A Study of ZN-c5 in Subjects With Breast Cancer

NCT ID: NCT03560531

Last Updated: 2024-08-09

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1/PHASE2

Total Enrollment

181 participants

Study Classification

INTERVENTIONAL

Study Start Date

2018-11-30

Study Completion Date

2022-12-22

Brief Summary

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This is a Phase 1/2, open-label, multicenter, dose-escalation and expansion study to evaluate the safety, tolerability, pharmacokinetics, and preliminary efficacy of ZN-c5 administered orally in subjects with advanced estrogen receptor positive, human epidermal growth factor receptor 2 negative (ER+/HER2-) breast cancer. ZN-c5 will be evaluated both as monotherapy and in combination with palbociclib (IBRANCE®).

Detailed Description

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Conditions

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Breast Cancer

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Dose escalation cohorts are planned in monotherapy and combination as well as monotherapy dose expansion, and monotherapy and combination Phase 2.
Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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ZN-c5 monotherapy

Dose escalation cohorts are planned to determine maximum tolerated dose(MTD) or recommended phase 2 dose (RP2D) of ZN-c5 as well as expansion cohorts and a Phase 2 cohort.

Group Type EXPERIMENTAL

ZN-c5

Intervention Type DRUG

ZN-c5 is a study drug

ZN-c5 + palbociclib combination therapy

Dose escalation cohorts are planned to determine maximum tolerated dose(MTD) or recommended phase 2 dose (RP2D) of ZN-c5 in combination with palbociclib as well as a Phase 2 cohort.

Group Type EXPERIMENTAL

ZN-c5

Intervention Type DRUG

ZN-c5 is a study drug

Palbociclib

Intervention Type DRUG

Palbociclib (IBRANCE®) is an approved drug

Interventions

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ZN-c5

ZN-c5 is a study drug

Intervention Type DRUG

Palbociclib

Palbociclib (IBRANCE®) is an approved drug

Intervention Type DRUG

Other Intervention Names

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IBRANCE®

Eligibility Criteria

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Inclusion Criteria

* Age ≥ 18 years of age

* Women can be postmenopausal, as defined by at least one of the following:
* Age ≥ 60 years;
* Age \< 60 years and cessation of regular menses for at least 12 consecutive months with no alternative pathological or physiological cause; and serum estradiol and follicle-stimulating hormone level within the laboratory's reference range for postmenopausal females;
* Documented bilateral oophorectomy; or can be peri- or premenopausal, however, they must receive a gonadotrophin-releasing hormone agonist beginning at least 4 weeks prior to the first dose of study medication.
* Histologically or cytologically confirmed diagnosis of advanced (metastatic or locoregionally recurrent) adenocarcinoma of the breast, not amenable to any potential curative intervention
* Estrogen Receptor (ER) positive disease
* Human Epidermal Growth Factor Receptor 2 (HER2) negative disease
* Documented prior response to endocrine therapy for metastatic disease (stable disease, partial response, or complete response by RECIST v1.1 criteria) lasting \> 6 months
* Evaluable or measurable disease by RECIST v1.1. Tumor lesions previously irradiated or subjected to other locoregional therapy will only be deemed measurable if progression at the treated site after completion of therapy is clearly documented.

Exclusion Criteria

* Prior anticancer or investigational drugs for the treatment of ER+/HER2 negative advanced breast cancer within the following windows:

* Tamoxifen, aromatase inhibitor, fulvestrant, or other anti-cancer endocrine therapy \< 14 days before first dose of study treatment
* Any chemotherapy \< 28 days before first dose of study, except for Phase 2 monotherapy which requires no prior chemotherapy treatment.
* Any investigational drug therapy \< 28 days or 5 half-lives (whichever is shorter) prior to first dose of study treatment
* Unexplained symptomatic endometrial disorders (including, but not limited to endometrial hyperplasia, dysfunctional uterine bleeding, or cysts)
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Zeno Alpha Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Zeno Alpha, Inc.

Role: STUDY_DIRECTOR

Zeno Alpha Inc.

Locations

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Site 3

Tucson, Arizona, United States

Site Status

Site 5

Los Angeles, California, United States

Site Status

Site 48

Bethesda, Maryland, United States

Site Status

Site 47

St Louis, Missouri, United States

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Site 7

New York, New York, United States

Site Status

Site 2

New York, New York, United States

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Site 50

Charleston, South Carolina, United States

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Site 4

Nashville, Tennessee, United States

Site Status

Site 1

Houston, Texas, United States

Site Status

Site 8

Houston, Texas, United States

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Site 6

Seattle, Washington, United States

Site Status

Site 46

Minsk, , Belarus

Site Status

Site 45

Vitebsk, , Belarus

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Site 10

Banja Luka, , Bosnia and Herzegovina

Site Status

Site 9

Sarajevo, , Bosnia and Herzegovina

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Site 11

Tuzla, , Bosnia and Herzegovina

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Site 29

Brno, , Czechia

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Site 28

Olomouc, , Czechia

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Site 30

Prague, , Czechia

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Site 51

Budapest, , Hungary

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Site 35

Kecskemét, , Hungary

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Site 37

Pécs, , Hungary

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Site 17

Kaunas, , Lithuania

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Site 16

Vilnius, , Lithuania

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Site 40

Nizhny Novgorod, , Russia

Site Status

Site 52

Omsk, , Russia

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Site 41

Pyatigorsk, , Russia

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Site 39

Saint Petersburg, , Russia

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Site 42

Yekaterinburg, , Russia

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Site 18

Belgrade, , Serbia

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Site 19

Belgrade, , Serbia

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Site 21

Niš, , Serbia

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Site 20

Novi Sad, , Serbia

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Site 25

Cherkasy, , Ukraine

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Site 27

Kharkiv, , Ukraine

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Site 24

Kropyvnytskyi, , Ukraine

Site Status

Site 26

Kryvyi Rih, , Ukraine

Site Status

Site 23

Kyiv, , Ukraine

Site Status

Countries

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United States Belarus Bosnia and Herzegovina Czechia Hungary Lithuania Russia Serbia Ukraine

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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ZN-c5-001

Identifier Type: -

Identifier Source: org_study_id

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