A Phase III Trial of ZD4054 (Zibotentan) (Endothelin A Antagonist) in Hormone Resistant Prostate Cancer With Bone Metastases

NCT ID: NCT00554229

Last Updated: 2016-02-08

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

View full results

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

896 participants

Study Classification

INTERVENTIONAL

Study Start Date

2007-11-30

Study Completion Date

2011-08-31

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

Enthuse M1 is a large phase III clinical trial studying the safety and efficacy of ZD4054 (Zibotentan) in patients with hormone resistant prostate cancer and bone metastases.

* This clinical trial will test if the Endothelin A Receptor Antagonist ZD4054 (Zibotentan) can improve survival compared with placebo.
* ZD4054(Zibotentan) is a new type of agent, which is thought to slow tumour growth and spread by blocking Endothelin A receptor activity. This trial will look at the effects of ZD4054 (Zibotentan) in hormone resistant prostate cancer patients with bone metastases.
* All patients participating in this clinical trial will receive existing standard prostate cancer treatments in addition to trial therapy.
* Half the patients will receive ZD4054 (Zibotentan), and half the patients will receive placebo in addition to standard prostate cancer therapy. By participating in this trial there is a 50% chance that patients will receive an agent that may slow the progression of the tumour.
* No patients will be deprived of standard prostate cancer therapy.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Prostate Cancer

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

ZD4054

ZD4054 10 mg oral tablet once daily

Group Type EXPERIMENTAL

ZD4054

Intervention Type DRUG

ZD4054 10 mg oral tablet once daily

Placebo

Matching Placebo, oral tablets once daily

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Matching placebo oral tablet once daily

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

ZD4054

ZD4054 10 mg oral tablet once daily

Intervention Type DRUG

Placebo

Matching placebo oral tablet once daily

Intervention Type DRUG

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

Zibotentan

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

Patients who answer TRUE to the following criteria may be eligible to participate in this trial.

1. Confirmed diagnosis of prostate cancer (adenocarcinoma of the prostate) that has spread to the bone (bone metastases)
2. Increasing Prostate Specific Antigen (PSA) over a one month period
3. No pain, or mild pain from prostate cancer
4. Currently receiving treatment with surgical or medical castration

Exclusion Criteria

Patients who answer TRUE to the following may NOT eligible to participate in this trial.

1. Currently using opiates based pain killers)
2. Previous treatment with chemotherapy (paclitaxel, docetaxel, and mitoxantrone)
3. Suffering from heart failure or had a myocardial infarction within last 6 months
4. A history of epilepsy or seizures
Minimum Eligible Age

18 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Martin Gleave, MD, FRCSC, FACS

