Study to Evaluate the Safety and Efficacy of E/C/F/TAF Versus E/C/F/TDF in HIV-1 Positive, Antiretroviral Treatment-Naive Adults

NCT ID: NCT01797445

Last Updated: 2020-03-02

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

View full results

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

872 participants

Study Classification

INTERVENTIONAL

Study Start Date

2013-03-12

Study Completion Date

2018-10-03

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

The primary objective of this study is to evaluate the efficacy of elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide (E/C/F/TAF) fixed-dose combination (FDC) versus elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate (E/C/F/TDF) in HIV-1 positive, antiretroviral treatment-naive adults.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

HIV HIV Infections

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

E/C/F/TAF (Double-Blind)

E/C/F/TAF plus E/C/F/TDF placebo for 144 weeks

After 144 weeks, participants will continue to take their blinded study drug until treatment assignments have been unblinded.

Group Type EXPERIMENTAL

E/C/F/TAF

Intervention Type DRUG

150/150/200/10 mg FDC tablet administered orally once daily

E/C/F/TDF Placebo

Intervention Type DRUG

Tablet administered orally once daily

E/C/F/TDF (Double-Blind)

E/C/F/TDF plus E/C/F/TAF placebo for 144 weeks

After 144 weeks, participants will continue to take their blinded study drug until treatment assignments have been unblinded.

Group Type ACTIVE_COMPARATOR

E/C/F/TDF

Intervention Type DRUG

150/150/200/300 mg FDC tablet administered orally once daily

E/C/F/TAF Placebo

Intervention Type DRUG

Tablet administered orally once daily

Open-Label E/C/F/TAF

After the unblinding visit, in countries where E/C/F/TAF is not commercially available, participants (except in UK) who complete 144 weeks of study will be given the option to receive open-label E/C/F/TAF and attend study visits every 12 weeks until it becomes commercially available, or until Gilead terminates the study in that country.

Group Type EXPERIMENTAL

E/C/F/TAF

Intervention Type DRUG

150/150/200/10 mg FDC tablet administered orally once daily

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

E/C/F/TAF

150/150/200/10 mg FDC tablet administered orally once daily

Intervention Type DRUG

E/C/F/TDF

150/150/200/300 mg FDC tablet administered orally once daily

Intervention Type DRUG

E/C/F/TDF Placebo

Tablet administered orally once daily

Intervention Type DRUG

E/C/F/TAF Placebo

Tablet administered orally once daily

Intervention Type DRUG

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

Genvoya® Stribild®

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Ability to understand and sign a written informed consent form, which must be obtained prior to initiation of study procedures
* Plasma HIV-1 RNA levels ≥ 1,000 copies/mL at screening
* No prior use of any approved or investigational antiretroviral drug for any length of time, except the use for pre-exposure prophylaxis (PREP), or post-exposure prophylaxis (PEP) up to 6 months prior to screening
* Screening genotype report must show sensitivity to elvitegravir, emtricitabine, tenofovir DF
* Normal electrocardiogram (ECG)
* Estimated glomerular filtration rate (eGFR) ≥ 50 mL/min according to the Cockcroft-Gault formula for creatinine clearance
* Hepatic transaminases (AST and ALT) ≤ 5 × upper limit of normal (ULN)
* Total bilirubin ≤ 1.5 mg/dL, or normal direct bilirubin
* Adequate hematologic function
* Serum amylase ≤ 5 × ULN
* Males and females of childbearing potential must agree to utilize highly effective contraception methods or be non-heterosexually active or practice sexual abstinence from screening throughout the duration of study treatment and for 30 days following the last dose of study drug
* Females who utilize hormonal contraceptive as one of their birth control methods must have used the same method for at least three months prior to study dosing
* Females who have stopped menstruating for ≥ 12 months but do not have documentation of ovarian hormonal failure must have a serum follicle stimulating hormone (FSH) level at screening within the post-menopausal range based on the Central Laboratory reference range
* Age ≥ 18 years

