A Phase III Trial of ZD4054 (Zibotentan) (Endothelin A Antagonist) and Docetaxel in Metastatic Hormone Resistant Prostate Cancer

NCT ID: NCT00617669

Last Updated: 2012-09-10

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

1494 participants

Study Classification

INTERVENTIONAL

Study Start Date

2008-01-31

Study Completion Date

2011-07-31

Brief Summary

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Enthuse M1C is a large phase III clinical trial studying the safety and efficacy of ZD4054 (Zibotentan) in combination with docetaxel (Taxotere) in patients with metastatic hormone resistant prostate cancer (HRPC).

This clinical trial will test if the Endothelin A Receptor Antagonist ZD4054 (Zibotentan) can further improve survival compared with docetaxel alone.

ZD4054 (Zibotentan) is a new type of agent, which is thought to slow tumour growth and spread by blocking Endothelin A receptor activity. This trial will look at the effects of ZD4054 (Zibotentan) in hormone resistant prostate cancer patients with bone metastases compared with docetaxel.

All patients participating in this clinical trial will receive docetaxel chemotherapy, which is a commonly used chemotherapy to treat prostate cancer in addition to other existing prostate cancer therapies.

Half the patients will receive ZD4054 (Zibotentan), and half the patients will receive placebo in addition to docetaxel and other prostate cancer therapy. By participating in this trial there is a 50% chance that patients will receive an agent that may further slow the progression of the tumour.

No patients will be deprived of standard prostate cancer therapy.

Detailed Description

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Conditions

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Prostate Cancer

Keywords

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Hormone Resistant Prostate Cancer Endothelin A Receptor Antagonist Endothelin A Endothelin A antagonist

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Caregivers Investigators

Study Groups

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Placebo + Docetaxel

placebo oral tablet once daily + docetaxel intravenous infusion every 3 weeks

Group Type ACTIVE_COMPARATOR

Docetaxel

Intervention Type DRUG

intravenous infusion given every three weeks

Placebo

Intervention Type DRUG

placebo oral tablet once daily

ZD4054 + Docetaxel

ZD4054 10 mg oral tablet once daily + docetaxel intravenous infusion every 3 weeks

Group Type EXPERIMENTAL

Docetaxel

Intervention Type DRUG

intravenous infusion given every three weeks

ZD4054

Intervention Type DRUG

10 mg oral once daily dose

Interventions

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Docetaxel

intravenous infusion given every three weeks

Intervention Type DRUG

ZD4054

10 mg oral once daily dose

Intervention Type DRUG

Placebo

placebo oral tablet once daily

Intervention Type DRUG

Other Intervention Names

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Taxotere® Zibotentan

Eligibility Criteria

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Inclusion Criteria

Patients who answer TRUE to the following criteria may be eligible to participate in this trial.

* Confirmed diagnosis of prostate cancer (adenocarcinoma of the prostate) that has spread to the bone (bone metastasis)
* Increasing Prostate Specific Antigen (PSA), collected within one year of enrollment
* Currently receiving treatment with surgical or medical castration

Exclusion Criteria

Patients who answer TRUE to the following ARE NOT eligible to participate in this trial.

* Previous treatment with chemotherapy (paclitaxel, docetaxel, and mitoxantrone). Prior targeted cancer therapies are permitted if received during a previous clinical trial.
* Suffering from heart failure or had a myocardial infarction within last 6 months
* A history of epilepsy or seizures
Minimum Eligible Age

18 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

No

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Karim Fizazi, MD, PhD

Role: PRINCIPAL_INVESTIGATOR

Gustave Roussy, Cancer Campus, Grand Paris

Judd W Moul, MD, FACS

Role: PRINCIPAL_INVESTIGATOR

Duke University

Locations

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Greenbrae, California, United States

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San Diego, California, United States

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Norwich, Connecticut, United States

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Washington D.C., District of Columbia, United States

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Fort Myers, Florida, United States

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Gainsville, Florida, United States

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Ocala, Florida, United States

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PORTUGALt Saint Lucie, Florida, United States

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Rockville, Maryland, United States

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Minneapolis, Minnesota, United States

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Lincoln, Nebraska, United States

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Omaha, Nebraska, United States

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Chapel Hill, North Carolina, United States

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Durham, North Carolina, United States

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Winston-Salem, North Carolina, United States

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Canton, Ohio, United States

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Cincinnati, Ohio, United States

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Pittsburgh, Pennsylvania, United States

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Charleston, South Carolina, United States

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Chattanooga, Tennessee, United States

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Nashville, Tennessee, United States

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San Antonio, Texas, United States

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Richmond, Virginia, United States

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Seattle, Washington, United States

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Milwaukee, Wisconsin, United States

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Bahía Blanca, Buenos Aires, Argentina

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Buenos Aires, Buenos Aires, Argentina

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Santa Fe, Santa Fe Province, Argentina

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Darlinghurst, New South Wales, Australia

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St Leonards, New South Wales, Australia

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Wollongong, New South Wales, Australia

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Redcliffe, Queensland, Australia

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Ashford, South Australia, Australia

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Footscray, Victoria, Australia

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Wodonga, Victoria, Australia

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Perth, Western Australia, Australia

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Subiaco, Western Australia, Australia

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Fortaleza, Ceara/ LA, Brazil

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Goiânia, Goias/ LA, Brazil

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Goiânia, Goiás, Brazil

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Belo Horizonte, Minas GERMANYais, Brazil

