A Study Comparing Upadacitinib (ABT-494) Monotherapy to Methotrexate (MTX) Monotherapy in Adults With Rheumatoid Arthritis (RA) Who Have an Inadequate Response to MTX (SELECT-MONOTHERAPY)

NCT ID: NCT02706951

Last Updated: 2024-01-30

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

648 participants

Study Classification

INTERVENTIONAL

Study Start Date

2016-03-23

Study Completion Date

2022-08-10

Brief Summary

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The study objective of Period 1 of this study is to compare the safety and efficacy (signs and symptoms) of upadacitinib 30 mg once daily (QD) alone and upadacitinib 15 mg QD alone versus continuing MTX alone adults with moderately to severely active rheumatoid arthritis (RA) with an inadequate response to MTX.

The study objective of Period 2 is to evaluate the long term safety, tolerability, and efficacy of upadacitinib 30 mg QD and 15 mg QD in adults with RA who had completed Period 1.

Detailed Description

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The study includes a 35-day screening period; a 14-week randomized, double-blind, parallel-group, controlled treatment period (Period 1); a 246-week blinded extension period (Period 2); and a 30-day follow-up visit.

Participants who met eligibility criteria were to be randomized in a 2:2:1:1 ratio to one of four treatment groups:

* Group 1: upadacitinib 30 mg QD (Period 1) → upadacitinib 30 mg QD (Period 2)
* Group 2: upadacitinib 15 mg QD (Period 1) → upadacitinib 15 mg QD (Period 2)
* Group 3: MTX (Period 1) → upadacitinib 30 mg QD (Period 2)
* Group 4: MTX (Period 1) → upadacitinib 15 mg QD (Period 2)

Starting with implementation of Protocol Amendment 5, all participants in the extension period will receive open-label upadacitinib 15 mg QD, including those currently on upadacitinib 30 mg QD.

Conditions

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Rheumatoid Arthritis

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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Upadacitinib 30 mg

Period 1: Participants receive upadacitnib 30 mg once daily and placebo to methotrexate once weekly for 14 weeks.

Period 2: Participants receive upadacitinib 30 mg once daily until implementation of Protocol Amendment 5 when participants begin to receive upadacitinib 15 mg once daily up to Week 260.

Group Type EXPERIMENTAL

Upadacitinib

Intervention Type DRUG

Tablet; Oral

Placebo Methotrexate

Intervention Type DRUG

Capsule; Oral

Upadacitinib 15 mg

Period 1: Participants receive upadacitnib 15 mg once daily and placebo to methotrexate once weekly for 14 weeks.

Period 2: Participants receive upadacitinib 15 mg once daily up to Week 260.

Group Type EXPERIMENTAL

Upadacitinib

Intervention Type DRUG

Tablet; Oral

Placebo Methotrexate

Intervention Type DRUG

Capsule; Oral

Methotrexate / Upadacitinib 30 mg

Period 1: Participants receive methotrexate once weekly and placebo to upadacitinib once daily for 14 weeks.

Period 2: Participants receive upadacitinib 30 mg once daily until implementation of Protocol Amendment 5 when participants begin to receive upadacitinib 15 mg once daily up to Week 260.

Group Type EXPERIMENTAL

Methotrexate

Intervention Type DRUG

Capsule; Oral

Upadacitinib

Intervention Type DRUG

Tablet; Oral

Placebo Upadacitinib

Intervention Type DRUG

Tablet; Oral

Placebo Methotrexate

Intervention Type DRUG

Capsule; Oral

Methotrexate / Upadacitinib 15 mg

Period 1: Participants receive methotrexate once weekly and placebo to upadacitinib for 14 weeks.

Period 2: Participants receive upadacitinib 15 mg once daily up to Week 260.

