A Study Evaluating the Effects of GLPG3667 Given as Oral Treatment for up to 24 Weeks in Adults With Dermatomyositis

NCT ID: NCT05695950

Last Updated: 2025-12-23

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE2

Total Enrollment

40 participants

Study Classification

INTERVENTIONAL

Study Start Date

2023-02-27

Study Completion Date

2026-04-30

Brief Summary

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The purpose of this study is to evaluate the efficacy, safety, tolerability, pharmacokinetics (PK), and pharmacodynamics (PD) of orally administered GLPG3667 once daily for 24 weeks in adult participants with dermatomyositis (DM), followed by an open-label extension (OLE) period until Week 48.

Detailed Description

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Conditions

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Dermatomyositis

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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GLPG3667 During DB + During OLE

Participants will receive GLPG3667 dose A orally once daily for 24 weeks in the double-blind (DB) treatment period. Eligible participants will roll-over to an open-label extension (OLE) period to receive the same dose for another 24 weeks.

Group Type EXPERIMENTAL

GLPG3667

Intervention Type DRUG

GLPG3667 capsules will be administered per dose and schedule specified in the arm description.

Placebo During DB + GLPG3667 During OLE

Participants will receive placebo matching to GLPG3667 orally once daily for 24 weeks in the DB treatment period. Eligible participants will roll-over to an OLE period to receive GLPG3667 dose A orally once daily for another 24 weeks.

Group Type PLACEBO_COMPARATOR

GLPG3667

Intervention Type DRUG

GLPG3667 capsules will be administered per dose and schedule specified in the arm description.

Placebo

Intervention Type DRUG

Placebo matching to GLPG3667 capsules will be administered per schedule specified in the arm description.

Interventions

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GLPG3667

GLPG3667 capsules will be administered per dose and schedule specified in the arm description.

Intervention Type DRUG

Placebo

Placebo matching to GLPG3667 capsules will be administered per schedule specified in the arm description.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Participant has probable or definite DM in accordance with the ACR/EULAR criteria for at least 3 months.
* Participant with DM diagnosed in the 3 years prior to screening must have undergone cancer screening (according to local standard of care or applicable guidelines) within 1 year prior to screening. Note: The evidence of cancer screening must be documented.
* Participant must present objective evidence of active disease as defined by fulfilling 1 of the criteria below (as confirmed by the sponsor):

* DM rash as defined by modified-Cutaneous Dermatomyositis Disease Area and Severity Index Activity Score (m-CDASI-A) ≥ 6 at screening, or
* Creatine kinase (CK) \> 4x upper limit of normal (ULN) at screening, or
* muscle biopsy evidence of active disease within 3 months prior to screening (defined as presence of active inflammation in muscle biopsy), or
* muscle magnetic resonance imaging showing active inflammation (edema) of the proximal skeletal muscles within 3 months prior to screening, or
* electromyography showing acute changes, such as spontaneous activity and myopathic changes not explained by other diseases within 3 months prior to screening, or
* any other clinical evidence of active disease as confirmed by the steering committee.
* Participant has reduced muscle strength (defined as Manual Muscle Test-8 \< 142/150) and at least 2 additional abnormal core set measurements out of the following 5 at screening:

* Physician's Global Disease Activity score \> 2/10 cm on the visual analog scale (VAS),
* Patient's Global Disease Activity score \> 2/10 cm on VAS,
* extra-muscular disease activity \> 2/10 cm on VAS,
* Health Assessment Questionnaire-Disability Index score \> 0.25,
* elevated muscle enzymes (e.g. aldolase, CK, ALT, AST, and lactate dehydrogenase) with at least 1 muscle enzyme \> 1.5x ULN.
* Participant previously demonstrated failure to or intolerance to first-line treatment (defined as oral corticosteroid\[s\] and at least 1 other immunosuppressant/ hydroxychloroquine) OR active disease despite treatment with first-line drugs. Currently, the participant is receiving maximum 3 treatments for DM (oral corticosteroid\[s\] and/or allowed immunosuppressant\[s\]/hydroxychloroquine) for at least 3 months and is on a stable dose (defined as no change in dose, type of administration, or dose regimen) for at least 4 weeks prior to screening and during screening within maximum allowed doses as specified in the study protocol. Note: Participants receiving 1 or no concomitant treatment for DM are also eligible.

