A Phase 3 Study to Compare Upadacitinib to Abatacept in Subjects With Rheumatoid Arthritis on Stable Dose of Conventional Synthetic Disease- Modifying Antirheumatic Drugs (csDMARDs) Who Have an Inadequate Response or Intolerance to Biologic DMARDs

NCT ID: NCT03086343

Last Updated: 2024-07-18

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

657 participants

Study Classification

INTERVENTIONAL

Study Start Date

2017-05-09

Study Completion Date

2023-06-06

Brief Summary

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The study objective of Period 1 was to compare the safety and efficacy of upadacitinib 15 mg once daily (QD) to abatacept on a background of conventional synthetic disease-modifying antirheumatic drugs (csDMARDs) for the treatment of signs and symptoms of rheumatoid arthritis (RA) in biologic disease-modifying antirheumatic drug (bDMARD)-inadequate response or bDMARD-intolerant participants with moderately to severely active RA. The study objective of Period 2 is to evaluate the long-term safety, tolerability, and efficacy of upadacitinib 15 mg QD in participants with RA who had completed Period 1.

Detailed Description

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This is a Phase 3 multicenter study with 2 periods. Period 1 was a 24-week, randomized, double-blind, parallel-group, active-controlled period designed to compare the safety and efficacy of upadacitinib 15 mg and abatacept for the treatment of signs and symptoms of participants with moderately to severely active RA who had an inadequate response to or intolerance to bDMARD therapy and were currently on a stable dose of csDMARD(s) and had never received abatacept. Period 2 is an open-label, long-term extension study to evaluate the long-term safety, tolerability, and efficacy of upadacitinib 15 mg once a day (QD) in participants with RA who had completed Period 1.

Conditions

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Rheumatoid Arthritis (RA)

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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Primary Cohort: Abatacept/Upadacitinib 15 mg QD

Period 1: 500 mg (for body weight \<60 kg); 750 mg (for body weight 60-100 kg); and 1000 mg (for body weight \>100 kg) IV infusion at Baseline, Week 2, Week 4, Week 8, Week 12, Week 16 and Week 20. Period 2: open label upadacitinib 15 mg QD for 192 weeks.

Group Type ACTIVE_COMPARATOR

Abatacept

Intervention Type DRUG

IV infusion

Upadacitinib

Intervention Type DRUG

15 mg extended release tablet

Placebo for upadacitinib

Intervention Type DRUG

Film-coated tablet

Primary Cohort: Upadacitinib 15 mg QD/Upadacitinib 15 mg QD

Period 1: One 15 mg upadacitinib oral tablet QD for 24 weeks. Period 2: open label upadacitinib 15 mg QD for 192 weeks.

Group Type EXPERIMENTAL

Placebo for abatacept (0.9% Sodium Chloride Injection or Solution for Infusion)

Intervention Type DRUG

IV infusion

Upadacitinib

Intervention Type DRUG

15 mg extended release tablet

30 mg Cohort: Upadacitinib 30 mg QD/Upadacitinib 30 mg QD

Period 1: One upadacitinib 30 mg oral tablet QD for 24 weeks. Period 2: open label upadacitinib 30 mg (reduced to 15 mg per Amendment 5) QD for 192 weeks.

Group Type EXPERIMENTAL

Placebo for abatacept (0.9% Sodium Chloride Injection or Solution for Infusion)

Intervention Type DRUG

IV infusion

Upadacitinib

Intervention Type DRUG

15 mg extended release tablet

30 mg Cohort: Abatacept/Upadacitinib 30 mg QD

Period 1: 500 mg (for body weight \<60 kg); 750 mg (for body weight 60-100 kg); and 1000 mg (for body weight \>100 kg) IV infusion at Baseline, Week 2, Week 4, Week 8, Week 12, Week 16 and Week 20. Period 2: open label upadacitinib 30 mg (reduced to 15 mg per Amendment 5) QD for 192 weeks.

