Efficacy of Oral Azacitidine Plus Best Supportive Care as Maintenance Therapy in Subjects With Acute Myeloid Leukemia (AML) in Complete Remission

NCT ID: NCT01757535

Last Updated: 2025-07-08

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

472 participants

Study Classification

INTERVENTIONAL

Study Start Date

2013-04-24

Study Completion Date

2024-06-18

Brief Summary

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This study enrolled 472 participants, aged 55 or older, with a diagnosis of de novo acute myeloid leukemia (AML) or AML secondary to prior myelodysplastic disease or chronic myelomonocytic leukemia (CMML), and who have achieved first complete remission (CR)/ complete remission with incomplete blood count recovery (CRi) following induction with or without consolidation chemotherapy.

The study is amended to include an extension phase (EP). The EP allows participants who are currently receiving oral azacitidine and who are demonstrating clinical benefit as assessed by the investigator, to continue receiving oral azacitidine after unblinding by sponsor until the participant meets the criteria for study discontinuation or until oral azacitidine becomes commercially available and reimbursed. In addition, all participants in the placebo arm and participants who had been discontinued from the treatment phase (irrespective of randomization arm) and continuing in the follow-up phase will be followed for survival in the EP.

Detailed Description

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This is an international, multicenter, placebo-controlled, Phase 3 study with a double-blind, randomized, parallel-group design in subjects with de novo AML or AML secondary to prior diagnosis of myelodysplastic syndromes (MDS) or chronic myelomonocytic leukemia (CMML) aged ≥ 55 years, who are in first CR/CRi following induction therapy with or without consolidation chemotherapy. The study consists of 3 phases; the pre-randomization phase (screening phase), the treatment phase, and the follow-up phase.

The study is amended to include an extension phase (EP). The EP allows participants who are currently receiving oral azacitidine and who are demonstrating clinical benefit as assessed by the Investigator, to continue receiving oral azacitidine after unblinding by sponsor until they meet the criteria for study discontinuation or until oral azacitidine becomes commercially available and reimbursed. In addition, all participants in the placebo arm and participants who had been discontinued from the treatment phase (irrespective of randomization arm) and continuing in the follow-up phase will be followed for survival in the EP.

Conditions

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Leukemia, Myeloid, Acute

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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Oral Azacitidine

300 mg oral azacitidine on days 1 to 14 of each 28-day treatment cycle.

Group Type EXPERIMENTAL

Oral Azacitidine

Intervention Type DRUG

300 mg oral azacitidine on days 1 to 14 of each 28-day treatment cycle.

Placebo

Identically matching placebo tablets on days 1 to 14 of each 28-day treatment cycle.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Identically matching placebo tablets on days 1 to 14 of each 28-day treatment cycle.

Interventions

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Oral Azacitidine

300 mg oral azacitidine on days 1 to 14 of each 28-day treatment cycle.

Intervention Type DRUG

Placebo

Identically matching placebo tablets on days 1 to 14 of each 28-day treatment cycle.

Intervention Type DRUG

Other Intervention Names

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CC-486; Onureg®

Eligibility Criteria

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Inclusion Criteria

1. Male or female participants ≥ 55 years of age
2. Newly diagnosed, histologically confirmed de novo acute myeloid leukemia (AML) or AML secondary to prior myelodysplastic disease or CMML (Chronic myelomonocytic leukemia)
3. First complete remission (CR)/ complete remission with incomplete blood count recovery (CRi) with induction therapy with intensive chemotherapy with or without consolidation therapy within 4 months (+/- 7 days of achieving CR or CRi)
4. Eastern Cooperative Oncology Group (ECOG) performance status - 0, 1, 2, 3


At the Investigator's discretion and with approval of the sponsor, participants meeting all of the following eligibility criteria are eligible to enter the extension phase:

1. All participants randomized into the oral azacitidine or placebo arm and are continuing in either the treatment phase or follow-up phase of the CC-486-AML-001 study;

