A Study of LOXO-783 in Patients With Breast Cancer/Other Solid Tumors

NCT ID: NCT05307705

Last Updated: 2026-01-21

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE1

Total Enrollment

193 participants

Study Classification

INTERVENTIONAL

Study Start Date

2022-05-11

Study Completion Date

2026-12-31

Brief Summary

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The main purpose of this study is to learn more about the safety, side effects, and effectiveness of LOXO-783. LOXO-783 may be used to treat breast cancer and other solid tumors that have a change in a particular gene (known as the PIK3CA gene). Participation could last up to 36 months (3 years) and possibly longer if the disease does not get worse.

Detailed Description

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Conditions

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Breast Cancer

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Phase 1A: LOXO-783 Monotherapy Dose Escalation

LOXO-783 administered orally

Group Type EXPERIMENTAL

LOXO-783

Intervention Type DRUG

Oral

Phase 1B: Part A

LOXO-783 administered orally in combination with fulvestrant intramuscularly, imlunestrant orally, or an aromatase inhibitor orally

Group Type EXPERIMENTAL

LOXO-783

Intervention Type DRUG

Oral

Fulvestrant

Intervention Type DRUG

Intramuscular

Imlunestrant

Intervention Type DRUG

Oral

Anastrozole, Exemestane, or Letrozole

Intervention Type DRUG

Oral

Phase 1B: Part B

LOXO-783 orally in combination with abemaciclib and either physician's choice aromatase inhibitor orally, fulvestrant intramuscularly, or imlunestrant orally

Group Type EXPERIMENTAL

LOXO-783

Intervention Type DRUG

Oral

Fulvestrant

Intervention Type DRUG

Intramuscular

Imlunestrant

Intervention Type DRUG

Oral

Abemaciclib

Intervention Type DRUG

Oral

Anastrozole, Exemestane, or Letrozole

Intervention Type DRUG

Oral

Phase 1B: Part C

LOXO-783 orally in combination with fulvestrant intramuscularly

Group Type EXPERIMENTAL

LOXO-783

Intervention Type DRUG

Oral

Fulvestrant

Intervention Type DRUG

Intramuscular

Phase 1B: Part D

LOXO-783 orally in combination with paclitaxel intravenously

Group Type EXPERIMENTAL

LOXO-783

Intervention Type DRUG

Oral

Paclitaxel

Intervention Type DRUG

Intravenous

Phase 1B: Part E

LOXO-783 orally

Group Type EXPERIMENTAL

LOXO-783

Intervention Type DRUG

Oral

Phase 1B: Part F

Multiple randomized dose levels of LOXO-783 orally with fulvestrant intramuscularly

Group Type EXPERIMENTAL

LOXO-783

Intervention Type DRUG

Oral

Fulvestrant

Intervention Type DRUG

Intramuscular

Interventions

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LOXO-783

Oral

Intervention Type DRUG

Fulvestrant

Intramuscular

Intervention Type DRUG

Imlunestrant

Oral

Intervention Type DRUG

Abemaciclib

Oral

Intervention Type DRUG

Anastrozole, Exemestane, or Letrozole

Oral

Intervention Type DRUG

Paclitaxel

Intravenous

Intervention Type DRUG

Other Intervention Names

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LY3849524 LY3484356 LY2835219

Eligibility Criteria

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Inclusion Criteria

* Have advanced breast cancer or another solid tumor with the presence of a phosphatidylinositol 3-kinase catalytic subunit alpha (PIK3CA) H1047R mutation (or other Sponsor and safety review committee (SRC)-approved, activating PIK3CA mutations other than H1047R mutation)
* Have adequate archival tumor tissue sample available or be approved by the Sponsor for enrollment if no tumor sample is available.
* Have stopped all cancer treatment and have recovered from the major side effects
* Have adequate organ function, as measured by blood tests
* Have a performance status of 0 or 1 on the Eastern Cooperative Oncology Group (ECOG) scale
* Patients must have

* Measurable disease

\--- Patients with non-breast tumor types must have at least 1 measurable lesion
* Non-measurable bone disease (at least 1 bone lesion in breast cancer patients only)
* For patients with an estrogen receptor (ER)+ breast cancer diagnosis:

* If female, must be postmenopausal
* If male, must agree to use hormone suppression
* Phase 1a:

\-- Dose escalation and backfill patients:
* Advanced solid tumor
* Patients may have had up to 5 prior regimens for advanced disease
* Phase 1b:

* Part A:

* ER+/human epidermal growth factor receptor 2 (HER2)- advanced breast cancer
* Patients may have had up to 5 prior regimens for advanced disease ---- Prior cyclin dependent kinase (CDK)4/6 inhibitor therapy required
* Part B:

* ER+/HER2- advanced breast cancer
* Patients may have had up to 2 prior regimens for advanced disease.
* Part C:

* ER+/HER2- advanced breast cancer
* Patients may have had up to 5 prior regimens for advanced disease.