Group Type ACTIVE_COMPARATOR

Abatacept

Intervention Type DRUG

IV infusion

Upadacitinib

Intervention Type DRUG

15 mg extended release tablet

Placebo for upadacitinib

Intervention Type DRUG

Film-coated tablet

Interventions

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Abatacept

IV infusion

Intervention Type DRUG

Placebo for abatacept (0.9% Sodium Chloride Injection or Solution for Infusion)

IV infusion

Intervention Type DRUG

Upadacitinib

15 mg extended release tablet

Intervention Type DRUG

Placebo for upadacitinib

Film-coated tablet

Intervention Type DRUG

Other Intervention Names

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ABT-494

Eligibility Criteria

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Inclusion Criteria

* Diagnosis of rheumatoid arthritis (RA) for ≥ 3 months who also fulfill the 2010 American College of Rheumatology (ACR)/European League Against Rheumatism (EULAR) classification criteria for RA
* Participants have been treated for ≥ 3 months prior to the screening visit with ≥ 1 bDMARD therapy, but continue to exhibit active RA or had to discontinue due to intolerability or toxicity, irrespective of treatment duration and have never received abatacept prior to the first dose of study drug
* Participants have been receiving csDMARD therapy ≥ 3 months and on a stable dose for ≥ 4 weeks prior to the first dose of study drug. The following csDMARDs are allowed: methotrexate (MTX), sulfasalazine, hydroxychloroquine, chloroquine, and leflunomide. A combination of up to two background csDMARDs is allowed except the combination of MTX and leflunomide
* Meets the following criteria: ≥ 6 swollen joints (based on 66 joint counts) and ≥ 6 tender joints (based on 68 joint counts) at Screening and Baseline Visits and high-sensitivity C-reactive protein (hsCRP) ≥ 3 mg/L at Screening

Exclusion Criteria

* Prior exposure to any Janus kinase (JAK) inhibitor (including but not limited to upadacitinib, tofacitinib, baricitinib and filgotinib)
* Prior exposure to abatacept
* History of any arthritis with onset prior to age 17 years or current diagnosis of inflammatory joint disease other than RA. Current diagnosis of secondary Sjogren's Syndrome is permitted
* Laboratory values meeting the following criteria within the Screening period prior to the first dose of study drug: serum aspartate transaminase \> 2 × upper limit of normal (ULN); serum alanine transaminase \> 2 × ULN; estimated glomerular filtration rate by simplified 4-variable Modification of Diet in Renal Disease formula \< 40 mL/minute/1.73 meter (m)\^2; total white blood cell count \< 2,500/ μL; absolute neutrophil count \< 1,500/μL; platelet count \< 100,000/μL; absolute lymphocyte count \< 800/μL; and hemoglobin \< 10 g/dL
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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AbbVie

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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AbbVie Inc.

Role: STUDY_DIRECTOR

AbbVie

Locations

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SunValley Arthritis Center, Lt /ID# 154558