Group Type EXPERIMENTAL

Methotrexate

Intervention Type DRUG

Capsule; Oral

Upadacitinib

Intervention Type DRUG

Tablet; Oral

Placebo Upadacitinib

Intervention Type DRUG

Tablet; Oral

Placebo Methotrexate

Intervention Type DRUG

Capsule; Oral

Interventions

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Methotrexate

Capsule; Oral

Intervention Type DRUG

Upadacitinib

Tablet; Oral

Intervention Type DRUG

Placebo Upadacitinib

Tablet; Oral

Intervention Type DRUG

Placebo Methotrexate

Capsule; Oral

Intervention Type DRUG

Other Intervention Names

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ABT-494 Rinvoq

Eligibility Criteria

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Inclusion Criteria

* Diagnosis of RA for \>= 3 months.
* Subjects must have been on oral or parenteral MTX therapy \>= 3 months and on a stable dose for \>= 4 weeks prior to first dose of study drug.
* Must have discontinued all conventional synthetic disease-modifying anti-rheumatic drugs (csDMARDs) (other than MTX) \>= 4 weeks prior to first dose of study drug.
* Meets the following minimum disease activity criteria: \>= 6 swollen joints (based on 66 joint counts) and \>= 6 tender joints (based on 68 joint counts) at Screening and Baseline Visits.

Exclusion Criteria

* Prior exposure to any Janus kinase (JAK) inhibitor (including but not limited to tofacitinib, baricitinib, and filgotinib).
* Prior exposure to any biological disease-modifying anti-rheumatic drugs (bDMARDs).
* Current diagnosis of inflammatory joint disease other than RA. Current diagnosis of secondary Sjogren's Syndrome is permitted.
Minimum Eligible Age

18 Years

Maximum Eligible Age

99 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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AbbVie

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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AbbVie Inc.

Role: STUDY_DIRECTOR

AbbVie

Locations

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Rheum Assoc of North Alabama /ID# 146009

