A Phase III Trial of ZD4054 (Zibotentan) (Endothelin A Antagonist) in Non-metastatic Hormone Resistant Prostate Cancer

NCT ID: NCT00626548

Last Updated: 2012-09-03

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE3

Total Enrollment

2577 participants

Study Classification

INTERVENTIONAL

Study Start Date

2008-01-31

Study Completion Date

2011-05-31

Brief Summary

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Enthuse M0 is a large phase III clinical trial studying the efficacy of ZD4054 (Zibotentan) in hormone resistant prostate cancer (HRPC).

This clinical trial will test if the Endothelin A Receptor Antagonist ZD4054 (Zibotentan) can improve progression-free survival and overall survival against a background of existing prostate cancer treatments.

ZD4054 (Zibotentan) is a new type of agent, which is thought to slow tumour growth and spread by blocking Endothelin receptor activity. This trial will look at the effects of ZD4054 (Zibotentan) in hormone resistant prostate cancer (HRPC) patients who have had rising PSA after surgical or medical castration but have no evidence of metastases.

All patients participating in this clinical trial will receive existing prostate cancer treatments in addition to trial therapy.

Half the patients will receive ZD4054 (Zibotentan) , and half the patients will receive placebo in addition to standard prostate cancer therapy. By participating in this trial there is a 50% chance that patients will receive an agent that may slow the progression of the tumour.

No patients will be deprived of standard prostate cancer therapy.

Detailed Description

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Conditions

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Prostate Cancer

Keywords

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Hormone Resistant Prostate Cancer Endothelin A Receptor Antagonist Endothelin A Endothelin A antagonist

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Caregivers Investigators

Study Groups

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Placebo

Matching Placebo

Group Type PLACEBO_COMPARATOR

Palcebo

Intervention Type DRUG

Matching Plcebo oral tablet once daily

ZD4054

ZD4054 (Zibotentan)

Group Type EXPERIMENTAL

ZD4054

Intervention Type DRUG

10 mg once daily oral dose

Interventions

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ZD4054

10 mg once daily oral dose

Intervention Type DRUG

Palcebo

Matching Plcebo oral tablet once daily

Intervention Type DRUG

Other Intervention Names

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Zibotentan

Eligibility Criteria

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Inclusion Criteria

Patients who answer TRUE to the following criteria may be eligible to participate in this study.

* Confirmed diagnosis of prostate cancer (adenocarcinoma of the prostate) that has NOT spread to the other parts of the body (metastases). Patients with lymph node involvement may be eligible if specified criteria is met.
* Increasing Prostate Specific Antigen (PSA), collected within one year of enrollment
* Currently receiving treatment with surgical or medical castration

Exclusion Criteria

Patients who answer TRUE to the following may NOT be eligible to participate in this study.

* Currently using opiate based pain killers for cancer related pain
* Previous treatment with chemotherapy (paclitaxel, docetaxel, and mitoxantrone). Prior targeted cancer therapies are permitted if received during a previous clinical trial
* Suffering from heart failure or had a myocardial infarction within last 6 months
* A history of epilepsy or seizures
Minimum Eligible Age

18 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

No

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Kurt Miller, Prof., M.D.

Role: PRINCIPAL_INVESTIGATOR

Charite University, Berlin, Germany

Tia Higano, MD

Role: PRINCIPAL_INVESTIGATOR

University of Washington

Locations

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Tucson, Arizona, United States

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Greenbrae, California, United States

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Los Angeles, California, United States

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San Diego, California, United States

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San Francisco, California, United States

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Denver, Colorado, United States

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Norwich, Connecticut, United States

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Washington D.C., District of Columbia, United States

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Boca Raton, Florida, United States

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Miami, Florida, United States

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Ocala, Florida, United States

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Port Saint Lucie, Florida, United States

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Atlanta, Georgia, United States

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Macon, Georgia, United States

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Kansas City, Kansas, United States

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New Orleans, Louisiana, United States

