Safety and Efficacy of Saxagliptin Plus Insulin With or Without Metformin

NCT ID: NCT00757588

Last Updated: 2015-06-01

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

455 participants

Study Classification

INTERVENTIONAL

Study Start Date

2008-11-30

Study Completion Date

2010-04-30

Brief Summary

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The purpose of this study is to compare the effects of saxagliptin with those of placebo as add-on therapy to insulin and insulin with metformin in improving glycemic control at 24 and 52 weeks.

Detailed Description

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Conditions

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Type 2 Diabetes

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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Saxagliptin, 5 mg + insulin

Saxagliptin, 5 mg, plus insulin, administered to participants with Type 2 diabetes inadequately controlled with insulin alone or with insulin plus metformin

Group Type EXPERIMENTAL

Saxagliptin, 5 mg + insulin

Intervention Type DRUG

Saxagliptin, 5-mg tablets (plus stable insulin dose), given orally once daily (24 weeks short-term, 28 weeks long-term); participants stratified by use of stable metformin dose; flexible insulin dose (as needed for rescue)

Placebo + insulin

Placebo administered to participants with Type 2 diabetes inadequately controlled with insulin alone or with insulin plus metformin

Group Type PLACEBO_COMPARATOR

Placebo + insulin

Intervention Type DRUG

Placebo tablets given orally once daily for 24 weeks (short-term period)+ insulin with metformin

Interventions

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Saxagliptin, 5 mg + insulin

Saxagliptin, 5-mg tablets (plus stable insulin dose), given orally once daily (24 weeks short-term, 28 weeks long-term); participants stratified by use of stable metformin dose; flexible insulin dose (as needed for rescue)

Intervention Type DRUG

Placebo + insulin

Placebo tablets given orally once daily for 24 weeks (short-term period)+ insulin with metformin

Intervention Type DRUG

Other Intervention Names

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BMS-477118

Eligibility Criteria

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Inclusion Criteria

* Type 2 diabetes mellitus
* Must have been taking a stable dose of basal or premixed insulin for 8 weeks or longer prior to screening
* If taking metformin, must have been taking the same daily dose for 8 weeks or longer prior to screening
* Insulin type should be intermediate- or long-acting (basal) or premixed (premixed formulation may include short- or rapid-acting insulin as 1 component).
* Inadequate glycemic control (A1C of 7.5% to 11.0%, inclusive)
* Body mass index of 45 kg/m² or lower
* Fasting C-peptide level of 0.8 ng/mL or higher

Exclusion Criteria

* Symptoms of poorly controlled diabetes, including but not limited to marked polyuria and polydipsia with greater than 10% weight loss during the last 3 months prior to screening or other signs and symptoms
* History of diabetic ketoacidosis or hyperosmolar nonketotic coma
* Women of childbearing potential unable or unwilling to use acceptable birth control
* Women who are pregnant or breastfeeding
* Active liver disease
* Anemia
* Chronic or repeated intermittent corticosteroid treatment (participants receiving stable doses of replacement corticosteroid (except dexamethasone) therapy may be enrolled)
* Use of short- or rapid-acting insulin
* Significant cardiovascular history defined as: myocardial infarction, coronary angioplasty or bypass graft, valvular disease or repair, unstable angina pectoris, transient ischemic attack, or cerebrovascular accident
* Congestive heart failure
* Unstable or rapidly progressing renal disease
* History of alcohol or drug abuse within the previous year
* History of hemoglobinopathies
* Unstable major psychiatric disorders
* Immunocompromised status
Minimum Eligible Age

18 Years

Maximum Eligible Age

78 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Bristol-Myers Squibb

Role: STUDY_DIRECTOR

Bristol-Myers Squibb

Locations

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Clinical Research Advantage, Inc

Tempe, Arizona, United States

Site Status

Valley Research

Fresno, California, United States

Site Status

Torrance-Lomita Medical Center

Lomita, California, United States

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Diabetes Medical Center Of California

Northridge, California, United States

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Ritchken & First M.D.'S

San Diego, California, United States

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Encompass Clinical Research

Spring Valley, California, United States

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Central Florida Clinical Trials, Inc.

Altamonte Springs, Florida, United States

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Family Care Associates Of Nw Florida

Chipley, Florida, United States

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Panhandle Family Care Assoc. & Coastal Palms Res. Grp Inc.

Marianna, Florida, United States

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Endocrine Research Solutions, Inc.

Roswell, Georgia, United States

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Danny W. Jackson P.A.

Rolling Fork, Mississippi, United States

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Southgate Medical Group

West Seneca, New York, United States

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Southeastern Research Associates, Inc.