* Participants randomized to oral azacitidine treatment arm and continuing in the treatment phase demonstrating clinical benefit as assessed by the investigator are eligible to receive oral azacitidine in the extension phase (EP);
* Participants randomized into placebo arm of the study will not receive oral azacitidine in the EP, but will be followed for survival in the EP;
* Participants currently in the follow-up phase will continue to be followed for survival in the EP;
2. Participants who have signed the informed consent for the EP of the study;
3. Participants who do not meet any of the criteria for study discontinuation

Exclusion Criteria

1. AML with inversion (inv)(16), translocation = t(8;21), t(16;16), t(15;17), or t(9;22) or molecular evidence of such translocations
2. Prior bone marrow or stem cell transplantation
3. Have achieved CR/CRi following therapy with hypomethylating agents
4. Diagnosis of malignant disease within the previous 12 months
5. Proven central nervous system (CNS) leukemia
Minimum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Celgene

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Bristol-Myers Squibb

Role: STUDY_DIRECTOR

Bristol-Myers Squibb

Locations

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Arizona Oncology Associates, P.C.

Phoenix, Arizona, United States

Site Status

Providence St Joseph Medical Center Cancer Center

Burbank, California, United States

Site Status

City Of Hope

Duarte, California, United States

Site Status

University of California San Francisco Fresno Campus

Fresno, California, United States

Site Status

University of Southern California Norris Cancer Center

Los Angeles, California, United States

Site Status

Local Institution - 006

Los Angeles, California, United States

Site Status

Local Institution - 050

Orange, California, United States

Site Status

Sharp Memorial Hospital

San Diego, California, United States

Site Status

Stanford Cancer Center

Stanford, California, United States

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Innovative Clinical Research Institute

Whittier, California, United States

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Rocky Mountain Cancer Center

Denver, Colorado, United States

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Local Institution - 010

Southington, Connecticut, United States

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George Washington University Cancer Center

Washington D.C., District of Columbia, United States

Site Status

Local Institution - 046

Gainesville, Florida, United States

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Mount Sinai Comprehensive Cancer Center

Miami Beach, Florida, United States

Site Status

Local Institution - 044

Orlando, Florida, United States

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Northwestern University Medical Center

Chicago, Illinois, United States

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Loyola University Chicago

Maywood, Illinois, United States

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Cancer Care and Hematology Specialists of Chicagoland, P.C. - Niles, IL

Niles, Illinois, United States

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Local Institution - 013

Indianapolis, Indiana, United States

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Franciscan St. Francis Health

Indianapolis, Indiana, United States

Site Status

Local Institution - 003

Westwood, Kansas, United States

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Local Institution - 049

Louisville, Kentucky, United States

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Local Institution - 058

Louisville, Kentucky, United States

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Local Institution - 047

New Orleans, Louisiana, United States

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Ochsner Medical Center - Jefferson Highway

New Orleans, Louisiana, United States

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Massachusetts General Hospital

Boston, Massachusetts, United States

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Beth Israel Deaconess Medical Center

Boston, Massachusetts, United States

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Local Institution - 015

Worcester, Massachusetts, United States

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Local Institution - 037

Rochester, Minnesota, United States

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Local Institution - 023

Kansas City, Missouri, United States

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Washington University School Of Medicine

St Louis, Missouri, United States

Site Status

Local Institution - 057

Omaha, Nebraska, United States

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John Theurer Cancer Center at Hackensack University Medical Center

Hackensack, New Jersey, United States

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Cancer Institute of New Jersey

New Brunswick, New Jersey, United States

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Winthrop University Hospital

Mineola, New York, United States

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Local Institution - 009

New York, New York, United States

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Columbia University Irving Medical Center

New York, New York, United States

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Local Institution - 002

New York, New York, United States

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Local Institution - 004

Rochester, New York, United States

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Local Institution - 014

Valhalla, New York, United States

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Duke University Medical Center

