A Study to Evaluate CIN-107 for the Treatment of Patients With Uncontrolled Hypertension and Chronic Kidney Disease

NCT ID: NCT05432167

Last Updated: 2025-05-20

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

View full results

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

195 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-04-29

Study Completion Date

2024-05-02

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

This study will evaluate the efficacy and safety of CIN-107 for the treatment of hypertension in patients with uncontrolled hypertension (uHTN) and Chronic Kidney Disease (CKD).

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

This randomized, double-blind, placebo-controlled will evaluate the efficacy and safety of CIN-107 in patients with uHTN and CKD. Approximately 200 patients will be randomized in a 1:1:1 ratio into 1 of the 3 treatment groups (placebo, low dose treatment strategy and high dose treatment strategy).

The study will consist of the following 3 periods:

* A Screening Period of up to 5 weeks;
* A Double-Blind Treatment Period of 26 weeks; and
* A Follow-Up Period of 2 weeks.

Patients will complete the study in approximately 8 months.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Uncontrolled Hypertension Chronic Kidney Diseases

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Low dose CIN-107

Patients will take oral tablets of CIN-107 for 26 weeks. The dose strength may be titrated within 6 weeks.

Group Type EXPERIMENTAL

CIN-107

Intervention Type DRUG

Patients will take CIN-107 tablets by mouth once daily.

High dose CIN-107

Patients will take oral tablets of CIN-107 for 26 weeks. The dose strength may be titrated within 6 weeks.

Group Type EXPERIMENTAL

CIN-107

Intervention Type DRUG

Patients will take CIN-107 tablets by mouth once daily.

Placebo

Patients will take oral tablets of Placebo for 26 weeks. The dose strength may be titrated within 6 weeks.

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Patients will take placebo tablets by mouth once daily.

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

CIN-107

Patients will take CIN-107 tablets by mouth once daily.

Intervention Type DRUG

Placebo

Patients will take placebo tablets by mouth once daily.

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Has a mean seated SBP ≥ 140 mmHg.
* Has a prior diagnosis of mild-to-severe CKD.
* Has an elevated UACR.
* Is currently taking an angiotensin-converting enzyme inhibitor (ACEi) or angiotensin receptor blocker (ARB) at the maximum tolerated daily dose.

Exclusion Criteria

* Have a documented diagnosis of type 1 diabetes.
* Are not willing or not able to discontinue a mineralocorticoid receptor antagonist (MRA) or a potassium sparing diuretic as part of an existing antihypertensive regimen.
* Have a single occurrence of mean seated SBP \>180 mmHg or DBP \>110 mmHg during the Screening Period.
* Has a body mass index (BMI) \>50 kg/m\^2.
* Has documented bilateral clinically relevant renal artery stenosis of ≥70%.
* Has had dialysis for acute kidney injury/acute renal failure within 12 weeks prior to the Screening Period or has a planned dialysis or kidney transplantation during the course of the study.
* Has known documented chronic heart failure New York Heart Association Class III or Class IV and/or hospitalization for heart failure within 6 months of Screening.
* Has had a stroke, transient ischemic attack, hypertensive encephalopathy, acute coronary syndrome, or hospitalization for heart failure within 6 months of Screening.
* Has known current severe left ventricular outflow obstruction, such as obstructive hypertrophic cardiomyopathy and/or severe aortic valvular disease.
* Has planned any major cardiac surgery during the study or had major cardiac surgery within 6 months of Screening.
* Has had a prior solid organ transplant or cell transplant.
* Has a known hypersensitivity to CIN-107 or drugs of the same class
* Has received immunotherapy for treatment of CKD within 6 months of Screening.
* Has any clinically relevant medical or surgical conditions including unstable conditions and/or conditions requiring regular transfusion or treatment with systemic immunosuppressants, including corticosteroids.
* Serum potassium \<3.5 mEq/L or \>5.0 mEq/L
* Serum sodium \<135 mEq/L
* Serum aspartate aminotransferase or alanine aminotransferase \>3 × upper limit of normal (ULN); or Total bilirubin \>2 × ULN, unless due to Gilbert's syndrome.
* GFR is \< 25 or \> 75 mL/min/1.73 m2
* Has uncontrolled diabetes with glycosylated hemoglobin \>10.5%.
* Is positive for Human immunodeficiency disease (HIV) antibody, hepatitis B surface antigen, or hepatitis C virus Ribonucleic acid (RNA).
* Has typical consumption of \>14 alcoholic drinks weekly.
Minimum Eligible Age

