A Study Measuring the Effectiveness, Safety, and Tolerability of BMS-986278 in Participants With Lung Fibrosis

NCT ID: NCT04308681

Last Updated: 2025-02-24

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

403 participants

Study Classification

INTERVENTIONAL

Study Start Date

2020-07-29

Study Completion Date

2023-09-22

Brief Summary

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The purpose of this study is to provide an initial evaluation of the effectiveness of BMS-986278 in participants with lung fibrosis, to demonstrate the safety of BMS-986278, and provide information on the drug levels of BMS-986278 in these participants.

Detailed Description

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Conditions

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Pulmonary Fibrosis

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Caregivers Investigators

Study Groups

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IPF Dose 1 + Post Treatment Follow-up or OTE

IPF (Idiopathic Pulmonary Fibrosis) OTE (Optional Treatment Extension)

Group Type EXPERIMENTAL

BMS-986278

Intervention Type DRUG

Specified Dose on Specified Days

IPF Dose 2 + Post Treatment Follow-up or OTE

Group Type EXPERIMENTAL

BMS-986278

Intervention Type DRUG

Specified Dose on Specified Days

IPF Placebo + Post Treatment Follow-up or OTE

Group Type PLACEBO_COMPARATOR

BMS-986278 Placebo

Intervention Type OTHER

Specified Dose on Specified Days

PF-ILD Dose 1 + Post Treatment Follow-up or OTE

PF-ILD (Progressive Fibrotic Interstitial Lung Disease)

Group Type EXPERIMENTAL

BMS-986278

Intervention Type DRUG

Specified Dose on Specified Days

PF-ILD Dose 2 + Post Treatment Follow-up or OTE

Group Type EXPERIMENTAL

BMS-986278

Intervention Type DRUG

Specified Dose on Specified Days

PF-ILD Placebo + Post Treatment Follow-up or OTE

Group Type PLACEBO_COMPARATOR

BMS-986278 Placebo

Intervention Type OTHER

Specified Dose on Specified Days

Interventions

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BMS-986278 Placebo

Specified Dose on Specified Days

Intervention Type OTHER

BMS-986278

Specified Dose on Specified Days

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

For the idiopathic pulmonary fibrosis (IPF) Cohort

* Diagnosis of IPF within 7 years of screening
* Female and males ≥ 40 years of age

For the progressive fibrotic interstitial lung disease (PF-ILD) Cohort

* Evidence of progressive ILD within the 24 months before screening
* Female and male ≥ 21 years of age.

Exclusion Criteria

* Women of childbearing potential (WOCBP)
* Active Smokers
* Current malignancy or previous malignancy up to 5 years prior to screening
* History of allergy to BMS-986278 or related compounds
Minimum Eligible Age

21 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Bristol-Myers Squibb

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Bristol-Myers Squibb

Role: STUDY_DIRECTOR

Bristol-Myers Squibb

Locations

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Local Institution - 0032

Birmingham, Alabama, United States

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Local Institution

Phoenix, Arizona, United States

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Local Institution - 0028

Los Angeles, California, United States

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Local Institution - 0043

Stanford, California, United States

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University of Colorado Anschutz Medical Campus-Department of Medicine

Aurora, Colorado, United States

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Local Institution - 0006

Denver, Colorado, United States

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Local Institution - 0171

New Haven, Connecticut, United States

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Local Institution - 0035

Gainesville, Florida, United States

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Local Institution - 0166

Orlando, Florida, United States

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Local Institution - 0078

Atlanta, Georgia, United States

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Local Institution - 0031

Kansas City, Kansas, United States

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Local Institution - 0154

Baltimore, Maryland, United States

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Local Institution - 0003

Boston, Massachusetts, United States

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Local Institution - 0030

Chesterfield, Missouri, United States

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Local Institution - 0036

St Louis, Missouri, United States

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Local Institution - 0029

Cincinnati, Ohio, United States

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Local Institution - 0164

Columbus, Ohio, United States

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Hershey, Pennsylvania, United States

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Nashville, Tennessee, United States

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Local Institution - 0096

Charlottesville, Virginia, United States

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Falls Church, Virginia, United States

