Pharmacokinetic-guided Dosing of Emicizumab

NCT ID: NCT06320626

Last Updated: 2024-03-20

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE4

Total Enrollment

95 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-09-08

Study Completion Date

2026-08-31

Brief Summary

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The goal of this multicentre, prospective, open-label, cross-over clinical study is to determine whether individualized PK-guided dosing of emicizumab is non-inferior to conventional dosing of emicizumab in the prevention of bleeding in congenital haemophilia A patients.

Detailed Description

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Haemophilia A is an X-linked hereditary bleeding disorder resulting from a deficiency or dysfunction of endogenous coagulation factor VIII (FVIII). Persons with haemophilia A (PwHA) suffer from spontaneous or provoked bleeding, predominantly into major joints, which eventually lead to painful and chronic disabling arthropathy. The primary goal in clinical management of haemophilia A is prevention of bleeding by self-administration of FVIII concentrates via intravenous injections.

Prophylaxis with FVIII concentrates has effectively reduced treated bleeds from an annual average of 20-30 to 1-4. However, in approximately 30% of PwHA anti-FVIII antibodies (known as inhibitors) develop that interfere with FVIII replacement therapy. PwHA who develop inhibitors require alternative suboptimal therapy with (costly) bypassing agents (BPA).

The first approved non-factor therapy is the bispecific, FVIII-mimicking antibody, emicizumab (Hemlibra®), which came available in the Netherlands in July 2018. Emicizumab is a humanized, bispecific antibody connecting factor IX and factor X enabling the activation of FX and subsequent thrombin generation. Emicizumab has shown to be highly effective prophylaxis in PwHA by achieving a complete eradication of treated bleeds in around 80% of PwHA (n = 374) during the second 24-week interval of treatment. Furter advantages of emicizumab are the subcutaneous administration and less frequent dosing intervals every 1, 2 or 4 weeks due to a long half-life (t ½: 28 days). Despite many PwHA are candidate for prophylaxis with emicizumab, cost limit widespread access.

Currently, emicizumab is approved by F. Hoffmann-La Roche® with a loading dose of 3 mg/kg/week for four weeks and a maintenance dose of 1.5 mg/kg/week, 3 mg/kg/2 weeks or 6 mg/kg/4 weeks. These dose regimens were based on a pharmacometric approach instead of a dose finding study, and targeted a trough concentration (Ctrough) of 45 µg/ml by using pharmacokinetic (PK)simulations. Meanwhile long-term bleed data from the phase III and IV studies by the pharmaceutical company were included in pharmacokinetic (PK) and pharmacodynamic (PD) modelling studies, and the effective Ctrough was suggested at 30 µg/ml.

Although this Ctrough of 30 µg/ml is substantially lower than the previous Ctrough (45 µg/ml), the dose regimens were not adjusted. Conventional dosing leads to mean concentrations of 55 µg/ml with two thirds of the observations between 40 and 70 µg/ml (i.e., SD of ±15 µg/ml). Emicizumab has been approved based on fixed body-weight-based dosing and therefore the concentration target might have been kept higher to avoid lower effectivity due to inter-patient variability. However, reduced dosing of emicizumab, either by extending the dosing interval or lowering the dose, without sacrificing its efficacy has been reported in small case series.

Therefore, the investigators hypothesized that lower dosing of emicizumab targeted at Ctrough 30 μg/mL, is equally as effective and less costly in preventing bleeds as conventional dosing of emicizumab, and designed the DosEmi study to investigate the hypothesis in a large prospective cohort of adult and paediatric PwHA.

Conditions

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Hemophilia A With Inhibitor Hemophilia A Without Inhibitor Hemophilia A, Severe Adolescent Child Adult

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

CROSSOVER

* PK-guided dosing - Intervention group (12M): Subjects with emicizumab concentration of ≥ 40 μg/mL will receive individualized PK-guided dose reduction of emicizumab targeted at a Ctrough of 30μg/mL. The validated population PK model is based on published population PK and PK/PD modelling studies. (9,10,15)
* PK-Guided dosing - Non-intervention group (12M): Subjects with emicizumab concentration of 25-39 μg/mL will continue on their current dose regimen and will be followed according to the same assessment schedule as the Intervention Group. Only subjects with emicizumab plasma concentration \< 25 μg/mL will be adjusted in dosing regimen according to local protocol. These subjects will be followed for selective safety data only.
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Conventional dosing - open label

Patients will be followed 6 months retrospectively and 6 months prospectively on conventional dosing.

