A Phase 2 Safety and Efficacy Study of INCB050465 in Subjects With Relapsed or Refractory Diffuse Large B-Cell Lymphoma (CITADEL-202)

NCT ID: NCT02998476

Last Updated: 2025-08-22

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

60 participants

Study Classification

INTERVENTIONAL

Study Start Date

2017-03-02

Study Completion Date

2021-02-05

Brief Summary

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The purpose of this study is to assess the safety and efficacy of parsaclisib in subjects with relapsed or refractory diffuse large B-cell lymphoma.

Detailed Description

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Conditions

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Lymphoma

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Group A Parsaclisib (no prior BTK inhibitor)

Parsaclisib in subjects who were not previously treated with a BTK inhibitor.

Group Type EXPERIMENTAL

Parsaclisib

Intervention Type DRUG

Parsaclisib once daily for 8 weeks followed by once weekly

Group B Parsaclisib (prior BTK inhibitor)

Parsaclisib in subjects who were previously treated with a BTK inhibitor.

Group Type EXPERIMENTAL

Parsaclisib

Intervention Type DRUG

Parsaclisib once daily for 8 weeks followed by once weekly

Interventions

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Parsaclisib

Parsaclisib once daily for 8 weeks followed by once weekly

Intervention Type DRUG

Other Intervention Names

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INCB050465

Eligibility Criteria

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Inclusion Criteria

* Eligible 19 years and older in South Korea
* Relapsed or refractory DLBCL, which has been histologically documented, defined as having received at least 2 but no more than 5 prior treatment regimens and ineligible for high-dose chemotherapy supported by autologous stem cell transplant.
* Must have ≥ 1 measurable lesion (≥2 cm in longest dimension) or ≥ 1 measurable extranodal lesion (≥1 cm in longest dimension) on computed tomography (CT) scan or magnetic resonance imaging (MRI).
* Subjects must be willing to undergo an incisional or excisional lymph node biopsy of accessible adenopathy or provide the most recent, available archived tumor biopsy.
* Eastern Cooperative Oncology Group performance status 0 to 2.

Exclusion Criteria

* Primary mediastinal (thymic) large B-cell lymphoma.
* Known brain or central nervous system metastases or history of uncontrolled seizures.
* Allogeneic stem cell transplant within the last 6 months, or active graft versus host disease following allogeneic transplant, or autologous stem cell transplant within the last 3 months.
* Use or expected use during the study of any prohibited medications, including potent cytochrome P450 3A4 inhibitors or inducers within 14 days or 5 half lives (whichever is longer) before the first dose of study drug.
* Prior treatment with the following:

* Group A: Prior treatment with a selective phosphatidylinositol 3-kinase (PI3K) δ inhibitor (eg, idelalisib), a pan-PI3K inhibitor, or a BTK inhibitor (eg, ibrutinib).
* Group B: Prior treatment with a selective PI3Kδ inhibitor (eg, idelalisib) or a pan PI3K inhibitor.
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Incyte Corporation

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Claudia Corrado, MD

Role: STUDY_DIRECTOR

Incyte Corporation

Locations

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University of Alabama at Birmingham