Exclusion Criteria

* Participant has cancer-associated myositis (defined as myositis diagnosed within 2 years of cancer diagnosis with the exception of basal cell carcinoma, squamous cell carcinoma of the skin, or in situ uterine cervical carcinoma that has been excised and cured). Note: At least 1 year for basal cell carcinoma and squamous cell carcinoma or 5 years for in situ uterine cervical carcinoma must have passed since the excision.
* Participant has other causes of myositis (e.g. connective tissue disease) associated DM, polymyositis, juvenile DM, inclusion body myositis, or necrotizing idiopathic inflammatory myopathies (with or without rash) with the exception of overlap with secondary Sjogren's syndrome.
* Participant has permanent muscle weakness due to muscle damage (e.g. participant is wheelchair bound or has significant muscle atrophy on magnetic resonance imaging \[MRI\]) or a non-DM cause (drug-induced myopathy, including glucocorticoid-induced myopathy as primary cause of muscle weakness), according to investigator's judgement.
* Participant has taken any prohibited therapies within the defined washout periods before screening, and during screening as listed in the study protocol.
* Open Label Extension : Participant meeting one or more of the criteria at Visit 8 as defined in the protocol, cannot be selected for the OLE period of this clinical study. 1. Participant has total bilirubin \>1.5x ULN; however, participant with an isolated increase in total bilirubin \<3 x ULN due to Gilbert's Syndrome, with normal direct bilirubin, can be enrolled in the OLE period. 2. Participant has AST or ALT \>1.5 x ULN (hepatic injury), or AST or ALT \>=5 x ULN if judged to be of muscular origin (and confirmed by the steering committee) at Visit 7 and Visit 8.
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Galapagos NV

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Galapagos Study Director

Role: STUDY_DIRECTOR

Galapagos NV

Locations

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HonorHealth Neurology

Scottsdale, Arizona, United States

Site Status

Inland Rheumatology Clinical Trials, Inc.

Upland, California, United States

Site Status

New Access Research and Medical Center

Kendall, Florida, United States

Site Status

Omega Research Orlando, LLC

Orlando, Florida, United States

Site Status

Augusta University

Augusta, Georgia, United States

Site Status

St. Paul Rheumatology

Eagan, Minnesota, United States

Site Status

Northwell Health, LLC PRIME

Lake Success, New York, United States

Site Status

Altoona Center for Clinical Research, P.C.

Duncansville, Pennsylvania, United States

Site Status

Fundacion Respirar Consultorios Médicos Dr. Doreski

Buenos Aires, , Argentina

Site Status

Hospital Cordoba

Córdoba, , Argentina

Site Status

Hospital Italiano de La Plata

La Plata, , Argentina

Site Status

Framingham Centro Medico

La Plata, , Argentina

Site Status

Instituto Medico CER

Quilmes, , Argentina

Site Status

UZ Leuven

Leuven, , Belgium

Site Status

Enroll SpA

Santiago, , Chile

Site Status

BioMedica Research Group Psicomedica Clinical and Research Group

Santiago, , Chile

Site Status

Clinica de la Costa S.A.S

Barranquilla, , Colombia

Site Status

Centro de Investigacion Medico Asistencial S.A.S

Barranquilla, , Colombia

Site Status

Healthy Medical Center

Zipaquirá, , Colombia

Site Status

Polyclinic Bonifarm

Zagreb, , Croatia

Site Status

Solmed Polyclinic

Zagreb, , Croatia

Site Status

Revmatologicky Ustav

Prague, , Czechia

Site Status

CHU de Nice Hôpital Pasteur 2 Centre de Réf des Maladies Neuromusculaires et SLA

Nice, , France

Site Status

Groupe Hospitalier Pitie-Salpetriere service de médecine interne et immunologie cliniqu

Paris, , France

Site Status

CHU Strasbourg - Hôpital Hautepierre service de rhumatologie

Strasbourg, , France

Site Status

Charité - Campus Charité Mitte - Klinik für Dermatologie, Venerologie und Allergologie