Group Type OTHER

Emicizumab - PK-guided dose reduction

Intervention Type OTHER

PK-guided dose reduction emicizumab targeted at a Ctrough of 30μg/mL.

Emicizumab - Dosis continuation group

Intervention Type OTHER

Continue on their current dose regimen

Emicizumab - Dose adjustment group

Intervention Type OTHER

Adjusted in dosing regimen according to local protocol

PK-guided dosing - open label

Patients with emicizumab concentration of ≥ 40 μg/mL will receive individualized PK-guided dose reduction of emicizumab targeted at a Ctrough of 30μg/mL. Patients will be followed for 12 months on reduced dosing.

Group Type OTHER

Emicizumab - PK-guided dose reduction

Intervention Type OTHER

PK-guided dose reduction emicizumab targeted at a Ctrough of 30μg/mL.

No intervention continuation - open label

Patients with emicizumab concentration of 25-39 μg/mL will continue on their current dose regimen. Patients will be followed for 12 months on current dosing.

Group Type OTHER

Emicizumab - Dosis continuation group

Intervention Type OTHER

Continue on their current dose regimen

No intervention adjusted - open label

Patients with emicizumab plasma concentration \< 25 μg/mL will be adjusted in dosing regimen according to local protocol. Patients will be followed for selective safety data only.

Group Type OTHER

Emicizumab - Dose adjustment group

Intervention Type OTHER

Adjusted in dosing regimen according to local protocol

Interventions

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Emicizumab - PK-guided dose reduction

PK-guided dose reduction emicizumab targeted at a Ctrough of 30μg/mL.

Intervention Type OTHER

Emicizumab - Dosis continuation group

Continue on their current dose regimen

Intervention Type OTHER

Emicizumab - Dose adjustment group

Adjusted in dosing regimen according to local protocol

Intervention Type OTHER

Other Intervention Names

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Hemlibra Hemlibra Hemlibra

Eligibility Criteria

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Inclusion Criteria

* Confirmed diagnosis of congenital haemophilia A, with a baseline endogenous FVIII of \<6 IU/ml
* Aged \> 1 year at inclusion (inclusion of children 1-16 years after favourable interim-analysis see protocol)
* Receiving conventional dosing of emicizumab (6 mg/kg/4 weeks with varying intervals) for a duration of at least 12 months prior to inclusion;
* Having good bleeding control, defined as:

i No spontaneous joint/muscle bleeds in the previous 6 months AND ii A maximum of two treated (traumatic) bleeds in the previous 6 months.

* Willing and able to provide written informed consent, either by the subject or its parents/legal guardian
* Willing to provide bleeding assessment information
* Willing to adhere to the medication regimen

Exclusion Criteria

* Acquired haemophilia A
Minimum Eligible Age

1 Year

Eligible Sex

MALE

Accepts Healthy Volunteers

No

Sponsors

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Erasmus Medical Center

OTHER

Sponsor Role collaborator

Amsterdam University Medical Center

OTHER

Sponsor Role collaborator

Leiden University Medical Center

OTHER

Sponsor Role collaborator

Radboud University Medical Center

OTHER

Sponsor Role collaborator

Maastricht University Medical Center

OTHER

Sponsor Role collaborator

University Medical Center Groningen

OTHER

Sponsor Role collaborator

HagaZiekenhuis

OTHER

Sponsor Role collaborator

Dutch Society of Haemophilia Patients

UNKNOWN

Sponsor Role collaborator

Kathelijn Fischer

OTHER

Sponsor Role lead

Responsible Party

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Kathelijn Fischer

Principal Investigator

Responsibility Role SPONSOR_INVESTIGATOR

Principal Investigators

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Study Officials Fischer, Dr, MD

