Open-Label Extension (OLE) Study to Assess Safety, Efficacy, and Tolerability of Lorundrostat in Subjects With Hypertension

NCT ID: NCT05968430

Last Updated: 2025-06-15

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE3

Total Enrollment

1400 participants

Study Classification

INTERVENTIONAL

Study Start Date

2023-07-14

Study Completion Date

2026-12-31

Brief Summary

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This study is to evaluate the long-term safety, efficacy and tolerability of lorundrostat (an aldosterone synthase inhibitor) in subjects with hypertension

Detailed Description

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The purpose of the study is to evaluate the long-term safety, efficacy, and tolerability of lorundrostat (an aldosterone synthase inhibitor) in subjects with hypertension.

This study consists of an open label treatment period of 52 weeks followed by a 2-week safety follow-up period. Eligible subjects for MLS-101-901 are those who were enrolled in one of the eligible parent studies, meet the eligibility criteria for this protocol, and agree, by signing an informed consent form (ICF), to transition to this open label extension (OLE) study at either the end-of-study (EoS) visit or the end-of-treatment (EoT) visit as required in the parent study protocol.

A Randomized Treatment Withdrawal (RTW) substudy will be performed in a subset of subjects meeting eligibility criteria.

Subjects who complete the open label treatment period will be invited to consent to an optional continuation period where they may remain on study until marketing authorization or early termination of the trial by the sponsor.

Conditions

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Hypertension

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Eligible subjects participating in the RTW will receive double-blind treatment with matching placebo. Upon completion, subjects will return to open-label treatment

Study Groups

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Open-Label Arm

lorundrostat once daily for 52 weeks depending on when the subject enrolled

Group Type EXPERIMENTAL

lorundrostat

Intervention Type DRUG

Tablet, administered orally

RTW Substudy

lorundrostat or placebo once daily for 4 weeks starting at week 12, in the double-blind randomized treatment withdrawal substudy

Optional for subjects from the MLS-101-301 parent study only

Group Type EXPERIMENTAL

lorundrostat

Intervention Type DRUG

Tablet, administered orally

Placebo

Intervention Type DRUG

Tablet, administered orally

Optional Continuation Period

lorundrostat once daily from week 52 or until marketing authorization or early termination of the trial by the sponsor

Group Type EXPERIMENTAL

lorundrostat

Intervention Type DRUG

Tablet, administered orally

Interventions

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lorundrostat

Tablet, administered orally

Intervention Type DRUG

Placebo

Tablet, administered orally

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Written informed consent signed by the participant, obtained before any study-related assessment is performed
2. At least 18 years of age at the time of signing the informed consent form (ICF)
3. Completed the EoT or EoS Visit (as applicable) in a lorundrostat study with the option of transitioning to the OLE study, in accordance with the parent study protocol
4. Fertile male subjects and female subjects of childbearing potential, and their partners, must agree to use an acceptable method of contraception from study entry to 28 days after the last dose of study drug
5. Willing and able to comply with the study instructions and attend all scheduled study visits

\[Randomized treatment withdrawal substudy only\]
6. Written informed consent to participate in the RTW substudy signed by the participant, obtained before any RTW study-related assessment is performed

Exclusion Criteria

1. Women who are pregnant, plan to become pregnant, or are breast-feeding
2. Use, or anticipated use during the course of the study, of a prohibited medication as listed in Section 6.7.1 of the protocol
3. In the opinion of the Investigator, any condition that will preclude participation in the study

\[Randomized treatment withdrawal substudy only\]
4. Non-compliance with study medication(s) (defined as taking \<75% or \>125% of the study drug provided) during the first 12 weeks of MLS-101-901
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Mineralys Therapeutics Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Accel Research Sites (ARS) - Birmingham Clinical Research Unit

Birmingham, Alabama, United States

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G & L Research LLC

Foley, Alabama, United States

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Chandler Clinical Trials

Chandler, Arizona, United States

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Arizona Kidney

Glendale, Arizona, United States

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AKDHC Medical Research Services, AZ

Phoenix, Arizona, United States

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Noble Clinical Research

Tucson, Arizona, United States

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Del Sol Research Management, LLC

Tucson, Arizona, United States

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Entertainment Medical Group, Inc

Beverly Hills, California, United States

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CA Institute of Renal Research, CA