Exclusion Criteria

* A new AIDS-defining condition diagnosed within the 30 days prior to screening
* Hepatitis B surface antigen (HBsAg) positive
* Hepatitis C antibody positive
* Individuals experiencing decompensated cirrhosis
* Females who are breastfeeding
* Positive serum pregnancy test
* Have an implanted defibrillator or pacemaker
* Current alcohol or substance use judged by the Investigator to potentially interfere with study compliance
* History of malignancy within the past 5 years or ongoing malignancy other than cutaneous Kaposi's sarcoma, basal cell carcinoma, or resected, noninvasive cutaneous squamous carcinoma
* Active, serious infections (other than HIV-1 infection) requiring parenteral antibiotic or antifungal therapy within 30 days prior to baseline
* Any other clinical condition or prior therapy that, in the opinion of the Investigator, would make the individual unsuitable for the study or unable to comply with dosing requirements
* Participation in any other clinical trial (including observational trials) without prior approval
* Receiving ongoing therapy with drugs not to be used with elvitegravir, cobicistat, emtricitabine, tenofovir DF, and TAF or participants with any known allergies to the excipients of E/C/F/TDF or E/C/F/TAF
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Gilead Sciences

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Gilead Study Director

Role: STUDY_DIRECTOR

Gilead Sciences

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

University of Alabama at Birmingham

Birmingham, Alabama, United States

Site Status

Spectrum Medical Group

Phoenix, Arizona, United States

Site Status

Kaiser Permanente - Los Angeles Medical Center

Los Angeles, California, United States

Site Status

University of Southern California AIDS Clinical Trials Group

Los Angeles, California, United States

Site Status

Peter J. Ruane, Inc.

Los Angeles, California, United States

Site Status

Anthony Mills MD Inc

Los Angeles, California, United States

Site Status

Alameda County Medical Center

Oakland, California, United States

Site Status

Stanford University

Palo Alto, California, United States

Site Status

University of California, Davis Medical Center

Sacramento, California, United States

Site Status

Kaiser Permanente Medical Group

Sacramento, California, United States

Site Status

La Playa Medical Group and Clinical Research

San Diego, California, United States

Site Status

Kaiser Permanente San Francisco

San Francisco, California, United States

Site Status

Kaiser Permanente

San Leandro, California, United States

Site Status

Los Angeles Biomedical Research Institute at Harbor - UCLA Medical Center

Torrance, California, United States

Site Status

University of Colorado

Aurora, Colorado, United States

Site Status

APEX Research LLC

Denver, Colorado, United States

Site Status

Greenwich Hospital

Greenwich, Connecticut, United States

Site Status

Yale University

New Haven, Connecticut, United States

Site Status

Dupont Circle Physicians Group

Washington D.C., District of Columbia, United States

Site Status

Whitman-Walker Health

Washington D.C., District of Columbia, United States

Site Status

Capital Medical Associates, PC

Washington D.C., District of Columbia, United States

Site Status

Medical Faculty Associates

Washington D.C., District of Columbia, United States

Site Status

Gary J. Richmond,M.D.,P.A.

Fort Lauderdale, Florida, United States

Site Status

Midway Immunology and Research Center

Ft. Pierce, Florida, United States

Site Status

AIDS Healthcare Foundation

Miami, Florida, United States

Site Status

AIDS Healthcare Foundation

Miami Beach, Florida, United States

Site Status

Orlando Immunology Center

Orlando, Florida, United States

Site Status

Idocf/Valuhealthmd

Orlando, Florida, United States

Site Status

Infectious Diseases Associates of NW FL

Sarasota, Florida, United States

Site Status

University of South Florida

Tampa, Florida, United States

Site Status

Infectious Disease Research Institute Inc.