Huntsville, Alabama, United States

Site Status

Alabama Medical Group, PC /ID# 153941

Mobile, Alabama, United States

Site Status

ArthroCare Arthritis Care & Re /ID# 143751

Gilbert, Arizona, United States

Site Status

Elite Clinical Studies, LLC /ID# 143760

Phoenix, Arizona, United States

Site Status

University of Arizona Cancer Center - North Campus /ID# 147175

Tucson, Arizona, United States

Site Status

NEA Baptist Womens Clinic /ID# 148904

Jonesboro, Arkansas, United States

Site Status

C.V. Mehta MD, Med Corporation /ID# 143762

Hemet, California, United States

Site Status

Arthritis Assoc & Osteo Ctr /ID# 147176

Colorado Springs, Colorado, United States

Site Status

Ctr Rheum, Immuno, Arthritis /ID# 143766

Fort Lauderdale, Florida, United States

Site Status

South Florida Research Ph I-IV /ID# 151983

Miami Springs, Florida, United States

Site Status

Advent Clinical Research /ID# 143767

Pinellas Park, Florida, United States

Site Status

Sarasota Arthritis Center /ID# 146011

Sarasota, Florida, United States

Site Status

W. Broward Rheum Assoc Inc. /ID# 146010

Tamarac, Florida, United States

Site Status

Clinical Research West FL /ID# 148726

Tampa, Florida, United States

Site Status

SW FL Clin Res Ctr, Tampa, FL /ID# 143763

Tampa, Florida, United States

Site Status

University of South Florida /ID# 146004

Tampa, Florida, United States

Site Status

BayCare Medical Group, Inc. /ID# 151985

Tampa, Florida, United States

Site Status

BayCare Medical Group, Inc. /ID# 163595

Tampa, Florida, United States

Site Status

Jefrey D. Lieberman, MD, P.C. /ID# 151816

Decatur, Georgia, United States

Site Status

Great Lakes Clinical Trials /ID# 150935

Chicago, Illinois, United States

Site Status

PRN Professional Research Network of Kansas, LLC /ID# 143761

Wichita, Kansas, United States

Site Status

Ochsner Clinic Foundation /ID# 153573

Baton Rouge, Louisiana, United States

Site Status

The Arthritis & Diabetes Clinic, Inc. /ID# 160809

Monroe, Louisiana, United States

Site Status

Vanguard Medical Research, LLC /ID# 153124

Shreveport, Louisiana, United States

Site Status

Mansfield Health Center /ID# 161627

Mansfield, Massachusetts, United States

Site Status

Quality Clinical Research Inc. /ID# 156415

Omaha, Nebraska, United States

Site Status

Dartmouth-Hitchcock Medical Center /ID# 146008

Lebanon, New Hampshire, United States

Site Status

Albuquerque Clinical Trials, Inc /ID# 147618

Albuquerque, New Mexico, United States

Site Status

Arthritis and Osteo Assoc /ID# 147177

Las Cruces, New Mexico, United States

Site Status

Coastal Carolina Health Care /ID# 149275

New Bern, North Carolina, United States

Site Status

STAT Research, Inc. /ID# 143770

Vandalia, Ohio, United States

Site Status

Health Research Oklahoma /ID# 159550

Oklahoma City, Oklahoma, United States

Site Status

Healthcare Research Consultant /ID# 147632

Tulsa, Oklahoma, United States

Site Status

Innovative Clinical Research /ID# 143757

Greenville, South Carolina, United States

Site Status

Nashville Arthritis and Rheumatology /ID# 162641

Nashville, Tennessee, United States

Site Status

Tekton Research, Inc. /ID# 159554

Austin, Texas, United States

Site Status

Diagnostic Group Integrated He /ID# 148725

Beaumont, Texas, United States

Site Status

Trinity Universal Res Assoc /ID# 150138

Carrollton, Texas, United States

Site Status

Arth and Osteo Clin Brazo Valley /ID# 160810

College Station, Texas, United States

Site Status

Adriana Pop-Moody MD Clinic PA /ID# 147627

Corpus Christi, Texas, United States

Site Status

Accurate Clinical Management /ID# 143768

Houston, Texas, United States

Site Status

Accurate Clinical Research /ID# 143769

Houston, Texas, United States

Site Status

Pioneer Research Solutions, Inc. /ID# 143765

Houston, Texas, United States

Site Status

P&I Clinical Research /ID# 151358

Lufkin, Texas, United States

Site Status

SW Rheumatology Res. LLC /ID# 147620

Mesquite, Texas, United States

Site Status

Sun Research Institute /ID# 159553

San Antonio, Texas, United States

Site Status

Arthritis Clinic of Central TX /ID# 149266

San Marcos, Texas, United States

Site Status

Adv Rheumatology of Houston /ID# 162609

The Woodlands, Texas, United States

Site Status

DM Clinical Research /ID# 151359

Tomball, Texas, United States

Site Status

Arthritis & Osteoporosis Clinic /ID# 143752

Waco, Texas, United States

Site Status

Ctr for Arth and Rheum Disease /ID# 143759

Chesapeake, Virginia, United States

Site Status

Aurora Rheumatology and Immunotherapy Center /ID# 160811

Franklin, Wisconsin, United States

Site Status

Mautalen Salud e Investigacion /ID# 145980

Buenos Aires, , Argentina

Site Status

Ctr Privado Med Familiar /ID# 149183

Buenos Aires, , Argentina

Site Status

Consultorio Reumatologic Pampa /ID# 145979

Buenos Aires, , Argentina

Site Status

Centro de Educación Médica e Investigaciones Clínicas "Norberto Quimo" - CEMIC /ID# 149176

