on PubMed)

Related Links

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Other Identifiers

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B1481006

Identifier Type: -

Identifier Source: org_study_id

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