A Phase 1 Study of Oral OP-1250 in Combination With Palbociclib in HR+/HER2- Breast Cancer Patients

NCT ID: NCT05266105

Last Updated: 2025-11-24

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE1

Total Enrollment

60 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-12-10

Study Completion Date

2026-03-31

Brief Summary

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This is an open-label, Phase 1b dose escalation and expansion study to determine the maximum tolerated dose (MTD) of OP-1250 in combination with palbociclib (Ibrance®️, Pfizer Inc.). Purpose of study is to evaluate the safety and pharmacokinetic (PK) profile, and estimate the preliminary anti-tumor activity of the combination in adult subjects with hormone receptor-positive (ER+ / HER2-) advanced or metastatic breast cancer (MBC).

Detailed Description

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Conditions

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Breast Cancer

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

SEQUENTIAL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Dose Escalation

This portion of the study will evaluate the safety and pharmacology of a range of OP-1250 doses administered daily with Palbociclib in subjects with advanced and/or metastatic hormone receptor (HR)-positive, HER2-negative breast cancer

Group Type EXPERIMENTAL

Palazestrant

Intervention Type DRUG

Complete Estrogen Receptor Antagonist

Palbociclib

Intervention Type DRUG

Palbociclib is an approved CDK 4/6 Inhibitor drug

Dose Expansion

This portion of the study further explores the clinical activity, safety and pharmacology of OP-1250 in combination with Palbociclib and estimates preliminary data of anti-tumor efficacy

Group Type EXPERIMENTAL

Palazestrant

Intervention Type DRUG

Complete Estrogen Receptor Antagonist

Palbociclib

Intervention Type DRUG

Palbociclib is an approved CDK 4/6 Inhibitor drug

Interventions

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Palazestrant

Complete Estrogen Receptor Antagonist

Intervention Type DRUG

Palbociclib

Palbociclib is an approved CDK 4/6 Inhibitor drug

Intervention Type DRUG

Other Intervention Names

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OP-1250 Ibrance®️

Eligibility Criteria

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Inclusion Criteria

* Confirmed and evaluable locally advanced or metastatic breast cancer
* Eastern Cooperative Oncology Group (ECOG) performance status of 0 or 1
* Must not have received prior oral endocrine or targeted therapy ≤ 2 weeks prior to first dose
* Must not have received prior chemotherapy, antibody therapy, or investigational therapy ≤ 4 weeks prior to the first dose
* Prior radiotherapy must have been completed 2 weeks prior to first dose
* Adequate safety laboratory tests
* Willingness to use effective contraception

Exclusion Criteria

* Gastrointestinal disease
* Significant hepatic disease
* Significant cardiovascular disease
* Significant ECG abnormalities
* History of pulmonary embolism or high risk of thrombosis
* Known HIV infection
* Active infection (requiring antimicrobial therapy)
* Pregnant
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role collaborator

Olema Pharmaceuticals, Inc.

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Sue Johnson

Role: STUDY_DIRECTOR

Olema Pharmaceuticals, Inc.

Locations

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Clinical Trial Site

Waratah, New South Wales, Australia

Site Status

Clinical Trial Site

Westmead, New South Wales, Australia

Site Status

Clinical Trial Site

South Brisbane, Queensland, Australia

Site Status

Clinical Trial Site

Southport, Queensland, Australia

Site Status

Clinical Trial Site

Clayton, Victoria, Australia

Site Status

Clinical Trial Site

Frankston, Victoria, Australia

Site Status

Clinical Trial Site

Geelong, Victoria, Australia

Site Status

Clinical Trial Site

Nedlands, Western Australia, Australia

Site Status

Countries

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Australia

Other Identifiers

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OP-1250-002

Identifier Type: -

Identifier Source: org_study_id

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