Tampa, Florida, United States

Site Status

St. Joseph's Comprehensive Research Institute

Tampa, Florida, United States

Site Status

Triple O Research Institute PA

West Palm Beach, Florida, United States

Site Status

AIDS Research Consortium of Atlanta

Atlanta, Georgia, United States

Site Status

Atlanta ID Group, PC

Atlanta, Georgia, United States

Site Status

Emory University

Atlanta, Georgia, United States

Site Status

Georgia Regents University

Augusta, Georgia, United States

Site Status

Infectious Disease Specialist of Atlanta

Decatur, Georgia, United States

Site Status

Mercer University

Macon, Georgia, United States

Site Status

University of Hawaii - Hawaii Center for AIDS

Honolulu, Hawaii, United States

Site Status

Rush University Medical Center, Section of Infectious Diseases

Chicago, Illinois, United States

Site Status

The Ruth M. Rothstein CORE Center

Chicago, Illinois, United States

Site Status

Community Research Initiative of New England

Boston, Massachusetts, United States

Site Status

The Research Institute

West Springfield, Massachusetts, United States

Site Status

Be Well Medical Center

Berkley, Michigan, United States

Site Status

Henry Ford Health System

Detroit, Michigan, United States

Site Status

Hennepin County Medical Center

Minneapolis, Minnesota, United States

Site Status

Central West Clinical Research

St Louis, Missouri, United States

Site Status

Southampton Healthcare, Inc.

St Louis, Missouri, United States

Site Status

ID Care

Hillsborough, New Jersey, United States

Site Status

Southwest CARE Center

Santa Fe, New Mexico, United States

Site Status

Albany Medical College

Albany, New York, United States

Site Status

Upstate ID Assoc

Albany, New York, United States

Site Status

North Shore University Hospital - Division of Infectious Diseases

Manhasset, New York, United States

Site Status

Chelsea Village Medical

New York, New York, United States

Site Status

Columbia University Medical Center

New York, New York, United States

Site Status

Weill Cornell Medical College

New York, New York, United States

Site Status

Jacobi Medical Center

The Bronx, New York, United States

Site Status

Montefiore Medical Center

The Bronx, New York, United States

Site Status

University of North Carolina AIDS Clinical Trials Unit

Chapel Hill, North Carolina, United States

Site Status

Carolinas Medical Center Myer's Park Clinic

Charlotte, North Carolina, United States

Site Status

Duke University Medical Center

Durham, North Carolina, United States

Site Status

East Carolina University The Brody School of Medicine

Greenville, North Carolina, United States

Site Status

Rosedale Infectious Disseases

Huntersville, North Carolina, United States

Site Status

Wake Forest University Health Sciences

Winston-Salem, North Carolina, United States

Site Status

University of Pennsylvania

Philadelphia, Pennsylvania, United States

Site Status

The Miriam Hospital

Providence, Rhode Island, United States

Site Status

Central Texas Clinical Research

Austin, Texas, United States

Site Status

St. Hope Foundation, Inc.

Bellaire, Texas, United States

Site Status

Trinity Health & Wellness Center / AIDS Arms, Inc.

Dallas, Texas, United States

Site Status

Southwest Infectious Disease Clinical Research, Inc.

Dallas, Texas, United States

Site Status

North Texas Infectious Diseases Consultants

Dallas, Texas, United States

Site Status

Tarrant County Infectious Disease Associates

Fort Worth, Texas, United States

Site Status

Therapeutic Concepts, PA

Houston, Texas, United States

Site Status

Gordon E. Crofoot, MD, PA

Houston, Texas, United States

Site Status

Research Access Network

Houston, Texas, United States

Site Status

DCOL Center for Clinical Research

Longview, Texas, United States

Site Status

Clinical Alliance for Research & Education - Infectious Diseases (CARE-ID)

Annandale, Virginia, United States

Site Status

Peter Shalit, MD

Seattle, Washington, United States

Site Status

Research Institute of McGill University Health Care

Montreal, Quebec, Canada

Site Status

Clinique Medicale L'actuel

Montreal, , Canada

Site Status

University Health Network/Toronto General Hospital

Toronto, , Canada

Site Status

Maple Leaf Research

Toronto, , Canada

Site Status

Spectrum Health Care

Vancouver, , Canada

Site Status

Instituto Dominicano de Estudios Virologicos--IDEV

Santo Domingo, , Dominican Republic

Site Status

Hopital de la Croix Rousse

Lyon, , France

Site Status

University Hospital of Montpellier (CHU-Gui de Chauliac)