Buenos Aires, , Argentina

Site Status

Cordis S.A. /Id# 152621

Salta, , Argentina

Site Status

Centro de Enfermedades /ID# 153543

Santa Fe, , Argentina

Site Status

Royal Prince Alfred Hospital /ID# 146028

Camperdown, New South Wales, Australia

Site Status

Rheuma-Zentrum Wien-Oberlaa /ID# 144728

Vienna, , Austria

Site Status

Algemeen Stedelijk Ziekenhuis /ID# 148720

Aalst, Oost-Vlaanderen, Belgium

Site Status

ReumaClinic Genk /ID# 146030

Genk, , Belgium

Site Status

Diag Consult Ctr 17 Sofia EOOD /ID# 144730

Sofia, , Bulgaria

Site Status

UMHAT Sv. Ivan Rilski /ID# 147351

Sofia, , Bulgaria

Site Status

Reg. Clinical Hosptial Concepcion /ID# 151267

Concepción, , Chile

Site Status

Quantum Research LTDA. /ID# 145984

Puerto Varas, , Chile

Site Status

Quantum Research Stgo. /ID# 145983

Santiago, , Chile

Site Status

CTCenter MaVe, s.r.o. /ID# 144823

Olomouc, Olomoucký kraj, Czechia

Site Status

Nuselská poliklinika, Revmatologie /ID# 145986

Prague, Praha 4, Czechia

Site Status

Thomayerova nemocnice /ID# 144736

Prague, Praha 4, Czechia

Site Status

RHEUMA s.r.o. /ID# 144737

Břeclav, , Czechia

Site Status

Medical Plus, s.r.o. /ID# 144821

Uherské Hradište, , Czechia

Site Status

MediTrials /ID# 159745

Tartu, Tartu, Estonia

Site Status

North Estonian Medical Centre /ID# 145455

Tallinn, , Estonia

Site Status

General Hospital of Athens "Ippokratio" /ID# 144739

Athens, , Greece

Site Status

Vital Medical Center Orvosi es /ID# 144740

Veszprém, Veszprém megye, Hungary

Site Status

Magyar Honvedseg Egeszsegugyi Kozpont /ID# 144743

Budapest, , Hungary

Site Status

Pest Megyei Flor Ferenc Korhaz /ID# 144742

Kistarcsa, , Hungary

Site Status

Fejer Megyei Szent Gyorgy Korh /ID# 144741

Székesfehérvár, , Hungary

Site Status

Barzilai Medical Center /ID# 144744

Ashkelon, , Israel

Site Status

Bnai Zion Medical Center /ID# 144745

Haifa, , Israel

Site Status

The Lady Davis Carmel MC /ID# 147174

Haifa, , Israel

Site Status

Sheba Medical Center /ID# 144824

Ramat Gan, , Israel

Site Status

Universita di Catanzaro Magna Graecia /ID# 144747

Catanzaro, Calabria, Italy

Site Status

A.O.U.I. di Verona Policlinico /ID# 144746

Verona, , Italy

Site Status

Kondo Clinic for Rheum & Ortho /ID# 148268

Fukuoka, Fukuoka, Japan

Site Status

NHO Kyushu Medical Center /ID# 148279

Fukuoka, Fukuoka, Japan

Site Status

NHO Kyushu Medical Center /ID# 148280

Fukuoka, Fukuoka, Japan

Site Status

Aso Iizuka Hospital /ID# 148272

Iizuka-shi, Fukuoka, Japan

Site Status

Inoue Hospital /ID# 148069

Takasaki, Gunma, Japan

Site Status

Bay Side Misato Medical Center /ID# 148281

Kochi, Kochi, Japan

Site Status

Center for Arthritis and Clinical Rheumatology Matsubara Clinic /ID# 148269

Kumamoto, Kumamoto, Japan

Site Status

Kumamoto Shinto General Hospital /ID# 148286

Kumamoto, Kumamoto, Japan

Site Status

Nagasaki University Hospital /ID# 149859

Nagasaki, Nagasaki, Japan

Site Status

Sasebo Chuo Hospital /ID# 148275

Sasebo, Nagasaki, Japan

Site Status

Osaka Red Cross Hospital /ID# 148267

Osaka, Osaka, Japan

Site Status

Seirei Hamamatsu General Hosp /ID# 148270

Hamamatsu, , Japan

Site Status

Ohira Orthopaedic Hospital /ID# 157944

Hyūga, , Japan

Site Status