18 Years

Maximum Eligible Age

130 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Parexel

INDUSTRY

Sponsor Role collaborator

AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Research Site

Birmingham, Alabama, United States

Site Status

Research Site

Huntsville, Alabama, United States

Site Status

Research Site

Beverly Hills, California, United States

Site Status

Research Site

Chula Vista, California, United States

Site Status

Research Site

Fountain Valley, California, United States

Site Status

Research Site

Granada Hills, California, United States

Site Status

Research Site

Lancaster, California, United States

Site Status

Research Site

Lincoln, California, United States

Site Status

Research Site

Los Angeles, California, United States

Site Status

Research Site

Lynwood, California, United States

Site Status

Research Site

Northridge, California, United States

Site Status

Research Site

Panorama City, California, United States

Site Status

Research Site

Pomona, California, United States

Site Status

Research Site

Rancho Cucamonga, California, United States

Site Status

Research Site

Riverside, California, United States

Site Status

Research Site

San Dimas, California, United States

Site Status

Research Site

South Gate, California, United States

Site Status

Research Site

Tarzana, California, United States

Site Status

Research Site

Vacaville, California, United States

Site Status

Research Site

Victorville, California, United States

Site Status

Research Site

Arvada, Colorado, United States

Site Status

Research Site

Littleton, Colorado, United States

Site Status

Research Site

Hollywood, Florida, United States

Site Status

Research Site

Orlando, Florida, United States

Site Status

Research Site

Orlando, Florida, United States

Site Status

Research Site

Tampa, Florida, United States

Site Status

Research Site

West Palm Beach, Florida, United States

Site Status

Research Site

Columbus, Georgia, United States

Site Status

Research Site

Decatur, Georgia, United States

Site Status

Research Site

Nampa, Idaho, United States

Site Status

Research Site

Chicago, Illinois, United States

Site Status

Research Site

Brownsburg, Indiana, United States

Site Status

Research Site

Lexington, Kentucky, United States

Site Status

Research Site

Metairie, Louisiana, United States

Site Status

Research Site

Monroe, Louisiana, United States

Site Status

Research Site

Silver Spring, Maryland, United States

Site Status

Research Site

New Bedford, Massachusetts, United States

Site Status

Research Site

Flint, Michigan, United States

Site Status

Research Site

Flint, Michigan, United States

Site Status

Research Site

Troy, Michigan, United States

Site Status

Research Site

Olive Branch, Mississippi, United States

Site Status

Research Site

Kansas City, Missouri, United States

Site Status

Research Site

Trenton, New Jersey, United States

Site Status

Research Site

The Bronx, New York, United States

Site Status

Research Site

Durham, North Carolina, United States

Site Status

Research Site

Greenville, North Carolina, United States

Site Status

Research Site

Kinston, North Carolina, United States

Site Status

Research Site

Morganton, North Carolina, United States

Site Status

Research Site

Oxford, North Carolina, United States

Site Status

Research Site

Wilmington, North Carolina, United States

Site Status

Research Site

Cincinnati, Ohio, United States

Site Status

Research Site

Bethany, Oklahoma, United States

Site Status

Research Site

Scottdale, Pennsylvania, United States

Site Status

Research Site

Smithfield, Pennsylvania, United States

Site Status

Research Site

Providence, Rhode Island, United States

Site Status

Research Site

Memphis, Tennessee, United States

Site Status

Research Site

Houston, Texas, United States

Site Status

Research Site

Lampasas, Texas, United States

Site Status

Research Site

Paris, Texas, United States

Site Status

Research Site

Red Oak, Texas, United States

Site Status

Research Site

San Antonio, Texas, United States

Site Status

Research Site

San Antonio, Texas, United States

Site Status

Research Site

Salt Lake City, Utah, United States

Site Status

Research Site

Burlington, Vermont, United States

Site Status

Research Site

Alexandria, Virginia, United States

Site Status

Research Site

Burke, Virginia, United States

Site Status

Research Site

Charlottesville, Virginia, United States

Site Status

Research Site

Manassas, Virginia, United States

Site Status

Research Site

Newport News, Virginia, United States

Site Status

Research Site

Salem, Virginia, United States

Site Status

Research Site

Kingwood, West Virginia, United States

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States

References

Explore related publications, articles, or registry entries linked to this study.

Dwyer JP, Maklad N, Vedin O, Monyak J, Myte R, Chertow GM, Heerspink HJL, Little DJ. Efficacy and Safety of Baxdrostat in Participants with CKD and Uncontrolled Hypertension: A Randomized, Double-Blind, Placebo-Controlled Trial. J Am Soc Nephrol. 2025 Sep 6. doi: 10.1681/ASN.0000000849. Online ahead of print. No abstract available.

Reference Type DERIVED
PMID: 40913594 (View on PubMed)

Townsend RR. Blocking Aldosterone Synthesis: Whose BrigHTN Idea Was That? Clin J Am Soc Nephrol. 2023 Dec 1;18(12):1631-1633. doi: 10.2215/CJN.0000000000000265. Epub 2023 Jul 24. No abstract available.

Reference Type DERIVED
PMID: 37490693 (View on PubMed)

Provided Documents

Download supplemental materials such as informed consent forms, study protocols, or participant manuals.

Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

D6972C00001

Identifier Type: OTHER

Identifier Source: secondary_id

CIN-107-123

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.