A Study of ABI-H2158-containing Regimens in Participants With Chronic Hepatitis B Virus Infection

NCT ID: NCT04398134

Last Updated: 2022-09-15

Study Results

Results available

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Basic Information

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Recruitment Status

TERMINATED

Clinical Phase

PHASE2

Total Enrollment

88 participants

Study Classification

INTERVENTIONAL

Study Start Date

2020-08-28

Study Completion Date

2021-12-28

Brief Summary

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This Phase 2a study will assess the safety, antiviral activity, and pharmacokinetics (PK) of ABI-H2158 administered once daily for up to 72 weeks in combination with entecavir (ETV) in participants with chronic hepatitis B virus (HBV) infection.

Detailed Description

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Conditions

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Chronic Hepatitis B

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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ABI-H2158 plus ETV

ABI-2158 300 mg tablet once daily for 72 weeks plus ETV 0.5 mg tablet once daily for 96 weeks

Group Type EXPERIMENTAL

ABI-H2158

Intervention Type DRUG

3 X 100 mg tablets for oral administration

Entecavir (ETV)

Intervention Type DRUG

0.5 mg tablet for oral administration

Placebo plus ETV

Placebo matching ABI-2158 300 mg tablet once daily for 72 weeks plus ETV 0.5 mg tablet once daily for 96 weeks

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Sugar pill manufactured to mimic the ABI-H2158 tablets

Entecavir (ETV)

Intervention Type DRUG

0.5 mg tablet for oral administration

Interventions

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ABI-H2158

3 X 100 mg tablets for oral administration

Intervention Type DRUG

Placebo

Sugar pill manufactured to mimic the ABI-H2158 tablets

Intervention Type DRUG

Entecavir (ETV)

0.5 mg tablet for oral administration

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Body mass index of 18 - 36 kg/m\^2 and body weight ≥45 kg
* HBeAg ≥500 IU/mL at Screening
* In good general health except for chronic HBV infection for ≥6 months documented, for example, by at least two measurements of HBsAg positivity and/or detectable HBV DNA ≥6 months apart
* Lack of cirrhosis or advanced liver disease

Exclusion Criteria

* Prior treatment for chronic HBV infection with lamivudine, telbivudine, adefovir, standard of care nucleoside or nucleotide analogue (NrtI), HBV core inhibitors, or an investigational agent for HBV infection
* History or evidence of advanced liver disease or hepatic decompensation (including jaundice, ascites, portal hypertension, gastrointestinal bleeding, esophageal varices, hepatic encephalopathy)
* History or presence of clinically significant medical conditions requiring frequent medical management or pharmacologic or surgical treatment
Minimum Eligible Age

18 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Assembly Biosciences

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Grace Wang

Role: STUDY_DIRECTOR

Assembly Biosciences

Locations

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Coalition of Inclusive Medicine

Los Angeles, California, United States

Site Status

California Liver Research Institute

Pasadena, California, United States

Site Status

Stanford University Medical Center

Redwood City, California, United States

Site Status

Research and Education Inc.

San Diego, California, United States

Site Status

Quest Clinical Research

San Francisco, California, United States

Site Status

University of Miami/Schiff Center for Liver Diseases

Miami, Florida, United States

Site Status

Johns Hopkins University

Baltimore, Maryland, United States

Site Status

New Discovery, LLC

Flushing, New York, United States

Site Status

Northwell Health Center for Liver Disease

Manhasset, New York, United States

Site Status

NYU Langone Health

New York, New York, United States

Site Status

Thomas Jefferson University

Philadelphia, Pennsylvania, United States

Site Status

American Research Corporation at the Texas Liver Institute

San Antonio, Texas, United States

Site Status

University of Washington

Seattle, Washington, United States

Site Status

Royal Prince Alfred Hospital

Camperdown, New South Wales, Australia

Site Status

St. Vincent's Hospital

Darlinghurst, New South Wales, Australia

Site Status

John Hunter Hospital

New Lambton, New South Wales, Australia

Site Status

Gallipoli Medical Research Foundation

Greenslopes, Queensland, Australia

Site Status

St. Vincent's Hospital

Fitzroy, Victoria, Australia

Site Status

Alfred Hospital

Melbourne, Victoria, Australia

Site Status

Melbourne Health

Parkville, Victoria, Australia

Site Status

(G.I.R.I.) GI Research Institute

Vancouver, British Columbia, Canada

Site Status

Toronto Liver Centre

Toronto, Ontario, Canada

Site Status

The First Hospital of Jilin University

Changchun, Jilin, China

Site Status

The Second Affliated Hospital of Chongqing Medical University

Chongqing, Yuzhong District, China

Site Status

Xiangya Hospital Central South University

Changsha, , China

Site Status

Nanfang Hospital

Guangzhou, , China

Site Status

Guangzhou Eighth People's Hospital - Guangzhou Infectious Diseases Hospital

Guangzhou, , China

Site Status

Prince of Wales Hospital

Shatin, New Territories, Hong Kong

Site Status

Queen Mary Hospital

Hong Kong, , Hong Kong

Site Status

Auckland Clinical Studies

Auckland, , New Zealand

Site Status

Waikato Hospital

Hamilton, , New Zealand

Site Status

Hallym University Chuncheon Sacred Heart Hospital

Chuncheon, Gangwon-do, South Korea

Site Status

Pusan National University Yangsan Hospital

Yangsan, Gyeongsangnam-do, South Korea

Site Status

Pusan National University Hospital

Busan, , South Korea

Site Status

Seoul National University Hospital

Seoul, , South Korea

Site Status

Severance Hospital, Yonsei University Health System

Seoul, , South Korea

Site Status

Asan Medical Center

Seoul, , South Korea

Site Status

SMG-SNU Boramae Medical Center

Seoul, , South Korea

Site Status

Kaohsiung Medical University Hospital

Kaohsiung City, Sanmin District, Taiwan

Site Status

China Medical University Hospital

Taichung, , Taiwan

Site Status

National Taiwan University Hospital

Taipei, , Taiwan

Site Status

Mackay Memorial Hospital Taipei Branch

Taipei, , Taiwan

Site Status

Chang Gung Memorial Hospital (CGMH) - Linkou Branch

Taoyuan District, , Taiwan

Site Status

King's College Hospital

London, , United Kingdom

Site Status

Countries

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United States Australia Canada China Hong Kong New Zealand South Korea Taiwan United Kingdom

Provided Documents

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Document Type: Study Protocol and Statistical Analysis Plan

View Document

Other Identifiers

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2019-004902-85

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

ABI-H2158-201

Identifier Type: -

Identifier Source: org_study_id

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