Durham, North Carolina, United States

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Local Institution - 025

Winston-Salem, North Carolina, United States

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Local Institution - 016

Cleveland, Ohio, United States

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University of Oklahoma Peggy and Charles Stephenson Cancer Center

Oklahoma City, Oklahoma, United States

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Kaiser Permanente Northwest Oncology Hematology

Portland, Oregon, United States

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Lancaster General Hospital

Lancaster, Pennsylvania, United States

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UPMC Cancer Pavillion

Pittsburgh, Pennsylvania, United States

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Greenville Hospital System

Greenville, South Carolina, United States

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Local Institution - 011

Nashville, Tennessee, United States

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Local Institution - 007

Nashville, Tennessee, United States

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Local Institution - 041

Dallas, Texas, United States

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Fort Sam Houston, Texas, United States

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Houston, Texas, United States

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Cancer Care Centers of South Texas - Loop

San Antonio, Texas, United States

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Local Institution - 039

San Antonio, Texas, United States

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Local Institution - 035

Richmond, Virginia, United States

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Swedish Cancer Inst

Seattle, Washington, United States

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Yakima Valley Memorial Hospital/ North Star Lodge

Yakima, Washington, United States

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Froedtert Hospital BMT Medical College of Wisconsin

Milwaukee, Wisconsin, United States

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Local Institution - 510

Wollongong, New South Wales, Australia

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Local Institution - 509

South Brisbane, Queensland, Australia

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Local Institution - 508

Adelaide, South Australia, Australia

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Bedford Park, South Australia, Australia

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Woodville South, South Australia, Australia

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Heidelberg, , Australia

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Hobart, , Australia

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Liverpool, , Australia

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Melbourne, , Australia

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Perth, , Australia

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Perth, , Australia

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St Leonards, , Australia

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Woolloongabba, , Australia

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Graz, , Austria

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Salzburg, , Austria

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Vienna, , Austria

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Vienna, , Austria

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Vienna, , Austria

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Bruges, , Belgium

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Charleroi, , Belgium

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Mons, , Belgium

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Curitiba, Paraná, Brazil

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Porto Alegre, Rio Grande do Sul, Brazil

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Rio de Janeiro, , Brazil

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São Paulo, , Brazil

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São Paulo, , Brazil

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Edmonton, Alberta, Canada

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Winnipeg, Manitoba, Canada

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Saint John, New Brunswick, Canada

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St. John's, Newfoundland and Labrador, Canada

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Halifax, Nova Scotia, Canada

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Toronto, Ontario, Canada

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Montreal, Quebec, Canada

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Montreal, Quebec, Canada

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Brno, South Moravian, Czechia

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Prague, , Czechia

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Prague, , Czechia

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Helsinki, , Finland

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Tampere, , Finland

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Turku, , Finland

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Amiens, , France

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Argenteuil, , France

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Bobigny, , France

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Boulognes Sur Mer, , France

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Clamart, , France

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Créteil, , France

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Le Chesnay, , France

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Lille, , France

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Limoges, , France

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Lyon, , France

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Paris, , France

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Paris, , France

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Paris, , France

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Pontoise, , France

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Rouen, , France

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Saint-Cloud, , France

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Villejuif, , France

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Dresden, Saxony, Germany

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Berlin, , Germany

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Bonn, , Germany

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Düsseldorf, , Germany

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Erlangen, , Germany

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Frankfurt am Main, , Germany