Role: PRINCIPAL_INVESTIGATOR

The Prostate Centre at Vancouver General Hospital

Joel B Nelson, MD

Role: PRINCIPAL_INVESTIGATOR

University of Pittsburgh

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Research Site

Tucson, Arizona, United States

Site Status

Research Site

Greenbrae, California, United States

Site Status

Research Site

Los Angeles, California, United States

Site Status

Research Site

Palm Springs, California, United States

Site Status

Research Site

San Mateo, California, United States

Site Status

Research Site

Norwich, Connecticut, United States

Site Status

Research Site

Washington D.C., District of Columbia, United States

Site Status

Research Site

Gainsville, Florida, United States

Site Status

Research Site

Port St.Lucie, Florida, United States

Site Status

Research Site

Des Moines, Iowa, United States

Site Status

Research Site

Canton, Ohio, United States

Site Status

Research Site

Pittsburgh, Pennsylvania, United States

Site Status

Research Site

Nashville, Tennessee, United States

Site Status

Research Site

Salt Lake City, Utah, United States

Site Status

Research Site

Burlington, Vermont, United States

Site Status

Research Site

Norfolk, Virginia, United States

Site Status

Research Site

Seattle, Washington, United States

Site Status

Research Site

Wheeling, West Virginia, United States

Site Status

Research Site

Milwaukee, Wisconsin, United States

Site Status

Research Site

Buenos Aires, Buenos Aires, Argentina

Site Status

Research Site

Santa Fe, Santa Fe Province, Argentina

Site Status

Research Site

Hornsby, New South Wales, Australia

Site Status

Research Site

St Leonards, New South Wales, Australia

Site Status

Research Site

Redcliffe, Queensland, Australia

Site Status

Research Site

Ashford, South Australia, Australia

Site Status

Research Site

Subiaco, Western Australia, Australia

Site Status

Research Site

Graz, Graz, Austria

Site Status

Research Site

Wels, Wels, Austria

Site Status

Research Site

Brussels, Brussels Capital, Belgium

Site Status

Research Site

Ghent, Gent, Belgium

Site Status

Research Site

Kortrijk, Kortrijk, Belgium

Site Status

Research Site

Leuven, Leuven, Belgium

Site Status

Research Site

Fortaleza, Ceará, Brazil

Site Status

Research Site

Goiânia, Goiás, Brazil

Site Status

Research Site

Belo Horizonte, Minas Gerais, Brazil

Site Status

Research Site

Curitiba, Paraná, Brazil

Site Status

Research Site

Porto Alegre, Rio Grande do Sul, Brazil

Site Status

Research Site

Ribeirão Preto, São Paulo, Brazil

Site Status

Research Site

Santo André, São Paulo, Brazil

Site Status

Research Site

São Paulo, São Paulo, Brazil

Site Status

Research Site

Calgary, Alberta, Canada

Site Status

Research Site

Edmonton, Alberta, Canada

Site Status

Research Site

Vancouver, British Columbia, Canada

Site Status

Research Site

Kentville, Nova Scotia, Canada

Site Status

Research Site

Barrie, Ontario, Canada

Site Status

Research Site

Burlington, Ontario, Canada

Site Status

Research Site

Hamilton, Ontario, Canada

Site Status

Research Site

Kitchener, Ontario, Canada

Site Status

Research Site

London, Ontario, Canada

Site Status

Research Site

Mississauga, Ontario, Canada

Site Status

Research Site

North York, Ontario, Canada

Site Status

Research Site

Oakville, Ontario, Canada

Site Status

Research Site

Ottawa, Ontario, Canada

Site Status

Research Site

Toronto, Ontario, Canada

Site Status

Research Site

Granby, Quebec, Canada

Site Status

Research Site

Laval, Quebec, Canada

Site Status

Research Site

Montreal, Quebec, Canada

Site Status

Research Site

Point-Claire, Quebec, Canada

Site Status

Research Site

Québec, Quebec, Canada

Site Status

Research Site

Haidian District, Beijing Municipality, China

Site Status

Research Site

XI Cheng District, Beijing Municipality, China

Site Status

Research Site

Xicheng District, Beijing Municipality, China

Site Status

Research Site

Wuhan, Hubei, China

Site Status

Research Site

Nanjing, Jiangsu, China

Site Status

Research Site

Pudong New Area, Shanghai Municipality, China

