A Phase III Study of BMS-512148 (Dapagliflozin) in Patients With Type 2 Diabetes Who Are Not Well Controlled on Metformin Alone

NCT ID: NCT00528879

Last Updated: 2015-10-20

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

915 participants

Study Classification

INTERVENTIONAL

Study Start Date

2007-09-30

Study Completion Date

2010-05-31

Brief Summary

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The purpose of this clinical research study is to learn whether dapagliflozin can help reduce blood sugar levels in participants with Type 2 diabetes that is not well controlled on metformin alone. The safety of this treatment will also be studied.

Detailed Description

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Conditions

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Type 2 Diabetes

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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Placebo + Metformin

Participants received dapagliflozin-matching placebo once daily plus open-label metformin ≥1500 mg per day for up to 102 weeks

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Dapagliflozin-matching placebo administered as tablets orally once daily for up to 102 weeks

Metformin

Intervention Type DRUG

Open-label metformin administered as ≥1500 mg per day for up to 102 weeks

Dapagliflozin, 2.5 mg + Metformin

Participants received dapagliflozin, 2.5 mg, once daily plus open-label metformin ≥1500 mg per day for up to 102 weeks

Group Type EXPERIMENTAL

Dapagliflozin

Intervention Type DRUG

Tablets administered orally as a 2.5-, 5-, or 10-mg dose once daily for up to 102 weeks

Metformin

Intervention Type DRUG

Open-label metformin administered as ≥1500 mg per day for up to 102 weeks

Dapagliflozin, 5 mg + Metformin

Participants received dapagliflozin, 5 mg, once daily plus open-label metformin ≥1500 mg per day for up to 102 weeks

Group Type EXPERIMENTAL

Dapagliflozin

Intervention Type DRUG

Tablets administered orally as a 2.5-, 5-, or 10-mg dose once daily for up to 102 weeks

Metformin

Intervention Type DRUG

Open-label metformin administered as ≥1500 mg per day for up to 102 weeks

Dapagliflozin, 10 mg + Metformin

Participants received dapagliflozin, 10 mg, once daily plus open-label metformin ≥1500 mg per day for up to 102 weeks

Group Type EXPERIMENTAL

Dapagliflozin

Intervention Type DRUG

Tablets administered orally as a 2.5-, 5-, or 10-mg dose once daily for up to 102 weeks

Placebo

Intervention Type DRUG

Dapagliflozin-matching placebo administered as tablets orally once daily for up to 102 weeks

Metformin

Intervention Type DRUG

Open-label metformin administered as ≥1500 mg per day for up to 102 weeks

Interventions

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Dapagliflozin

Tablets administered orally as a 2.5-, 5-, or 10-mg dose once daily for up to 102 weeks

Intervention Type DRUG

Placebo

Dapagliflozin-matching placebo administered as tablets orally once daily for up to 102 weeks

Intervention Type DRUG

Metformin

Open-label metformin administered as ≥1500 mg per day for up to 102 weeks

Intervention Type DRUG

Other Intervention Names

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BMS-512148

Eligibility Criteria

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Inclusion Criteria

* Males and females, 18 to 77 years old, with type 2 diabetes and inadequate glycemic control
* Participants who have been receiving metformin at a total daily dose ≥1500 mg per day for at least 8 weeks
* C-peptide ≥1.0 ng/mL
* Body mass index ≤45.0 kg/m\^2
* Serum creatinine level \<1.50 mg/dL for men or \<1.40 mg/dL for women.

Exclusion Criteria

* Aspartate aminotransferase and/or alanine aminotransferase level \>3.0 times the upper limit of normal
* Serum total bilirubin level \>2 mg/dL
* Creatinine kinase level \>3 times upper limit of normal
* Symptoms of severely uncontrolled diabetes
* Serum creatinine level ≥1.50 mg/dL for men or ≥1.40 mg/dL for women
* Currently unstable or serious cardiovascular, renal, hepatic, hematologic, oncologic, endocrine, psychiatric, or rheumatic diseases
Minimum Eligible Age

18 Years

Maximum Eligible Age

77 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Bristol-Myers Squibb

INDUSTRY

Sponsor Role collaborator

AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Bristol-Myers Squibb

Role: STUDY_DIRECTOR

Bristol-Myers Squibb

Locations

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Clinical Research Advantage / Desert Clinical Res, Llc

Tempe, Arizona, United States

Site Status

Medical Group Of Encino

Encino, California, United States

Site Status

Valley Research

Fresno, California, United States

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Randall Shue, D.O.