\---- Prior CDK4/6 inhibitor therapy required.
* Have a diagnosis of diabetes mellitus Type 2
* Part D:

* Advanced breast cancer
* Patients may have had up to 5 prior regimens for advanced disease.
* Part E:

* Advanced solid tumor
* Patients may have had up to 3 prior regimens for advanced disease advanced disease
* Part F:

* ER+/HER2- advanced breast cancer
* Patients may have had up to 5 prior regimens for advanced disease

* Prior cyclin dependent kinase (CDK)4/6 inhibitor therapy required

Exclusion Criteria

* Medical Conditions

* Colorectal cancer
* Endometrial cancers with specific concurrent oncogenic alterations
* A history of known active or suspected

* Diabetes mellitus Type 1 or
* Diabetes mellitus Type 2 requiring antidiabetic medication (Phase 1a and all parts of Phase 1b except Part C).
* Serious concomitant systemic disorder
* Known or suspected history of untreated or uncontrolled central nervous system (CNS) involvement.
* Active uncontrolled systemic bacterial, viral, fungal, or parasitic infection, or other clinically significant active disease process
* Prior exposure to phosphatidylinositol 3-kinase/protein kinase B/mammalian target of rapamycin (PI3K/AKT/mTOR) inhibitor(s), except in certain circumstances
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Eli Lilly and Company

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Call 1-877-CTLILLY (1-877-285-4559) or 1-317-615-4559 Mon - Fri 9 AM - 5 PM Eastern time (UTC/GMT - 5 hours, EST)

Role: STUDY_DIRECTOR

Eli Lilly and Company

Locations

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Mayo Clinic of Scottsdale

Scottsdale, Arizona, United States

Site Status

UCLA Medical Center

Los Angeles, California, United States

Site Status

UCSF Medical Center at Mission Bay

San Francisco, California, United States

Site Status

Stanford University Hospital

Stanford, California, United States

Site Status

Mayo Clinic

Jacksonville, Florida, United States

Site Status

Winship Cancer Center Emory University

Atlanta, Georgia, United States

Site Status

Massachusetts General Hospital

Boston, Massachusetts, United States

Site Status

Dana-Farber Cancer Institute

Boston, Massachusetts, United States

Site Status

Mayo Clinic

Rochester, Minnesota, United States

Site Status

Washington University Medical School

St Louis, Missouri, United States

Site Status

Memorial Sloan Kettering Cancer Center

New York, New York, United States

Site Status

Wilmot Cancer Institute

Rochester, New York, United States

Site Status

Tennessee Oncology PLLC

Nashville, Tennessee, United States

Site Status

Texas Oncology-Baylor Charles A. Sammons Cancer Center

Dallas, Texas, United States

Site Status

UT Southwestern Medical Center

Dallas, Texas, United States

Site Status

University of Texas MD Anderson Cancer Center

Houston, Texas, United States

Site Status

South Texas Accelerated Research Therapeutics (START)

San Antonio, Texas, United States

Site Status

Cancer Research SA

Adelaide, , Australia

Site Status

Peter Maccallum Cancer Institute Erb

East Melbourne, , Australia

Site Status

St Vincent's Hospital

Sydney, , Australia

Site Status

Institut Jules Bordet

Anderlecht, , Belgium

Site Status

Universitaire Ziekenhuizen Leuven - Campus Gasthuisberg

Leuven, , Belgium

Site Status

Princess Margaret Hospital (Hong Kong)

Toronto, , Canada

Site Status

BC Cancer Vancouver

Vancouver, , Canada

Site Status

Beijing Cancer hospital

Beijing, , China

Site Status

The Third Hospital of Nanchang

Nanchang, , China

Site Status

Fudan University Shanghai Cancer Center

Shanghai, , China

Site Status

Centre Leon Berard

Lyon, , France

Site Status

Institut Curie

Paris, , France

Site Status

Institut de Cancérologie de l'Ouest

Saint-Herblain, , France

Site Status

ICANS_Institut de Cancerologie Strasbourg Europe

Strasbourg, , France

Site Status

Gustave Roussy

Villejuif, , France

Site Status

Universitätsklinikum Erlangen

Erlangen, , Germany

Site Status

National Cancer Center Hospital

Chūōku, , Japan

Site Status

The Cancer Institute Hospital of JFCR

Kōtō City, , Japan

Site Status

Kyoto University Hospital

Kyoto, , Japan

Site Status

Aichi Cancer Center Hospital

Nagoya, , Japan

Site Status

National Cancer Centre Singapore

Singapore, , Singapore

Site Status

Samsung Medical Center

Seoul, , South Korea

Site Status

Asan Medical Center

Seoul, , South Korea

Site Status

Hospital Universitario Quiron Dexeus

Barcelona, , Spain

Site Status

Hospital Universitari Vall d'Hebron

Barcelona, , Spain

Site Status

Hospital Clinic de Barcelona

Barcelona, , Spain

Site Status

Hospital General Universitario Gregorio Maranon

Madrid, , Spain

Site Status

Hospital Universitario 12 de Octubre

Madrid, , Spain

Site Status

Hospital Quironsalud Madrid

Pozuelo de Alarcón, , Spain

Site Status

Hospital Clinico Universitario de Valencia

Valencia, , Spain

Site Status

Hospital Arnau de Vilanova Valencia

Valencia, , Spain

Site Status

Royal Marsden NHS Trust

London, , United Kingdom

Site Status

Royal Marsden Hospital (Sutton)

Sutton, , United Kingdom

Site Status

Countries

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United States Australia Belgium Canada China France Germany Japan Singapore South Korea Spain United Kingdom

Related Links

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https://trials.lilly.com/en-US/trial/338185

A Study of LOXO-783 in Patients With Breast Cancer/Other Solid Tumors

Other Identifiers

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2022-000175-40

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

J4C-OX-JZUA

Identifier Type: OTHER

Identifier Source: secondary_id

LOXO-PIK-21001

Identifier Type: OTHER

Identifier Source: secondary_id

18394

Identifier Type: -

Identifier Source: org_study_id

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