Safety and Efficacy of Combination Saxagliptin & Dapagliflozin Added to Metformin to Treat Subjects With Type 2 Diabetes

NCT ID: NCT01606007

Last Updated: 2017-05-15

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

1282 participants

Study Classification

INTERVENTIONAL

Study Start Date

2012-07-31

Study Completion Date

2014-01-31

Brief Summary

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The purpose of this study is to learn if a combination of BMS-477118 (Saxagliptin) and BMS -512148 (Dapagliflozin) added to Metformin can improve (decrease) Glycosylated Hemoglobin (Hemoglobin A1c) in patients with type 2 diabetes after 24 weeks of treatment. The safety of this treatment will also be studied.

Detailed Description

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Conditions

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Type 2 Diabetes

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Caregivers Investigators

Study Groups

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Arm 1: Saxagliptin+Metformin XR+Placebo

Group Type ACTIVE_COMPARATOR

Saxagliptin

Intervention Type DRUG

Tablets, Oral, 5mg , Once daily, 24 weeks

Metformin XR

Intervention Type DRUG

Tablets, Oral, ≥ 1500mg/≤ 2000mg, Once daily, 24 weeks

Placebo matching with Dapagliflozin

Intervention Type DRUG

Tablets, Oral, 0mg, Once daily, 24 weeks

Arm 2: Dapagliflozin+Metformin XR+Placebo

Group Type ACTIVE_COMPARATOR

Metformin XR

Intervention Type DRUG

Tablets, Oral, ≥ 1500mg/≤ 2000mg, Once daily, 24 weeks

Dapagliflozin

Intervention Type DRUG

Tablets, Oral, 10mg , Once daily, 24 weeks

Placebo matching with Saxagliptin

Intervention Type DRUG

Tablets, Oral, 0mg, Once daily, 24 weeks

Arm 3: Saxagliptin+Dapagliflozin+Metformin XR

Group Type EXPERIMENTAL

Saxagliptin

Intervention Type DRUG

Tablets, Oral, 5mg , Once daily, 24 weeks

Metformin XR

Intervention Type DRUG

Tablets, Oral, ≥ 1500mg/≤ 2000mg, Once daily, 24 weeks

Dapagliflozin

Intervention Type DRUG

Tablets, Oral, 10mg , Once daily, 24 weeks

Interventions

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Saxagliptin

Tablets, Oral, 5mg , Once daily, 24 weeks

Intervention Type DRUG

Metformin XR

Tablets, Oral, ≥ 1500mg/≤ 2000mg, Once daily, 24 weeks

Intervention Type DRUG

Dapagliflozin

Tablets, Oral, 10mg , Once daily, 24 weeks

Intervention Type DRUG

Placebo matching with Dapagliflozin

Tablets, Oral, 0mg, Once daily, 24 weeks

Intervention Type DRUG

Placebo matching with Saxagliptin

Tablets, Oral, 0mg, Once daily, 24 weeks

Intervention Type DRUG

Other Intervention Names

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Onglyza Glucophage XR BMS-512148

Eligibility Criteria

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Inclusion Criteria

* Subjects with Type 2 diabetes mellitus (T2DM) with HbA1c ≥ 8.0% and ≤ 12.0%
* Stable metformin therapy dose of ≥ 1500mg for at least 8 weeks prior to screening
* Body mass index (BMI) ≤ 45.0kg/m2

Exclusion Criteria

* Estimated glomerular filtration rate (eGFR) \< 60mL/min/1,73m2 and Serum Creatinine (Scr) ≥ 1.5 mg/dL in males or ≥ 1.4 mg/dL in females
* Uncontrolled hypertension Systolic Blood Pressure (SBP) ≥ 160mmHg and/or Diastolic Blood Pressure (DBP) ≥ 100mmHg
* Hepatic disease
* Cardiovascular disease within 3 months
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Bristol-Myers Squibb

Role: STUDY_DIRECTOR

Bristol-Myers Squibb

Locations

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Central Alabama Research

Birmingham, Alabama, United States

Site Status

Central Alabama Research

Homewood, Alabama, United States

Site Status

Terence T. Hart, Md

Muscle Shoals, Alabama, United States

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International Institute Of Clinical Research

Ozark, Alabama, United States

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Clinical Research Advantage

Mesa, Arizona, United States

Site Status

Elite Clinical Studies, Llc

Phoenix, Arizona, United States

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Genova Clinical Research

Tucson, Arizona, United States

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Medical Investigations, Inc.

Little Rock, Arkansas, United States

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Aureus Research, Inc.