Peoria, Arizona, United States

Site Status

AZ Arthritis & Rheum Research /ID# 156539

Sun City, Arizona, United States

Site Status

AZ Arth & Rheum Res /ID# 167161

Tucson, Arizona, United States

Site Status

CHI St. Vincent Medical Group /ID# 154561

Hot Springs, Arkansas, United States

Site Status

Saint Jude Heritage /ID# 158833

Fullerton, California, United States

Site Status

Kotha and Kotha /ID# 154573

La Mesa, California, United States

Site Status

Denver Arthritis Clinic /ID# 159195

Denver, Colorado, United States

Site Status

Arthritis and Rheum Clin N. CO /ID# 155673

Fort Collins, Colorado, United States

Site Status

Scientia Medical Research /ID# 159189

Lakewood, Colorado, United States

Site Status

Clinical Res of West FL, Inc. /ID# 154576

Clearwater, Florida, United States

Site Status

Advanced Clin Res of Orlando /ID# 154580

Ocoee, Florida, United States

Site Status

Gulf Region Clinical Res Inst /ID# 154597

Pensacola, Florida, United States

Site Status

W. Broward Rheum Assoc Inc. /ID# 158835

Tamarac, Florida, United States

Site Status

Lovelace Scientific Resources /ID# 154600

Venice, Florida, United States

Site Status

Jefrey D. Lieberman, MD, P.C. /ID# 157178

Decatur, Georgia, United States

Site Status

Advanced Clinical Research /ID# 154603

Meridian, Idaho, United States

Site Status

PMG Research of Christie Clini /ID# 154569

Champaign, Illinois, United States

Site Status

Bluegrass Community Research /ID# 154604

Lexington, Kentucky, United States

Site Status

Four Rivers Clinical Research /ID# 154606

Paducah, Kentucky, United States

Site Status

Ochsner Clinic Foundation /ID# 154585

Baton Rouge, Louisiana, United States

Site Status

The Center for Rheumatology & Bone Research /ID# 158723

Wheaton, Maryland, United States

Site Status

West Michigan Rheumatology /ID# 154551

Grand Rapids, Michigan, United States

Site Status

Advanced Rheumatology, PC /ID# 154589

Lansing, Michigan, United States

Site Status

Clinvest Research LLC /ID# 154554

Springfield, Missouri, United States

Site Status

Overlook Medical Center /ID# 154794

Summit, New Jersey, United States

Site Status

Atlantic Coast Research /ID# 155234

Toms River, New Jersey, United States

Site Status

Ocean Rheumatology, PA /ID# 162980

Toms River, New Jersey, United States

Site Status

Arthritis and Osteo Assoc /ID# 154560

Las Cruces, New Mexico, United States

Site Status

The Center for Rheumatology /ID# 162979

Albany, New York, United States

Site Status

NYU Langone Rheum Assoc /ID# 155236

Lake Success, New York, United States

Site Status

NYU Langone Medical Center /ID# 158829

New York, New York, United States

Site Status

Physicians East, PA /ID# 154565

Greenville, North Carolina, United States

Site Status

PMG Research of Salisbury /ID# 154605

Salisbury, North Carolina, United States

Site Status

PMG Research of Wilmington LLC /ID# 154584

Wilmington, North Carolina, United States

Site Status

Wake Forest Baptist Medical Center /ID# 154586

Winston-Salem, North Carolina, United States

Site Status

Oregon Health and Science University /ID# 163822

Portland, Oregon, United States

Site Status

East Penn Rheumatology Assoc /ID# 159193

Bethlehem, Pennsylvania, United States

Site Status

Altoona Ctr Clinical Res /ID# 154572

Duncansville, Pennsylvania, United States

Site Status

University of Pittsburgh MC /ID# 157434

Pittsburgh, Pennsylvania, United States

Site Status

West Tennessee Research Inst /ID# 158721

Jackson, Tennessee, United States

Site Status

Adriana Pop-Moody MD Clinic PA /ID# 154607

Corpus Christi, Texas, United States

Site Status

P&I Clinical Research /ID# 159191

Lufkin, Texas, United States

Site Status

DM Clinical Research /ID# 158722

Tomball, Texas, United States

Site Status

Care Access Research /ID# 158098

Salt Lake City, Utah, United States

Site Status

Aprillus Asistencia e Investig /ID# 159173

Capital Federal, Buenos Aires, Argentina

Site Status

Ctr Privado Med Familiar /ID# 158814

Buenos Aires, , Argentina

Site Status

Atencion Integral en Reuma /ID# 155696

Buenos Aires, , Argentina

Site Status

Hospital General de Agudos /ID# 167117

Buenos Aires, , Argentina

Site Status

Inst. de Rehab. Psicofisica /ID# 167768

CABA, , Argentina

Site Status

Inst. Rheumatologic Strusberg /ID# 159021

Córdoba, , Argentina

Site Status

Instituto Medico DAMIC /ID# 167770

Córdoba, , Argentina

Site Status

DIM Clinica Privada /ID# 167769

Ramos Mejía, , Argentina

Site Status

Instituto CAICI SRL /ID# 159022

Rosario, Santa FE, , Argentina

Site Status

Rheumatology Research Unit /ID# 159174

Maroochydore, Queensland, Australia

Site Status

The Queen Elizabeth Hospital /ID# 159175

Woodville, South Australia, Australia

Site Status

Western Health Footscray Hospi /ID# 157968

Footscray, Victoria, Australia

Site Status

CHU UCL Namur /ID# 157628

Namur, , Belgium

Site Status

CEDOES-Centro de Diagnóstico e Pesquisa da Osteoporose do Espírito Santo LTDA /ID# 155228

