Evaluation of Oral Tofacitinib in Children Aged 2 to 17 Years Old Suffering From Moderate to Severe Ulcerative Colitis

NCT ID: NCT04624230

Last Updated: 2025-10-24

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE3

Total Enrollment

120 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-08-12

Study Completion Date

2029-05-15

Brief Summary

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This study, A3921210 is designed to evaluate the efficacy, safety and pharmacokinetics (PK) of tofacitinib in pediatric participants with moderately to severely active UC. In the US and EU, patients with prior TNFi failure or intolerance will be enrolled. Outside of the US or EU, patients having had inadequate response or intolerance to oral or IV corticosteroids or azathioprine or 6-mercaptopurine or TNFi will be enrolled.

All eligible participants will initially receive open label tofacitinib at a dose expected to produce equivalent systemic exposure to that observed in adults receiving 5 mg BID with the option for individual dose increase to 10 mg BID adult dose equivalent if dose escalation criteria are met.

The primary objective of this study is to evaluate the efficacy of tofacitinib based on remission in pediatric participants with moderately to severely active UC. The primary endpoint is remission by central read Mayo score following 44 weeks in the maintenance phase. Remission is defined by a Mayo score of 2 points or lower, with no individual subscore exceeding 1 point and a rectal bleeding subscore of 0.

The study Design is an open-label Phase 3 study that includes a screening period of up to 4-weeks duration, an 8-week or 16-week induction phase, a 44-week maintenance phase, and a 24-month extension phase for pediatric participants with moderately to severely active UC. Participants will have a follow-up visit 4 weeks after the last dose of study intervention and a telephone contact 8 weeks later to assess for any adverse events (AEs)/serious adverse events (SAEs). The total maximum duration of this study will be up to 180 weeks.

Detailed Description

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Conditions

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Ulcerative Colitis

Study Design

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Allocation Method

NA

Intervention Model

SEQUENTIAL

Single Group
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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tofacitinib

Open label tofacitinib 5 mg BID weight based adult equivalent with the option for individual dose increase to 10 mg BID weight based adult equivalent for a limited time if dose escalation criteria are met, prior to returning to 5 mg BID.

Group Type EXPERIMENTAL

tofacitinib

Intervention Type DRUG

Open label tofacitinib 5 mg BID weight based adult equivalent with the option for individual dose increase to 10 mg BID weight based adult equivalent for a limited time if dose escalation criteria are met, prior to returning to 5 mg BID.

Interventions

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tofacitinib

Open label tofacitinib 5 mg BID weight based adult equivalent with the option for individual dose increase to 10 mg BID weight based adult equivalent for a limited time if dose escalation criteria are met, prior to returning to 5 mg BID.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Evidence of a personally signed and dated informed consent document and assent document.
* Males and females 2 to less than18 years old and weighing at least 10 kg.
* Having a pathology report that confirms colonic inflammation consistent with UC with a clinical diagnosis of UC for at least 12 weeks prior to baseline, with biopsy report supporting the diagnosis of UC.
* Participants diagnosed with UC at age less than 6 years old, must have had testing and be negative for monogenic disorders associated with very early onset IBD.
* Moderately to severely active UC as defined (via screening colonoscopy) by a Mayo score of at least 6, with a rectal bleeding score of at least 1 and an endoscopic subscore of at least 2.
* Pediatric Ulcerative Colitis Activity Index (PUCAI) score greater or equal to 35 .
* No history of dysplasia or colon cancer.
* No evidence or history of untreated or inadequately treated active or latent infection with Mycobacterium Tuberculosis.
* For participants outside of the United States or the European Union: have had an inadequate response or been intolerant to at least one prior therapy as listed below or have a medical contraindication to such therapies:

* Oral or intravenous (IV) corticosteroids;
* Azathioprine or 6-mercaptopurine;
* TNF inhibitors or anti integrin therapy.
* For participants in the United States and the European Union: have had an inadequate response or intolerance to TNF inhibitors.
* Stable doses of the following therapies for UC:

* Oral 5 Aminosalicyclic acids (ASA) or sulfasalazine
* Oral corticosteroids equivalent to prednisone at most 1 mg/kg up to a maximum of 20 mg/day or budesonide up to 9 mg/day.
* female participant is eligible if she is not pregnant or breastfeeding, If she is a woman of child bearing potential, she needs to be using a contraceptive method that is highly effective (with a failure rate of \<1% per year).