Chula Vista, California, United States

Site Status

Amicis Research Center - Vacaville

Fairfield, California, United States

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Amicis Research Center - Granada Hills

Granada Hills, California, United States

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Marvel Clinical Research 002, LLC

Huntington Beach, California, United States

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University of California San Diego (UCSD) - Altman Clinical and Translational Research Institute (ACTRI)

La Jolla, California, United States

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Clinical Trials Research (CTR) - Lincoln

Lincoln, California, United States

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Academic Medical Research Institute (AMRI) - Los Angeles

Los Angeles, California, United States

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Cedars-Sinai Medical Center

Los Angeles, California, United States

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Amicis Research Center - Mission Hills

Northridge, California, United States

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Amicis Research Center-Northridge

Northridge, California, United States

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Northridge Clinical Trials

Northridge, California, United States

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Pasadena Clinical Trials

Pasadena, California, United States

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Empire Clinical Research

Pomona, California, United States

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Clinical Trials Research (CTR) - Sacramento

Sacramento, California, United States

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Triwest Research Associates

San Diego, California, United States

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San Jose Clinical Trials

San Jose, California, United States

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Amicis Research Center - Valencia

Valencia, California, United States

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Kidney & Hypertension Center - Victorville

Victorville, California, United States

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Blue Coast Research Center (BCRC)

Vista, California, United States

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Accelerated Enrollment Solutions (AES) -Vista/Synexus (Radiant Research)

Vista, California, United States

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Colorado Kidney (Denver) Nephrology

Denver, Colorado, United States

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CMR of Greater New Haven

Hamden, Connecticut, United States

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Qway Research

Hialeah, Florida, United States

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Indago Research and Health Center

Hialeah, Florida, United States

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Clinical Neuroscience Solutions, Inc

Jacksonville, Florida, United States

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Nuovida Research Center Corp

Miami, Florida, United States

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Clinical Neuroscience Solutions, Inc

Orlando, Florida, United States

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Nephrology Associates of Central Florida

Orlando, Florida, United States

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AES - Orlando

Orlando, Florida, United States

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Pines Care Research Center

Pembroke Pines, Florida, United States

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Patron Medical - Andres Patron D.O. (Patron Ventures, LLC)

Pembroke Pines, Florida, United States

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Progressive Medical Research

Port Orange, Florida, United States

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Infigo Clinical Research (Mid Florida)

Sanford, Florida, United States

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Clinical Research of West Florida, Inc.

Tampa, Florida, United States

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AES The Villages

The Villages, Florida, United States

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Palm Beach Diabetes and Endocrine Specialists, PA (PBDES) - West Palm Beach Office)

West Palm Beach, Florida, United States

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American Clinical Trials

Acworth, Georgia, United States

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Morehouse School of Medicine

Atlanta, Georgia, United States

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Coastal Medical

Brunswick, Georgia, United States

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Accel Research Sites

Decatur, Georgia, United States

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Georgia Clinical Research, LLC

Lawrenceville, Georgia, United States

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Alta Pharmaceutical Research Center

Peachtree Corners, Georgia, United States

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Elite Clinical Trials

Blackfoot, Idaho, United States

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Meridian Family Medicine

Meridian, Idaho, United States

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AES Chicago/Synexus Clinical Research

Chicago, Illinois, United States

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Eagle Clinical Research

Chicago, Illinois, United States

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The University of Chicago Medicine

Chicago, Illinois, United States

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Healthcare Research Network - Chicago

Flossmoor, Illinois, United States

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Koch Family Medicine, S.C

Morton, Illinois, United States

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Southern Illinois School of Medicine

Springfield, Illinois, United States

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Hendricks Regional Health Medical Group - Lizton Family Medicine

Brownsburg, Indiana, United States

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AES Evansville/Synexus Clinical Research

Evansville, Indiana, United States

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ASHA Clinical Research- Munster, LLC

Hammond, Indiana, United States

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The Research Group of Lexington, LLC

Lexington, Kentucky, United States

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Nephrology Associates of Kentuckiana

Louisville, Kentucky, United States

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Alliance for Multispecialty Research, LLC

New Orleans, Louisiana, United States

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Northwest Louisiana Nephrology, LLC - Shreveport

Shreveport, Louisiana, United States

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Boston Clinical Trials

Boston, Massachusetts, United States

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ActiveMed Practices & Research LLC