Site Status

Research Site

Shanghai, Shanghai Municipality, China

Site Status

Research Site

Xuhui District, Shanghai Municipality, China

Site Status

Research Site

Xi’an, Shanxi, China

Site Status

Research Site

Brno, Brno, Czechia

Site Status

Research Site

Olomouc, Olomouc, Czechia

Site Status

Research Site

Prague, Prague, Czechia

Site Status

Research Site

Ústí nad Labem, Usti nad Labem, Czechia

Site Status

Research Site

Aalborg, Aalborg, Denmark

Site Status

Research Site

Aarhus, Aarhus, Denmark

Site Status

Research Site

Herlev, Herlev, Denmark

Site Status

Research Site

Copenhagen, Kobenhavn, Denmark

Site Status

Research Site

Joensuu, Joensuu, Finland

Site Status

Research Site

Kajaanintie, Kajaanintie, Finland

Site Status

Research Site

Tampere, Pirkanmaa, Finland

Site Status

Research Site

Montpellier, Montpellier, France

Site Status

Research Site

Paris, Paris, France

Site Status

Research Site

Poitiers, Poitiers Cedex, France

Site Status

Research Site

Suresnes, Suresnes, France

Site Status

Research Site

Toulouse, Toulouse, France

Site Status

Research Site

Villejuif, Villejuif, France

Site Status

Research Site

Augsburg, Augsburg, Germany

Site Status

Research Site

Bad Gegeberg, Bad Gegeberg, Germany

Site Status

Research Site

Emmendingen, Emmendingen, Germany

Site Status

Research Site

Leipzig, Leipzig, Germany

Site Status

Research Site

Lübeck, Luebeck, Germany

Site Status

Research Site

Mannheim, Mannheim, Germany

Site Status

Research Site

München, Muenchen, Germany

Site Status

Research Site

Planegg, Muenchen, Germany

Site Status

Research Site

Reutlingen, Reutlingen, Germany

Site Status

Research Site

Berlin, State of Berlin, Germany

Site Status

Research Site

Kirchheim, Teck, Germany

Site Status

Research Site

Hong Kong, Hong Kong, Hong Kong

Site Status

Research Site

Tuenmen, Hong Kong, Hong Kong

Site Status

Research Site

Shatin, Shatin, Hong Kong

Site Status

Research Site

Budapest, Budapest, Hungary

Site Status

Research Site

Debrecen, Debrecen, Hungary

Site Status

Research Site

Miskolc, Miskolc, Hungary

Site Status

Research Site

Nyíregyháza, Nyiregyhaza, Hungary

Site Status

Research Site

Szeged, Szeged, Hungary

Site Status

Research Site

Gujarat, Gujarat, India

Site Status

Research Site

Trivandrum, Kerala, India

Site Status

Research Site

Bhopal, Madhya Pradesh, India

Site Status

Research Site

Mumbai, Maharashtra, India

Site Status

Research Site

Rohini, National Capital Territory of Delhi, India

Site Status

Research Site

New Delhi, New Delhi, India

Site Status

Research Site

Chandigarh, Punjab, India

Site Status

Research Site

Ludhiana, Punjab, India

Site Status

Research Site

Bikaner, Rajasthan, India

Site Status

Research Site

Jaipur, Rajasthan, India

Site Status

Research Site

Kolkota, West Bengal, India

Site Status

Research Site

Milan, Milan, Italy

Site Status

Research Site

Rome, Rome, Italy

Site Status

Research Site

Asahi, Chiba, Japan

Site Status

Research Site

Chiba, Chiba, Japan

Site Status

Research Site

Narashino, Chiba, Japan

Site Status

Research Site

Matsuyama, Ehime, Japan

Site Status

Research Site

Fukuoka, Fukuoka, Japan

Site Status

Research Site

Maebashi, Gunma, Japan

Site Status

Research Site

Ōtake, Hiroshima, Japan

Site Status

Research Site

Sapporo, Hokkaido, Japan

Site Status

Research Site

Kobe, Hyōgo, Japan

Site Status

Research Site

Tsukuba, Ibaraki, Japan

Site Status

Research Site

Kita-gun, Kagawa-ken, Japan

Site Status

Research Site

Sagamihara, Kanagawa, Japan

Site Status

Research Site

Kyoto, Kyoto, Japan

Site Status

Research Site

Sendai, Miyagi, Japan

Site Status

Research Site

Nagasaki, Nagasaki, Japan

Site Status

Research Site

Ōita, Oita Prefecture, Japan

Site Status

Research Site

Osaka, Osaka, Japan

Site Status

Research Site

Ōsaka-sayama, Osaka, Japan

Site Status

Research Site

Suita, Osaka, Japan

Site Status

Research Site

Wako, Saitama, Japan

Site Status

Research Site

Hamamatsu, Shizuoka, Japan

Site Status

Research Site

Sunto-gun, Shizuoka, Japan