Berlin, , Germany

Site Status

Helios Fachklinik Vogelsang-Gommern

Gommern, , Germany

Site Status

Universitätsklinikum Tübingen - Universitäts-Hautklinik

Tübingen, , Germany

Site Status

Azienda Socio Sanitaria Territoriale degli Spedali Civili di Brescia (Presidio Spedali Civili) Medicina Interna

Brescia, , Italy

Site Status

Azienda Ospedaliero Universitaria Policlinico. PO San Marco

Catania, , Italy

Site Status

Ospedale San Raffaele U.O. di Medicina Gen. Ind. Immunologico-Clinica

Milan, , Italy

Site Status

Azienda Ospedaliero Universitaria Pisana U.O. Reumatologia Universitaria

Pisa, , Italy

Site Status

Fondazione Policlinico Universitario Agostino Gemelli IRCCS

Roma, , Italy

Site Status

Istituto Clinico Humanitas U.O. Reumatologia

Rozzano, , Italy

Site Status

Ospedale San Giovanni Bosco

Torino, , Italy

Site Status

Medical Care & Research SA de CV

Mérida, , Mexico

Site Status

Centro de Investigacion Clínica GRAMEL S.C

México, , Mexico

Site Status

Consultorio de Reumatologia Hospital Angeles Lindavista

México, , Mexico

Site Status

Centro de Alta Especialidad en Reumatología e Investigación del Potosí S.C.

San Luis Potosí City, , Mexico

Site Status

Nova Reuma Domysławska i Rusiłowicz, Spółka Partnerska Lekarza Reumatologa i Fizjoterapeuty

Bialystok, , Poland

Site Status

Centrum Medyczne Plejady

Krakow, , Poland

Site Status

Zespol Poradni Specjalistycznych Reumed

Lublin, , Poland

Site Status

Klinika Ambroziak ESTEDERM

Warsaw, , Poland

Site Status

Spitalul Clinic Colentina parent

Bucharest, , Romania

Site Status

Spitalul Clinic 'Sf. Maria' Clinica de Medicina Interna si Reumatologie

Bucharest, , Romania

Site Status

Sc Medaudio-Optica SRL

Râmnicu Vâlcea, , Romania

Site Status

Hospital Universitari Vall d'Hebron Internal Medicine Dept.

Barcelona, , Spain

Site Status

Hospital Clinic de Barcelona Servicio de Medicina Interna

Barcelona, , Spain

Site Status

Hospital Universitari de Bellvitge Servicio de Cardiologia

L'Hospitalet de Llobregat, , Spain

Site Status

Hospital Universitario Fundacion Jimenez Diaz

Madrid, , Spain

Site Status

St. Peter´s Hospital Dept of Rheumatology

Chertsey, , United Kingdom

Site Status

Western General Hospital Dept of Rheumatology

Edinburgh, , United Kingdom

Site Status

King's College Hospital Dept of Rheumatology

London, , United Kingdom

Site Status

Salford Care Organisation Dept of Rheumatology

Salford, , United Kingdom

Site Status

Countries

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Bulgaria United States Argentina Belgium Chile Colombia Croatia Czechia France Germany Italy Mexico Poland Romania Spain United Kingdom

References

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Mammoliti O, Martina S, Claes P, Coti G, Blanque R, Jagerschmidt C, Shoji K, Borgonovi M, De Vos S, Marsais F, Oste L, Quinton E, Lopez-Ramos M, Amantini D, Brys R, Jimenez JM, Galien R, van der Plas S. Discovery of GLPG3667, a Selective ATP Competitive Tyrosine Kinase 2 Inhibitor for the Treatment of Autoimmune Diseases. J Med Chem. 2024 Jun 13;67(11):8545-8568. doi: 10.1021/acs.jmedchem.4c00769. Epub 2024 May 28.

Reference Type DERIVED
PMID: 38805213 (View on PubMed)

Other Identifiers

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2022-501097-19-00

Identifier Type: CTIS

Identifier Source: secondary_id

GLPG3667-CL-214

Identifier Type: -

Identifier Source: org_study_id