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Goch, , Germany

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Hanover, , Germany

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Heilbronn, , Germany

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Jena, , Germany

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Keil, , Germany

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Mannheim, , Germany

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München, , Germany

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München, , Germany

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Oldenburg, , Germany

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Schweiler, , Germany

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Ulm, , Germany

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Dublin, , Ireland

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Galway, , Ireland

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Beersheba, , Israel

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Haifa, , Israel

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Jerusalem, , Israel

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Petah Tikva, , Israel

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Alessandria, , Italy

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Bari, , Italy

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Bologna, , Italy

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Cagliari, , Italy

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Cremona, , Italy

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Florence, , Italy

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Genova, , Italy

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Lecce, , Italy

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Milan, , Italy

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Milan, , Italy

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Monza, , Italy

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Naples, , Italy

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Naples, , Italy

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Orbassano (TO), , Italy

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Palermo, , Italy

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Palermo, , Italy

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Pesaro, , Italy

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Reggio Calabria, , Italy

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Roma, , Italy

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Roma, , Italy

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Roma, , Italy

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Rome, , Italy

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Torino, , Italy

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Torino, , Italy

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Udine, , Italy

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Varese, , Italy

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Klaipėda, , Lithuania

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Huixquilucan de Degollado, , Mexico

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México, , Mexico

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Monterrey, , Mexico

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Bydgoszcz, , Poland

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Gdansk, , Poland

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Lodz, , Poland

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Warsaw, , Poland

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Wroclaw, , Poland

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Coimbra, , Portugal

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Lisbon, , Portugal

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Lisbon, , Portugal

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Porto, , Portugal

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Porto, , Portugal

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Moscow, , Russia

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Nizhny Novgorod, , Russia

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Saint Petersburg, , Russia

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Saint Petersburg, , Russia

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Busan, , South Korea

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Daegu, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Palma de Mallorca, Balearic Islands, Spain

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A Coruña, , Spain

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Badalona (Barcelona), , Spain

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Barcelona, , Spain

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Barcelona, , Spain

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Cáceres, , Spain

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Córdoba, , Spain

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Madrid, , Spain

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Madrid, , Spain

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Madrid, , Spain

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Oviedo, , Spain

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Salamanca, , Spain

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Seville, , Spain

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Valencia, , Spain

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Beitou District, Taipei City, , Taiwan

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Niaosong District Kaohsiung City, , Taiwan

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Taichung, Northern Dist., , Taiwan

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Tainan, Taiana, , Taiwan

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Taipei, Zhongzheng Dist., , Taiwan

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Ankara, , Turkey (Türkiye)

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Ankara, , Turkey (Türkiye)

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Local Institution - 651

Istanbul, , Turkey (Türkiye)

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Samsun, , Turkey (Türkiye)

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Local Institution - 904

Nottingham, Nottinghamshire, United Kingdom

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Local Institution - 907

Boston, , United Kingdom

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Brighton East Sussex, , United Kingdom

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Canterbury Kent, , United Kingdom

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London, , United Kingdom

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London, , United Kingdom

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London, , United Kingdom

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Maidstone, , United Kingdom

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Local Institution - 900

Manchester, , United Kingdom

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Local Institution - 906

Romford, Essex, , United Kingdom

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Countries

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United States Australia Austria Belgium Brazil Canada Czechia Finland France Germany Ireland Israel Italy Lithuania Mexico Poland Portugal Russia South Korea Spain Taiwan Turkey (Türkiye) United Kingdom

References

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Roboz GJ, Montesinos P, Selleslag D, Wei A, Jang JH, Falantes J, Voso MT, Sayar H, Porkka K, Marlton P, Almeida A, Mohan S, Ravandi F, Garcia-Manero G, Skikne B, Kantarjian H. Design of the randomized, Phase III, QUAZAR AML Maintenance trial of CC-486 (oral azacitidine) maintenance therapy in acute myeloid leukemia. Future Oncol. 2016 Feb;12(3):293-302. doi: 10.2217/fon.15.326. Epub 2016 Jan 19.

Reference Type BACKGROUND
PMID: 26785287 (View on PubMed)

Ravandi F, Dohner H, Wei AH, Montesinos P, Pfeilstocker M, Papayannidis C, Lai Y, Wang K, See WL, de Menezes DL, Petrlik E, Prebet T, Roboz GJ. Survival outcomes in patients with acute myeloid leukaemia who received subsequent therapy for relapse in QUAZAR AML-001. Br J Haematol. 2024 Mar;204(3):877-886. doi: 10.1111/bjh.19202. Epub 2023 Nov 12.