Shirahama Hamayu Hospital /ID# 148277

Nishimura, , Japan

Site Status

Sanuki Municipal Hospital /ID# 158080

Sanuki, , Japan

Site Status

Hokkaido University Hospital /ID# 148285

Sapporo, , Japan

Site Status

Hokkaido Medical Center for Rheumatic Diseases /ID# 148274

Sapporo, , Japan

Site Status

Miyasato Clinic /ID# 148271

Shūnan, , Japan

Site Status

Takaoka Rheumatic Orthopedic Clinic /ID# 148068

Takaoka, , Japan

Site Status

Matsuta Clinic /ID# 148278

Tokyo, , Japan

Site Status

National Hospital Organization Shimoshizu National Hospital /ID# 148273

Yotsukaidō, , Japan

Site Status

Desarrollos Biomedicos y Biotc /ID# 147379

Monterrey, Nuevo León, Mexico

Site Status

Cryptex Investigación Clínica S.A de C.V /ID# 147095

Mexico City, , Mexico

Site Status

Medyczne Centrum Hetmanska /ID# 144751

Poznan, Greater Poland Voivodeship, Poland

Site Status

WroMedica I. Bielicka, A. Strzalkowska s.c. /ID# 157622

Wroclaw, Lower Silesian Voivodeship, Poland

Site Status

REUMED Sp.z o.o. Filia nr 1 /ID# 144752

Lublin, Lublin Voivodeship, Poland

Site Status

Centralny Szpital Kliniczny MSWiA w Warszawie /ID# 149521

Warsaw, Masovian Voivodeship, Poland

Site Status

Osteo-Medic spolka cywilna /ID# 144753

Bialystok, Podlaskie Voivodeship, Poland

Site Status

Centrum Badań Klinicznych Pi-House /ID# 149520

Gdansk, Pomeranian Voivodeship, Poland

Site Status

NZOZ Centrum Reumatologiczne /ID# 144749

Elblag, Warmian-Masurian Voivodeship, Poland

Site Status

Instituto Portugues De Reumatologia /ID# 149281

Lisbon, Lisbon District, Portugal

Site Status

Centro Hospitalar De Vila Nova /ID# 146036

Vila Nova de Gaia, Porto District, Portugal

Site Status

Centro Hospitalar Lisboa Norte, EPE /ID# 146035

Lisbon, , Portugal

Site Status

Centro Hospitalar Baixo Vouga /ID# 152916

Porto, , Portugal

Site Status

Dr. Ramon L. Ortega-Colon, MD /ID# 145989

Carolina, , Puerto Rico

Site Status

Ponce School of Medicine /ID# 145990

Ponce, , Puerto Rico

Site Status

Spitalul Municipal Ploiesti /ID# 144756

Ploieşti, , Romania

Site Status

Clinical Hospital No.1 n.a. N.I.Pirogov /ID# 147255

Moscow, Moscow, Russia

Site Status

LLC Medical Center /ID# 144758

Novosibirsk, Novosibirsk Oblast, Russia

Site Status

Perm Clinical Center of FMBA /ID# 145993

Perm, Permskiy Kray, Russia

Site Status

Tver Regional Clinical Hosp. /ID# 147254

Tver', Tver Oblast, Russia

Site Status

Сity Clinical Hospital 4 /ID# 145994

Ivanovo, , Russia

Site Status

City Clinical Hospital Botkina /ID# 145995

Moscow, , Russia

Site Status

City Clinical Hospital #5 /ID# 149832

Nizhny Novgorod, , Russia

Site Status

Orenburg State Medical Academy /ID# 145992

Orenburg, , Russia

Site Status

Republican Clin Hos n.a. Baran /ID# 147251

Petrozavodsk, , Russia

Site Status

Samara Regional Clinical Hosp /ID# 150934

Samara, , Russia

Site Status

Reg Clin Hosp n.a. Kuvatova G. /ID# 144757

Ufa, , Russia

Site Status

Yaroslavi State Medical Univer /ID# 147253

Yaroslavl, , Russia

Site Status

Institute for Rheumatology /ID# 144759

Belgrade, Beograd, Serbia

Site Status

Institute for Rheumatology /ID# 144761

Belgrade, Beograd, Serbia

Site Status

Institute for Rheumatology /ID# 144762

Belgrade, Beograd, Serbia

Site Status