Exclusion Criteria

* Diagnosis of indeterminate colitis, isolated proctitis, microscopic colitis, infectious colitis, Crohn's disease, or clinical findings suggestive of Crohn's disease.
* History of symptomatic obstructive intestinal strictures or active ostomy, or history of colectomy, extensive small bowel resection ( greater than100 centimetres) or short bowel syndrome, or hospitalization for UC related reason(s) within 2 weeks of baseline visit.
* Any factors or clinical characteristics potentially related to the risk of venous thromboembolism that may increase the risk associated with study participation or study intervention administration or may interfere with the interpretation of study results and, in the judgment of the investigator, would make the participant inappropriate for entry into this study.
* Participants who have previously received tofacitinib or another Janus Kinase inhibitor.
* Vaccination or exposure to a live or attenuated vaccine within the 6 weeks prior to the first dose of study drug, or who are expected to be vaccinated or to have household exposure to these vaccines during treatment or during the 6 weeks following discontinuation of study drug.
* Participants having received azathioprine, 6-mercaptopurine, methotrexate, thioguanine, infliximab, adalimumab, golimumab, ustekinumab, interferon, cyclosporine, mycophenolate, tacrolimus, IV or rectally administered corticosteroids, natalizumab, vedolizumab, other antiadhesion molecules, or investigational drugs during the specified time periods prior to baseline whereby they may still have pharmacokinetic and/or pharmacodynamic effect in the body of the participant.
* Previous treatment by leukocyte apheresis including selective lymphocyte, monocyte, or granulocyte apheresis, or plasma exchange within 6 months prior to baseline.
* Treatment by specified prohibited concomitant medications, including moderate to potent CYP3A inducers or inhibitors in the specified time periods prior to the first dose of study drug or are expected to receive any of these medications during the study period.
* Chronic and frequent use of antimotility agents for control of diarrhea (ie, diphenoxylate hydrochloride with atropine sulfate or loperamide).
* History of bowel surgery, including cholecystectomy within 6 months prior to baseline, history of appendectomy within 3 months prior to baseline, or significant trauma or major surgery within 4 weeks of screening visit are excluded.
* Participants with the following laboratory values at screening:

* Hemoglobin level lower than 9.0 g/Dl.
* Absolute white blood cell (WBC) count lower than 3000/mm3.
* Absolute neutrophil count lower than 1200/mm3.
* Absolute lymphocyte count lower than 750/mm3.
* Thrombocytopenia as defined by a platelet count lower than 100,000/mm3.
* Estimated bedside Schwartz Glomerular filtration rate (GFR) lower or equal to 40 mL/min/1.73 m2.
* Total bilirubin, aspartate aminostransferase (AST) or alanine aminotransferase (ALT) more than 1.5 times the upper limit of normal.
* Positive stool examinations for enteric pathogens, pathogenic ova or parasites, or C. difficile toxin at screening.
* Participants infected with human immunodeficiency virus (HIV) or hepatitis B or C viruses.
* History of more than one episode of HZ, a history of disseminated HZ or disseminated herpes simplex.
* History or current symptoms of any lymphoproliferative disorder (eg, Epstein Barr Virus (EBV) related lymphoproliferative disorder, lymphoma, leukemia, myeloproliferative disorders, multiple myeloma, or signs and symptoms suggestive of currently lymphatic disease).
* Clinically significant infections currently or within 3 months prior to baseline (eg, those requiring hospitalization or parenteral antimicrobial therapy or opportunistic infections), a history of any infection requiring antimicrobial therapy within 2 weeks of baseline, or a history of any infection otherwise judged by the investigator to have the potential for exacerbation by participation in the study.
* Any malignancies or with a history of malignancies, with the exception of adequately treated or excised nonmetastatic basal cell or squamous cell cancer of the skin.
* Investigator site staff members directly involved in the conduct of the study and their family members, site staff members otherwise supervised by the investigator, or participants who are employees of the Sponsor, including their family members, directly involved in the conduct of the study.
* Participation in other studies involving investigational drug(s) within 2 months prior to study entry and/or during study participation.
* Other acute or chronic medical or psychiatric condition including recent (within the past year) or active suicidal ideation or behavior or laboratory abnormality that may increase the risk associated with study participation or study intervention administration or may interfere with the interpretation of study results and, in the judgment of the investigator, would make the participant inappropriate for entry into this study.
* Pregnant female participants; breastfeeding female participants; fertile female participants of childbearing potential who are unwilling or unable to use a highly effective method of contraception as outlined in this protocol for the duration of the study and through the telephone follow up visit.
* History of allergies, intolerance or hypersensitivity to lactose or tofacitinib, or any other excipients of the investigational medicinal products, including placebos.
Minimum Eligible Age

