Single-dose to Evaluate the Pharmacokinetics of GTX-101 and Subcutaneous Injectable Bupivacaine in Healthy Subjects

NCT ID: NCT05517486

Last Updated: 2023-01-23

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

UNKNOWN

Clinical Phase

PHASE1

Total Enrollment

48 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-07-26

Study Completion Date

2023-05-03

Brief Summary

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This is a single-center, randomized, single-dose, active-controlled study in healthy male and female subjects.

The study will enroll subjects to evaluate the PK of 3 dose strengths (50 mg, 100 mg and 200 mg) of GTX-101 compared to Subcutaneous injection in healthy adult subjects.

Blood samples for PK assessments will be collect at specified time points. Safety assessments will also be performed throughout the study.

Detailed Description

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Conditions

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Postherpetic Neuralgia

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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50 mg GTX-101

Group Type EXPERIMENTAL

GTX-101

Intervention Type DRUG

Bupivacaine HCl metered spray

100 mg GTX-101

Group Type EXPERIMENTAL

GTX-101

Intervention Type DRUG

Bupivacaine HCl metered spray

200 mg GTX-101

Group Type EXPERIMENTAL

GTX-101

Intervention Type DRUG

Bupivacaine HCl metered spray

Bupivacaine subcutaneous injection

Group Type ACTIVE_COMPARATOR

Bupivacaine HCl subcutaneous injection

Intervention Type DRUG

Bupivacaine HCl, 50 mg/10 mL

Interventions

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GTX-101

Bupivacaine HCl metered spray

Intervention Type DRUG

Bupivacaine HCl subcutaneous injection

Bupivacaine HCl, 50 mg/10 mL

Intervention Type DRUG

Other Intervention Names

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Bupivacaine HCl metered spray

Eligibility Criteria

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Inclusion Criteria

* Provision of signed and dated informed consent form (ICF)
* Healthy adult male or female, aged 18 to 55 years, inclusive, at Screening
* Body mass index (BMI) within 18.0 kg/m2 to 30.0 kg/m2, inclusively at Screening
* Have no clinically significant diseases captured in the medical/surgical history or evidence of clinically significant findings on the physical examination (including vital signs), weight and/or clinical laboratory tests and/or ECG, as determined by an Investigator

Exclusion Criteria

* History of significant hypersensitivity to bupivacaine, local anesthetic agents of amide type, or any related products (including excipients of the formulations) as well as severe hypersensitivity reactions (like angioedema) to any drugs
* Presence of significant gastrointestinal, liver or kidney disease, or any other conditions known to interfere with the absorption, distribution, metabolism or excretion of drugs or known to potentiate or predispose to undesired effects
* History of significant gastrointestinal, liver or kidney disease that may affect drug bioavailability
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Grace Therapeutics Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Eric Sicard, MD

Role: PRINCIPAL_INVESTIGATOR

Clinical Research Unit

Locations

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Clinical Research Unit

Montreal, , Canada

Site Status

Countries

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Canada

Other Identifiers

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GTX-101-004

Identifier Type: -

Identifier Source: org_study_id

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