ZD4054 (Zibotentan) in Pain-free or Mildly Symptomatic Patients With Prostate Cancer and Bone Metastases Who Have Rising Serum Prostate Specific Antigen (PSA)

NCT ID: NCT00090363

Last Updated: 2013-01-08

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

447 participants

Study Classification

INTERVENTIONAL

Study Start Date

2004-07-31

Study Completion Date

2011-08-31

Brief Summary

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This study is being carried out to see if ZD4054 (Zibotentan) is effective in treating prostate cancer and spread of cancer to the bone, and if so, how it compares with placebo (sugar pill). The study will also provide further information on the safety of ZD4054 (Zibotentan).

Detailed Description

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Conditions

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Prostate Cancer

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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Placebo

Matching placebo oral tablet once daily, with best supportive care

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

ZD4054 10 mg

ZD4054 10 mg oral tablet once daily, with best supportive care

Group Type EXPERIMENTAL

ZD4054 10 mg

Intervention Type DRUG

10mg oral tablet once daily

ZD4054 15 mg

ZD4054 15 mg oral tablet once daily, with best supportive care

Group Type EXPERIMENTAL

ZD4054 15 mg

Intervention Type DRUG

15 mg oral tablet once daily

Interventions

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ZD4054 15 mg

15 mg oral tablet once daily

Intervention Type DRUG

Placebo

Intervention Type DRUG

ZD4054 10 mg

10mg oral tablet once daily

Intervention Type DRUG

Other Intervention Names

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Zibotentan (Zibotentan)

Eligibility Criteria

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Inclusion Criteria

* Surgically or medically castrated
* Bone metastasis
* Rising PSA

Exclusion Criteria

* Opiate use
* Prior chemotherapy
Minimum Eligible Age

18 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

No

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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AstraZeneca Emerging Oncology Medical Science Director, MD

Role: STUDY_DIRECTOR

AstraZeneca

Locations

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Research Site

Tucson, Arizona, United States

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Los Angeles, California, United States

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Gainsville, Florida, United States

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Chicago, Illinois, United States

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Baltimore, Maryland, United States

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Cleveland, Ohio, United States

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Simpsonville, South Carolina, United States

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Wolloongabba, Queensland, Australia

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Ashford, South Australia, Australia

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Wodonga, Victoria, Australia

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Nedlands, , Australia

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Brussels, , Belgium

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Ghent, , Belgium

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Leuven, , Belgium

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Vancouver, British Columbia, Canada

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London, Ontario, Canada

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Toronto, Ontario, Canada

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Montreal, Quebec, Canada

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Québec, Quebec, Canada

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Aarhus, , Denmark

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Herlev, , Denmark

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Helsinki, , Finland

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Joensuu, , Finland

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OYS, , Finland

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Seinäjoki, , Finland

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Tampere, , Finland

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Lille, , France

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Montpellier, , France

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Paris, , France

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Pontoise, , France

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Toulouse, , France

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Jakarta, , Indonesia

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Eindhoven, , Netherlands

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Groningen, , Netherlands

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Heerlen, , Netherlands

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Leiden, , Netherlands

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Rotterdam, , Netherlands

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Utrecht, , Netherlands

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Bergen, , Norway

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Fredrikstad, , Norway

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Moelv, , Norway

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Oslo, , Norway

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Tromsø, , Norway

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Trondheim, , Norway

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Tønsberg, , Norway

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Bydgoszcz, , Poland

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Katowice, , Poland

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Warsaw, , Poland

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Gothenburg, , Sweden

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Malmo, , Sweden

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Stockholm, , Sweden

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Geneva, , Switzerland

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Locarno, , Switzerland

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Birmingham, , United Kingdom

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Leeds, , United Kingdom

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London, , United Kingdom

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Maidstone, , United Kingdom

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Manchester, , United Kingdom

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Newcastle, , United Kingdom

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York, , United Kingdom

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Countries

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United States Australia Belgium Canada Denmark Finland France Indonesia Netherlands Norway Poland Sweden Switzerland United Kingdom

References

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James ND, Caty A, Borre M, Zonnenberg BA, Beuzeboc P, Morris T, Phung D, Dawson NA. Safety and efficacy of the specific endothelin-A receptor antagonist ZD4054 in patients with hormone-resistant prostate cancer and bone metastases who were pain free or mildly symptomatic: a double-blind, placebo-controlled, randomised, phase 2 trial. Eur Urol. 2009 May;55(5):1112-23. doi: 10.1016/j.eururo.2008.11.002. Epub 2008 Nov 29.

Reference Type DERIVED
PMID: 19042080 (View on PubMed)

Other Identifiers

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Trial 6

Identifier Type: -

Identifier Source: secondary_id

ZD4054

Identifier Type: -

Identifier Source: secondary_id

D4320C00006

Identifier Type: -

Identifier Source: org_study_id

NCT00107146

Identifier Type: -

Identifier Source: nct_alias

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