Montpellier, , France

Site Status

Archet 1 CHU de Nice, Department of Infectiology

Nice, , France

Site Status

Saint Louis Hospital of Infectious Diseases

Paris, , France

Site Status

Hopital Saint Antoine

Paris, , France

Site Status

Hôpital Bichat Claude Bernard

Paris, , France

Site Status

Hopital Tenon

Paris, , France

Site Status

Hopital Pitie Salpetriere

Paris, , France

Site Status

CH Tourcoing

Tourcoing, , France

Site Status

Universitaria di Bologna-Policlicnico S' Orsola Malpighi

Bologna, , Italy

Site Status

IRCCS Ospedale San Raffaele

Milan, , Italy

Site Status

Hospital Civil de Guadalajara

Guadalajara, , Mexico

Site Status

Insituto Nacional De Enfermedades Respiratorias "Ismael Cosio Villegas"

Mexico City, , Mexico

Site Status

Onze Lieve Vrouwe Gasthuis

Amsterdam, , Netherlands

Site Status

Serviço de Doenças Infecciosas, HUC-CHUC, EPE

Coimbra, , Portugal

Site Status

Hospital Santo Antonio dos Capuchos

Lisbon, , Portugal

Site Status

Hospital de Santa Maria - CHLN, EPE

Lisbon, , Portugal

Site Status

Centro Hospitalar do Porto - Hospital Joaquim Urbano

Porto, , Portugal

Site Status

Hope Clinical Research

San Juan, , Puerto Rico

Site Status

University of Puerto Rico ACTU

San Juan, , Puerto Rico

Site Status

Venhalsan / Sodersjukhuset

Stockholm, , Sweden

Site Status

Karolinska University Hospital, Huddinge

Stockholm, , Sweden

Site Status

Whittall Street Clinic

Birmingham, , United Kingdom

Site Status

Heart Of England NHS Foundation Trust

Birmingham, , United Kingdom

Site Status

Brighton and Sussex University Hospitals NHS Trust

Brighton, , United Kingdom

Site Status

Brownlee Centre, Gartnavel General Hospital

Glasgow, , United Kingdom

Site Status

Barts Health NHS Trust

London, , United Kingdom

Site Status

Royal Free London NHS Foundation Trust

London, , United Kingdom

Site Status

Kings College Hospital

London, , United Kingdom

Site Status

Chelsea and Westminster

London, , United Kingdom

Site Status

Mortimer Market Centre

London, , United Kingdom

Site Status

North Manchester General Hospital

Manchester, , United Kingdom

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States Canada Dominican Republic France Italy Mexico Netherlands Portugal Puerto Rico Sweden United Kingdom

References

Explore related publications, articles, or registry entries linked to this study.

Sax PE, Wohl D, Yin MT, Post F, DeJesus E, Saag M, Pozniak A, Thompson M, Podzamczer D, Molina JM, Oka S, Koenig E, Trottier B, Andrade-Villanueva J, Crofoot G, Custodio JM, Plummer A, Zhong L, Cao H, Martin H, Callebaut C, Cheng AK, Fordyce MW, McCallister S; GS-US-292-0104/0111 Study Team. Tenofovir alafenamide versus tenofovir disoproxil fumarate, coformulated with elvitegravir, cobicistat, and emtricitabine, for initial treatment of HIV-1 infection: two randomised, double-blind, phase 3, non-inferiority trials. Lancet. 2015 Jun 27;385(9987):2606-15. doi: 10.1016/S0140-6736(15)60616-X. Epub 2015 Apr 15.