Vitória, Espírito Santo, Brazil

Site Status

Santa Casa de Belo Horizonte /ID# 154631

Belo Horizonte, Minas Gerais, Brazil

Site Status

CMiP - Centro Mineiro de Pesquisa Ltda - ME /ID# 154564

Juiz de Fora, Minas Gerais, Brazil

Site Status

Ceti - Centro de Estudos Em Terapias Inovadoras Ltda /Id# 154634

Curitiba, Paraná, Brazil

Site Status

Hospital de Clinicas de Porto Alegre /ID# 161211

Porto Alegre, Rio Grande do Sul, Brazil

Site Status

LMK Sevicos Medicos S/S /ID# 159176

Porto Alegre, Rio Grande do Sul, Brazil

Site Status

CEMEC - Centro Multidisciplinar de Estudos Clínicos /ID# 154632

Santo André, São Paulo, Brazil

Site Status

CEPIC - Centro Paulista de Investigação Clínica e Serviços Médicos Ltda /ID# 159587

São Paulo, São Paulo, Brazil

Site Status

MHAT Trimontsium /ID# 155226

Plovdiv, , Bulgaria

Site Status

Diag Consult Ctr 17 Sofia EOOD /ID# 169298

Sofia, , Bulgaria

Site Status

UMHAT Sv. Ivan Rilski /ID# 155000

Sofia, , Bulgaria

Site Status

Medical Centre Synexus Sofia /ID# 201807

Sofia, , Bulgaria

Site Status

The Waterside Clinic /ID# 159178

Barrie, Ontario, Canada

Site Status

Adachi Medicine Prof. Corp /ID# 158024

Hamilton, Ontario, Canada

Site Status

Institut de Rhum. de Montreal /ID# 155001

Montreal, Quebec, Canada

Site Status

Groupe de Recherche en Maladies Osseuses /ID# 154601

Sainte-Foy, Quebec, Canada

Site Status

Revmatologicky ustav Praha /ID# 154612

Prague, Praha 2, Czechia

Site Status

Medical Plus, s.r.o. /ID# 155230

Uherské Hradište, , Czechia

Site Status

Uniklinik Koln /ID# 156047

Cologne, North Rhine-Westphalia, Germany

Site Status

Praxis fuer Rheumatologie /ID# 156156

Berlin, , Germany

Site Status

Rheumaforschungszentrum II /ID# 157177

Hamburg, , Germany

Site Status

Welcker, Planegg, DE /ID# 160185

Planegg, , Germany

Site Status

University General Hospital of Heraklion "PA.G.N.I" /ID# 163916

Heraklion, , Greece

Site Status

Budai Irgalmasrendi Korhaz /ID# 154457

Budapest, , Hungary

Site Status

Obudai Egeszsegugyi Centrum Kft. /ID# 156159

Budapest, , Hungary

Site Status

Debreceni Egyetem Kenezy Gyula Egyetemi Korhaz /ID# 159183

Debrecen, , Hungary

Site Status

Markhot Ferenc Oktatokorhaz es Rendelointezet /ID# 159689

Eger, , Hungary

Site Status

MAV Korhaz ess Rendelointezet /ID# 154455

Szolnok, , Hungary

Site Status

Our Lady's Hospital /ID# 161149

Manorhamilton, , Ireland

Site Status

Barzilai Medical Center /ID# 161685

Ashkelon, , Israel

Site Status

The Lady Davis Carmel MC /ID# 161686

Haifa, , Israel

Site Status

Meir Medical Center /ID# 162774

Kfar Saba, , Israel

Site Status

Sheba Medical Center /ID# 163154

Ramat Gan, , Israel

Site Status

Istituto Clinico Humanitas /ID# 154999

Rozzano, Milano, Italy

Site Status

AOU Citta della Salute Scienza /ID# 154577

Turin, Piedmont, Italy

Site Status

Presidio Columbus, Fondazione Policlinico Gemelli Universita Cattolica S. Cuore /ID# 162252

