Evaluate the Drug-drugs Interaction Between Lobeglitazone and Empagliflozin

NCT ID: NCT02854748

Last Updated: 2016-08-09

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

UNKNOWN

Clinical Phase

PHASE1

Total Enrollment

30 participants

Study Classification

INTERVENTIONAL

Study Start Date

2016-08-31

Study Completion Date

2016-09-30

Brief Summary

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This study is a randomized, open-label, multiple dosing, crossover study to evaluate the drug-drugs interaction between Lobeglitazone and Empagliflozin in healthy male volunteers

Detailed Description

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To healthy male subjects of 30, following treatments are administered dosing in each 3 period(Lobeglitazone or Empagliflozin or Lobe.+Empa.) and wash-out period is a minimum of 7 days.

Test Drug 1: Lobeglitazone 0.5mg 1T

Test Drug 2: Empagliflozin 25mg 1T

Pharmacokinetic blood samples are collected up to 24hrs.

Safety, pharmacokinetic and the drug-drugs interaction are assessed.

Conditions

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Diabetes Mellitus, Type II

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Empagliflozin / Lobeglitazone / Empa.+Lobe.

Period 1: Empagliflozin 25 mg QD for 5 days Period 2: Lobeglitazone 0.5 mg QD for 5 days Period 3: Empagliflozin 25 mg + Lobeglitazone 0.5 mg QD for 5 days

Group Type EXPERIMENTAL

Empagliflozin 25mg

Intervention Type DRUG

Empagliflozin 25 mg QD for 5 days

Lobeglitazone 0.5mg

Intervention Type DRUG

Lobeglitazone 0.5mg QD for 5 days

Empagliflozin 25mg/Lobeglitazone 0.5mg

Intervention Type DRUG

Empagliflozin 25 mg + Lobeglitazone 0.5mg QD for 5 days

Empagliflozin / Empa.+Lobe. / Lobeglitazone

Period 1: Empagliflozin 25 mg QD for 5 days Period 2: Empagliflozin 25 mg + Lobeglitazone 0.5 mg QD for 5 days Period 3: Lobeglitazone 0.5 mg QD for 5 days

Group Type EXPERIMENTAL

Empagliflozin 25mg

Intervention Type DRUG

Empagliflozin 25 mg QD for 5 days

Lobeglitazone 0.5mg

Intervention Type DRUG

Lobeglitazone 0.5mg QD for 5 days

Empagliflozin 25mg/Lobeglitazone 0.5mg

Intervention Type DRUG

Empagliflozin 25 mg + Lobeglitazone 0.5mg QD for 5 days

Lobeglitazone / Empagliflozin / Empa.+Lobe.

Period 1: Lobeglitazone 0.5 mg QD for 5 days Period 2: Empagliflozin 25 mg QD for 5 days Period 3: Empagliflozin 25 mg + Lobeglitazone 0.5 mg QD for 5 days

Group Type EXPERIMENTAL

Empagliflozin 25mg

Intervention Type DRUG

Empagliflozin 25 mg QD for 5 days

Lobeglitazone 0.5mg

Intervention Type DRUG

Lobeglitazone 0.5mg QD for 5 days

Empagliflozin 25mg/Lobeglitazone 0.5mg

Intervention Type DRUG

Empagliflozin 25 mg + Lobeglitazone 0.5mg QD for 5 days

Lobeglitazone / Empa.+Lobe. / Empagliflozin

Period 1: Lobeglitazone 0.5 mg QD for 5 days Period 2: Empagliflozin 25 mg + Lobeglitazone 0.5 mg QD for 5 days Period 3: Empagliflozin 25 mg QD for 5 days

Group Type EXPERIMENTAL

Empagliflozin 25mg

Intervention Type DRUG

Empagliflozin 25 mg QD for 5 days

Lobeglitazone 0.5mg

Intervention Type DRUG

Lobeglitazone 0.5mg QD for 5 days

Empagliflozin 25mg/Lobeglitazone 0.5mg

Intervention Type DRUG

Empagliflozin 25 mg + Lobeglitazone 0.5mg QD for 5 days

Empa.+Lobe. / Empagliflozin / Lobeglitazone

Period 1: Empagliflozin 25 mg + Lobeglitazone 0.5 mg QD for 5 days Period 2: Empagliflozin 25 mg QD for 5 days Period 3: Lobeglitazone 0.5 mg QD for 5 days

Group Type EXPERIMENTAL

Empagliflozin 25mg

Intervention Type DRUG

Empagliflozin 25 mg QD for 5 days

Lobeglitazone 0.5mg

Intervention Type DRUG

Lobeglitazone 0.5mg QD for 5 days

Empagliflozin 25mg/Lobeglitazone 0.5mg

Intervention Type DRUG

Empagliflozin 25 mg + Lobeglitazone 0.5mg QD for 5 days

Empa.+Lobe. / Lobeglitazone / Empagliflozin

Period 1: Empagliflozin 25 mg + Lobeglitazone 0.5 mg QD for 5 days Period 2: Lobeglitazone 0.5 mg QD for 5 days Period 3: Empagliflozin 25 mg QD for 5 days