Birmingham, Alabama, United States

Site Status

Banner MD Anderson Cancer Center

Gilbert, Arizona, United States

Site Status

Arizona Oncology Associates, PC - HAL

Tempe, Arizona, United States

Site Status

Sutter Gould Medical Foundation

Modesto, California, United States

Site Status

Sharp Memorial Hospital

San Diego, California, United States

Site Status

Advanced Pharma CR, LLC

Miami, Florida, United States

Site Status

Asclepes Research Centers

Weeki Wachee, Florida, United States

Site Status

Advocate Medical Group Niles Milwaukee Ave

Niles, Illinois, United States

Site Status

Indiana BMT

Beech Grove, Indiana, United States

Site Status

Parkview Research Center

Fort Wayne, Indiana, United States

Site Status

University of Kentucky Hospital

Lexington, Kentucky, United States

Site Status

St. Agnes Hospital

Baltimore, Maryland, United States

Site Status

Karmanos Cancer Institute

Detroit, Michigan, United States

Site Status

St. John Hospital and Medical Center

Detroit, Michigan, United States

Site Status

CHI Health - St. Francis Medical Center

Grand Island, Nebraska, United States

Site Status

Summit Medical Group

Morristown, New Jersey, United States

Site Status

Rutgers Cancer Institute of New Jersey

New Brunswick, New Jersey, United States

Site Status

Clinical Research Alliance

Lake Success, New York, United States

Site Status

Abington Memorial Hospital

Abington, Pennsylvania, United States

Site Status

Utah Cancer Specialists- Network

Salt Lake City, Utah, United States

Site Status

St Vincent's Hospital Sydney

Darlinghurst, New South Wales, Australia

Site Status

Westmead Hospital

Westmead, New South Wales, Australia

Site Status

Flinders Medical Centre

Bedford Park, South Australia, Australia

Site Status

Ballarat Base Hospital

Ballarat, Victoria, Australia

Site Status

Sunshine Hospital

St Albans, Victoria, Australia

Site Status

Fiona Stanley Hospital

Murdoch, Western Australia, Australia

Site Status

ZNA Stuivenberg

Antwerp, , Belgium

Site Status

Cliniques Universitaires Ucl Saint-Luc

Brussels, , Belgium

Site Status

UZ Leuven

Leuven, , Belgium

Site Status

AZ Delta

Roeselare, , Belgium

Site Status

LHSC - Victoria Hospital

London, Ontario, Canada

Site Status

Fakultni nemocnice Brno

Brno, , Czechia

Site Status

Fakultni nemocnice Hradec Kralove

Hradec Králové, , Czechia

Site Status

University Hospital Ostrava

Ostrava, , Czechia

Site Status

Fakultni nemocnice v Motole

Prague, , Czechia

Site Status

Centre Antoine Lacassagne

Nice, Alpes Maritimes, France

Site Status

Centre Francois Baclesse

Caen, Calvados, France

Site Status

CHU Dijon - Hopital du Bocage

Dijon, Cote dÝOr, France

Site Status

Centre Hospitalier Libourne

Libourne, Gironde, France

Site Status

CHU de Grenoble - Hôpital Albert Michallon

Grenoble, Isere, France

Site Status

Centre Hospitalier d'Angers

Angers, Maine Et Loire, France

Site Status

Hopital Claude Huriez - CHU Lille

Lille, Nord, France

Site Status

Hôpital Saint-Louis

Paris, Paris, France

Site Status

Clinique Victor Hugo - Centre Jean Bernard

Le Mans, Sarthe, France

Site Status

Hôpital Henri Mondor

Créteil, Val De Marne, France

Site Status

Chu de Grenoble - Hopital Albert Michallon

Grenoble, , France

Site Status

Groupe Hospitalier Pitie-Salpetriere

Paris, , France

Site Status

Chu Vandoeuvre-Les-Nancy Hopital Brabois

Vandœuvre-lès-Nancy, , France

Site Status

Institut Gustave Roussy

Villejuif, , France

Site Status

IRCCS Ospedale Casa Sollievo della Sofferenza

San Giovanni Rotondo, Foggia, Italy

Site Status

Istituto Tumori Giovanni Paolo II IRCCS Ospedale Oncologico Bari

Bari, , Italy

Site Status

Istituto Scientifico Romagnolo Per Lo Studio E La Cura Dei Tumori

Meldola, , Italy

Site Status

Policlinico Universitario Agostino Gemelli Universita Cattolica Del Sacro Cuore

Rome, , Italy

Site Status

Szpital Specjalistyczny W Brzozowie, Podkarpacki Osrodek Onkologiczny Im.Ks.B.Markiewicza

Brzozów, , Poland

Site Status

Uniwersyteckie Centrum Kliniczne

Gdansk, , Poland

Site Status

Malopolskie Centrum Medyczne s.c.

Krakow, , Poland

Site Status

Seoul National University Hospital

Seoul, , South Korea

Site Status

Severance Hospital, Yonsei University

Seoul, , South Korea

Site Status

Asan Medical Center

Seoul, , South Korea

Site Status

Samsung Medical Center

Seoul, , South Korea

Site Status

ICO l´Hospitalet - Hospital Duran i Reynals

L'Hospitalet de Llobregat, Barcelona, Spain

Site Status

Hospital del Mar

Barcelona, , Spain

Site Status

Hospital General Universitario Gregorio Marañon

Madrid, , Spain

Site Status

Hospital Universitario Ramon y Cajal

Madrid, , Spain

Site Status

Clinica Universidad de Navarra (Cun)

Pamplona, , Spain

Site Status

Hospital Universitario Nuestra Señora de Valme

Seville, , Spain

Site Status

Hospital Txagorritxu

Vitoria-Gasteiz, , Spain

Site Status

The Christie

Manchester, Greater Manchester, United Kingdom

Site Status

Southend University Hospital

Southend-on-Sea, , United Kingdom

Site Status

Royal Marsden Hospital

Sutton, , United Kingdom

Site Status

Countries

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United States Australia Belgium Canada Czechia France Italy Poland South Korea Spain United Kingdom

References

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Coleman M, Belada D, Casasnovas RO, Gressin R, Lee HP, Mehta A, Munoz J, Verhoef G, Corrado C, DeMarini DJ, Zhao W, Li J, Fay K. Phase 2 study of parsaclisib (INCB050465), a highly selective, next-generation PI3Kdelta inhibitor, in relapsed or refractory diffuse large B-cell lymphoma (CITADEL-202). Leuk Lymphoma. 2021 Feb;62(2):368-376. doi: 10.1080/10428194.2020.1832660. Epub 2020 Nov 3.

Reference Type DERIVED
PMID: 33140664 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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Parsaclisib

Identifier Type: OTHER

Identifier Source: secondary_id

2016-002205-19

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

INCB 50465-202/CITADEL-202

Identifier Type: -

Identifier Source: org_study_id

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