A Two-Stage Phase 1 Dose Escalation Pharmacokinetic Study of Tarceva in Patients With Stage IIIB/IV Non-small Cell Lung Cancer Who Continue to Smoke After Failure of One or Two Prior Chemotherapy Regimens

NCT ID: NCT00294736

Last Updated: 2012-08-08

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

57 participants

Study Classification

INTERVENTIONAL

Study Start Date

2005-11-30

Study Completion Date

2007-09-30

Brief Summary

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This is a multicenter, open-label, randomized phase 1 study of escalating doses of Tarceva in patients with advanced NSCLC who currently smoke.

Part I will establish the maximum tolerated dose (MTD) of Tarceva in current smokers.

In Part II, patients will be randomized 1:1 to two treatment groups: Arm A (Tarceva MTD established in Part I) and Arm B (150 mg Tarceva daily). Patients in both arms will be treated for two weeks and then have pharmacokinetic samples collected on day 14. Part II is open as of Nov-2006.

Detailed Description

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Conditions

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NSCLC

Keywords

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lung cancer erlotinib NSCLC smokers

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Arm A

Arm A (Tarceva MTD established in Part I)

Group Type EXPERIMENTAL

Tarceva

Intervention Type DRUG

Dose Escalation: 150-350+ mg/day

Arm B

Arm B (150 mg Tarceva daily).

Group Type EXPERIMENTAL

Tarceva

Intervention Type DRUG

Dose Escalation: 150-350+ mg/day

Interventions

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Tarceva

Dose Escalation: 150-350+ mg/day

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Histologically or cytologically confirmed diagnosis of stage IIIB/IV NSCLC;
* Must have received 1 or 2 prior chemotherapy regimens for advanced NSCLC and now have progressive disease;
* Must have recovered from any treatment-related toxicities prior to registration, except for alopecia, grade 1 fatigue, or grade 1 neurotoxicity;
* A current cigarette smoker (minimum of 10 cigarettes per day for \>= 1 year and have a positive test for cotinine) despite advice and support to quit;
* Age \>= 18 years;
* ECOG PS 0-1 and predicted life expectancy \>= 12 weeks;
* Previous surgery is permitted provided that wound healing has occurred prior to registration;
* Adequate hematopoietic, hepatic and renal function defined as follows: ANC \>= 1.5 x 10\^9/L, platelets \>= 100 x 10\^9/L, bilirubin \<= 1.5 x ULN, ALT \<= 2.5 x ULN (or 5 x ULN in case of liver metastases), creatinine \<= 1.5 x ULN;
* No prior treatment with Tarceva or gefitinib (or other drug with significant activity against EGFR (eg, cetuximab and/or ZD6474));
* Patients with reproductive potential must practice effective contraceptive measures throughout the study. Women of child-bearing potential must provide a negative pregnancy test within 14 days prior to registration;
* Accessible for repeat dosing and follow-up.

Exclusion Criteria

* Any concurrent anticancer cytostatic or cytotoxic chemotherapy;
* Concomitant CYP3A4 or CYP1A2 inducers/inhibitors (or during 14 days prior to study) with the exception of tobacco;
* Other active malignancies, unless disease-free and without cancer-specific therapy for at least the last 5 years. Basal or squamous cell skin cancers are not excluded;
* Significant history of cardiac disease unless the disease is well-controlled;
* Active or uncontrolled infections or serious illnesses or medical conditions that could interfere with the patient's ongoing participation in the study;
* History of any psychiatric condition that might impair the patient's ability to understand or comply with the requirements; of the study or to provide informed consent.
* Gastrointestinal abnormalities, including inability to take oral medication, requirement for IV alimentation, active peptic ulcer or prior surgical procedures affecting absorption;
* Clinically significant ophthalmologic abnormalities;
* Pregnant or breast-feeding females. Males or females not practicing effective birth control;
* Symptomatic brain metastases which are not stable, require steroids, or that have required radiation within the last 28 days;
* History of allergic reactions attributed to compounds of similar chemical or biologic composition to the study drug;
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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OSI Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Medical Monitor

Role: STUDY_DIRECTOR

OSI Pharmaceuticals

Locations

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Comprehensive Blood and Cancer Center

Bakersfield, California, United States

Site Status

Wake Forest University Comprehensive Cancer Center

Winston-Salem, North Carolina, United States

Site Status

University of Edinburgh,Division of Oncology,

Edinburgh, Scotland, United Kingdom

Site Status

Aberdeen Royal Infirmary

Aberdeen, , United Kingdom

Site Status

Ninewells Hospital

Dundee, , United Kingdom

Site Status

Beatson West of Scotland Cancer Centre

Glasgow, , United Kingdom

Site Status

Sir Bobby Robson Cancer Trials Research Centre

Newcastle upon Tyne, , United Kingdom

Site Status

Department of Oncology

Sheffield, , United Kingdom

Site Status

Royal Marsden Hospital

Sutton, , United Kingdom

Site Status

Countries

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United States United Kingdom

Other Identifiers

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2005-003883-46

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

OSI-774-107

Identifier Type: -

Identifier Source: org_study_id