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Baltimore, Maryland, United States

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Rockville, Maryland, United States

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Minneapolis, Minnesota, United States

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Lincoln, Nebraska, United States

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Las Vegas, Nevada, United States

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Brooklyn, New York, United States

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Chapel Hill, North Carolina, United States

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Bismarck, North Dakota, United States

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Canton, Ohio, United States

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Cincinnati, Ohio, United States

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Philadelphia, Pennsylvania, United States

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Pittsburgh, Pennsylvania, United States

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Charleston, South Carolina, United States

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Mystle Beach, South Carolina, United States

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Raleigh, South Carolina, United States

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Memphis, Tennessee, United States

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Nashville, Tennessee, United States

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San Antonio, Texas, United States

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Burlington, Vermont, United States

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Seattle, Washington, United States

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Wenatchee, Washington, United States

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Milwaukee, Wisconsin, United States

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Ciudad Autonoma de Buenos Aires, Buenos Aires, Argentina

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Rosario, Santa Fe Province, Argentina

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Santa Fe, Santa Fe Province, Argentina

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Darlinghurst, New South Wales, Australia

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Hornsby, New South Wales, Australia

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Westmead, New South Wales, Australia

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Wollongong, New South Wales, Australia

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Wodonga, Victoria, Australia

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Nedlands, Western Australia, Australia

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Sydney, , Australia

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Graz, , Austria

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Innsbruck, , Austria

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Wels, , Austria

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(Wilrijk) Antwerpen, , Belgium

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Brussels, , Belgium

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Edegem, , Belgium

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Ghent, , Belgium

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Kortrijk, , Belgium

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Leuven, , Belgium

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Liège, , Belgium

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Goiânia, Goiás, Brazil

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Belo Horizonte, Minas Gerais, Brazil

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Curitiba, Paraná, Brazil

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Londrina, Paraná, Brazil

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Rio de Janeiro, Rio de Janeiro, Brazil

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Porto Alegre, Rio Grande do Sul, Brazil

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Santo André, São Paulo, Brazil

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São Paulo, São Paulo, Brazil

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Calgary, Alberta, Canada

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Edmonton, Alberta, Canada

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Vancouver, British Columbia, Canada

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Victoria, British Columbia, Canada

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Winnipeg, Manitoba, Canada

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Burlington, Ontario, Canada

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Hamilton, Ontario, Canada

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Kingston, Ontario, Canada

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Kitchener, Ontario, Canada

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London, Ontario, Canada

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North York, Ontario, Canada

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Oakville, Ontario, Canada

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Toronto, Ontario, Canada

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Greenfeild Park, Quebec, Canada

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Montreal, Quebec, Canada

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Point-Claire, Quebec, Canada

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Québec, Quebec, Canada

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Sherbrooke, Quebec, Canada

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La Serena, , Chile

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Santiago, , Chile

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Temuco, , Chile

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Viña del Mar, , Chile

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Nanjing, Jiangsu, China

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Hangzhou, Zhejiang, China

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Beijing, , China

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Chongqing, , China

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Guangzhou, , China

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Hubei, , China

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Jiangsu, , China

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Shanghai, , China

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Shanxi, , China

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Tianjin, , China

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Zejiang, , China

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Bogotá, , Colombia

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Medellín, , Colombia

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Brno, , Czechia

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Hradec Králové, , Czechia

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Jablonec nad Nisou, , Czechia

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Kroměříž, , Czechia

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Olomouc, , Czechia

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Prague, , Czechia

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Ústí nad Labem, , Czechia

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Aalborg, , Denmark

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Copenhagen, , Denmark

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Frederiksberg, , Denmark

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Herlev, , Denmark

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Holstebro, , Denmark

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Odense, , Denmark

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Roskilde, , Denmark

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Helsinki, , Finland

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Joensuu, , Finland

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Oulu, , Finland

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Seinäjoki, , Finland

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Tampere, , Finland

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Caen, , France

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Créteil, , France

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Lille, , France

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Lyon, , France

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Marseille, , France

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Montpellier, , France

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Orléans, , France

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Paris, , France

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Pierre-Bénite, , France

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Poitiers, , France

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Reims, , France

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Rennes, , France

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Rouen, , France

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Suresnes, , France

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Toulouse, , France

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Vandœuvre-lès-Nancy, , France