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Local Institution - 0049

Buenos Aires, Distrito Federal, Argentina

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Local Institution - 0103

Rosario, Santa Fe Province, Argentina

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Local Institution - 0097

San Miguel de Tucumán, Tucumán Province, Argentina

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Local Institution - 0115

Buenos Aires, , Argentina

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Local Institution - 0048

Buenos Aires, , Argentina

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Local Institution - 0122

Mendoza, , Argentina

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Local Institution - 0045

Camperdown, New South Wales, Australia

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Local Institution - 0025

Westmead, New South Wales, Australia

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Local Institution - 0026

Brisbane, Queensland, Australia

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Local Institution - 0046

Greenslopes, Queensland, Australia

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Local Institution - 0022

Adelaide, South Australia, Australia

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Local Institution - 0023

Heidelberg, Victoria, Australia

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Local Institution - 0021

Murdoch, Western Australia, Australia

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Local Institution - 0044

Nedlands, Western Australia, Australia

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Local Institution - 0074

Brussels, , Belgium

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Local Institution - 0065

Leuven, , Belgium

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Local Institution - 0051

Liège, , Belgium

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Porto Alegre, Rio Grande do Sul, Brazil

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São Paulo, São Paulo, Brazil

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São Paulo, São Paulo, Brazil

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Local Institution - 0076

São Paulo, , Brazil

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Local Institution - 0141

Vancouver, British Columbia, Canada

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Vancouver, British Columbia, Canada

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Local Institution - 0134

Toronto, Ontario, Canada

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Local Institution - 0094

Montreal, Quebec, Canada

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Local Institution - 0127

Québec, Quebec, Canada

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Local Institution - 0144

Sherbrooke, Quebec, Canada

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Local Institution - 0108

Curicó, Maule Region, Chile

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Local Institution - 0054

Talca, Maule Region, Chile

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Local Institution - 0038

Quillota, Región de Valparaíso, Chile

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Local Institution - 0187

Beijing, Beijing Municipality, China

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Local Institution - 0183

Beijing, Beijing Municipality, China

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Local Institution - 0188

Wuhan, Hubei, China

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Local Institution - 0189

Shanghai, Shanghai Municipality, China

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Local Institution - 0120

Bobigny, , France

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Local Institution - 0066

Bron, , France

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Local Institution - 0136

Dijon, , France

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Local Institution - 0162

Marseille, , France

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Hopital Europeen Georges Pompidou

Paris, , France

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Local Institution - 0143

Paris, , France

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Local Institution - 0067

Rennes, , France

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Local Institution - 0132

Toulouse, , France

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Local Institution - 0111

Hanover, Lower Saxony, Germany

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Local Institution - 0107

Essen, , Germany

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Freiburg im Breisgau, , Germany

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Local Institution - 0093

Großhansdorf, , Germany

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Local Institution - 0110

Heidelberg, , Germany

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Local Institution - 0121

Munich, , Germany

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Local Institution - 0119

Stuttgart, , Germany

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Local Institution - 0145

Tel Aviv, Tel Aviv, Israel

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Local Institution - 0113

Haifa, , Israel

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Local Institution - 0149

Jerusalem, , Israel

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Local Institution - 0114

Petah Tikva, , Israel

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Ramat Gan, , Israel

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Local Institution - 0073

Catania, , Italy

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Modena, , Italy

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Local Institution - 0089

Monza, , Italy

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Roma, , Italy

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Local Institution - 0155

Seto, Aichi-ken, Japan

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Local Institution - 0106

Kōriyama, Fukushima, Japan

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Local Institution - 0180

Sapporo, Hokkaido, Japan

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Local Institution - 0095

Kobe, Hyōgo, Japan

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Local Institution - 0169

Kobe, Hyōgo, Japan

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Local Institution - 0071

Yokohama, Kanagawa, Japan

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Local Institution - 0112

Sakai, Osaka, Japan

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Local Institution - 0128

Izumo, Shimane, Japan

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Local Institution - 0064

Hamamatasu, Shizuoka, Japan

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Local Institution - 0080

Bunkyo-ku, Tokyo, Japan

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Local Institution - 0153

Minato-ku, Tokyo, Japan

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Local Institution - 0177

Shinjyuku-ku, Tokyo, Japan

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Local Institution - 0117

Kumamoto, , Japan

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Local Institution - 0146

Nagasaki, , Japan

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Local Institution - 0170

Saitama, , Japan

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Local Institution - 0173

Tokyo, , Japan

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Mexico City, Mexico City, Mexico