Role: PRINCIPAL_INVESTIGATOR

UMC Utrecht

Locations

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Radboud University Medical Center

Nijmegen, Gelderland, Netherlands

Site Status RECRUITING

Maastricht University Medical Center

Maastricht, Limburg, Netherlands

Site Status RECRUITING

Amsterdam University Medical Center

Amsterdam, North Holland, Netherlands

Site Status RECRUITING

Leids Universitair Medisch Centrum

Leiden, South Holland, Netherlands

Site Status RECRUITING

Erasmus University Medical Center

Rotterdam, South Holland, Netherlands

Site Status RECRUITING

HagaZiekenhuis

The Hague, South Holland, Netherlands

Site Status RECRUITING

University Medical Center Groningen

Groningen, , Netherlands

Site Status RECRUITING

University Medical Center Utrecht

Utrecht, , Netherlands

Site Status RECRUITING

Countries

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Netherlands

Central Contacts

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Kathelijn Fischer, Dr, MD.

Role: CONTACT

+318 875 584 50

Konrad VD van der Zwet, MD

Role: CONTACT

+31650124691

Facility Contacts

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Saskia Schols, Dr, MD

Role: primary

+310 24 361 8823

Floor Moenen, Dr, MD

Role: primary

+31433876543

Michiel Coppens, Dr, MD

Role: primary

+31(0)20 566 5964

Paul den Exter, Dr, MD

Role: primary

+31 (0)71 526 1850

Marjon Cnossen, Dr., MD

Role: primary

+31107040113

Paula Ypma, MD

Role: primary

+310702102620

Louise Hooimeijer, MD

Role: primary

+310-503612740

Kathelijn Fischer, Dr, MD

Role: primary

+31887558450

Konrad van der Zwet, MD

Role: backup

+31650124691

References

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Donners A, van der Zwet K, Egberts ACG, Fijnvandraat K, Mathot R, Kruis I, Cnossen MH, Schutgens R, Urbanus RT, Fischer K. DosEmi study protocol: a phase IV, multicentre, open-label, crossover study to evaluate non-inferiority of pharmacokinetic-guided reduced dosing compared with conventional dosing of emicizumab in people with haemophilia A. BMJ Open. 2023 Jun 26;13(6):e072363. doi: 10.1136/bmjopen-2023-072363.

Reference Type BACKGROUND
PMID: 37369395 (View on PubMed)

Berntorp E, Fischer K, Hart DP, Mancuso ME, Stephensen D, Shapiro AD, Blanchette V. Haemophilia. Nat Rev Dis Primers. 2021 Jun 24;7(1):45. doi: 10.1038/s41572-021-00278-x.

Reference Type BACKGROUND
PMID: 34168126 (View on PubMed)

Blanchette VS, Key NS, Ljung LR, Manco-Johnson MJ, van den Berg HM, Srivastava A; Subcommittee on Factor VIII, Factor IX and Rare Coagulation Disorders of the Scientific and Standardization Committee of the International Society on Thrombosis and Hemostasis. Definitions in hemophilia: communication from the SSC of the ISTH. J Thromb Haemost. 2014 Nov;12(11):1935-9. doi: 10.1111/jth.12672. Epub 2014 Sep 3. No abstract available.

Reference Type BACKGROUND
PMID: 25059285 (View on PubMed)

Srivastava A, Santagostino E, Dougall A, Kitchen S, Sutherland M, Pipe SW, Carcao M, Mahlangu J, Ragni MV, Windyga J, Llinas A, Goddard NJ, Mohan R, Poonnoose PM, Feldman BM, Lewis SZ, van den Berg HM, Pierce GF; WFH Guidelines for the Management of Hemophilia panelists and co-authors. WFH Guidelines for the Management of Hemophilia, 3rd edition. Haemophilia. 2020 Aug;26 Suppl 6:1-158. doi: 10.1111/hae.14046. Epub 2020 Aug 3. No abstract available.