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Villejuif, , France

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Augsburg, , Germany

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Bad Ems, , Germany

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Berlin, , Germany

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Bonn, , Germany

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Borken, , Germany

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Chemnitz, , Germany

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Emmendingen, , Germany

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Fürth, , Germany

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Gelsenkirchen-Buer, , Germany

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Germering, , Germany

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Göttingen, , Germany

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Holzminden, , Germany

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Kirchheim/Teck, , Germany

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Leipzig, , Germany

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Lübeck, , Germany

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Mannheim, , Germany

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Muehlheim An Der Ruhr, , Germany

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Muenchen-Planegg, , Germany

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Mühlacker, , Germany

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München, , Germany

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Münster, , Germany

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Reutlingen, , Germany

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Rostock, , Germany

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Tübingen, , Germany

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Waltshut-Tiengen, , Germany

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Wuppertal, , Germany

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Budapest, , Hungary

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Debrecen, , Hungary

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Győr, , Hungary

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Miskolc, , Hungary

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Nyíregyháza, , Hungary

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Szeged, , Hungary

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Székesfehérvár, , Hungary

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Ahmedabad, Gujarat, India

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Nadiād, Gujarat, India

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Kochi, Kerala, India

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Pune, Maharashtra, India

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Chennai, Tamil Nadu, India, India

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Lucknow, Uttar Pradesh, India

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Kolkota, West Bengal, India

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New Delhi, , India

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Dublin, , Ireland

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Beersheba, , Israel

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Be’er Ya‘aqov, , Israel

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Haifa, , Israel

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Holon, , Israel

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Jeruslaem, , Israel

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Petah Tikva, , Israel

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Tel-HaShomer - Ramat Gan, , Israel

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Ancona, , Italy

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Bari, , Italy

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Bergamo, , Italy

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Bologna, , Italy

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Catania, , Italy

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Como, , Italy

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Florence, , Italy

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Genova, , Italy

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Messina, , Italy

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Milan, , Italy

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Pisa, , Italy

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Rome, , Italy

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Terni, , Italy

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Varese, , Italy

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Hirosaki, Aomori, Japan

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Chiba, Chiba, Japan

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Narashino, Chiba, Japan

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Matsuyama, Ehime, Japan

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Fukuoka, Fukuoka, Japan

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Maebashi, Gunma, Japan

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Ōtake, Hiroshima, Japan

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Sapporo, Hokkaido, Japan

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Kobe, Hyōgo, Japan

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Ibaraki-machi, Ibaraki, Japan

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Mito, Ibaraki, Japan

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Tsukuba, Ibaraki, Japan

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Kita-gun, Kagawa-ken, Japan

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Sagamihara, Kanagawa, Japan

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Kamigyō-ku, Kyoto, Japan

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Kyoto, Kyoto, Japan

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Sendai, Miyagi, Japan

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Ueda, Nagano, Japan

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Nagasaki, Nagasaki, Japan

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Kashihara, Nara, Japan

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Ōita, Oita Prefecture, Japan

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Kurashiki, Okayama-ken, Japan

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Osaka, Osaka, Japan

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Ōsaka-sayama, Osaka, Japan

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Suita, Osaka, Japan

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Wako, Saitama, Japan

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Hamamatsu, Shizuoka, Japan

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Sunto-gun, Shizuoka, Japan

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Bunkyo-ku, Tokyo, Japan

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Fuchu_city, Tokyo, Japan

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Itabashi-Ku, Tokyo, Japan

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Meguro-ku, Tokyo, Japan

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Minato-Ku, Tokyo, Japan

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Mitaka, Tokyo, Japan

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Shinjuku-ku, Tokyo, Japan

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Liepāja, , Latvia

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Riga, , Latvia

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Distrito Federal, Mexico City, Mexico