Site Status

Research Site

Bunkyo-ku, Tokyo, Japan

Site Status

Research Site

Fuchu_city, Tokyo, Japan

Site Status

Research Site

Itabashi-Ku, Tokyo, Japan

Site Status

Research Site

Meguro-ku, Tokyo, Japan

Site Status

Research Site

Mitaka, Tokyo, Japan

Site Status

Research Site

Shinjuku-ku, Tokyo, Japan

Site Status

Research Site

Mexico City, Mexico City, Mexico

Site Status

Research Site

Distrito Federal Ciudad, Mexico, Mexico

Site Status

Research Site

Metepec, State of Mexico, Mexico

Site Status

Research Site

Amsterdam, Amsterdam, Netherlands

Site Status

Research Site

Eindhoven, Eindhoven, Netherlands

Site Status

Research Site

Nijmegen, Nijmegen, Netherlands

Site Status

Research Site

Groningen, Provincie Groningen, Netherlands

Site Status

Research Site

Bialystok, Bialystok, Poland

Site Status

Research Site

Kościerzyna, Koscierzyna, Poland

Site Status

Research Site

Krakow, Krakow, Poland

Site Status

Research Site

Rzeszów, Rzeszow, Poland

Site Status

Research Site

Warsaw, Warszawa, Poland

Site Status

Research Site

Wroclaw, Wroclaw, Poland

Site Status

Research Site

Coimbra, Coimbra District, Portugal

Site Status

Research Site

Lisbon, Lisbon District, Portugal

Site Status

Research Site

Porto, Porto District, Portugal

Site Status

Research Site

Barnaul, Barnaul, Russia

Site Status

Research Site

Stary Oskol, Belgorod Oblast, Russia

Site Status

Research Site

Izhevsk, Izhevsk, Russia

Site Status

Research Site

Kursk, Kursk Oblast, Russia

Site Status

Research Site

Moscow, Moscow, Russia

Site Status

Research Site

Saint Petersgurg, Saint Petersgurg, Russia

Site Status

Research Site

Sochi, Sochi, Russia

Site Status

Research Site

Voronezh, Voronezh Oblast, Russia

Site Status

Research Site

Belgrade, Belgrade, Serbia

Site Status

Research Site

Niš, Nis, Serbia

Site Status

Research Site

Novi Sad, Novi Sad, Serbia

Site Status

Research Site

Singapore, Singapore, Singapore

Site Status

Research Site

Bloemfontein, Bloemfontein, South Africa

Site Status

Research Site

Tygerberg, Cape Town, South Africa

Site Status

Research Site

Pietermaritzburg, Pietermaritzburg, South Africa

Site Status

Research Site

Port Elizabeth, Port Elizabeth, South Africa

Site Status

Research Site

Seo-gu, Busan, South Korea

Site Status

Research Site

Seongnam-si, Gyeonggi-do, South Korea

Site Status

Research Site

Heungduk-gu Cheongju, North Chungcheong, South Korea

Site Status

Research Site

Gangnam-gu, Seoul, South Korea

Site Status

Research Site

Songpa-gu, Seoul, South Korea

Site Status

Research Site

Gothenburg, Goteborg, Sweden

Site Status

Research Site

Gothenburg, Gothenburg, Sweden

Site Status

Research Site

Stockholm, Stockholm County, Sweden

Site Status

Research Site

Basel, Basel, Switzerland

Site Status

Research Site

Bern, Canton of Bern, Switzerland

Site Status

Research Site

Locarno, Locarno, Switzerland

Site Status

Research Site

Sursee, Sursee, Switzerland

Site Status

Research Site

Kaohsiung City, Kaohsiung, Taiwan

Site Status

Research Site

Taipei, Taipei, Taiwan

Site Status

Research Site

Taoyuan District, Taiwan, Taiwan

Site Status

Research Site

Reading, Berkshire, United Kingdom

Site Status

Research Site

Cambridge, Cambridgeshire, United Kingdom

Site Status

Research Site

Maidstone, Kent, United Kingdom

Site Status

Research Site

London, London, United Kingdom

Site Status

Research Site

Huddersfield, Yorkshire, United Kingdom

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States Argentina Australia Austria Belgium Brazil Canada China Czechia Denmark Finland France Germany Hong Kong Hungary India Italy Japan Mexico Netherlands Poland Portugal Russia Serbia Singapore South Africa South Korea Sweden Switzerland Taiwan United Kingdom

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

2007-003227-20

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

D4320C00014

Identifier Type: -

Identifier Source: org_study_id

NCT00707395

Identifier Type: -

Identifier Source: nct_alias

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.