TL-895 and KRT-232 Study in Acute Myeloid Leukemia

NCT ID: NCT04669067

Last Updated: 2023-02-17

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE1/PHASE2

Total Enrollment

18 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-03-31

Study Completion Date

2025-11-30

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

This study evaluates TL-895, a potent, orally available and highly selective irreversible tyrosine kinase inhibitor combined with navtemadlin (KRT-232), a novel oral small molecule inhibitor of MDM2 for the treatment of adults with FLT3 mutated Acute Myeloid Leukemia. Participants must be relapsed/refractory (e.g., having failed prior therapy) to be eligible for this study.

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Acute Myeloid Leukemia

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

NON_RANDOMIZED

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

Phase 1b - Dose Level 1

KRT-232 240mg QD, orally administered on days 1 through 7 of each 28-day cycle in combination with TL-895 150mg BID continuously for each 28-day cycle.

Group Type EXPERIMENTAL

TL-895

Intervention Type DRUG

TL-895 is an experimental tyrosine kinase inhibitor anticancer drug taken by mouth.

KRT-232

Intervention Type DRUG

KRT-232 is an experimental MDM2 inhibitor anticancer drug taken by mouth.

Phase 1b - Dose Level 2

KRT-232 300mg QD, orally administered on days 1 through 7 of each 28-day cycle in combination with TL-895 150mg BID continuously for each 28-day cycle.

Group Type EXPERIMENTAL

TL-895

Intervention Type DRUG

TL-895 is an experimental tyrosine kinase inhibitor anticancer drug taken by mouth.

KRT-232

Intervention Type DRUG

KRT-232 is an experimental MDM2 inhibitor anticancer drug taken by mouth.

Phase 1b - Dose Level 3

Cycle 1 only: KRT-232 360 mg QD orally administered on Days 1 through 7 of the first 28-day cycle in combination with TL-895 150 mg BID continuously for the first 28-day cycle

Cycle 2 and beyond: KRT-232 300 mg QD orally administered on Days 1 through 7 of each 28-day cycle in combination with TL-895 150 mg BID continuously for each 28-day cycle.

Group Type EXPERIMENTAL

TL-895

Intervention Type DRUG

TL-895 is an experimental tyrosine kinase inhibitor anticancer drug taken by mouth.

KRT-232

Intervention Type DRUG

KRT-232 is an experimental MDM2 inhibitor anticancer drug taken by mouth.

Phase 1b - Dose Level 4

Cycle 1 only: KRT-232 360 mg QD orally administered on Days 1 through 7 of the first 28-day cycle in combination with TL-895 300 mg BID continuously for the first 28-day cycle.

Cycle 2 and beyond: KRT-232 300 mg QD orally administered on Days 1 through 7 of each 28-day cycle in combination with TL-895 300 mg BID continuously for each 28-day cycle.

Group Type EXPERIMENTAL

TL-895

Intervention Type DRUG

TL-895 is an experimental tyrosine kinase inhibitor anticancer drug taken by mouth.

KRT-232

Intervention Type DRUG

KRT-232 is an experimental MDM2 inhibitor anticancer drug taken by mouth.

Phase 1b - Dose Level 5

Cycle 1 only: KRT-232 360 mg QD orally administered on Days 1 through 7 of the first 28-day cycle in combination with TL-895 450 mg BID continuously for the first 28-day cycle.

Cycle 2 and beyond: KRT-232 300 mg QD orally administered on Days 1 through 7 of each 28-day cycle in combination with TL-895 450 mg BID continuously for each 28-day cycle.

Group Type EXPERIMENTAL

TL-895

Intervention Type DRUG

TL-895 is an experimental tyrosine kinase inhibitor anticancer drug taken by mouth.

KRT-232

Intervention Type DRUG

KRT-232 is an experimental MDM2 inhibitor anticancer drug taken by mouth.

Phase 2 - Dose Expansion

Dose expansion of the recommended phase 2 dose of TL-895 in combination with KRT-232 as determined in Phase 1b.

Group Type EXPERIMENTAL

TL-895

Intervention Type DRUG

TL-895 is an experimental tyrosine kinase inhibitor anticancer drug taken by mouth.

KRT-232

Intervention Type DRUG

KRT-232 is an experimental MDM2 inhibitor anticancer drug taken by mouth.