Rome, Roma, Italy

Site Status

A.O. Univ. Ospedali Riuniti /ID# 161707

Ancona, The Marches, Italy

Site Status

Azienda Ospedaliero Universitaria Policlinico Vittorio Emanuele /ID# 161172

Catania, , Italy

Site Status

ASST G. Pini /ID# 162223

Milan, , Italy

Site Status

D.Saulites-Kandevicas PP /ID# 154578

Liepāja, , Latvia

Site Status

Riga East Clinical Univ Hosp /ID# 155024

Riga, , Latvia

Site Status

Morales Vargas Centro de Investigacion S.C. /ID# 200800

León, Guanajuato, Mexico

Site Status

Centro Integral en Reumatología S.A de C.V /ID# 204493

Guadalajara, Jalisco, Mexico

Site Status

CINTRE, Centro de Investigación y Tratamiento Reumatológico SC /ID# 154579

Mexico City, Mexico City, Mexico

Site Status

RM Pharma Specialists S.A de C.V /ID# 159588

Mexico City, , Mexico

Site Status

Centro Especializado en Diabetes, Obesidad y Prevención de Enfermedades Cardiova /ID# 160126

Mexico City, , Mexico

Site Status

Antonius Ziekenhuis /ID# 155737

Sneek, Provincie Friesland, Netherlands

Site Status

Reade /ID# 161002

Amsterdam, , Netherlands

Site Status

Spaarne Gasthuis /ID# 161003

Haarlem, , Netherlands

Site Status

Medisch Centrum Leeuwarden /ID# 156043

Leeuwarden, , Netherlands

Site Status

Timaru Medical Specialists Ltd /ID# 159184

Timaru, , New Zealand

Site Status

Wellington Hospital (Capital and Coast District Health Board) /ID# 154591

Wellington, , New Zealand

Site Status

Medyczne Centrum Hetmanska /ID# 155746

Poznan, Greater Poland Voivodeship, Poland

Site Status

Malopolskie Centrum Kliniczne /ID# 157180

Krakow, Lesser Poland Voivodeship, Poland

Site Status

Centrum Medyczne AMED Warszawa Targowek /ID# 159589

Warsaw, Masovian Voivodeship, Poland

Site Status

Gabinet Internistyczno Reum. /ID# 157433

Bialystok, Podlaskie Voivodeship, Poland

Site Status

ClinicMed Daniluk, Nowak Sp.j. /ID# 202998

Bialystok, Podlaskie Voivodeship, Poland

Site Status

Synexus Polska Sp. z o.o. Oddzial w Gdyni /ID# 202472

Gdynia, Pomeranian Voivodeship, Poland

Site Status

Centrum Med Amed Oddzial Lodzi /ID# 154458

Lodz, , Poland

Site Status

Salve Medica Sp. z o.o. S.K. /ID# 202473

Lodz, Łódź Voivodeship, Poland

Site Status

Instituto Portugues De Reumatologia /ID# 155698

Lisbon, Lisbon District, Portugal

Site Status

Centro Hospitalar Lisboa Ocidental, EPE /ID# 200035

Lisbon, Lisbon District, Portugal

Site Status

Hospital Garcia de Orta, E.P.E /ID# 164056

Almada, Setúbal District, Portugal

Site Status

Centro Hospitalar Lisboa Norte, EPE /ID# 200037

Lisbon, , Portugal

Site Status

Unidade Local De Saude Do Alto Minho /ID# 200036

Viana do Castelo, , Portugal

Site Status

Centro Hosp de Tondela-Viseu /ID# 155699

Viseu, , Portugal

Site Status

Dr. Ramon L. Ortega-Colon, MD /ID# 158097

Carolina, , Puerto Rico

Site Status

GCM Medical Group /ID# 156158

San Juan, , Puerto Rico

Site Status

Spitalul Clinic Dr. I. Cantacuzino /ID# 155893

Bucharest, București, Romania

Site Status

Spitalul Clinic Sf. Maria /ID# 167245

Bucharest, , Romania

Site Status

Family Outpatient clinic#4 LLC /ID# 203524

Korolev, Moscow, Russia

Site Status

LLC Medical Center /ID# 203523

Novosibirsk, Novosibirsk Oblast, Russia