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Curitiba, Parana/ Brazil, Brazil

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Londrina, Paraná, Brazil

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Rio de Janeiro, Rio de Janeiro, Brazil

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PORTUGALto Alegre, Rio Grande Do Sul/ LA, Brazil

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Ribeirão Preto, Sao Paulo/ LA, Brazil

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Santo André, São Paulo, Brazil

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São Paulo, São Paulo, Brazil

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Winnipeg, Manitoba, Canada

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Halifax, Nova Scotia, Canada

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London, Ontario, Canada

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Toronto, Ontario, Canada

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Québec, Quebec, Canada

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Sherbrooke, Quebec, Canada

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Olomouc, Czech Republic, Czechia

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Prague, Czech Republic, Czechia

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Ústí nad Labem, Czech Republic, Czechia

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Brno, Czechoslovakia Republic, Czechia

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Jablonec nad Nisou, , Czechia

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Kroměříž, , Czechia

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Prague, , Czechia

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Helsinki, Finland, Finland

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Joensuu, , Finland

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Seinäjoki, , Finland

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La Roche-sur-Yon, FRANCEnce, France

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Marseille, FRANCEnce, France

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Paris, FRANCEnce, France

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Reims, FRANCEnce, France

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Villejuif, FRANCEnce, France

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Paris, Paris, France

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Saint-Herblain, Saint Herblain, France

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Paris, , France

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Hanover, GERMANYmany, Germany

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Berlin, , Germany

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Bonn, , Germany

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Dresden, , Germany

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Emmendingen, , Germany

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Kirchheim-Teck, , Germany

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Leipzig, , Germany

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Lübeck, , Germany

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Münster, , Germany

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Tübingen, , Germany

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Wuppertal, , Germany

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Budapest, HUNGARYary, Hungary

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Győr, HUNGARYary, Hungary

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Miskolc, HUNGARYary, Hungary

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Ny Regyh Za, HUNGARYary, Hungary

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Szeged, HUNGARYary, Hungary

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Bangalore, Karnataka, India

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Trivandrum, Kerala, India

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Bhopal, Madhya Pradesh, India

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Pune, Maharashtra, India

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Bikaner, Rajasthan, India

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Jaipur, Rajasthan, India

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Vellore, Tamil Nadu, India

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Kolkata, West Bengal, India

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Kolkota, West Bengal, India

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Delhi, , India

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New Delhi, , India

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Genoa, Italy, Italy

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Lugo (RA), Italy, Italy

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Rome, Italy, Italy

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Nijmegen, , Netherlands

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Cercado de Arequipa, Arequipa, Peru

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Cercado, Arequipa, Peru

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Callao, , Peru

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Lima, , Peru

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Lublin, POLANDand, Poland

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Swidnica, POLANDand, Poland

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Warszaa, POLANDand, Poland

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Kościerzyna, , Poland

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Wroclaw, , Poland

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Coimbra, PORTUGALtugal, Portugal

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PORTUGALto, PORTUGALtugal, Portugal

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Bucharest, , Romania

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Sibiu, , Romania

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Timișoara, , Romania

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Barnaul, RUSSIAsia, Russia

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Izhevsk, RUSSIAsia, Russia

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Kursk, RUSSIAsia, Russia

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Sochi, RUSSIAsia, Russia

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Voronezh, RUSSIAsia, Russia

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Belgrade, SERBIAbia, Serbia

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Niš, SERBIAbia, Serbia

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Panorama, Cape Town, South Africa

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TyGERberg, Cape Town, South Africa

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Overport, Durban, South Africa

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Bloemfontein, , South Africa

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Port Elizabeth, , South Africa

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Ilsandong-gu, Goyang-si, Gyeonggi-do, South Korea

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Cheongju-si, North Chungcheong, South Korea

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Nowon-gu, Seoul, South Korea

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Seodaemun-gu, Seoul, South Korea

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Songpa-gu, Seoul, South Korea

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Madrid, Spain, Spain

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Valencia, Spain, Spain

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Stockholm, Sweden, Sweden

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Uppsala, , Sweden

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Aarau, , Switzerland

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Locarno, , Switzerland

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Sursee, , Switzerland

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Kaohsiung City, TAIWANwan, Taiwan

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TAIWANpei, TAIWANwan, Taiwan

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Reading, Berkshire, United Kingdom

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Manchester, Manchester, United Kingdom

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Westgate Road, Newcastle Upon Tyne, United Kingdom

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London, , United Kingdom

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Countries

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Norway Singapore United States Argentina Australia Brazil Canada Czechia Finland France Germany Hungary India Italy Netherlands Peru Poland Portugal Romania Russia Serbia South Africa South Korea Spain Sweden Switzerland Taiwan United Kingdom

References

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Fizazi K, Higano CS, Nelson JB, Gleave M, Miller K, Morris T, Nathan FE, McIntosh S, Pemberton K, Moul JW. Phase III, randomized, placebo-controlled study of docetaxel in combination with zibotentan in patients with metastatic castration-resistant prostate cancer. J Clin Oncol. 2013 May 10;31(14):1740-7. doi: 10.1200/JCO.2012.46.4149. Epub 2013 Apr 8.

Reference Type DERIVED
PMID: 23569308 (View on PubMed)

Other Identifiers

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D4320C00033

Identifier Type: -

Identifier Source: org_study_id