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

TL-895

TL-895 is an experimental tyrosine kinase inhibitor anticancer drug taken by mouth.

Intervention Type DRUG

KRT-232

KRT-232 is an experimental MDM2 inhibitor anticancer drug taken by mouth.

Intervention Type DRUG

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* TP53 wildtype AML
* Relapsed/Refractory to at least one prior therapy, one of which must have included a FLT-3 inhibitor
* FLT3 mutation (FLT3-TKD or FLT3-ITD)
* ECOG 0-2
* Adequate hematologic, hepatic, and renal functions

Exclusion Criteria

* AML subtype 3
* Prior treatment with MDM2 antagonist therapies
* Eligible for HSCT
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Kartos Therapeutics, Inc.

INDUSTRY

Sponsor Role collaborator

Telios Pharma, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Keck School of Medicine

Los Angeles, California, United States

Site Status

University of California, Irvine Medical Center

Orange, California, United States

Site Status

Georgia Cancer Center

Augusta, Georgia, United States

Site Status

Northwestern Memorial Hospital

Chicago, Illinois, United States

Site Status

Rush University Medical Center, Division of Hematology Oncology and Cell Therapy

Chicago, Illinois, United States

Site Status

Karmanos Cancer Institute

Detroit, Michigan, United States

Site Status

Weill Cornell Medical College

New York, New York, United States

Site Status

University of Cincinnati

Cincinnati, Ohio, United States

Site Status

Thomas Jefferson University, Sidney Kimmel Cancer Center, Clinical Research Organization

Philadelphia, Pennsylvania, United States

Site Status

UT Southwestern Medical Center, Harold C. Simmons Cancer Center

Dallas, Texas, United States

Site Status

Seattle Cancer Care Alliance

Seattle, Washington, United States

Site Status

University of Sunshine Coast-Sippy Downs

Sippy Downs, , Australia

Site Status

Westmead Hospital

Sydney, , Australia

Site Status

Ordensklinikum Linz GmbH Elisabethinen

Linz, , Austria

Site Status

Medical University Vienna, Department of Internal Medicine I, Clinical Department of Hematology and Hemostaseology

Vienna, , Austria

Site Status

Claude Huriez Hospital

Lille, , France

Site Status

South Lyon Hospital Center

Lyon, , France

Site Status

Paoli-Calmettes Institute

Marseille, , France

Site Status

University Hospital of Nantes

Nantes, , France

Site Status

Hospital Center Universitaire De Nice

Nice, , France

Site Status

Saint-Louis Hospital

Paris, , France

Site Status

University Hospital Halle (Saale), Department of Internal Medicine IV - Hematology and Oncology

Halle, Saxony-Anhalt, Germany

Site Status

University Duisburg-Essen, University Hospital Essen, Department of Internal Medicine

Essen, , Germany

Site Status

University Hospital Hamburg-Eppendorf, Department of Internal Medicine II

Hamburg, , Germany

Site Status

Hannover Medical School, Center for Internal Medicine, Clinic of Hematology, Hemostaseology, Oncology and Stem Cell Transplantation

Hanover, , Germany

Site Status

University Hospital Jena, Clinic of Internal Medicine II, Department of Hematology and Medical Oncology

Jena, , Germany

Site Status

University Hospital - Ospedali Riuniti Umberto I - GM Lancisi - G Salesi of Ancona, Haematology Clinic

Ancona, , Italy

Site Status

Polyclinic S. Orsola-Malpighi, Operative Unit of Hematology

Bologna, , Italy

Site Status

Romagnolo Scientific Institute of Meldola (IRST) S.r.l., Department of Oncology and Clinical and Experimental Haematology

Meldola, , Italy

Site Status

Gachon University Gil Medical Center

Incheon, , South Korea

Site Status

Seoul National University Hospital, Department of Hemato-Oncology

Seoul, , South Korea

Site Status

University Hospital Germans Trias i Pujol, Department of Clinical Hematology

Badalona, , Spain

Site Status

University Hospital Vall d'Hebron

Barcelona, , Spain

Site Status

University Clinical Hospital of Valencia, Department of Hematology and Medical Oncology

Valencia, , Spain

Site Status

Hospital Universitario y Politécnico de La Fe

Valencia, , Spain

Site Status

Countries

Review the countries where the study has at least one active or historical site.

United States Australia Austria France Germany Italy South Korea Spain

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

TL-895-203

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.