Open Label Safety Study in Acute Treatment of Migraine

NCT ID: NCT03266588

Last Updated: 2023-02-16

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2/PHASE3

Total Enrollment

3019 participants

Study Classification

INTERVENTIONAL

Study Start Date

2017-08-30

Study Completion Date

2019-07-15

Brief Summary

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The purpose of this study is to evaluate safety and tolerability of BHV-3000 (rimegepant).

Detailed Description

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Conditions

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Migraine, With or Without Aura

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Rimegepant

Group Type EXPERIMENTAL

Rimegepant

Intervention Type DRUG

75 mg oral tablet

Interventions

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Rimegepant

75 mg oral tablet

Intervention Type DRUG

Other Intervention Names

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BHV-3000

Eligibility Criteria

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Inclusion Criteria

* Subjects with 2-8 moderate to severe migraines/month
* Age of onset of migraines prior to 50 years of age
* Migraine attacks, on average, lasting 4-72 hours if untreated
* Ability to distinguish migraine attacks from tension/cluster headaches
* Patients with contraindications for use of triptans may be included provided they meet all other study entry criteria

Exclusion Criteria

* History of basilar migraine or hemiplegic migraine
* History of HIV disease
* History with current evidence of uncontrolled, unstable or recently diagnosed cardiovascular disease, such as ischemic heart disease, coronary artery vasospasm, and cerebral ischemia.
* Uncontrolled hypertension or uncontrolled diabetes (however, patients can be included who have stable hypertension and /or diabetes for 3 months prior to screening
* History of gastric or small intestinal surgery or has a disease that causes malabsorption
* BMI ≥ 30
* HbA1c ≥ 6.5%
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Central Research Associates, Inc

Birmingham, Alabama, United States

Site Status

Coastal Clinical Research, Inc.

Mobile, Alabama, United States

Site Status

Thunderbird Internal Medicine / Radiant Research, Inc

Glendale, Arizona, United States

Site Status

Neurological Physicians of Arizona

Tempe, Arizona, United States

Site Status

Clinical Research Consortium Arizona

Tempe, Arizona, United States

Site Status

Woodland International Research Group, LLC

Little Rock, Arkansas, United States

Site Status

Woodland Research Northwest, LLC

Rogers, Arkansas, United States

Site Status

Pharmacology Research Institute

Encino, California, United States

Site Status

eStudySite

La Mesa, California, United States

Site Status

Collaborative Neuroscience Network, LLC

Long Beach, California, United States

Site Status

Pharmacology Research Institute

Los Alamitos, California, United States

Site Status

Pharmacology Research Institute

Newport Beach, California, United States

Site Status

Pacific Research Partners LLC

Oakland, California, United States

Site Status

National Research Institute

Panorama City, California, United States

Site Status

Optimus Medical Group

San Francisco, California, United States

Site Status

California Medical Clinic for Headache

Santa Monica, California, United States

Site Status

California Neuroscience Research Medical Group, Inc.

Sherman Oaks, California, United States

Site Status

Diablo Clinical Research, Inc

Walnut Creek, California, United States

Site Status

Clinical Trials of the Rockies

Denver, Colorado, United States

Site Status

AGA Clinical Trials

Hialeah, Florida, United States

Site Status

Clinical Neuroscience Solutions, Inc.

Jacksonville, Florida, United States

Site Status

Multi-Specialty Research Associates, Inc

Lake City, Florida, United States

Site Status

Renstar Medical Research

Ocala, Florida, United States

Site Status

Clinical Neuroscience Solutions, Inc

Orlando, Florida, United States

Site Status

Compass Research, LLC

Orlando, Florida, United States

Site Status

Ormond Medical Arts Pharmaceutical Research

Ormond Beach, Florida, United States

Site Status

Meridien Research

Tampa, Florida, United States

Site Status

Radiant Research, Inc.

Atlanta, Georgia, United States

Site Status

Meridian Clinical Research

Savannah, Georgia, United States

Site Status

Savannah Neurology Specialists

Savannah, Georgia, United States

Site Status

Christie Clinic, LLC

Champaign, Illinois, United States

Site Status

PMG Research of McFrland Clinic

Ames, Iowa, United States

Site Status

Heartland Research Associates, LLC

Augusta, Kansas, United States

Site Status

Heartland Research Associates, LLC

Newton, Kansas, United States

Site Status

Heartland Research Associates, LLC

Wichita, Kansas, United States

Site Status

Heartland Research Associates, LLC

Wichita, Kansas, United States

Site Status

Benchmark Research

Metairie, Louisiana, United States

Site Status

MedPharmics, LLC

Metairie, Louisiana, United States

Site Status

New Orleans Center for Clinical Research

New Orleans, Louisiana, United States

Site Status

Boston Clinical Trials, Inc.