Los Angeles, California, United States

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Diabetes Medical Center Of California

Northridge, California, United States

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Ritchken & First M.D.'S

San Diego, California, United States

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Encompass Clinical Research

Spring Valley, California, United States

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Raikhel, Marina

Torrance, California, United States

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Express Care Clinical Res

Colorado Springs, Colorado, United States

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Denver Internal Medicine

Denver, Colorado, United States

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New West Physicians

Golden, Colorado, United States

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Central Florida Clinical Trials, Inc.

Altamonte Springs, Florida, United States

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Family Care Associates Of Nw Florida

Chipley, Florida, United States

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Health Partners Research Foundation

Minneapolis, Minnesota, United States

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Woodlake Research

Chesterfield, Missouri, United States

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Nevada Alliance Against Diabetes

Las Vegas, Nevada, United States

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Diabetes & Endocrinology Consultants, Pc

Morehead City, North Carolina, United States

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Newark Physician Associates

Newark, Ohio, United States

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Integris Family Care S. Penn

Oklahoma City, Oklahoma, United States

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Cumberland Valley Endocrinology Center, Llc

Carlisle, Pennsylvania, United States

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Banksville Medical Pc

Pittsburgh, Pennsylvania, United States

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Palmetto Clinical Research

Summerville, South Carolina, United States

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Southeastern Research Assoc

Taylors, South Carolina, United States

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Texas Center For Drug Development, P.A.

Houston, Texas, United States

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Diabetes & Glandular Disease Research Associates, Inc.

San Antonio, Texas, United States

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S.A.M. Clinical Research Center

San Antonio, Texas, United States

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Optimum Clinical Research

Salt Lake City, Utah, United States

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Office Of Dr. Gray

Spokane, Washington, United States

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Local Institution

Buenos Aires, Buenos Aires, Argentina

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Local Institution

Capital Federal, Buenos Aires, Argentina

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Capital Federal, Buenos Aires, Argentina

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Capital Federal, Buenos Aires, Argentina

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Capital Federal, Buenos Aires, Argentina

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Ciudad Auton., Buenos Aires, Argentina

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Ciudad Auton, Buenos Aires, Argentina

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Mar del Plata, Buenos Aires, Argentina

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Zárate, Buenos Aires, Argentina

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Córdoba, Córdoba Province, Argentina

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Villa Carlos Paz, Córdoba Province, Argentina

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Fortaleza, Ceará, Brazil

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Itajubá, Minas Gerais, Brazil

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Belém, Pará, Brazil

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Rio de Janeiro, Rio de Janeiro, Brazil

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Caxias do Sul, Rio Grande do Sul, Brazil

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Porto Alegre, Rio Grande do Sul, Brazil

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Porto Alegre, Rio Grande do Sul, Brazil

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Marília, São Paulo, Brazil

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Calgary, Alberta, Canada

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Kelowna, British Columbia, Canada

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Winnipeg, Manitoba, Canada

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Bathurst, New Brunswick, Canada

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Mount Pearl, Newfoundland and Labrador, Canada

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St. John's, Newfoundland and Labrador, Canada

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Sarnia, Ontario, Canada

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Thornhill, Ontario, Canada

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Toronto, Ontario, Canada

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Toronto, Ontario, Canada

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Charlottetown, Prince Edward Island, Canada

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Drummondville, Quebec, Canada

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Granby, Quebec, Canada

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L'Ancienne-Lorette, Quebec, Canada

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Mirabel, Quebec, Canada

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Saint-Léonard, Quebec, Canada