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Mexico City, Mexico City, Mexico

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's-Hertogenbosch, , Netherlands

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Amsterdam, , Netherlands

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Arnhem, , Netherlands

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Eindhoven, , Netherlands

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Nijmegen, , Netherlands

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Rotterdam, , Netherlands

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Tilburg, , Netherlands

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Trondheim, , Norway

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Tønsberg, , Norway

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Arequipa, , Peru

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Bellavista, , Peru

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Jesus Maria, , Peru

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Lima, , Peru

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Gdynia, , Poland

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Kielce, , Poland

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Kościerzyna, , Poland

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Szczecin, , Poland

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Warsaw, , Poland

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Wroclaw, , Poland

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Coimbra, , Portugal

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Porto, , Portugal

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Timișoara, Timiș County, Romania

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Bucharest, , Romania

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Cluj-Napoca, , Romania

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Omsk, Omsk Oblast, Russia

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Izhevsk, Russia, Russia

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Tomsk, Tomsk Oblast, Russia

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Barnaul, , Russia

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Kursk, , Russia

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Moscow, , Russia

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Saint Petersburg, , Russia

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Sochi, , Russia

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Voronezh, , Russia

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Belgrade, , Serbia

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Niš, , Serbia

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Novi Sad, , Serbia

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Observatory, Cape Town, South Africa

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Tygerberg, Cape Town, South Africa

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Overport, Durban, South Africa

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Parktown, Johannesburg, South Africa

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Pietermaritzburg, , South Africa

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Pretoria, , South Africa

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Seo-gu, Busan, South Korea

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Bundang-Gu, Seongnam-si, Gyeonggi-do, South Korea

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Gangnam-gu, Seoul, South Korea

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Seodaemun-gu, Seoul, South Korea

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Seongbuk-gu, Seoul, South Korea

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Songpa-gu, Seoul, South Korea

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Elche, Alicante, Spain

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Barakaldo, Bizkaia, Spain

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Bilbao, Vizcaya, Spain

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A Corunna, , Spain

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Barcelona, , Spain

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Madrid, , Spain

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Seville, , Spain

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Valencia, , Spain

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Gothenburg, , Sweden

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Helsingborg, , Sweden

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Jönköping, , Sweden

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Örebro, , Sweden

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Stockholm, , Sweden

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Uppsala, , Sweden

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Aarau, , Switzerland

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Ch-4031 Basel, , Switzerland

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Locarno, , Switzerland

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Zurich, , Switzerland

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Taipei, , Taiwan

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Ankara, , Turkey (Türkiye)

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Istanbul, , Turkey (Türkiye)

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Izmir, , Turkey (Türkiye)

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Reading, Berkshire, United Kingdom

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Cottingham, East Yorkshire, United Kingdom

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Stevenage, Hertfordshire, United Kingdom

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Maidstone, Kent, United Kingdom

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Guildford, Surrey, United Kingdom

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Cambridge, , United Kingdom

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Coventry, , United Kingdom

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Glasgow, , United Kingdom

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Huddersfield, , United Kingdom

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Liverpool, , United Kingdom

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London, , United Kingdom

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Manchester, , United Kingdom

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Newcastle upon Tyne, , United Kingdom

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Countries

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Serbia and Montenegro United States Argentina Australia Austria Belgium Brazil Canada Chile China Colombia Czechia Denmark Finland France Germany Hungary India Ireland Israel Italy Japan Latvia Mexico Netherlands Norway Peru Poland Portugal Romania Russia Serbia South Africa South Korea Spain Sweden Switzerland Taiwan Turkey (Türkiye) United Kingdom

Other Identifiers

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D4320C00015

Identifier Type: -

Identifier Source: org_study_id