Filgotinib Alone and in Combination With Methotrexate (MTX) in Adults With Moderately to Severely Active Rheumatoid Arthritis Who Are Naive to MTX Therapy

NCT ID: NCT02886728

Last Updated: 2021-06-01

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

1252 participants

Study Classification

INTERVENTIONAL

Study Start Date

2016-08-08

Study Completion Date

2019-05-08

Brief Summary

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The primary objective of this study is to evaluate the effects of filgotinib in combination with methotrexate (MTX) versus MTX alone in adults with active rheumatoid arthritis (RA).

Detailed Description

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Conditions

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Rheumatoid Arthritis

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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Filgotinib 200 mg + MTX

Filgotinib 200 mg + placebo to match filgotinib 100 mg + MTX up to 20 mg

Group Type EXPERIMENTAL

Filgotinib

Intervention Type DRUG

Tablet(s) administered orally once daily

Placebo to match filgotinib

Intervention Type DRUG

Tablet(s) administered orally once daily

MTX

Intervention Type DRUG

Capsule(s) administered orally once weekly

Filgotinib 100 mg + MTX

Filgotinib 100 mg + placebo to match filgotinib 200 mg + MTX up to 20 mg

Group Type EXPERIMENTAL

Filgotinib

Intervention Type DRUG

Tablet(s) administered orally once daily

Placebo to match filgotinib

Intervention Type DRUG

Tablet(s) administered orally once daily

MTX

Intervention Type DRUG

Capsule(s) administered orally once weekly

Filgotinib 200 mg Monotherapy

Filgotinib 200 mg + placebo to match filgotinib 100 mg + placebo to match MTX

Group Type EXPERIMENTAL

Filgotinib

Intervention Type DRUG

Tablet(s) administered orally once daily

Placebo to match filgotinib

Intervention Type DRUG

Tablet(s) administered orally once daily

Placebo to match MTX

Intervention Type DRUG

Capsule(s) administered orally once weekly

MTX Monotherapy

Placebo to match filgotinib 200 mg + placebo to match filgotinib 100 mg + MTX up to 20 mg

Group Type ACTIVE_COMPARATOR

Placebo to match filgotinib

Intervention Type DRUG

Tablet(s) administered orally once daily

MTX

Intervention Type DRUG

Capsule(s) administered orally once weekly

Interventions

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Filgotinib

Tablet(s) administered orally once daily

Intervention Type DRUG

Placebo to match filgotinib

Tablet(s) administered orally once daily

Intervention Type DRUG

MTX

Capsule(s) administered orally once weekly

Intervention Type DRUG

Placebo to match MTX

Capsule(s) administered orally once weekly

Intervention Type DRUG

Other Intervention Names

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GS-6034 GLPG0634

Eligibility Criteria

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Inclusion Criteria

* Have a diagnosis of RA (2010 American College of Rheumatology \[ACR\]/European League Against Rheumatism \[EULAR\] criteria) and are ACR functional class I-III.
* Have ≥ 6 swollen joints (from a swollen joint count based on 66 joints (SJC66)) and ≥ 6 tender joints (from a tender joint count based on 68 joints (TJC68)) at both screening and Day 1.
* Limited or no prior treatment with MTX

Exclusion Criteria

* Previous treatment with any janus kinase (JAK) inhibitor
* Previous therapy for longer than 3 months with conventional synthetic disease modifying antirheumatic drugs (csDMARDs) other than MTX or hydroxychloroquine
* Use of any licensed or investigational biologic disease-modifying antirheumatic drugs (DMARDs)
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Galapagos NV

INDUSTRY

Sponsor Role collaborator

Gilead Sciences

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Gilead Study Director

Role: STUDY_DIRECTOR

Gilead Sciences

Locations

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Huntsville, Alabama, United States

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Phoenix, Arizona, United States

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Tucson, Arizona, United States

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Covina, California, United States

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Los Angeles, California, United States

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Palm Desert, California, United States

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Victorville, California, United States

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Whittier, California, United States

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DeBary, Florida, United States

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Jacksonville, Florida, United States

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Miami, Florida, United States

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Orlando, Florida, United States

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Plantation, Florida, United States

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Springfield, Illinois, United States

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Wichita, Kansas, United States

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Elizabethtown, Kentucky, United States

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Cumberland, Maryland, United States

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Wheaton, Maryland, United States

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Worcester, Massachusetts, United States

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Saint Clair Shores, Michigan, United States

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Eagan, Minnesota, United States

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Hattiesburg, Mississippi, United States

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Tupelo, Mississippi, United States

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St Louis, Missouri, United States

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Lincoln, Nebraska, United States

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Lebanon, New Hampshire, United States

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Freehold, New Jersey, United States

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Toms River, New Jersey, United States

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Albuquerque, New Mexico, United States

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Charlotte, North Carolina, United States

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Oklahoma City, Oklahoma, United States

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Tulsa, Oklahoma, United States

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Bethlehem, Pennsylvania, United States

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Duncansville, Pennsylvania, United States

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Wyomissing, Pennsylvania, United States

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Charleston, South Carolina, United States

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Orangeburg, South Carolina, United States