Reference Type BACKGROUND
PMID: 32744769 (View on PubMed)

Callaghan MU, Negrier C, Paz-Priel I, Chang T, Chebon S, Lehle M, Mahlangu J, Young G, Kruse-Jarres R, Mancuso ME, Niggli M, Howard M, Bienz NS, Shima M, Jimenez-Yuste V, Schmitt C, Asikanius E, Levy GG, Pipe SW, Oldenburg J. Long-term outcomes with emicizumab prophylaxis for hemophilia A with or without FVIII inhibitors from the HAVEN 1-4 studies. Blood. 2021 Apr 22;137(16):2231-2242. doi: 10.1182/blood.2020009217.

Reference Type BACKGROUND
PMID: 33512413 (View on PubMed)

Yoneyama K, Schmitt C, Kotani N, Levy GG, Kasai R, Iida S, Shima M, Kawanishi T. A Pharmacometric Approach to Substitute for a Conventional Dose-Finding Study in Rare Diseases: Example of Phase III Dose Selection for Emicizumab in Hemophilia A. Clin Pharmacokinet. 2018 Sep;57(9):1123-1134. doi: 10.1007/s40262-017-0616-3.

Reference Type BACKGROUND
PMID: 29214439 (View on PubMed)

Retout S, Schmitt C, Petry C, Mercier F, Frey N. Population Pharmacokinetic Analysis and Exploratory Exposure-Bleeding Rate Relationship of Emicizumab in Adult and Pediatric Persons with Hemophilia A. Clin Pharmacokinet. 2020 Dec;59(12):1611-1625. doi: 10.1007/s40262-020-00904-z.

Reference Type BACKGROUND
PMID: 32504271 (View on PubMed)

Jonsson F, Schmitt C, Petry C, Mercier F, Frey N, Retout S. Exposure-Bleeding Count Modeling of Emicizumab for the Prophylaxis of Bleeding in Persons with Hemophilia A with/Without Inhibitors Against Factor VIII. Clin Pharmacokinet. 2021 Jul;60(7):931-941. doi: 10.1007/s40262-021-01006-0. Epub 2021 Mar 12.

Reference Type BACKGROUND
PMID: 33709296 (View on PubMed)

Donners AAMT, Rademaker CMA, Bevers LAH, Huitema ADR, Schutgens REG, Egberts TCG, Fischer K. Pharmacokinetics and Associated Efficacy of Emicizumab in Humans: A Systematic Review. Clin Pharmacokinet. 2021 Nov;60(11):1395-1406. doi: 10.1007/s40262-021-01042-w. Epub 2021 Aug 13.

Reference Type BACKGROUND
PMID: 34389928 (View on PubMed)

Lehtinen AE, Lassila R. Do we need all that emicizumab? Haemophilia. 2022 Mar;28(2):e53-e55. doi: 10.1111/hae.14483. Epub 2021 Dec 30. No abstract available.

Reference Type BACKGROUND
PMID: 34970820 (View on PubMed)

Chuansumrit A, Sirachainan N, Jaovisidha S, Jiravichitchai T, Kadegasem P, Kempka K, Panuwannakorn M, Rotchanapanya W, Nuntiyakul T. Effectiveness of monthly low dose emicizumab prophylaxis without 4-week loading doses among patients with haemophilia A with and without inhibitors: A case series report. Haemophilia. 2023 Jan;29(1):382-385. doi: 10.1111/hae.14707. Epub 2022 Nov 29. No abstract available.

Reference Type BACKGROUND
PMID: 36446746 (View on PubMed)

Bansal S, Donners AAMT, Fischer K, Kshirsagar S, Rangarajan S, Phadke V, Mhatre S, Sontate B, Silva M, Ansari S, Shetty S. Low dose emicizumab prophylaxis in haemophilia a patients: A pilot study from India. Haemophilia. 2023 May;29(3):931-934. doi: 10.1111/hae.14785. Epub 2023 Apr 8. No abstract available.

Reference Type BACKGROUND
PMID: 37029771 (View on PubMed)

Study Documents

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Document Type: Study Protocol

Published study protocol

View Document

Other Identifiers

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22-571

Identifier Type: -

Identifier Source: org_study_id

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