A Study of YL242 in Subjects With Advanced Solid Tumors

NCT ID: NCT07197827

Last Updated: 2025-12-24

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1/PHASE2

Total Enrollment

424 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-09-22

Study Completion Date

2028-11-30

Brief Summary

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This is a multicenter, open-label study to evaluate the safety and tolerability of YL242 monotherapy and combination in participants with advanced solid malignant tumors.

Detailed Description

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Conditions

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Advanced Solid Tumor

Keywords

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Oncology VEGF Antibody drug conjugate Developmental Phase I/II

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Part 1 and Part 2: Mono Dose Escalation & Expansion

Participants receive YL242 administered via intravenous (IV) solution per protocol defined dose level and frequency.

Group Type EXPERIMENTAL

YL242

Intervention Type DRUG

The YL242 drug product is provided as a lyophilized powder containing 200 mg of YL242 in a glass vial. The initial dose of YL242 will be infused IV into each patient for 90±10 minutes. If there is no infusion-related reaction after the initial dose, the second and subsequent doses of YL242 will be infused IV into each patient for 60±10 minutes.

Part 3 and 4: Combination Dose Escalation & Expansion

Participants receive YL242 at protocol defined dose level, in combination with Pembrolizumab (200 mg), administered via intravenous (IV) solution at protocol defined dose level and frequency.

Group Type EXPERIMENTAL

YL242; Pembrolizumab

Intervention Type DRUG

The YL242 drug product is provided as a lyophilized powder containing 200 mg of YL242 in a glass vial. The initial dose of YL242 will be infused IV into each patient for 90±10 minutes. If there is no infusion-related reaction after the initial dose, the second and subsequent doses of YL242 will be infused IV into each patient for 60±10 minutes. Pembrolizumab will be administered subsequent to YL242.

Part 5: Combination Dose Optimization and Expansion

Participants receive YL242, 5-FU and LV, administered via intravenous (IV) solution.

Group Type EXPERIMENTAL

YL242; 5-FU; LV

Intervention Type DRUG

The YL242 drug product is provided as a lyophilized powder containing 200 mg of YL242 in a glass vial. The initial dose of YL242 will be infused IV into each patient for 90±10 minutes. If there is no infusion-related reaction after the initial dose, the second and subsequent doses of YL242 will be infused IV into each patient for 60±10 minutes.

LV and 5-FU will be sequentially administered following YL242.

Part 6: Combination Dose Optimization and Expansion

Participants receive YL242, pembrolizumab and 5-FU, administered via intravenous (IV) solution at protocol defined frequency.

Group Type EXPERIMENTAL

YL242; Pembrolizumab; 5-FU

Intervention Type DRUG

The YL242 drug product is provided as a lyophilized powder containing 200 mg of YL242 in a glass vial. YL242 will be administered via Intravenous (IV) Infusion.

Pembrolizumab and 5-FU will be administered in sequence after YL242.

Interventions

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YL242

The YL242 drug product is provided as a lyophilized powder containing 200 mg of YL242 in a glass vial. The initial dose of YL242 will be infused IV into each patient for 90±10 minutes. If there is no infusion-related reaction after the initial dose, the second and subsequent doses of YL242 will be infused IV into each patient for 60±10 minutes.

Intervention Type DRUG

YL242; Pembrolizumab

The YL242 drug product is provided as a lyophilized powder containing 200 mg of YL242 in a glass vial. The initial dose of YL242 will be infused IV into each patient for 90±10 minutes. If there is no infusion-related reaction after the initial dose, the second and subsequent doses of YL242 will be infused IV into each patient for 60±10 minutes. Pembrolizumab will be administered subsequent to YL242.

Intervention Type DRUG

YL242; 5-FU; LV

The YL242 drug product is provided as a lyophilized powder containing 200 mg of YL242 in a glass vial. The initial dose of YL242 will be infused IV into each patient for 90±10 minutes. If there is no infusion-related reaction after the initial dose, the second and subsequent doses of YL242 will be infused IV into each patient for 60±10 minutes.

LV and 5-FU will be sequentially administered following YL242.

Intervention Type DRUG

YL242; Pembrolizumab; 5-FU

The YL242 drug product is provided as a lyophilized powder containing 200 mg of YL242 in a glass vial. YL242 will be administered via Intravenous (IV) Infusion.

Pembrolizumab and 5-FU will be administered in sequence after YL242.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Aged ≥18 years.
* Eastern Cooperative Oncology Group performance status (ECOG PS) of 0 or 1
* Adequate organ and bone marrow function
* Tumor type:

Part 1-3: Advanced/unresectable or metastatic solid malignant tumor; Have received at least one prior line of systemic anti-tumor therapy

Part 4: locally advanced or metastatic non-sq NSCLC without AGA and HCC; Have not received any systemic anti-tumor therapy;

Part 5: mCRC, have received at least one (5a) or one (5b) prior line of systemic anti-tumor therapy

Part 6: advanced or metastatic HER2-negative G/GEJ; have received at least one (6a) or one (6b) prior line of systemic anti-tumor therapy

Exclusion Criteria

* Be intolerant to prior treatment with a topoisomerase I inhibitor or an ADC that consists of a topoisomerase I inhibitor
* Uncontrolled or clinically significant cardiovascular and cerebrovascular diseases
* Clinically significant concomitant pulmonary disease
* A history of leptomeningeal carcinomatosis or carcinomatous meningitis
* Any illness, medical condition, organ system dysfunction, or social situation, including but not limited to mental illness or substance/alcohol abuse, deemed by the investigator to be likely to interfere with a patient's ability to sign informed consent, adversely affect the patient's ability to cooperate and participate in the study, or compromise the interpretation of study results
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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MediLink Therapeutics (Suzhou) Co., Ltd.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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US-201

New Haven, Connecticut, United States

Site Status NOT_YET_RECRUITING

US-202

Sarasota, Florida, United States

Site Status RECRUITING

US-204

Boston, Massachusetts, United States

Site Status NOT_YET_RECRUITING

US-206

Grand Rapids, Michigan, United States

Site Status RECRUITING

US-205

Nashville, Tennessee, United States

Site Status RECRUITING

US-203

Houston, Texas, United States

Site Status NOT_YET_RECRUITING

US-207

San Antonio, Texas, United States

Site Status NOT_YET_RECRUITING

AUS-101

Liverpool, New South Wales, Australia

Site Status NOT_YET_RECRUITING

AUS-102

Darlinghurst, Victoria, Australia

Site Status RECRUITING

AUS-104

Fitzroy, Victoria, Australia

Site Status NOT_YET_RECRUITING

AUS-103

Heidelberg, Victoria, Australia

Site Status NOT_YET_RECRUITING

AUS-105

Nedlands, Western Australia, Australia

Site Status NOT_YET_RECRUITING

CN-303

Harbin, Heilongjiang, China

Site Status RECRUITING

CN-301

Shanghai, Shanghai Municipality, China

Site Status RECRUITING

CN-302

Hangzhou, Zhejiang, China

Site Status RECRUITING

Countries

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United States Australia China

Central Contacts

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Medilink Study Team

Role: CONTACT

Phone: +86 0512-62858368

Email: [email protected]

Facility Contacts

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study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

study coordinator

Role: primary

Other Identifiers

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YL242-INT-101-01

Identifier Type: -

Identifier Source: org_study_id