Absorption and Pharmacokinetics of Nitroglycerin to a New Formulation

NCT ID: NCT03777605

Last Updated: 2018-12-19

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

UNKNOWN

Clinical Phase

PHASE4

Total Enrollment

10 participants

Study Classification

INTERVENTIONAL

Study Start Date

2018-12-23

Study Completion Date

2020-12-23

Brief Summary

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The study evaluate the absorption rate of different sublingual formulation of nitroglycerine (NTG) either in the form of available tablets or a new rapid absorbable gelation capsule formulation "NTG1523" by determining T-max and area under the response curve of nitoglycerine in blood concentration as well as from clinical effects after intake. Data is entered on data sheet in anonymous form and processed. The results are presented in anonymous form by publication and lecture. Experts are given the supplement: "The applicant's rights in a biomedical research project

Detailed Description

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Ten healthy young volunteers are recruited,, and the experiments begin at 07:45 after an overneight fast. BMI and blod pressure are recorded and a catheter is inserted in an anticubical vein for blood samples.

At 08.00 a sublingual tablet (Takeda, nitroglycerin 0.4 milligrams) tablet or a "NTG1523" capsule with 0.4 milligrams of nitroglycerine is placed under the tongue in random order. Subsequently, blood samples are taken every minute for 10 minutes, then every 10 minutes the following two hours. In addition, blood pressure and puls rate are measured every second minute the first ten minutes, and then every 10 minutes.Side effects and time to the participants registrate any effect of the drugs are assessed in a prefabricated scheme.

The disadvantages associated with the experiment are sought monitored by adverse event registration which ends at the end of the trial. The trial day lasts 2 hours in which blood samples are taken as described above, and blood pressure and records are stored .

Conditions

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Angina Pectoris

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

A randomized, cross over design
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

All tablets are processed, marked and coded by a pharmacist,

Study Groups

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"NTG1523", rapid absorbable capsule

Nitroglycerine 0.4 milligram taken as ordinary tablets or "NTG1523" rapid absorbable capsule once in the morning, and subsequently blood samples and observations for 2 hours are performed

Group Type EXPERIMENTAL

Nitroglycerin 0.4 MG

Intervention Type DRUG

The study evaluate absorption rate of nitroglycerine 0.4 milligrams as tablets or a quickly absorbable capsuel "NTG1523" determined by T-max and area under the response curve in the blood of NTG as well as from clinical effects.

Data is entered on data sheet in anonymous form and processed. The results are presented in anonymous form by publication and lecture. Experts are given the supplement: "The applicant's rights in a biomedical research project

Interventions

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Nitroglycerin 0.4 MG

The study evaluate absorption rate of nitroglycerine 0.4 milligrams as tablets or a quickly absorbable capsuel "NTG1523" determined by T-max and area under the response curve in the blood of NTG as well as from clinical effects.

Data is entered on data sheet in anonymous form and processed. The results are presented in anonymous form by publication and lecture. Experts are given the supplement: "The applicant's rights in a biomedical research project

Intervention Type DRUG

Other Intervention Names

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"NTG1523"

Eligibility Criteria

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Inclusion Criteria

* Normal healthy volunteers
* Must be able to swallow tablets

Exclusion Criteria

* Insulin dependent diabetes
* Thyroid disease
* any medial treatment
Minimum Eligible Age

18 Years

Maximum Eligible Age

28 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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Kolding Sygehus

OTHER

Sponsor Role lead

Responsible Party

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Ole Winther Rasmussen

Clinical professor

Responsibility Role PRINCIPAL_INVESTIGATOR

Principal Investigators

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ole W Rasmussen, M.D. Dr.Sci

Role: PRINCIPAL_INVESTIGATOR

Medical Dept.,Kolding Hospital, SLB, Denmark

Locations

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Kolfding Sygehus, SLB

Kolding, , Denmark

Site Status

Countries

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Denmark

Central Contacts

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ole W Rasmussen, M.D., Dr.Sci

Role: CONTACT

Phone: +4550506930

Email: [email protected]

Poul H Madsen, M.D., Ph.D.

Role: CONTACT

Phone: +45 76362000

Email: [email protected]

References

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Nakashima E, Rigod JF, Lin ET, Benet LZ. Pharmacokinetics of nitroglycerin and its dinitrate metabolites over a thirtyfold range of oral doses. Clin Pharmacol Ther. 1990 May;47(5):592-8. doi: 10.1038/clpt.1990.80.

Reference Type BACKGROUND
PMID: 2111749 (View on PubMed)

McAllister A, Mosberg H, Settlage JA, Steiner JA. Plasma levels of nitroglycerin generated by three nitroglycerin patch preparations, Nitradisc, Transiderm-Nitro and Nitro-Dur and one ointment formulation, Nitrobid. Br J Clin Pharmacol. 1986 Apr;21(4):365-9. doi: 10.1111/j.1365-2125.1986.tb05208.x.

Reference Type RESULT
PMID: 3085698 (View on PubMed)

Other Identifiers

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Nitroglycerine1523 (NTG1523)

Identifier Type: -

Identifier Source: org_study_id