First-In-Human Study To Evaluate Safety, Tolerability, And Pharmacokinetics Following Single Ascending And Multiple Ascending Doses of PF-07304814 In Hospitalized Participants With COVID-19.

NCT ID: NCT04535167

Last Updated: 2023-05-03

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

26 participants

Study Classification

INTERVENTIONAL

Study Start Date

2020-09-09

Study Completion Date

2021-06-07

Brief Summary

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It is Phase 1b, 2-part, double-blind, placebo-controlled study to evaluate safety, tolerability, and pharmacokinetics of PF-07304814, in patients hospitalized with SARS-CoV-2 virus infection.

Detailed Description

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It is a 2-part study in hospitalized COVID-19 patients.

* Part 1 is to evaluate safety, tolerability, PK and markers of clinical activity of escalating doses of PF-07304814 given as 24-hour IV infusion.

2 planned and 3 optional cohorts with 8 participants each are planned.
* Part 2 is to evaluate safety, tolerability, PK and markers of clinical activity of escalating doses of PF- 07304814 given as 120-hour infusion.

2 planned and 2 optional cohorts with 8 participants each are planned

Conditions

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Viral Disease

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

FACTORIAL

Part 1 will have 2 planned cohorts. Each escalating cohort will be initiated for enrollment after assessment of safety, tolerability and PK data from previous cohorts by an independent IRC and is deemed acceptable.

Part 2 will have 2 planned cohort and each escalating cohort will be initiated after all safety, tolerability and PK data from previous cohort is evaluated and is deemed acceptable by a competent regulatory authority.
Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Caregivers Investigators

Study Groups

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PF-07304814

Part 1:

Cohort 1-5

Part 2:

Cohort 6-9

Group Type EXPERIMENTAL

PF-07304814

Intervention Type DRUG

PF-07304814 is an anti-viral, formulated for intravenous delivery

Placebo

Part 1:

Cohort 1-5

Part 2:

Cohort 6-9

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Placebo will be formulated for intravenous delivery

Interventions

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PF-07304814

PF-07304814 is an anti-viral, formulated for intravenous delivery

Intervention Type DRUG

Placebo

Placebo will be formulated for intravenous delivery

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Male or female participants between the ages of 18 and 79 years.
2. Confirmed SARS-CoV-2 infection.
3. Hospitalized for COVID-19.
4. Symptoms consistent with COVID-19 indicated by at least 1 of the following: fever, cough, sore throat, malaise, headache, muscle pain, shortness of breath, new loss of taste and smell, nausea, chills, fatigue, rhinorrhea, diarrhea, vomiting or radiographic infiltrates by imaging consistent with COVID-19
5. Total body weight \>=50 kg (110 lb), BMI \<40 kg/m2; BMI \<35 kg/m2 for 76- 79 years.

Exclusion Criteria

1. Evidence of critical illness, defined by at least one of the following: Respiratory failure, Multi-organ dysfunction/failure, Cardiac failure or septic shock
2. Participants that are anticipated by the study Investigator to progress to critical disease, including mechanical ventilation, within 24 hours of enrolment
3. Participants with pre-existing moderate to severe cardiovascular disease, uncontrolled diabetes, or severe asthma or severe COPD.

3.Participants with a known medical history of recent acute or chronic liver disease (other than NASH), chronic or active hepatitis B or C infection, or primary biliary cirrhosis.

4.Participants with a known medical history of ischemic heart disease, heart failure, dysrhythmia or other pre-existing cardiac condition.

5\. Participants with known HIV infection, acute or chronic history of hepatitis B or C.

6.Participants with a known medical history of recurrent seizures. 7. Participants with history of venous thromboembolic event, including deep venous thrombosis or pulmonary embolism 8.Confirmed concurrent active systemic infection other than COVID-19. 9.Current diagnosis of cancer, unless in remission and untreated. 10.Other medical or psychiatric condition including recent or active suicidal ideation/behavior or laboratory abnormality that may increase the risk of study participation 11.Females who are pregnant or breastfeeding.
Minimum Eligible Age

18 Years

Maximum Eligible Age

79 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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El Camino Health

Mountain View, California, United States

Site Status

Palo Alto Medical Foundation

Mountain View, California, United States

Site Status

Hoag Memorial Hospital Presbyterian

Newport Beach, California, United States

Site Status

UC Davis Health Investigational Drug Pharmacy

Sacramento, California, United States

Site Status

UC Davis Medical Center

Sacramento, California, United States

Site Status

Massachusetts General Hospital Translational and Clinical Research Center

Boston, Massachusetts, United States

Site Status

Massachusetts General Hospital, Clinical Trials Pharmacy

Boston, Massachusetts, United States

Site Status

Massachusetts General Hospital

Boston, Massachusetts, United States

Site Status

Regional One Health

Memphis, Tennessee, United States

Site Status

University Hospital Brugmann

Brussels, , Belgium

Site Status

Santa Casa De Misericórdia de Belo Horizonte

Belo Horizonte, Minas Gerais, Brazil

Site Status

Hospital Universitario Fundacion Jimenez Diaz

Madrid, , Spain

Site Status

Hospital Universitario Virgen Del Rocio

Seville, , Spain

Site Status

Countries

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United States Belgium Brazil Spain

References

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Robinson P, Toussi SS, Aggarwal S, Bergman A, Zhu T, Hackman F, Sathish JG, Updyke L, Loudon P, Krishna G, Clevenbergh P, Hernandez-Mora MG, Cisneros Herreros JM, Albertson TE, Dougan M, Thacker A, Baniecki ML, Soares H, Whitlock M, Nucci G, Menon S, Anderson AS, Binks M. Safety, Tolerability, and Pharmacokinetics of Single and Multiple Ascending Intravenous Infusions of PF-07304814 (Lufotrelvir) in Participants Hospitalized With COVID-19. Open Forum Infect Dis. 2023 Jul 10;10(8):ofad355. doi: 10.1093/ofid/ofad355. eCollection 2023 Aug.

Reference Type DERIVED
PMID: 37559753 (View on PubMed)

Crosas-Molist E, Samain R, Kohlhammer L, Orgaz JL, George SL, Maiques O, Barcelo J, Sanz-Moreno V. Rho GTPase signaling in cancer progression and dissemination. Physiol Rev. 2022 Jan 1;102(1):455-510. doi: 10.1152/physrev.00045.2020. Epub 2021 Sep 20.

Reference Type DERIVED
PMID: 34541899 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Related Links

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https://pmiform.com/clinical-trial-info-request?StudyID=C4611001

To obtain contact information for a study center near you, click here.

Other Identifiers

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2020-003905-73

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

C4611001

Identifier Type: -

Identifier Source: org_study_id

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