Taylors, South Carolina, United States

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Texas Center For Drug Development

Houston, Texas, United States

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Dgd Research, Inc.

San Antonio, Texas, United States

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Aurora Advanced Healthcare

Milwaukee, Wisconsin, United States

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Local Institution

Calgary, Alberta, Canada

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Vancouver, British Columbia, Canada

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Bathurst, New Brunswick, Canada

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London, Ontario, Canada

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Charlottetown, Prince Edward Island, Canada

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Gatineau, Quebec, Canada

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Laval, Quebec, Canada

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Sherbrooke, Quebec, Canada

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Regina, Saskatchewan, Canada

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Besançon, , France

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Montpellier, , France

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Nantes, , France

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Valenciennes, , France

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Balatonfüred, , Hungary

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Budapest, , Hungary

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Budapest, , Hungary

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Budapest, , Hungary

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Szentes, , Hungary

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Zalaegerszeg-Pozva, , Hungary

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Indore, Madhya Pradesh, India

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Hariyāna, , India

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Mumbai, , India

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Pune, , India

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Pune, , India

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Pune, , India

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Vellore, , India

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Aguascalientes, Aguascalientes, Mexico

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Aguascalientes, Aguascalientes, Mexico

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Zapopan, Jal., Jalisco, Mexico

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Mexico City, Mexico City, Mexico

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Mexico City, Mexico City, Mexico

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Monterrey, Nuevo León, Mexico

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Monterrey, Nuevo León, Mexico

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Monterrey, Nuevo León, Mexico

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Monterrrey, Nuevo León, Mexico

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Veracruz, Veracruz, Mexico

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Elblag, , Poland

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Gdansk, , Poland

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Krakow, , Poland

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Lodz, , Poland

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Lublin, , Poland

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Sopot, , Poland

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Szczecin, , Poland

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Wroclaw, , Poland

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Zabrze, , Poland

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Kursk, , Russia

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Saint Petersburg, , Russia

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Saint Petersburg, , Russia

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Saint Petersburg, , Russia

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Saint Petersburg, , Russia

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Saint Petersburg, , Russia

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Saratov, , Russia

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Smolensk, , Russia

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Yaroslaval, , Russia

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Parktown, Gauteng, South Africa

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Durban, KwaZulu-Natal, South Africa

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Umhlanga, KwaZulu-Natal, South Africa

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Goodwood, Western Cape, South Africa

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Tygerberg, Western Cape, South Africa

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Middlesbrough, Cleveland, United Kingdom

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Salford, Greater Manchester, United Kingdom

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Newcastle upon Tyne, Tyne and Wear, United Kingdom

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Birmingham, West Midlands, United Kingdom

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Sheffield, Yorkshire, United Kingdom

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Countries

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United States Canada France Hungary India Mexico Poland Russia South Africa United Kingdom

References

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Perl S, Cook W, Wei C, Iqbal N, Hirshberg B. Saxagliptin Efficacy and Safety in Patients With Type 2 Diabetes and Moderate Renal Impairment. Diabetes Ther. 2016 Sep;7(3):527-35. doi: 10.1007/s13300-016-0184-9. Epub 2016 Jul 11.

Reference Type DERIVED
PMID: 27402391 (View on PubMed)

Cook W, Minervini G, Bryzinski B, Hirshberg B. Saxagliptin efficacy and safety in patients with type 2 diabetes mellitus stratified by cardiovascular disease history and cardiovascular risk factors: analysis of 3 clinical trials. Postgrad Med. 2014 Oct;126(6):19-32. doi: 10.3810/pgm.2014.10.2818.

Reference Type DERIVED
PMID: 25414932 (View on PubMed)

Barnett AH, Charbonnel B, Li J, Donovan M, Fleming D, Iqbal N. Saxagliptin add-on therapy to insulin with or without metformin for type 2 diabetes mellitus: 52-week safety and efficacy. Clin Drug Investig. 2013 Oct;33(10):707-17. doi: 10.1007/s40261-013-0107-8.

Reference Type DERIVED
PMID: 23949898 (View on PubMed)

Barnett AH, Charbonnel B, Donovan M, Fleming D, Chen R. Effect of saxagliptin as add-on therapy in patients with poorly controlled type 2 diabetes on insulin alone or insulin combined with metformin. Curr Med Res Opin. 2012 Apr;28(4):513-23. doi: 10.1185/03007995.2012.665046. Epub 2012 Mar 1.

Reference Type DERIVED
PMID: 22313154 (View on PubMed)

Related Links

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Other Identifiers

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Eudract-2008-001089-10

Identifier Type: -

Identifier Source: secondary_id

CV181-057

Identifier Type: -

Identifier Source: org_study_id

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