Site Status

Alliance Biomedical Ural Group /ID# 154609

Izhevsk, Udmurtiya Republic, Russia

Site Status

State Budget Healthcare Instit /ID# 154593

Moscow, , Russia

Site Status

Nort-Western State Medical Uni /ID# 154610

Saint Petersburg, , Russia

Site Status

Novamed,spol.s.r.o. /ID# 157928

Banská Bystrica, , Slovakia

Site Status

Univerzitna Nemocnica Bratislava /ID# 161143

Bratislava, , Slovakia

Site Status

Narodny ustav reumatickych chorob Piestany /ID# 156864

Pieštany, , Slovakia

Site Status

SMG-SNU Boramae Medical Center /ID# 155788

Seoul, Seoul Teugbyeolsi, South Korea

Site Status

The Catholic University of Korea, Yeouido St. Mary's Hospital /ID# 155231

Seoul, Seoul Teugbyeolsi, South Korea

Site Status

Asan Medical Center /ID# 154639

Seoul, , South Korea

Site Status

Hospital Universitario Reina S /ID# 155701

Córdoba, , Spain

Site Status

Hospital General Univ de Elche /ID# 158825

Elche, , Spain

Site Status

Hospital Universitario La Paz /ID# 163636

Madrid, , Spain

Site Status

Corp Sanitaria Parc Tauli /ID# 163634

Sabadell, Barcelona, , Spain

Site Status

Complejo Hospitalario /ID# 155700

Santiago de Compostela, , Spain

Site Status

Hospital Infanta Luisa /ID# 154641

Seville, , Spain

Site Status

Skanes Universitetssjukhus /ID# 165133

Malmo, Skåne County, Sweden

Site Status

Akademiskt specialistcentrum Centrum for reumatologi /ID# 156046

Stockholm, Stockholm County, Sweden

Site Status

Sahlgrenska University Hosp /ID# 162775

Gothenburg, , Sweden

Site Status

Vastmanlands Sjukhus /ID# 159186

Västerås, , Sweden

Site Status

Hopitaux Universitaires de Geneve /ID# 159083

Geneva, Canton of Geneva, Switzerland

Site Status

Kantonsspital St. Gallen /ID# 155232

Sankt Gallen, Canton of St. Gallen, Switzerland

Site Status

University Hospital of Basel /ID# 160860

Basel, , Switzerland

Site Status

HFR Fribourg - Hopital Canton /ID# 160970

Fribourg, , Switzerland

Site Status

Hacettepe University Medical Faculty /ID# 167995

Ankara, , Turkey (Türkiye)

Site Status

Ankara Univ Medical Faculty /ID# 162691

Ankara, , Turkey (Türkiye)

Site Status

Akdeniz University Faculty /ID# 163153

Antalya, , Turkey (Türkiye)

Site Status

Istanbul Fizik Tedavi Rehabilitasyon Egitim ve Arastırma Hastanesi /ID# 169479

Istanbul, , Turkey (Türkiye)

Site Status

Whipps Cross Univ Hospital /ID# 205985

London, London, City of, United Kingdom

Site Status

Ninewells Hospital /ID# 156050

Dundee, , United Kingdom

Site Status

Altnagelvin Area Hospital /ID# 156540

Londonderry, , United Kingdom

Site Status

Lancashire Care NHS Foundation /ID# 156042

Preston, , United Kingdom

Site Status

Royal Cornwall Hospital /ID# 157785

Truro, , United Kingdom

Site Status

Countries

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United States Argentina Australia Belgium Brazil Bulgaria Canada Czechia Germany Greece Hungary Ireland Israel Italy Latvia Mexico Netherlands New Zealand Poland Portugal Puerto Rico Romania Russia Slovakia South Korea Spain Sweden Switzerland Turkey (Türkiye) United Kingdom

References

Explore related publications, articles, or registry entries linked to this study.