2 Years

Maximum Eligible Age

17 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Children's Hospital Los Angeles

Los Angeles, California, United States

Site Status RECRUITING

University of California, San Francisco Benioff Children's Hospital

San Francisco, California, United States

Site Status RECRUITING

University of California, San Francisco Pediatric Clinical Research Center (PCRC)

San Francisco, California, United States

Site Status RECRUITING

Connecticut Children's Ambulatory Surgical Center

Farmington, Connecticut, United States

Site Status ACTIVE_NOT_RECRUITING

Connecticut Children's Infusion Center

Farmington, Connecticut, United States

Site Status ACTIVE_NOT_RECRUITING

Connecticut Children's Medical Center

Hartford, Connecticut, United States

Site Status ACTIVE_NOT_RECRUITING

Nicklaus Children's Hospital

Miami, Florida, United States

Site Status RECRUITING

Center for Advanced Pediatrics

Atlanta, Georgia, United States

Site Status RECRUITING

Children's Healthcare of Atlanta - Arthur M. Blank Hospital

Atlanta, Georgia, United States

Site Status RECRUITING

Boston Children's Hospital

Boston, Massachusetts, United States

Site Status RECRUITING

Atlantic Children's Health-Pediatric Gastroenterology & Nutrition

Morristown, New Jersey, United States

Site Status RECRUITING

Goryeb Children's Hospital (Endoscopy only)

Morristown, New Jersey, United States

Site Status RECRUITING

Atlantic Health System- Morristown Medical Center (Pharmacy)

Morristown, New Jersey, United States

Site Status RECRUITING

Northwell Health - Cohen Children's Medical Center

Lake Success, New York, United States

Site Status ACTIVE_NOT_RECRUITING

Northwell Health - Cohen Children's Medical Center

New Hyde Park, New York, United States

Site Status ACTIVE_NOT_RECRUITING

Columbia University Irving Medical Center

New York, New York, United States

Site Status RECRUITING

CUIMC Research Pharmacy - Milstein Hospital (Pharmacy Only)

New York, New York, United States

Site Status RECRUITING

Morgan Stanley Children's Hospital, CUIMC

New York, New York, United States

Site Status RECRUITING

Cincinnati Children's Hospital Medical Center

Cincinnati, Ohio, United States

Site Status RECRUITING

Buerger Center for Advanced Pediatric Care

Philadelphia, Pennsylvania, United States

Site Status ACTIVE_NOT_RECRUITING

Children's Hospital of Philadelphia

Philadelphia, Pennsylvania, United States

Site Status ACTIVE_NOT_RECRUITING

Roberts Center for Pediatric Research

Philadelphia, Pennsylvania, United States

Site Status ACTIVE_NOT_RECRUITING

Texas Children's Hospital

Houston, Texas, United States

Site Status RECRUITING

Seattle Children's Hospital

Seattle, Washington, United States

Site Status RECRUITING

The Royal Children's Hospital

Parkville, Victoria, Australia

Site Status ACTIVE_NOT_RECRUITING

Universitaire Ziekenhuizen Leuven

Leuven, Vlaams Brabant, Belgium

Site Status RECRUITING

Hôpital Universitaire Des Enfants Reine Fabiola

Brussels, , Belgium

Site Status RECRUITING

Universitair Ziekenhuis Brussel

Brussels, , Belgium

Site Status RECRUITING

Cliniques Universitaires Saint-Luc

Brussels, , Belgium

Site Status RECRUITING

Stollery Children's Hospital University of Alberta

Edmonton, Alberta, Canada

Site Status RECRUITING

British Columbia Children's Hospital

Vancouver, British Columbia, Canada

Site Status RECRUITING

IWK Health Centre

Halifax, Nova Scotia, Canada

Site Status RECRUITING

London Health Sciences Centre - Children's Hospital

London, Ontario, Canada

Site Status RECRUITING

The Hospital for Sick Children - Division of Gastroenterology, Hepatology and Nutrition

Toronto, Ontario, Canada

Site Status ACTIVE_NOT_RECRUITING

CHU Sainte-Justine

Montreal, Quebec, Canada

Site Status RECRUITING

Tampereen yliopistollinen sairaala

Tampere, , Finland

Site Status RECRUITING

CHU de Lyon - Hôpital Femme Mère Enfant

Bron, , France

Site Status RECRUITING

Hôpital Necker Enfants Malades

Paris, , France

Site Status RECRUITING

Dr. von Haunersches Kinderspital, LMU

Munich, Bavaria, Germany

Site Status RECRUITING

Debreceni Egyetem Klinikai Kozpont

Debrecen, Hajdú-Bihar, Hungary

Site Status RECRUITING

Szegedi Tudomanyegyetem Szent-Gyorgyi Albert Klinikai Kozpont

Szeged, , Hungary

Site Status RECRUITING

Shamir Medical Center (Assaf Harofeh)