Boston, Massachusetts, United States

Site Status

NECCR Primacare Research, LLC

Fall River, Massachusetts, United States

Site Status

Milford Emergency Associates, Inc.

Marlborough, Massachusetts, United States

Site Status

Michigan Head Pain and Neurological Institute

Ann Arbor, Michigan, United States

Site Status

Clinical Research Institute, Inc.

Minneapolis, Minnesota, United States

Site Status

Clinical Research Insitute

Plymouth, Minnesota, United States

Site Status

The Center for Pharmaceutical Research

Kansas City, Missouri, United States

Site Status

Sundance Clinical Research, LLC

St Louis, Missouri, United States

Site Status

Meridian Clinical Research -Norfolk

Norfolk, Nebraska, United States

Site Status

Meridian Clinical Research, LLC

Omaha, Nebraska, United States

Site Status

Clinical Research Consortium- Las Vegas

Las Vegas, Nevada, United States

Site Status

Hassman Research Institute, LLC

Berlin, New Jersey, United States

Site Status

Albuquerque Neuroscience, Inc.

Albuquerque, New Mexico, United States

Site Status

United Medical Associates

Binghamton, New York, United States

Site Status

SPRI Clinical Trials, LLC

Brooklyn, New York, United States

Site Status

Regional Clinical Research, Inc.

Endwell, New York, United States

Site Status

Radiant Research, Inc.

Jamaica, New York, United States

Site Status

Central New York Clinical Research

Manlius, New York, United States

Site Status

Fieve Clinical Research

New York, New York, United States

Site Status

Rochester Clinical Research, Inc

Rochester, New York, United States

Site Status

Montefiore Heachache Center

The Bronx, New York, United States

Site Status

PMG Research of Charlotte, LLC

Charlotte, North Carolina, United States

Site Status

PharmQuest, LLC

Greensboro, North Carolina, United States

Site Status

PMG Research of Raleigh, LLC

Raleigh, North Carolina, United States

Site Status

Wake Research Associates, LLC

Raleigh, North Carolina, United States

Site Status

PMG Research of Wilmington, LLC

Wilmington, North Carolina, United States

Site Status

CTI Clinical Research Center

Cincinnati, Ohio, United States

Site Status

Radiant Research, Inc.

Cincinnati, Ohio, United States

Site Status

Radiant Research, Inc.

Columbus, Ohio, United States

Site Status

Midwest Clinical Research Center

Dayton, Ohio, United States

Site Status

Neurology Diagnostics, Inc.

Dayton, Ohio, United States

Site Status

Aventiv Research, Inc.

Dublin, Ohio, United States

Site Status

Summit Research Network (Oregon), Inc.

Portland, Oregon, United States

Site Status

Oregon Center for Clinical Investigations, Inc

Salem, Oregon, United States

Site Status

Clinical Research of Philadelphia, LLC

Philadelphia, Pennsylvania, United States

Site Status

Fieve Clinical Research

Scranton, Pennsylvania, United States

Site Status

Preferred Primary Care Physicians

Uniontown, Pennsylvania, United States

Site Status

Omega Medical Research

Warwick, Rhode Island, United States

Site Status

Radiant Research, Inc.

Anderson, South Carolina, United States

Site Status

Coastal Carolina Research Center

Mt. Pleasant, South Carolina, United States

Site Status

Meridian Clinical Research

Dakota Dunes, South Dakota, United States

Site Status

PMG Research of Bristol, LLC

Bristol, Tennessee, United States

Site Status

Clinical Neuroscience Solutions, Inc

Memphis, Tennessee, United States

Site Status

Clinical Research Associates, Inc.