Special Hospital for Rheuma /ID# 144760

Novi Sad, Vojvodina, Serbia

Site Status

Wits Clinical Research Site /ID# 149835

Johannesburg, Gauteng, South Africa

Site Status

University of Pretoria /ID# 148740

Pretoria, Gauteng, South Africa

Site Status

Synexus Helderberg Clinical Tr /ID# 148724

Cape Town, Western Cape, South Africa

Site Status

Tiervlei Trial Centre /ID# 153086

Cape Town, Western Cape, South Africa

Site Status

Hospital Plató /ID# 145999

Barcelona, , Spain

Site Status

Hospital Univ Germans Trias I /ID# 146037

Barcelona, , Spain

Site Status

Hospital Infanta Luisa /ID# 144771

Seville, , Spain

Site Status

Hospital Universitario de Valm /ID# 144770

Seville, , Spain

Site Status

Hospital Universitario La Fe /ID# 158013

Valencia, , Spain

Site Status

Uludağ Üniversitesi Atatürk Rehabilitasyon Uygulama ve Araştırma Merkezi /ID# 144772

Osmangazi, Bursa, Turkey (Türkiye)

Site Status

Lviv Regional Clinical Hospita /ID# 154448

Lviv, Lviv Oblast, Ukraine

Site Status

Vinnytsia Regional Clinical Hospital n.a. M.I.Pyrogov /ID# 146002

Vinnytsia, Vinnytsia Oblast, Ukraine

Site Status

Regional Clinical Hospital /ID# 152007

Ivano-Frankivsk, , Ukraine

Site Status

NSC-Strazhesko Ist Cardiology /ID# 152004

Kiev, , Ukraine

Site Status

Zaporizhzhia Regional Clinical /ID# 146000

Zaporizhia, , Ukraine

Site Status

Countries

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United States Argentina Australia Austria Belgium Bulgaria Chile Czechia Estonia Greece Hungary Israel Italy Japan Mexico Poland Portugal Puerto Rico Romania Russia Serbia South Africa Spain Turkey (Türkiye) Ukraine

References

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Rubbert-Roth A, Kakehasi AM, Takeuchi T, Schmalzing M, Palac H, Coombs D, Liu J, Anyanwu SI, Lippe R, Curtis JR. Malignancy in the Upadacitinib Clinical Trials for Rheumatoid Arthritis, Psoriatic Arthritis, Ankylosing Spondylitis, and Non-radiographic Axial Spondyloarthritis. Rheumatol Ther. 2024 Feb;11(1):97-112. doi: 10.1007/s40744-023-00621-6. Epub 2023 Nov 20.

Reference Type DERIVED
PMID: 37982966 (View on PubMed)

Charles-Schoeman C, Choy E, McInnes IB, Mysler E, Nash P, Yamaoka K, Lippe R, Khan N, Shmagel AK, Palac H, Suboticki J, Curtis JR. MACE and VTE across upadacitinib clinical trial programmes in rheumatoid arthritis, psoriatic arthritis and ankylosing spondylitis. RMD Open. 2023 Nov;9(4):e003392. doi: 10.1136/rmdopen-2023-003392.

Reference Type DERIVED
PMID: 37945286 (View on PubMed)

Fleischmann R, Curtis JR, Charles-Schoeman C, Mysler E, Yamaoka K, Richez C, Palac H, Dilley D, Liu J, Strengholt S, Burmester G. Safety profile of upadacitinib in patients at risk of cardiovascular disease: integrated post hoc analysis of the SELECT phase III rheumatoid arthritis clinical programme. Ann Rheum Dis. 2023 Sep;82(9):1130-1141. doi: 10.1136/ard-2023-223916. Epub 2023 Jun 12.

Reference Type DERIVED
PMID: 37308218 (View on PubMed)

Conaghan PG, Pavelka K, Hsieh SC, Bonnington TL, Kent TC, Marchbank K, Edwards CJ. Evaluating the efficacy of upadacitinib in patients with moderate rheumatoid arthritis: a post-hoc analysis of the SELECT phase 3 trials. Rheumatol Adv Pract. 2023 Feb 8;7(1):rkad017. doi: 10.1093/rap/rkad017. eCollection 2023.