Be’er Ya‘aqov, , Israel

Site Status RECRUITING

Lady Davis Carmel Medical Center

Haifa, , Israel

Site Status RECRUITING

Shaare Zedek Medical Center

Jerusalem, , Israel

Site Status RECRUITING

Schneider Children's Medical Center of Israel

Petah Tikva, , Israel

Site Status RECRUITING

Tel-Aviv Sourasky Medical Center

Tel Aviv, , Israel

Site Status RECRUITING

ASST Papa Giovanni XXIII Epatologia e Gastroenterologia Pediatrica e dei Trapianti

Bergamo, BG, Italy

Site Status RECRUITING

A.O.U. Federico II

Napoli, Naples, Italy

Site Status RECRUITING

Azienda Ospedaliero - Universitaria Policlinico Umberto I di Roma

Roma, RM, Italy

Site Status RECRUITING

Azienda USL di Bologna - IRCCS ISNB - Programma Gastroenterologia Pediatrica

Bologna, , Italy

Site Status ACTIVE_NOT_RECRUITING

Aichi Children's Health and Medical Center

Obu-shi, Aichi-ken, Japan

Site Status RECRUITING

Kurume University Hospital

Kurume-shi, Fukuoka, Japan

Site Status RECRUITING

Gunma University Hospital

Maebashi, Gunma, Japan

Site Status RECRUITING

Miyagi Children's Hospital

Sendai, Miyagi, Japan

Site Status RECRUITING

Osaka Women's and Children's Hospital

Izumi, Osaka, Japan

Site Status RECRUITING

Osaka Medical and Pharmaceutical University Hospital

Takatsuki-shi, Osaka, Japan

Site Status RECRUITING

Saitama Prefectural Children's Medical Center

Saitama-shi, Saitama, Japan

Site Status RECRUITING

Jichi Medical University Hospital

Shimotsuke, Tochigi, Japan

Site Status RECRUITING

Juntendo University Hospital

Bunkyo-ku, Tokyo, Japan

Site Status RECRUITING

National Center for Child Health and Development

Setagaya-ku, Tokyo, Japan

Site Status RECRUITING

Amsterdam UMC location AMC

Amsterdam, North Holland, Netherlands

Site Status RECRUITING

Amsterdam UMC, location VUmc Boelelaan

Amsterdam, , Netherlands

Site Status RECRUITING

Erasmus Medical Center - Sophia Children's Hospital

Rotterdam, , Netherlands

Site Status RECRUITING

Medical Network Spółka z o.o. WIP Warsaw IBD Point Profesor Kierkuś

Warsaw, Masovian Voivodeship, Poland

Site Status RECRUITING

Instytut "Centrum Zdrowia Matki Polki"

Lodz, , Poland

Site Status RECRUITING

Korczowski Bartosz, Gabinet Lekarski

Rzeszów, , Poland

Site Status RECRUITING

Instytut "Pomnik - Centrum Zdrowia Dziecka"

Warsaw, , Poland

Site Status RECRUITING

Uniwersytecki Szpital Kliniczny im. Jana Mikulicza-Radeckiego we Wroclawiu

Wroclaw, , Poland

Site Status RECRUITING

Narodny ustav detskych chorob

Bratislava, , Slovakia

Site Status ACTIVE_NOT_RECRUITING

Hospital Infantil Universitario Niño Jesus

Madrid, , Spain

Site Status RECRUITING

Sahlgrenska Universitetssjukhuset

Gothenburg, , Sweden

Site Status RECRUITING

Sachsska Children's and Youth Hospital/South General Hospital

Stockholm, , Sweden

Site Status RECRUITING

Karolinska Universitetssjukhuset Barngastroenterologi, hepatologi och nutrition

Stockholm, , Sweden

Site Status RECRUITING

King's College Hospital NHS Foundation Trust

London, Greater London, United Kingdom

Site Status RECRUITING

Birmingham Women's and Children's NHS Foundation Trust

Birmingham, WEST Midlands, United Kingdom

Site Status RECRUITING

NHS Lothian

Edinburgh, , United Kingdom

Site Status RECRUITING

Bart's Health NHS Trust

London, , United Kingdom

Site Status RECRUITING

Countries

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United States Australia Belgium Canada Finland France Germany Hungary Israel Italy Japan Netherlands Poland Slovakia Spain Sweden United Kingdom