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Memphis, Tennessee, United States

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Beaumont, Texas, United States

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Carrollton, Texas, United States

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Corpus Christi, Texas, United States

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Mesquite, Texas, United States

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Plano, Texas, United States

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San Antonio, Texas, United States

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Webster, Texas, United States

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Buenos Aires, , Argentina

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Caba, , Argentina

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Mendoza, , Argentina

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Quilmes, , Argentina

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San Fernando, , Argentina

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San Juan, , Argentina

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San Miguel de Tucumán, , Argentina

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Maroochydore, Queensland, Australia

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Hobart, Tasmania, Australia

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Victoria Park, Western Australia, Australia

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Leuven, Flemish Brabant, Belgium

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Genk, , Belgium

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Hasselt, , Belgium

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Merksem, , Belgium

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Dobrich, , Bulgaria

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Haskovo, , Bulgaria

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Plovdiv, , Bulgaria

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Sofia, , Bulgaria

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Varna, , Bulgaria

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Vidin, , Bulgaria

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Barrie, Ontario, Canada

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Trois-Rivières, Quebec, Canada

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Santiago, , Chile

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Temuco, , Chile

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Ostrava, , Czechia

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Prague, , Czechia

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Uherské Hradiště, , Czechia

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Aachen, , Germany

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Hamburg, , Germany

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Ratingen, , Germany

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Hong Kong, , Hong Kong

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Tuenmen, , Hong Kong

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Kalocsa, Bács-Kiskun county, Hungary

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Székesfehérvár, Fejér, Hungary

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Budapest, , Hungary

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Kistarcsa, , Hungary

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Ahmedabad, , India

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Bangalore, , India

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Delhi, , India

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Jaipur, , India

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Kolkata, , India

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Lucknow, , India

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Mangalore, , India

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Mysuru, , India

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Nagpur, , India

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New Delhi, , India

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Pune, , India

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Secunderabad, , India

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Srikakulam, , India

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Surat, , India

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Vadodara, , India

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Visakhapatnam, , India

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Dublin, , Ireland

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Petah Tikva, , Israel

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Bologna, , Italy

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Reggio Emilia, , Italy

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Fukuoka, , Japan

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Hamamatsu, , Japan

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Hiroshima, , Japan

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Kagoshima, , Japan

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Katō, , Japan

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Kawagoe, , Japan

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Miyagi, , Japan

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Nagaoka, , Japan

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Nagasaki, , Japan

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Okayama, , Japan

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Ōme, , Japan

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Sanuki, , Japan

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Sapporo, , Japan

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Sasebo, , Japan

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Sayama, , Japan

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Tokyo, , Japan

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Batu Caves, , Malaysia

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Kuala Lumpur, , Malaysia

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Mérida, Yucatán, Mexico

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Chihuahua City, , Mexico

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Distrito Federal, , Mexico

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Mérida, , Mexico

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Monterrey, , Mexico

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Morelia, , Mexico

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Timaru, Canterbury, New Zealand

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Hamilton, , New Zealand

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Newtown, , New Zealand

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Papatoetoe, , New Zealand

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Bialystok, , Poland

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Bydgoszcz, , Poland

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Bytom, , Poland

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Dąbrówka, , Poland

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Elblag, , Poland

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Gdynia, , Poland

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Katowice, , Poland

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Krakow, , Poland

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Nowa Sól, , Poland

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Poznan, , Poland

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Torun, , Poland

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Warsaw, , Poland

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Târgu Mureş, Mureș County, Romania

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Bucharest, , Romania

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Oradea, , Romania

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Barnaul, , Russia

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Kemerovo, , Russia

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Moscow, , Russia

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Nizhny Novgorod, , Russia

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Saratov, , Russia

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Yaroslavl, , Russia

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Belgrade, , Serbia

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Bratislava, , Slovakia

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Prievidza, , Slovakia

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Topoľčany, , Slovakia

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Cape Town, , South Africa

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Durban, , South Africa

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Anyang-si, , South Korea

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Daegu, , South Korea

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Daejeon, , South Korea

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Incheon, , South Korea

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Seoul, , South Korea

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Sabadell, Barcelona, Spain

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A Coruña, , Spain

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Barakaldo, , Spain

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Málaga, , Spain

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Sabadell, , Spain

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Santiago de Compostela, , Spain

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Valencia, , Spain

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Kaohsiung City, , Taiwan

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Taichung, , Taiwan

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Tainan City, , Taiwan

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Taipei, , Taiwan

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Taoyuan District, , Taiwan

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Bangkok, , Thailand

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Chiang Mai, , Thailand

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Songkhla, , Thailand

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Dnipro, , Ukraine

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Kharkiv, , Ukraine

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Kherson, , Ukraine

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Kyiv, , Ukraine

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Lviv, , Ukraine

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Vinnitsa, , Ukraine

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Vinnytsia, , Ukraine

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Zaporizhzhya, , Ukraine

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Edinburgh, , United Kingdom

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Newcastle upon Tyne, , United Kingdom

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Countries

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United States Argentina Australia Belgium Bulgaria Canada Chile Czechia Germany Hong Kong Hungary India Ireland Israel Italy Japan Malaysia Mexico New Zealand Poland Romania Russia Serbia Slovakia South Africa South Korea Spain Taiwan Thailand Ukraine United Kingdom

References

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Westhovens R, Rigby W, van der Heijde D, Ching D, Bartok B, Matzkies F, et al. Efficacy and safety of filgotinib for patients with rheumatoid arthritis naive to methotrexate therapy: FINCH 3 primary outcome results. Ann Rheum Dis 2019; 78 (supplement 2): A259.