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Saskatoon, Saskatchewan, Canada

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Saskatoon, Saskatchewan, Canada

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Durango, Durango, Mexico

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Guadalajara, Jalisco, Mexico

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Guadalajara, Jalisco, Mexico

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Df, Mexico City, Mexico

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Guadalajara, Mexico City, Mexico

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Zapopan, Mexico City, Mexico

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Monterrey, Nuevo León, Mexico

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Monterrey, Nuevo León, Mexico

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Monterrrey, Nuevo León, Mexico

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Tampico, Tamaulipas, Mexico

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Countries

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United States Argentina Brazil Canada Mexico

References

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Natale P, Tunnicliffe DJ, Toyama T, Palmer SC, Saglimbene VM, Ruospo M, Gargano L, Stallone G, Gesualdo L, Strippoli GF. Sodium-glucose co-transporter protein 2 (SGLT2) inhibitors for people with chronic kidney disease and diabetes. Cochrane Database Syst Rev. 2024 May 21;5(5):CD015588. doi: 10.1002/14651858.CD015588.pub2.

Reference Type DERIVED
PMID: 38770818 (View on PubMed)

Shah M, Stolbov L, Yakovleva T, Tang W, Sokolov V, Penland RC, Boulton D, Parkinson J. A model-based approach to investigating the relationship between glucose-insulin dynamics and dapagliflozin treatment effect in patients with type 2 diabetes. Diabetes Obes Metab. 2021 Apr;23(4):991-1000. doi: 10.1111/dom.14305. Epub 2021 Jan 25.

Reference Type DERIVED
PMID: 33368935 (View on PubMed)

Bailey CJ, Del Prato S, Wei C, Reyner D, Saraiva G. Durability of glycaemic control with dapagliflozin, an SGLT2 inhibitor, compared with saxagliptin, a DPP4 inhibitor, in patients with inadequately controlled type 2 diabetes. Diabetes Obes Metab. 2019 Nov;21(11):2564-2569. doi: 10.1111/dom.13841. Epub 2019 Aug 26.

Reference Type DERIVED
PMID: 31364269 (View on PubMed)

Mellander A, Billger M, Johnsson E, Traff AK, Yoshida S, Johnsson K. Hypersensitivity Events, Including Potentially Hypersensitivity-Related Skin Events, with Dapagliflozin in Patients with Type 2 Diabetes Mellitus: A Pooled Analysis. Clin Drug Investig. 2016 Nov;36(11):925-933. doi: 10.1007/s40261-016-0438-3.

Reference Type DERIVED
PMID: 27461213 (View on PubMed)

Kohan DE, Fioretto P, Johnsson K, Parikh S, Ptaszynska A, Ying L. The effect of dapagliflozin on renal function in patients with type 2 diabetes. J Nephrol. 2016 Jun;29(3):391-400. doi: 10.1007/s40620-016-0261-1. Epub 2016 Feb 19.

Reference Type DERIVED
PMID: 26894924 (View on PubMed)

Bailey CJ, Gross JL, Hennicken D, Iqbal N, Mansfield TA, List JF. Dapagliflozin add-on to metformin in type 2 diabetes inadequately controlled with metformin: a randomized, double-blind, placebo-controlled 102-week trial. BMC Med. 2013 Feb 20;11:43. doi: 10.1186/1741-7015-11-43.

Reference Type DERIVED
PMID: 23425012 (View on PubMed)

Bailey CJ, Gross JL, Pieters A, Bastien A, List JF. Effect of dapagliflozin in patients with type 2 diabetes who have inadequate glycaemic control with metformin: a randomised, double-blind, placebo-controlled trial. Lancet. 2010 Jun 26;375(9733):2223-33. doi: 10.1016/S0140-6736(10)60407-2.

Reference Type DERIVED
PMID: 20609968 (View on PubMed)

Other Identifiers

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MB102-014

Identifier Type: OTHER

Identifier Source: secondary_id

MB102-014 LT

Identifier Type: -

Identifier Source: org_study_id

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