Nashville, Tennessee, United States

Site Status

FutureSearch Trials of Neurology, LP

Austin, Texas, United States

Site Status

Tekton Research- Austin

Austin, Texas, United States

Site Status

FutureSearch Trials of Neurology, LP

Dallas, Texas, United States

Site Status

Ventavia Research Group, LLC

Fort Worth, Texas, United States

Site Status

Texas Center for Drug Development

Houston, Texas, United States

Site Status

Red Star Research, LLC

Lake Jackson, Texas, United States

Site Status

FMC Science

Lampasas, Texas, United States

Site Status

PCP for Life

Magnolia, Texas, United States

Site Status

Research Across America - Mesquite

Mesquite, Texas, United States

Site Status

Doctors of Internal Medicine, LTD / Radiant Research Inc.

Plano, Texas, United States

Site Status

DM Clinical Research

Tomball, Texas, United States

Site Status

J.Lewis Research Inc / Foothill Family Clinic South

Salt Lake City, Utah, United States

Site Status

Tidewater Integrated Medical Research

Virginia Beach, Virginia, United States

Site Status

Northwest Clinical Research Center

Bellevue, Washington, United States

Site Status

Seattle Women's:Health, Research & Gynecology

Seattle, Washington, United States

Site Status

Countries

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United States

References

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Ailani J, Pavlovic J, Pixton GC, Fullerton T. Rimegepant safety and patient-reported outcomes among triptan-naive, triptan-using, and triptan-failure participants: Subgroup analysis of an open-label, multicenter study. Cephalalgia. 2025 Jul;45(7):3331024251343309. doi: 10.1177/03331024251343309. Epub 2025 Jul 9.

Reference Type DERIVED
PMID: 40629887 (View on PubMed)

Kudrow D, Hutchinson S, Pixton GC, Fullerton T. Safety of Rimegepant in Adults with Migraine and Anxiety, Depression, or Using Antidepressants: Analysis of a Multicenter, Long-Term, Open-Label Study. Pain Ther. 2025 Feb;14(1):237-255. doi: 10.1007/s40122-024-00675-6. Epub 2024 Nov 9.

Reference Type DERIVED
PMID: 39520634 (View on PubMed)

True D, Mullin K, Croop R. Safety of Rimegepant in Adults with Migraine and Cardiovascular Risk Factors: Analysis of a Multicenter, Long-Term, Open-Label Study. Pain Ther. 2024 Oct;13(5):1203-1218. doi: 10.1007/s40122-024-00626-1. Epub 2024 Jul 10.

Reference Type DERIVED
PMID: 38985436 (View on PubMed)

Fullerton T, Pixton G. Long-Term Use of Rimegepant 75 mg for the Acute Treatment of Migraine is Associated with a Reduction in the Utilization of Select Analgesics and Antiemetics. J Pain Res. 2024 May 15;17:1751-1760. doi: 10.2147/JPR.S456006. eCollection 2024.

Reference Type DERIVED
PMID: 38764606 (View on PubMed)

Croop R, Berman G, Kudrow D, Mullin K, Thiry A, Lovegren M, L'Italien G, Lipton RB. A multicenter, open-label long-term safety study of rimegepant for the acute treatment of migraine. Cephalalgia. 2024 Apr;44(4):3331024241232944. doi: 10.1177/03331024241232944.

Reference Type DERIVED
PMID: 38659334 (View on PubMed)

Johnston K, Harris L, Powell L, Popoff E, Coric V, L'Italien G, Schreiber CP. Monthly migraine days, tablet utilization, and quality of life associated with Rimegepant - post hoc results from an open label safety study (BHV3000-201). J Headache Pain. 2022 Jan 17;23(1):10. doi: 10.1186/s10194-021-01378-5.

Reference Type DERIVED
PMID: 35038983 (View on PubMed)

Johnston KM, L'Italien G, Popoff E, Powell L, Croop R, Thiry A, Harris L, Coric V, Lipton RB. Mapping Migraine-Specific Quality of Life to Health State Utilities in Patients Receiving Rimegepant. Adv Ther. 2021 Oct;38(10):5209-5220. doi: 10.1007/s12325-021-01897-2. Epub 2021 Aug 29.

Reference Type DERIVED
PMID: 34455556 (View on PubMed)

Mullin K, Kudrow D, Croop R, Lovegren M, Conway CM, Coric V, Lipton RB. Potential for treatment benefit of small molecule CGRP receptor antagonist plus monoclonal antibody in migraine therapy. Neurology. 2020 May 19;94(20):e2121-e2125. doi: 10.1212/WNL.0000000000008944. Epub 2020 Jan 13.

Reference Type DERIVED
PMID: 31932515 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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BHV3000-201

Identifier Type: -

Identifier Source: org_study_id

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