Central Contacts

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Pfizer CT.gov Call Center

Role: CONTACT

1-800-718-1021

References

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Benchimol EI, Bernstein CN, Bitton A, Carroll MW, Singh H, Otley AR, Vutcovici M, El-Matary W, Nguyen GC, Griffiths AM, Mack DR, Jacobson K, Mojaverian N, Tanyingoh D, Cui Y, Nugent ZJ, Coulombe J, Targownik LE, Jones JL, Leddin D, Murthy SK, Kaplan GG. Trends in Epidemiology of Pediatric Inflammatory Bowel Disease in Canada: Distributed Network Analysis of Multiple Population-Based Provincial Health Administrative Databases. Am J Gastroenterol. 2017 Jul;112(7):1120-1134. doi: 10.1038/ajg.2017.97. Epub 2017 Apr 18.

Reference Type RESULT
PMID: 28417994 (View on PubMed)

Konstantinides SV, Meyer G, Becattini C, Bueno H, Geersing GJ, Harjola VP, Huisman MV, Humbert M, Jennings CS, Jimenez D, Kucher N, Lang IM, Lankeit M, Lorusso R, Mazzolai L, Meneveau N, Ni Ainle F, Prandoni P, Pruszczyk P, Righini M, Torbicki A, Van Belle E, Zamorano JL; ESC Scientific Document Group. 2019 ESC Guidelines for the diagnosis and management of acute pulmonary embolism developed in collaboration with the European Respiratory Society (ERS). Eur Heart J. 2020 Jan 21;41(4):543-603. doi: 10.1093/eurheartj/ehz405. No abstract available.

Reference Type RESULT
PMID: 31504429 (View on PubMed)

Kelsen JR, Sullivan KE, Rabizadeh S, Singh N, Snapper S, Elkadri A, Grossman AB. North American Society for Pediatric Gastroenterology, Hepatology, and Nutrition Position Paper on the Evaluation and Management for Patients With Very Early-onset Inflammatory Bowel Disease. J Pediatr Gastroenterol Nutr. 2020 Mar;70(3):389-403. doi: 10.1097/MPG.0000000000002567.

Reference Type RESULT
PMID: 32079889 (View on PubMed)

Turner D, Otley AR, Mack D, Hyams J, de Bruijne J, Uusoue K, Walters TD, Zachos M, Mamula P, Beaton DE, Steinhart AH, Griffiths AM. Development, validation, and evaluation of a pediatric ulcerative colitis activity index: a prospective multicenter study. Gastroenterology. 2007 Aug;133(2):423-32. doi: 10.1053/j.gastro.2007.05.029. Epub 2007 May 21.

Reference Type RESULT
PMID: 17681163 (View on PubMed)

Otley A, Smith C, Nicholas D, Munk M, Avolio J, Sherman PM, Griffiths AM. The IMPACT questionnaire: a valid measure of health-related quality of life in pediatric inflammatory bowel disease. J Pediatr Gastroenterol Nutr. 2002 Oct;35(4):557-63. doi: 10.1097/00005176-200210000-00018.

Reference Type RESULT
PMID: 12394384 (View on PubMed)

Marcovitch L, Nissan A, Mack D, Otley A, Hussey S, Mclean B, Lewis M, Croft N, Barakat FM, Griffiths AM, Turner D. Item Generation and Reduction Toward Developing a Patient-reported Outcome for Pediatric Ulcerative Colitis (TUMMY-UC). J Pediatr Gastroenterol Nutr. 2017 Mar;64(3):373-377. doi: 10.1097/MPG.0000000000001259.

Reference Type RESULT
PMID: 27159210 (View on PubMed)

Taylor SJ, Whincup PH, Hindmarsh PC, Lampe F, Odoki K, Cook DG. Performance of a new pubertal self-assessment questionnaire: a preliminary study. Paediatr Perinat Epidemiol. 2001 Jan;15(1):88-94. doi: 10.1046/j.1365-3016.2001.00317.x.

Reference Type RESULT
PMID: 11237120 (View on PubMed)

Related Links

Access external resources that provide additional context or updates about the study.

https://pmiform.com/clinical-trial-info-request?StudyID=A3921210

To obtain contact information for a study center near you, click here.

Other Identifiers

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OVATION

Identifier Type: OTHER

Identifier Source: secondary_id

2023-509694-22-00

Identifier Type: REGISTRY

Identifier Source: secondary_id

A3921210

Identifier Type: -

Identifier Source: org_study_id

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