Reference Type RESULT
PMID: 25890673 (View on PubMed)

Margot N, Cox S, Das M, McCallister S, Miller MD, Callebaut C. Rare emergence of drug resistance in HIV-1 treatment-naive patients receiving elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide for 144 weeks. J Clin Virol. 2018 Jun;103:37-42. doi: 10.1016/j.jcv.2018.03.012. Epub 2018 Apr 2.

Reference Type RESULT
PMID: 29627709 (View on PubMed)

Arribas JR, Thompson M, Sax PE, Haas B, McDonald C, Wohl DA, DeJesus E, Clarke AE, Guo S, Wang H, Callebaut C, Plummer A, Cheng A, Das M, McCallister S. Brief Report: Randomized, Double-Blind Comparison of Tenofovir Alafenamide (TAF) vs Tenofovir Disoproxil Fumarate (TDF), Each Coformulated With Elvitegravir, Cobicistat, and Emtricitabine (E/C/F) for Initial HIV-1 Treatment: Week 144 Results. J Acquir Immune Defic Syndr. 2017 Jun 1;75(2):211-218. doi: 10.1097/QAI.0000000000001350.

Reference Type RESULT
PMID: 28282300 (View on PubMed)

Margot N, Cox S, Das M, McCallister S, Miller MD, Callebaut C. Infrequent development of drug resistance in HIV-1-infected treatment-naive subjects after 96 weeks of treatment with elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide or elvitegravir/cobicistat/emtricitabine/tenofovir disoproxil fumarate. Antivir Ther. 2017;22(5):443-446. doi: 10.3851/IMP3125. Epub 2017 Jan 11.

Reference Type RESULT
PMID: 28076335 (View on PubMed)

Margot NA, Kitrinos KM, Fordyce M, McCallister S, Miller MD, Callebaut C. Rare emergence of drug resistance in HIV-1 treatment-naive patients after 48 weeks of treatment with elvitegravir/cobicistat/emtricitabine/tenofovir alafenamide. HIV Clin Trials. 2016 Mar;17(2):78-87. doi: 10.1080/15284336.2016.1142731.

Reference Type RESULT
PMID: 26892863 (View on PubMed)

Funderburg NT, McComsey GA, Kulkarni M, Bannerman T, Mantini J, Thornton B, Liu HC, Zhang Y, Song Q, Fang L, Dinoso J, Cheng A, McCallister S, Fordyce MW, Das M. Equivalent Decline in Inflammation Markers with Tenofovir Disoproxil Fumarate vs. Tenofovir Alafenamide. EBioMedicine. 2016 Nov;13:321-327. doi: 10.1016/j.ebiom.2016.10.009. Epub 2016 Oct 11.

Reference Type RESULT
PMID: 27742226 (View on PubMed)

Wohl D, Oka S, Clumeck N, Clarke A, Brinson C, Stephens J, Tashima K, Arribas JR, Rashbaum B, Cheret A, Brunetta J, Mussini C, Tebas P, Sax PE, Cheng A, Zhong L, Callebaut C, Das M, Fordyce M; GS-US-2,92-01040111 and Study Team. Brief Report: A Randomized, Double-Blind Comparison of Tenofovir Alafenamide Versus Tenofovir Disoproxil Fumarate, Each Coformulated With Elvitegravir, Cobicistat, and Emtricitabine for Initial HIV-1 Treatment: Week 96 Results. J Acquir Immune Defic Syndr. 2016 May 1;72(1):58-64. doi: 10.1097/QAI.0000000000000940.

Reference Type RESULT
PMID: 26829661 (View on PubMed)

Custodio JM, Garner W, Callebaut C, Fordyce M, Plummer A, Zhong L, et al. The Pharmacokinetics of Tenofovir and Tenofovir Diphosphate Following Administration of Tenofovir Alafenamide vs Tenofovir Disoproxil Fumarate [Oral Abstract #6]. The 16th International Workshop on Clinical Pharmacology of HIV & Hepatitis Therapy. Washington DC, USA, May 26-28, 2015.

Reference Type RESULT

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

2013-000102-37

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

GS-US-292-0111

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.