Methuen, Massachusetts, United States

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Hattiesburg Clinic

Petal, Mississippi, United States

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Healthcare Research Network-Hazelwood

Hazelwood, Missouri, United States

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Clinical Research Consultants (CRC) - Kansas City

Kansas City, Missouri, United States

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Quality Clinical Research

Omaha, Nebraska, United States

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AES - Nevada

Henderson, Nevada, United States

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Henderson Clinical Trials

Henderson, Nevada, United States

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Sierra Clinical Research

Las Vegas, Nevada, United States

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Oasis Clinical Trials

Las Vegas, Nevada, United States

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Las Vegas Clinical Trials

North Las Vegas, Nevada, United States

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Renown Regional Medical Center

Reno, Nevada, United States

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Albany Medical College

Albany, New York, United States

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Erie County Medical Center

Buffalo, New York, United States

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AES New York/Synexus Clinical Research

New York, New York, United States

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Columbia University

New York, New York, United States

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Triad Internal Medicine

Asheboro, North Carolina, United States

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East Carolina University (ECU) Physicians - East Carolina Heart Institute - East Carolina University Location

Greenville, North Carolina, United States

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Physician's East Endocrinology

Greenville, North Carolina, United States

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Carteret Medical Group

Morehead City, North Carolina, United States

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Lucas Research

New Bern, North Carolina, United States

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Research Innovations (Elligo Health Research)

Beavercreek, Ohio, United States

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Diabetes & Endocrinology Associates of Stark County

Canton, Ohio, United States

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Intrepid Research

Cincinnati, Ohio, United States

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Cleveland Clinic - Main Campus

Cleveland, Ohio, United States

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Arthritis & Osteoarthritis Center of SW Ohio/ dba STAT Research

Vandalia, Ohio, United States

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Lynn Institute of Norman (LION Research)

Norman, Oklahoma, United States

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Willamette Valley Clinical Studies

Eugene, Oregon, United States

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AMS Cardiology (Elligo)

Horsham, Pennsylvania, United States

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University of Pennsylvania

Philadelphia, Pennsylvania, United States

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Preferred Primary Care Physicians

Pittsburgh, Pennsylvania, United States

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Accelerated Enrollment Solutions (AES) - Anderson

Anderson, South Carolina, United States

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Wake Research - Notus Clinical Trials, LLC

Charleston, South Carolina, United States

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Coastal Carolina Research Center

North Charleston, South Carolina, United States

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Chattanooga Medical Research

Chattanooga, Tennessee, United States

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AMR - Knoxville

Knoxville, Tennessee, United States

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Clinical Neuroscience Solutions, Inc

Memphis, Tennessee, United States

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Lifedoc Research

Memphis, Tennessee, United States

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Vanderbilt University Medical Center (VUMC)

Nashville, Tennessee, United States

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Punzi Medical Center

Carrollton, Texas, United States

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AES - Dallas Fort Worth

Dallas, Texas, United States

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David Turbay, MD, PLLC (Elligo Health Research)

El Paso, Texas, United States

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Synergy Groups Medical - Bissonet Site

Houston, Texas, United States

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Juno Research, LLC

Houston, Texas, United States

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Gulf Coast Clinical Research

Houston, Texas, United States

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Medical Colleagues of Texas, LLP (Elligo Health Research)

Katy, Texas, United States

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R & H Clinical Research

Katy, Texas, United States

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Gamma Medical Research, Inc

McAllen, Texas, United States

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Office of Audrey L. Jones, DO

McAllen, Texas, United States

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PRX Research - Mesquite

Mesquite, Texas, United States

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Synergy Groups Medical - Missouri City

Missouri City, Texas, United States

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ACRC Trials - Legacy Medical Village Location

Plano, Texas, United States

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Clinical Investigations of Texas (CIT)

Plano, Texas, United States

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ACRC Trials - Legacy Medical Village

Plano, Texas, United States

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Sun Research Institute (SRI) - San Antonio

San Antonio, Texas, United States

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San Antonio ClinicalTrials

San Antonio, Texas, United States

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Discovery Clinical Trials

San Antonio, Texas, United States

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Sugar Lakes Family Practice (Elligo Health Research)

Sugar Land, Texas, United States

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The University of Utah

Salt Lake City, Utah, United States

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Velocity Clinical Research

West Jordan, Utah, United States

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Burke Internal Medicine

Burke, Virginia, United States

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Eastern VA Medical School

Norfolk, Virginia, United States

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Office of Ramon Mendez

Woodbridge, Virginia, United States

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Renal Research - Gosford

Gosford, New South Wales, Australia

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Castle Hill Medical Centre

Castle Hill, , Australia

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The University of Western Australia - School of Medicine and Pharmacology - Royal Perth Hospital Unit.