Rubbert-Roth A, Enejosa J, Pangan AL, Haraoui B, Rischmueller M, Khan N, Zhang Y, Martin N, Xavier RM. Trial of Upadacitinib or Abatacept in Rheumatoid Arthritis. N Engl J Med. 2020 Oct 15;383(16):1511-1521. doi: 10.1056/NEJMoa2008250.

Reference Type BACKGROUND
PMID: 33053283 (View on PubMed)

Burmester GR, Deodhar A, Irvine AD, Panaccione R, Winthrop KL, Vleugels RA, Levy G, Suravaram S, Palac H, Wegrzyn L, Ford S, Meerwein S, Guttman-Yassky E. Safety Profile of Upadacitinib: Descriptive Analysis in Over 27,000 Patient-Years Across Rheumatoid Arthritis, Psoriatic Arthritis, Axial Spondyloarthritis, Atopic Dermatitis, and Inflammatory Bowel Disease. Adv Ther. 2025 Oct;42(10):5215-5237. doi: 10.1007/s12325-025-03328-y. Epub 2025 Aug 28.

Reference Type DERIVED
PMID: 40875187 (View on PubMed)

Rubbert-Roth A, Kato K, Haraoui B, Rischmueller M, Liu Y, Khan N, Camp HS, Xavier RM. Safety and Efficacy of Upadacitinib in Patients with Rheumatoid Arthritis Refractory to Biologic DMARDs: Results Through Week 216 from the SELECT-CHOICE Study. Rheumatol Ther. 2024 Oct;11(5):1197-1215. doi: 10.1007/s40744-024-00694-x. Epub 2024 Jul 20.

Reference Type DERIVED
PMID: 39031276 (View on PubMed)

Rubbert-Roth A, Kakehasi AM, Takeuchi T, Schmalzing M, Palac H, Coombs D, Liu J, Anyanwu SI, Lippe R, Curtis JR. Malignancy in the Upadacitinib Clinical Trials for Rheumatoid Arthritis, Psoriatic Arthritis, Ankylosing Spondylitis, and Non-radiographic Axial Spondyloarthritis. Rheumatol Ther. 2024 Feb;11(1):97-112. doi: 10.1007/s40744-023-00621-6. Epub 2023 Nov 20.

Reference Type DERIVED
PMID: 37982966 (View on PubMed)

Charles-Schoeman C, Choy E, McInnes IB, Mysler E, Nash P, Yamaoka K, Lippe R, Khan N, Shmagel AK, Palac H, Suboticki J, Curtis JR. MACE and VTE across upadacitinib clinical trial programmes in rheumatoid arthritis, psoriatic arthritis and ankylosing spondylitis. RMD Open. 2023 Nov;9(4):e003392. doi: 10.1136/rmdopen-2023-003392.

Reference Type DERIVED
PMID: 37945286 (View on PubMed)

Fleischmann R, Curtis JR, Charles-Schoeman C, Mysler E, Yamaoka K, Richez C, Palac H, Dilley D, Liu J, Strengholt S, Burmester G. Safety profile of upadacitinib in patients at risk of cardiovascular disease: integrated post hoc analysis of the SELECT phase III rheumatoid arthritis clinical programme. Ann Rheum Dis. 2023 Sep;82(9):1130-1141. doi: 10.1136/ard-2023-223916. Epub 2023 Jun 12.

Reference Type DERIVED
PMID: 37308218 (View on PubMed)

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Kakehasi AM, Radominski SC, Baravalle MD, Palazuelos FCI, Garcia-Garcia C, Arruda MS, Curi M, Liu J, Qiao M, Velez-Sanchez P, Vargas JI. Safety of upadacitinib in Latin American patients with rheumatoid arthritis: an integrated safety analysis of the SELECT phase 3 clinical program. Clin Rheumatol. 2023 May;42(5):1249-1258. doi: 10.1007/s10067-023-06513-y. Epub 2023 Jan 30.

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Provided Documents

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Document Type: Study Protocol

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Document Type: Statistical Analysis Plan

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Other Identifiers

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2016-000933-37

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

M15-925

Identifier Type: -

Identifier Source: org_study_id

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