Reference Type DERIVED
PMID: 37952982 (View on PubMed)

Wei AH, Roboz GJ, Dombret H, Dohner H, Schuh AC, Montesinos P, Selleslag D, Bondarenko SN, Prebet T, Lai Y, Skikne B, Beach CL, Ravandi F. Survival outcomes with oral azacitidine maintenance in patients with acute myeloid leukemia in remission by receipt of initial chemotherapy: subgroup analyses from the phase III QUAZAR AML-001 trial. Haematologica. 2023 Oct 1;108(10):2820-2825. doi: 10.3324/haematol.2022.282296. No abstract available.

Reference Type DERIVED
PMID: 36951156 (View on PubMed)

Dohner H, Wei AH, Roboz GJ, Montesinos P, Thol FR, Ravandi F, Dombret H, Porkka K, Sandhu I, Skikne B, See WL, Ugidos M, Risueno A, Chan ET, Thakurta A, Beach CL, Lopes de Menezes D. Prognostic impact of NPM1 and FLT3 mutations in patients with AML in first remission treated with oral azacitidine. Blood. 2022 Oct 13;140(15):1674-1685. doi: 10.1182/blood.2022016293.

Reference Type DERIVED
PMID: 35960871 (View on PubMed)

Zhu J, Wu Q, Wang J, Niu T. Cost-effectiveness analysis of azacitidine maintenance therapy in patients with acute myeloid leukemia. Expert Rev Hematol. 2022 Apr;15(4):375-382. doi: 10.1080/17474086.2022.2061456. Epub 2022 May 11.

Reference Type DERIVED
PMID: 35437111 (View on PubMed)

Roboz GJ, Ravandi F, Wei AH, Dombret H, Thol F, Voso MT, Schuh AC, Porkka K, La Torre I, Skikne B, Zhong J, Beach CL, Risueno A, Menezes DL, Ossenkoppele G, Dohner H. Oral azacitidine prolongs survival of patients with AML in remission independently of measurable residual disease status. Blood. 2022 Apr 7;139(14):2145-2155. doi: 10.1182/blood.2021013404.

Reference Type DERIVED
PMID: 34995344 (View on PubMed)

Ravandi F, Roboz GJ, Wei AH, Dohner H, Pocock C, Selleslag D, Montesinos P, Sayar H, Musso M, Figuera-Alvarez A, Safah H, Tse W, Sohn SK, Hiwase D, Chevassut T, Pierdomenico F, La Torre I, Skikne B, Bailey R, Zhong J, Beach CL, Dombret H. Management of adverse events in patients with acute myeloid leukemia in remission receiving oral azacitidine: experience from the phase 3 randomized QUAZAR AML-001 trial. J Hematol Oncol. 2021 Aug 28;14(1):133. doi: 10.1186/s13045-021-01142-x.

Reference Type DERIVED
PMID: 34454540 (View on PubMed)

Wei AH, Dohner H, Pocock C, Montesinos P, Afanasyev B, Dombret H, Ravandi F, Sayar H, Jang JH, Porkka K, Selleslag D, Sandhu I, Turgut M, Giai V, Ofran Y, Kizil Cakar M, Botelho de Sousa A, Rybka J, Frairia C, Borin L, Beltrami G, Cermak J, Ossenkoppele GJ, La Torre I, Skikne B, Kumar K, Dong Q, Beach CL, Roboz GJ; QUAZAR AML-001 Trial Investigators. Oral Azacitidine Maintenance Therapy for Acute Myeloid Leukemia in First Remission. N Engl J Med. 2020 Dec 24;383(26):2526-2537. doi: 10.1056/NEJMoa2004444.

Reference Type DERIVED
PMID: 33369355 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Related Links

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Other Identifiers

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2012-003457-28

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

CC-486-AML-001

Identifier Type: -

Identifier Source: org_study_id

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