Study of MK-4464 as Monotherapy and in Combination With Pembrolizumab in Participants With Advanced/Metastatic Solid Tumors (MK-4464-001)

NCT ID: NCT05514444

Last Updated: 2025-10-09

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

64 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-09-25

Study Completion Date

2025-09-18

Brief Summary

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The purpose of this study is to assess the safety, pharmacokinetics, and preliminary efficacy of MK-4464 as monotherapy and in combination with pembrolizumab in participants with advanced/metastatic solid tumors.

Detailed Description

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Conditions

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Advanced/Metastatic Solid Tumors Neoplasms

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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MK-4464

Participants will receive an intravenous (IV) infusion of MK-4464 administered in escalating doses every 3 weeks for up to 35 cycles. Escalation to subsequent MK-4464 doses will be based on safety of previous dose.

Group Type EXPERIMENTAL

MK-4464

Intervention Type BIOLOGICAL

MK-4464 administered as an IV infusion every three weeks according to allocation and dose escalation.

MK-4464 + Pembrolizumab

Participants will receive an IV infusion of MK-4464 administered in escalating doses and a 200 mg IV infusion of Pembrolizumab every 3 weeks for up to 35 cycles. Escalation to subsequent MK-4464 doses will be based on safety of MK-4464 monotherapy arm.

Group Type EXPERIMENTAL

MK-4464

Intervention Type BIOLOGICAL

MK-4464 administered as an IV infusion every three weeks according to allocation and dose escalation.

Pembrolizumab

Intervention Type BIOLOGICAL

Pembrolizumab 200 mg administered as an IV infusion every three weeks.

MK-4464 + Pembrolizumab + Zirconium 89 (89Zr)-MK-4464

Participants will receive an IV infusion of 89Zr-MK-4464 + IV infusion of MK-4464 on Cycle 1 Day 1, followed by an IV infusion of MK-4464 + a 200 mg IV infusion of pembrolizumab starting on Cycle 2 Day 1 and every 3 weeks for up to 35 cycles. Each cycle=3 weeks. MK-4464 doses will be based on safety of MK-4464 monotherapy arm. Participants may receive a 200 mg IV infusion of pembrolizumab on cycle 36.

Group Type EXPERIMENTAL

MK-4464

Intervention Type BIOLOGICAL

MK-4464 administered as an IV infusion every three weeks according to allocation and dose escalation.

Pembrolizumab

Intervention Type BIOLOGICAL

Pembrolizumab 200 mg administered as an IV infusion every three weeks.

89Zr-MK-4464

Intervention Type DRUG

89ZR-MK-4464 administered as an IV infusion on C1D1.

Interventions

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MK-4464

MK-4464 administered as an IV infusion every three weeks according to allocation and dose escalation.

Intervention Type BIOLOGICAL

Pembrolizumab

Pembrolizumab 200 mg administered as an IV infusion every three weeks.

Intervention Type BIOLOGICAL

89Zr-MK-4464

89ZR-MK-4464 administered as an IV infusion on C1D1.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Have a histologically or cytologically confirmed advanced/metastatic solid tumor by pathology report and have received, been intolerant to, been ineligible for, or refused all treatment known to confer clinical benefit
* Must submit a baseline tumor sample for analysis
* Have a performance status of 0 or 1 on the Eastern Cooperative Oncology Group (ECOG) Performance Scale
* Human immunodeficiency virus (HIV) infected participants must have well controlled HIV on antiretroviral therapy (ART)
* Participants who are HBsAg positive are eligible if they have received HBV antiviral therapy for at least 4 weeks, and have undetectable HBV viral load before randomization.

Exclusion Criteria

* Has had chemotherapy, definitive radiation, or biological cancer therapy within 4 weeks (2 weeks for palliative radiation) before the first dose of study intervention or has not recovered to CTCAE Grade 1 or better from any AEs that were due to cancer therapeutics administered more than 4 weeks earlier
* Has a history of a second malignancy, unless potentially curative treatment has been completed with no evidence of malignancy for 2 years
* Has clinically active central nervous system (CNS) metastases and/or carcinomatous meningitis
* Has an active infection requiring therapy
* History of an allogenic stem cell transplant or a solid organ transplant
* Has a history of (noninfectious) pneumonitis/interstitial lung disease that required steroids or has current pneumonitis/interstitial lung disease
* Has an active autoimmune disease that has required systemic treatment in the past 2 years
* HIV-infected participants with a history of Kaposi's sarcoma and/or Multicentric Castleman's Disease
* Has known psychiatric or substance abuse disorders that would interfere with the participant's ability to cooperate with the requirements of the study
* Has not fully recovered from any effects of major surgery without significant detectable infection
* Has received radiation therapy to the lung that is \>30 gray (Gy) within 6 months of the first dose of study treatment
* Received a live or live-attenuated vaccine within 30 days before the first dose of study intervention
* Is currently participating and receiving study intervention in a study of an investigational agent or has participated and received study intervention in a study of an investigational agent or has used an investigational device within 28 days
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Merck Sharp & Dohme LLC

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Medical Director

Role: STUDY_DIRECTOR

Merck Sharp & Dohme LLC

Locations

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The University of Louisville, James Graham Brown Cancer Center ( Site 0100)

Louisville, Kentucky, United States

Site Status

Princess Margaret Cancer Centre-Division of Medical Oncology and Hematology ( Site 0201)

Toronto, Ontario, Canada

Site Status

Rambam Health Care Campus-Oncology Division ( Site 0300)

Haifa, , Israel

Site Status

Hadassah Medical Center-Oncology ( Site 0302)

Jerusalem, , Israel

Site Status

Nederlands Kanker Instituut - Antoni van Leeuwenhoek - NKI-AVL ( Site 0401)

Amsterdam, North Holland, Netherlands

Site Status

Amsterdam UMC, locatie VUmc ( Site 0400)

Amsterdam, North Holland, Netherlands

Site Status

Countries

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United States Canada Israel Netherlands

Related Links

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Other Identifiers

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MK-4464-001

Identifier Type: OTHER

Identifier Source: secondary_id

2023-504855-28-00

Identifier Type: REGISTRY

Identifier Source: secondary_id

U1111-1290-2697

Identifier Type: REGISTRY

Identifier Source: secondary_id

2021-005882-42

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

4464-001

Identifier Type: -

Identifier Source: org_study_id

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