Little Rock, Arkansas, United States

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Southland Clinical Research Center, Inc.

Fountain Valley, California, United States

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Torrance Clinical Research

Lomita, California, United States

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National Research Inst

Los Angeles, California, United States

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Providence Clinical Research

North Hollywood, California, United States

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Diabetes Medical Center Of California

Northridge, California, United States

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Mehrdad Kevin Ariani Md, Inc.

Northridge, California, United States

Site Status

Lucita M. Cruz,Md.,Inc.

Norwalk, California, United States

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Center For Clinical Trials, Llc.

Paramount, California, United States

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Center For Clinical Trials Of Sacramento, Inc.

Sacramento, California, United States

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Trinitas Research, Inc

San Jose, California, United States

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Orange County Research Center

Tustin, California, United States

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Clinical Research Advantage

Colorado Springs, Colorado, United States

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Infocus Clinical Research

Denver, Colorado, United States

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Lynn Institute Of Denver

Denver, Colorado, United States

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Southeast Clinical Research, Llc

Chiefland, Florida, United States

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Clinical Therapeutics Corporation

Coral Gables, Florida, United States

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Southeast Clinical Research, Llc

Jacksonville, Florida, United States

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Fpa Clinical Research

Kissimmee, Florida, United States

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Clinical Research Of Miami, Inc.

Miami, Florida, United States

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Advanced Pharma Cr, Llc

Miami, Florida, United States

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Newphase Clinical Trials, Inc.

Miami Beach, Florida, United States

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Omega Research Consultants, Llc

Orlando, Florida, United States

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Palm Harbor Medical Associates

Palm Harbor, Florida, United States

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Andres Patron, Do Pa

Pembroke Pines, Florida, United States

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Endocrine Research Solutions, Inc.

Roswell, Georgia, United States

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Cedar Crosse Research Center

Chicago, Illinois, United States

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Deerbrook Medical Associates

Vernon Hills, Illinois, United States

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Clinical Research Advantage

Council Bluffs, Iowa, United States

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Horizon Research Group Of Opelousas, Llc

Eunice, Louisiana, United States

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Associated Internal Medicine Specialists

Battle Creek, Michigan, United States

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Harris And Associates, P.C.

Detroit, Michigan, United States

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Patterson Medical Clinic

Florissant, Missouri, United States

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Bellevue Family Practice

Bellevue, Nebraska, United States

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Clinical Research Advantage

Elkhorn, Nebraska, United States

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Clinical Research Advantage

Fremont, Nebraska, United States

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Clinical Research Advantage

Omaha, Nebraska, United States

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South Jersey Medical Associates, P.A.

Blackwood, New Jersey, United States

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Central Jersey Health And Medical Research

Elizabeth, New Jersey, United States

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Southgate Medical Group

West Seneca, New York, United States

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Metrolina Internal Medicine

Charlotte, North Carolina, United States

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Triad Clinical Trials, Llc

Greensboro, North Carolina, United States

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Diabetes & Endocrinology Consultants

Morehead City, North Carolina, United States

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Pmg Research Of Winston-Salem, Llc

Winston-Salem, North Carolina, United States

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Daystar Clinical Resarch, Inc.

Akron, Ohio, United States

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Sterling Research Grp, Ltd.

Cincinnati, Ohio, United States

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Rapid Medical Research, Inc.

Cleveland, Ohio, United States

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Primed Clinical Research

Dayton, Ohio, United States

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Physicians Research, Inc.

Zanesville, Ohio, United States

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Lynn Institute Of Norman

Norman, Oklahoma, United States

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Willamette Valley Clinical Studies

Eugene, Oregon, United States

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Oregon Clinical Research

Portland, Oregon, United States

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Heritage Valley Medical Group

Beaver, Pennsylvania, United States

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Wellmon Family Practice

Shippensburg, Pennsylvania, United States

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Tlm Medical Services

Columbia, South Carolina, United States

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Palmetto Clinical Trial Services Llc

Fountain Inn, South Carolina, United States

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Holston Medical Group

Bristol, Tennessee, United States

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Holston Medical Group

Kingsport, Tennessee, United States

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Pmg Research Of Knoxville

Knoxville, Tennessee, United States

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Arlington Family Research Center, Inc.

Arlington, Texas, United States

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Padre Coast Clinical Research

Corpus Christi, Texas, United States

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Dallas Diabetes & Endocrine Center

Dallas, Texas, United States

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Excel Clinical Research, Llc

Houston, Texas, United States

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North Hills Medical Research, Inc.