Reference Type DERIVED
PMID: 36794283 (View on PubMed)

Smolen JS, Pangan AL, Emery P, Rigby W, Tanaka Y, Vargas JI, Zhang Y, Damjanov N, Friedman A, Othman AA, Camp HS, Cohen S. Upadacitinib as monotherapy in patients with active rheumatoid arthritis and inadequate response to methotrexate (SELECT-MONOTHERAPY): a randomised, placebo-controlled, double-blind phase 3 study. Lancet. 2019 Jun 8;393(10188):2303-2311. doi: 10.1016/S0140-6736(19)30419-2. Epub 2019 May 23.

Reference Type BACKGROUND
PMID: 31130260 (View on PubMed)

Burmester GR, Deodhar A, Irvine AD, Panaccione R, Winthrop KL, Vleugels RA, Levy G, Suravaram S, Palac H, Wegrzyn L, Ford S, Meerwein S, Guttman-Yassky E. Safety Profile of Upadacitinib: Descriptive Analysis in Over 27,000 Patient-Years Across Rheumatoid Arthritis, Psoriatic Arthritis, Axial Spondyloarthritis, Atopic Dermatitis, and Inflammatory Bowel Disease. Adv Ther. 2025 Oct;42(10):5215-5237. doi: 10.1007/s12325-025-03328-y. Epub 2025 Aug 28.

Reference Type DERIVED
PMID: 40875187 (View on PubMed)

Smolen JS, Emery P, Rigby W, Tanaka Y, Vargas JI, Jain M, Kato K, Carter KM, Khan N, Phillips C, Meerwein S, Cohen SB. Upadacitinib as monotherapy in patients with rheumatoid arthritis and prior inadequate response to methotrexate: results at 260 weeks from the SELECT-MONOTHERAPY randomised study. RMD Open. 2025 May 11;11(2):e005051. doi: 10.1136/rmdopen-2024-005051.

Reference Type DERIVED
PMID: 40350200 (View on PubMed)

Burmester GR, Cohen SB, Winthrop KL, Nash P, Irvine AD, Deodhar A, Mysler E, Tanaka Y, Liu J, Lacerda AP, Palac H, Shaw T, Mease PJ, Guttman-Yassky E. Safety profile of upadacitinib over 15 000 patient-years across rheumatoid arthritis, psoriatic arthritis, ankylosing spondylitis and atopic dermatitis. RMD Open. 2023 Feb;9(1):e002735. doi: 10.1136/rmdopen-2022-002735.

Reference Type DERIVED
PMID: 36754548 (View on PubMed)

Kakehasi AM, Radominski SC, Baravalle MD, Palazuelos FCI, Garcia-Garcia C, Arruda MS, Curi M, Liu J, Qiao M, Velez-Sanchez P, Vargas JI. Safety of upadacitinib in Latin American patients with rheumatoid arthritis: an integrated safety analysis of the SELECT phase 3 clinical program. Clin Rheumatol. 2023 May;42(5):1249-1258. doi: 10.1007/s10067-023-06513-y. Epub 2023 Jan 30.

Reference Type DERIVED
PMID: 36715850 (View on PubMed)

Bergman M, Buch MH, Tanaka Y, Citera G, Bahlas S, Wong E, Song Y, Zueger P, Ali M, Strand V. Routine Assessment of Patient Index Data 3 (RAPID3) in Patients with Rheumatoid Arthritis Treated with Long-Term Upadacitinib Therapy in Five Randomized Controlled Trials. Rheumatol Ther. 2022 Dec;9(6):1517-1529. doi: 10.1007/s40744-022-00483-4. Epub 2022 Sep 20.

Reference Type DERIVED
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Provided Documents

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Document Type: Study Protocol

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Document Type: Statistical Analysis Plan

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Related Links

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Other Identifiers

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2015-003376-75

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

M15-555

Identifier Type: -

Identifier Source: org_study_id

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