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Local Institution - 0081

Monterrey, Nuevo León, Mexico

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Local Institution - 0109

Monterrey, N.l., Nuevo León, Mexico

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Local Institution - 0083

San Nicolás de los Garza, Nuevo León, Mexico

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Local Institution - 0156

Oaxaca City, Oaxaca, Mexico

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Local Institution - 0087

Seoul, , South Korea

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Local Institution - 0086

Seoul, , South Korea

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Seoul, , South Korea

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Barcelona, , Spain

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Local Institution - 0116

Barcelona, , Spain

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Local Institution - 0140

L'Hospitalet de Llobregat, , Spain

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Madrid, , Spain

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Local Institution - 0137

Madrid, , Spain

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Marbella Málaga, , Spain

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Pozuelo de Alarcón, , Spain

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Santander, , Spain

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Local Institution - 0176

Kaohsiung City, , Taiwan

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Local Institution - 0174

Taipei, , Taiwan

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Local Institution - 0175

Taipei, , Taiwan

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Local Institution - 0050

Cambridge, , United Kingdom

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Local Institution - 0163

Edinburgh, , United Kingdom

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Local Institution - 0041

London, , United Kingdom

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Local Institution - 0092

London, , United Kingdom

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London, , United Kingdom

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Countries

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United States Argentina Australia Belgium Brazil Canada Chile China France Germany Israel Italy Japan Mexico South Korea Spain Taiwan United Kingdom

References

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Kreuter M, Maher TM, Wuyts WA, Valenzuela C, Hamblin M, Kim S, Patel A, Elpers B, Richeldi L. Effect of Admilparant, a Lysophosphatidic Acid Receptor 1 Antagonist, on Disease Progression in Pulmonary Fibrosis. Chest. 2025 Sep;168(3):677-687. doi: 10.1016/j.chest.2025.04.003. Epub 2025 Apr 8.

Reference Type DERIVED
PMID: 40210090 (View on PubMed)

Corte TJ, Behr J, Cottin V, Glassberg MK, Kreuter M, Martinez FJ, Ogura T, Suda T, Wijsenbeek M, Berkowitz E, Elpers B, Kim S, Watanabe H, Fischer A, Maher TM. Efficacy and Safety of Admilparant, an LPA1 Antagonist, in Pulmonary Fibrosis: A Phase 2 Randomized Clinical Trial. Am J Respir Crit Care Med. 2025 Feb;211(2):230-238. doi: 10.1164/rccm.202405-0977OC.

Reference Type DERIVED
PMID: 39393084 (View on PubMed)

Corte TJ, Lancaster L, Swigris JJ, Maher TM, Goldin JG, Palmer SM, Suda T, Ogura T, Minnich A, Zhan X, Tirucherai GS, Elpers B, Xiao H, Watanabe H, Smith RA, Charles ED, Fischer A. Phase 2 trial design of BMS-986278, a lysophosphatidic acid receptor 1 (LPA1) antagonist, in patients with idiopathic pulmonary fibrosis (IPF) or progressive fibrotic interstitial lung disease (PF-ILD). BMJ Open Respir Res. 2021 Dec;8(1):e001026. doi: 10.1136/bmjresp-2021-001026.

Reference Type DERIVED
PMID: 34969771 (View on PubMed)

Cheng PTW, Kaltenbach RF 3rd, Zhang H, Shi J, Tao S, Li J, Kennedy LJ, Walker SJ, Shi Y, Wang Y, Dhanusu S, Reddigunta R, Kumaravel S, Jusuf S, Smith D, Krishnananthan S, Li J, Wang T, Heiry R, Sum CS, Kalinowski SS, Hung CP, Chu CH, Azzara AV, Ziegler M, Burns L, Zinker BA, Boehm S, Taylor J, Sapuppo J, Mosure K, Everlof G, Guarino V, Zhang L, Yang Y, Ruan Q, Xu C, Apedo A, Traeger SC, Cvijic ME, Lentz KA, Tirucherai G, Sivaraman L, Robl J, Ellsworth BA, Rosen G, Gordon DA, Soars MG, Gill M, Murphy BJ. Discovery of an Oxycyclohexyl Acid Lysophosphatidic Acid Receptor 1 (LPA1) Antagonist BMS-986278 for the Treatment of Pulmonary Fibrotic Diseases. J Med Chem. 2021 Nov 11;64(21):15549-15581. doi: 10.1021/acs.jmedchem.1c01256. Epub 2021 Oct 28.

Reference Type DERIVED
PMID: 34709814 (View on PubMed)

Provided Documents

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Document Type: Study Protocol and Statistical Analysis Plan

View Document

Related Links

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Other Identifiers

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2019-003992-21

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

IM027-040

Identifier Type: -

Identifier Source: org_study_id

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