Reference Type RESULT

Taylor PC, Downie B, Han L, Hawtin R, Hertz A, Moots RJ, Takeuchi T. Patients with High Baseline Neutrophil-to-Lymphocyte Ratio Exhibit Better Response to Filgotinib as Treatment for Rheumatoid Arthritis. Rheumatol Ther. 2024 Oct;11(5):1383-1392. doi: 10.1007/s40744-024-00695-w. Epub 2024 Jul 10.

Reference Type DERIVED
PMID: 38985247 (View on PubMed)

Curtis JR, Emery P, Downie B, Zhong Y, Liu J, Han L, Hawtin RE, Burmester GR. Filgotinib Demonstrates Efficacy in Rheumatoid Arthritis Independent of Smoking Status: Post Hoc Analysis of Phase 3 Trials and Claims-Based Analysis. Rheumatol Ther. 2024 Feb;11(1):177-189. doi: 10.1007/s40744-023-00619-0. Epub 2023 Dec 6.

Reference Type DERIVED
PMID: 38057656 (View on PubMed)

Balsa A, Wassenberg S, Tanaka Y, Tournadre A, Orzechowski HD, Rajendran V, Lendl U, Stiers PJ, Watson C, Caporali R, Galloway J, Verschueren P. Effect of Filgotinib on Body Mass Index (BMI) and Effect of Baseline BMI on the Efficacy and Safety of Filgotinib in Rheumatoid Arthritis. Rheumatol Ther. 2023 Dec;10(6):1555-1574. doi: 10.1007/s40744-023-00599-1. Epub 2023 Sep 25.

Reference Type DERIVED
PMID: 37747626 (View on PubMed)

Tanaka Y, Atsumi T, Aletaha D, Bartok B, Pechonkina A, Han L, Emoto K, Kano S, Rajendran V, Takeuchi T. Benefit of Filgotinib, a JAK1 Preferential Inhibitor, in Rheumatoid Arthritis Patients with Previous Rapid Radiographic Progression: Post Hoc Analysis of Two Trials. Rheumatol Ther. 2023 Feb;10(1):161-185. doi: 10.1007/s40744-022-00503-3. Epub 2022 Nov 3.

Reference Type DERIVED
PMID: 36327094 (View on PubMed)

Combe B, Besuyen R, Gomez-Centeno A, Matsubara T, Sancho Jimenez JJ, Yin Z, Buch MH. Geographic Analysis of the Safety and Efficacy of Filgotinib in Rheumatoid Arthritis. Rheumatol Ther. 2023 Feb;10(1):35-51. doi: 10.1007/s40744-022-00494-1. Epub 2022 Oct 7.

Reference Type DERIVED
PMID: 36205910 (View on PubMed)

Bingham CO 3rd, Walker D, Nash P, Lee SJ, Ye L, Hu H, Khalid JM, Combe B. The impact of filgotinib on patient-reported outcomes and health-related quality of life for patients with active rheumatoid arthritis: a post hoc analysis of Phase 3 studies. Arthritis Res Ther. 2022 Jan 3;24(1):11. doi: 10.1186/s13075-021-02677-7.

Reference Type DERIVED
PMID: 34980223 (View on PubMed)

Aletaha D, Westhovens R, Gaujoux-Viala C, Adami G, Matsumoto A, Bird P, Messina OD, Buch MH, Bartok B, Yin Z, Guo Y, Hendrikx T, Burmester GR. Efficacy and safety of filgotinib in methotrexate-naive patients with rheumatoid arthritis with poor prognostic factors: post hoc analysis of FINCH 3. RMD Open. 2021 Aug;7(2):e001621. doi: 10.1136/rmdopen-2021-001621.

Reference Type DERIVED
PMID: 34385364 (View on PubMed)

Westhovens R, Rigby WFC, van der Heijde D, Ching DWT, Stohl W, Kay J, Chopra A, Bartok B, Matzkies F, Yin Z, Guo Y, Tasset C, Sundy JS, Jahreis A, Mozaffarian N, Messina OD, Landewe RB, Atsumi T, Burmester GR. Filgotinib in combination with methotrexate or as monotherapy versus methotrexate monotherapy in patients with active rheumatoid arthritis and limited or no prior exposure to methotrexate: the phase 3, randomised controlled FINCH 3 trial. Ann Rheum Dis. 2021 Jun;80(6):727-738. doi: 10.1136/annrheumdis-2020-219213. Epub 2021 Jan 15.

Reference Type DERIVED
PMID: 33452004 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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2016-000570-37

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

GS-US-417-0303

Identifier Type: -

Identifier Source: org_study_id

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