North Richland Hills, Texas, United States

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Med-Olam Clinical Research

Pasadena, Texas, United States

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Sam Clinical Research Center

San Antoinio, Texas, United States

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Covenant Clinical Research, Pa

San Antonio, Texas, United States

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Hillcrest Family Health Center

Waco, Texas, United States

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Val R. Hansen, M.D.

Bountiful, Utah, United States

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Highland Clinical Research

Salt Lake City, Utah, United States

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Southwestern Vermont Med Cntr

Bennington, Vermont, United States

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Hampton Roads Center For Clinical Research, Inc.

Suffolk, Virginia, United States

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Local Institution

Coquitlam, British Columbia, Canada

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Winnipeg, Manitoba, Canada

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Brampton, Ontario, Canada

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Smiths Falls, Ontario, Canada

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Toronto, Ontario, Canada

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Granby, Quebec, Canada

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Québec, Quebec, Canada

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Saskatoon, Saskatchewan, Canada

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Aguascalientes, Aguascalientes, Mexico

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Chihuahua City, Chihuahua, Mexico

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Durango, Durango, Mexico

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Guadalajara, Jalisco, Mexico

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Cuautla, Morelos, Mexico

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Monterrey, Nuevo León, Mexico

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Monterrey, Nuevo León, Mexico

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Mérida, Yucatán, Mexico

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Gdansk, , Poland

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Katowice, , Poland

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Katowice, , Poland

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Krakow, , Poland

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Lodz, , Poland

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Opole, , Poland

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Poznan, , Poland

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Puławy, , Poland

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Warsaw, , Poland

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Cidra, , Puerto Rico

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Manatí, , Puerto Rico

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Ponce, , Puerto Rico

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San Juan, , Puerto Rico

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San Juan, , Puerto Rico

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San Juan, , Puerto Rico

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Villa Fontana, , Puerto Rico

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Galati, Galați County, Romania

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Ploieşti, Prahova, Romania

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Ploieşti, Prahova, Romania

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Timișoara, Timiș County, Romania

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Bucharest, , Romania

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Bucharest, , Romania

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Bucharest, , Romania

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Bucharest, , Romania

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Cluj Napoca Cluj, , Romania

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Craiova, , Romania

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Soweto, Gauteng, South Africa

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Gauteng, Johannesburg, South Africa

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Johannesburg, Johannesburg, South Africa

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Durban, KwaZulu-Natal, South Africa

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Cape Town, Western Cape, South Africa

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Goodwood, Western Cape, South Africa

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Paarl, Western Cape, South Africa

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Rondebosch, Western Cape, South Africa

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Somerset West, Western Cape, South Africa

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Johannesburg, , South Africa

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Bucheon-si, Gyeonggi-do, South Korea

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Sungnam-si, Gyeonggi-do, South Korea

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Daegu, , South Korea

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Incheon, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Seoul, , South Korea

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Countries

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United States Canada Mexico Poland Puerto Rico Romania South Africa South Korea

References

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Rosenstock J, Hansen L, Zee P, Li Y, Cook W, Hirshberg B, Iqbal N. Dual add-on therapy in type 2 diabetes poorly controlled with metformin monotherapy: a randomized double-blind trial of saxagliptin plus dapagliflozin addition versus single addition of saxagliptin or dapagliflozin to metformin. Diabetes Care. 2015 Mar;38(3):376-83. doi: 10.2337/dc14-1142. Epub 2014 Oct 28.

Reference Type RESULT
PMID: 25352655 (View on PubMed)

Bailey CJ, Del Prato S, Wei C, Reyner D, Saraiva G. Durability of glycaemic control with dapagliflozin, an SGLT2 inhibitor, compared with saxagliptin, a DPP4 inhibitor, in patients with inadequately controlled type 2 diabetes. Diabetes Obes Metab. 2019 Nov;21(11):2564-2569. doi: 10.1111/dom.13841. Epub 2019 Aug 26.

Reference Type DERIVED
PMID: 31364269 (View on PubMed)

Rosenstock J, Mathieu C, Chen H, Garcia-Sanchez R, Saraiva GL. Dapagliflozin versus saxagliptin as add-on therapy in patients with type 2 diabetes inadequately controlled with metformin. Arch Endocrinol Metab. 2018 Aug;62(4):424-430. doi: 10.20945/2359-3997000000056.

Reference Type DERIVED
PMID: 30304106 (View on PubMed)

Other Identifiers

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2012-000679-18

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

CV181-169

Identifier Type: -

Identifier Source: org_study_id

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