Group Type EXPERIMENTAL

Empagliflozin 25mg

Intervention Type DRUG

Empagliflozin 25 mg QD for 5 days

Lobeglitazone 0.5mg

Intervention Type DRUG

Lobeglitazone 0.5mg QD for 5 days

Empagliflozin 25mg/Lobeglitazone 0.5mg

Intervention Type DRUG

Empagliflozin 25 mg + Lobeglitazone 0.5mg QD for 5 days

Interventions

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Empagliflozin 25mg

Empagliflozin 25 mg QD for 5 days

Intervention Type DRUG

Lobeglitazone 0.5mg

Lobeglitazone 0.5mg QD for 5 days

Intervention Type DRUG

Empagliflozin 25mg/Lobeglitazone 0.5mg

Empagliflozin 25 mg + Lobeglitazone 0.5mg QD for 5 days

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. A healthy person whose age is in between 19 to 45 during the screening tests
2. Whose weight is more than 55 kg, BMI is over 18.5 and under 29.9 during the screening test. (BMI (kg/m2) = weight (kg) / {height (m)}2)
3. A male with no congenital or chronic disease in three years, no history of symptoms in internal treatment, or no knowledge in the area
4. Due to the special characteristics of drugs, the participators must be qualified to do the clinical screening tests
5. The participants must have an ability and willingness to participate throughout the entire trials

Exclusion Criteria

1. A person who has a history of clinically significant cardiovascular, respiratory, liver, kidney, endocrine system, immune system, urinary system diseases, blood-tumor diseases, mental illness.
2. Who had a history of gastrointestinal related disease which can be affected the drug absorption (esophageal achalasia, esophagostenosis, esophageal disease, or Crohn's disease) or surgeries (except a simple appendectomy or herniotomy)
3. Who has a history of hypersensitivity reactions to Empagliflozin or Lobeglitazone or similar series or other excipient ingredients (aspirin, fibrate, antibiotics, etc.)
4. A person whose electrocardiogram value includes QTc \> 450 msec, PR interval \> 200 msec, QRS duration \> 120 msec after screening, or who show clinically significant opinion.
5. Who falls under the following results

1. Liver Function Test (AST, ALT) are exceeded over 1.5x the upper limit of the normal range
2. eGFR \< 60mL/min/1.73m2
6. Who shows the vital sign values of more than 150 mmHg or less than 90 mmHg in systolic pressure or more than 95 mmHg or less than 60 mmHg in diastolic blood pressure
7. Who has history of drug abuses or shows a positive result in the urinary drug screen
8. Who took any prescribed drugs, medicinal plants within the 2 weeks before the first day of dosing or takes any over-the-counter drugs or vitamin supplements within 1 week (but, if other conditions are met, they can still participate in the clinical test through the researcher's judgment)
9. Who took other investigational drugs or bioequivalence drugs within 3 months before the first day of dosing
10. Who participated in whole blood donation within 2 months before the first of dosing, or platelet donations within 1 months. Who received blood a month before the first day of dosing
11. Who constantly drinks alcohol (over 21 units/week, 1 unit = 10 g of pure alcohol) or cannot stop drinking alcohol during the clinical test.
12. Who smokes more than 10 cigarettes per day within 3 months , or who cannot quit smoking when hospitalized
13. Who cannot limit intake of grapefruit or grapefruit containing foods in 48hrs from the first dosing of clinical testing drug to collect pharmacokinetic blood samples
14. Who absorb caffeinated drinks (coffee, tea (black or green tea), soda, coffee flavored milk, energy drinks, etc.) or cannot stop absorbing them 24 hours before hospitalization until discharging
15. Not using a reliable contraception, planning a pregnancy during the study
16. Who has Galactose intolerance, LAPP lactose intolerance, glucose-galactose malabsorption or genetic disorders
17. Person who is not determined unsuitable to participate in this test by the researchers
Minimum Eligible Age

19 Years

Maximum Eligible Age

45 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

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Chong Kun Dang Pharmaceutical

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Dong A University Hospital

Seo-gu, Busan, South Korea

Site Status

Countries

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South Korea

References

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Kim YK, Hwang JG, Park MK. No Relevant Pharmacokinetic Drug-Drug Interaction Between the Sodium-Glucose Co-Transporter-2 Inhibitor Empagliflozin and Lobeglitazone, a Peroxisome Proliferator-Activated Receptor-gamma Agonist, in Healthy Subjects. Drug Des Devel Ther. 2021 Apr 28;15:1725-1734. doi: 10.2147/DDDT.S302215. eCollection 2021.

Reference Type DERIVED
PMID: 33953542 (View on PubMed)

Other Identifiers

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19DDI16005

Identifier Type: -

Identifier Source: org_study_id

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