Perth, , Australia

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University of Sunshine Coast Clinical Trial Centre

Sippy Downs, , Australia

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AusTrials - Taringa

Taringa, , Australia

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Medical Center New Polyclinic Gabrovo Ltd.

Gabrovo, , Bulgaria

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Medical Center

Pleven, , Bulgaria

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ASOMHIDC - Individual practice Cardio Tonus EOOD

Sofia, , Bulgaria

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DCC 1 - Veliko Tarnovo" EOOD

Veliko Tarnovo, , Bulgaria

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Centre Medical L'Acadie - Montreal

Montreal, Quebec, Canada

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Centre Hospitalier Annecy Genevois - Site d'Annecy

Annecy, , France

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Emovis GmbH

Berlin, , Germany

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MVZ Jung GbR

Deggingen, , Germany

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Klinische Forschung Dresden GmbH

Dresden, , Germany

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Uniklinik Leipzig, Klinik und Poliklinik für Kardiologie

Leipzig, , Germany

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Herzzentrum Leipzig

Leipzig, , Germany

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IRCCS AOU di Bologna - Policlinico S. Orsola

Bologna, , Italy

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IRCCS Ospedale Policlinico San Martino

Genova, , Italy

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University of Messina

Messina, , Italy

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Azienda Ospedaliero Universitaria Pisana

Pisa, , Italy

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University of Rome Sapienza, AO Sant'Andrea

Roma, , Italy

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Amsterdam AMC

Amsterdam, , Netherlands

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Samodzielny Publiczny Szpital Kliniczny im. Andrzeja Mielęckiego (SPSKM)

Katowice, , Poland

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Futuremeds Lodz

Lodz, , Poland

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Futuremeds Olsztyn

Olsztyn, , Poland

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Etyka Osrodek Badan Klinicznych

Olsztyn, , Poland

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Clinmedica Research

Skierniewice, , Poland

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ETG Warszawa

Warsaw, , Poland

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Latin Clinical Trial Center

San Juan, , Puerto Rico

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Centrul Medical Unirea SRL Brasov (Regina Maria)

Brasov, , Romania

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Delta Health Care SRL Bucuresti - Spitalul Academic Ponderas (Regina Maria)

Bucharest, , Romania

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Spitalul Clinic Judetean de Urgenta Targu Mures

Târgu Mureş, , Romania

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MEDICALI'S SRL Timisoara

Timișoara, , Romania

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Spitalul Clinic Judetean de Urgenta "Pius Branzeu" Timisoara

Timișoara, , Romania

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Complejo Hospitalario Universitario de Badajoz (CHUB) (Hospital Infanta Cristina)

Badajoz, , Spain

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Hospital Universitario Reina Sofia

Córdoba, , Spain

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Hospital Universitario Virgen de las Nieves

Granada, , Spain

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Hospital Clínico Universitario Valencia

Valencia, , Spain

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Newquay Health Centre

Newquay, Cornwall, United Kingdom

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Fowey River Practice

Fowey, England, United Kingdom

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Queen Elizabeth University Hospital

Glasgow, Scotland, United Kingdom

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Rowden Surgery Rowden Medical Partnership

Chippenham, wilts, United Kingdom

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Cambridge University Hospitals NHS Foundation Trust

Cambridge, , United Kingdom

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Epsom and St Helier University Hospitals NHS Trust

Carshalton, , United Kingdom

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Barts Health Nhs Trust

London, , United Kingdom

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Knowle House Surgery

Plymouth, , United Kingdom

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Rame Medical Limited

Torpoint, , United Kingdom

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Countries

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United States Australia Bulgaria Canada France Germany Italy Netherlands Poland Puerto Rico Romania Spain United Kingdom

Other Identifiers

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MLS-101-901

Identifier Type: -

Identifier Source: org_study_id

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