CKD-391 DDI : Atorvastatin and Ezetimibe in Healthy Volunteers

NCT ID: NCT02288338

Last Updated: 2015-03-10

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

36 participants

Study Classification

INTERVENTIONAL

Study Start Date

2014-11-30

Study Completion Date

2015-02-28

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

A randomized open-label, multiple dose, three-treatment, three-period, six-sequence, crossover study to investigate the pharmacokinetic drug interaction between Atorvastatin and Ezetimibe after oral administration in healthy volunteers

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Outcome Measures

1. Primary endpoint AUCτ,ss, Cmax,ss of atorvastatin and free ezetimibe
2. Second endpoint 1) AUCinf,ss, Cavg,ss, %fluctuation, tmax,ss, t1/2, CL/Fss, Vd/Fss of atorvastatin and free ezetimibe 2) AUCτ,ss, AUCinf,ss, Cmax,ss, tmax,ss, t1/2, metabolic ratio of 2-hydroxy atorvastatin and free ezetimibe

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Healthy

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

1(Lipitor®>Ezetrol®>Lipitor®, Ezetrol®)

Three treatment

1. atorvastatin calcium 40mg will be administration to healthy volunteers during 7days
2. after 11days withdrawal period, ezetimibe 10mg will be administered to healthy volunteers during 7days
3. after 11days withdrawal period, atorvastatin calcium 40mg and ezetimibe 10mg will be administered to healthy volunteers during 7days

Group Type EXPERIMENTAL

1 (Lipitor®)

Intervention Type DRUG

atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

1 (Ezetrol®)

Intervention Type DRUG

After 11days withdrawal period, ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

1 (Lipitor®, Ezetrol®)

Intervention Type DRUG

After 11days withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

2(Ezetrol®>Lipitor®, Ezetrol®>Lipitor®)

Three treatment

1. ezetimibe 10mg will be administered to healthy volunteers during 7days
2. after 11days withdrawal period, atorvastatin calcium 40mg and ezetimibe 10mg will be administered to healthy volunteers during 7days
3. after 11days withdrawal period, atorvastatin calcium 40mg will be administered to healthy volunteers during 7days

Group Type EXPERIMENTAL

2 (Ezetrol®)

Intervention Type DRUG

ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

2(Lipitor®, Ezetrol®)

Intervention Type DRUG

After 11days withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

2 (Lipitor®)

Intervention Type DRUG

After 11day withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

3(Lipitor®, Ezetrol®>Lipitor®>Ezetrol®)

Three treatment

1. atorvastatin calcium 40mg and ezetimibe 10mg will be administered to healthy volunteers during 7days
2. after 11days withdrawal period, atorvastatin calcium 40mg will be administered to healthy volunteers during 7days
3. after 11days withdrawal period, ezetimibe 10mg will be administered to healthy volunteers during 7days

Group Type EXPERIMENTAL

3(Lipitor®, Ezetrol®)

Intervention Type DRUG

atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

3 (Lipitor®)

Intervention Type DRUG

After 11day withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

3 (Ezetrol®)

Intervention Type DRUG

After 11day withdrawal period, ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

4(Lipitor®>Lipitor®, Ezetrol®>Ezetrol®)

1. atorvastatin calcium 40mg will be administered to healthy volunteers during 7days
2. after 11days withdrawal period, atorvastatin calcium 40mg and ezetimibe 10mg will be administered to healthy volunteers during 7days
3. after 11days withdrawal period, ezetimibe 10mg will be administered to healthy volunteers during 7days

Group Type EXPERIMENTAL

4 (Lipitor®)

Intervention Type DRUG

atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

4(Lipitor®, Ezetrol®)

Intervention Type DRUG

After 11days withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

4 (Ezetrol®)

Intervention Type DRUG

After 11day withdrawal period, ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

5(Ezetrol®>Lipitor®>Lipitor®, Ezetrol®)

1. ezetimibe 10mg will be administered to healthy volunteers during 7days
2. after 11days withdrawal period, atorvastatin calcium 40mg will be administered to healthy volunteers during 7days
3. after 11days withdrawal period, atorvastatin calcium 40mg and ezetimibe 10mg will be administered to healthy volunteers during 7days

Group Type EXPERIMENTAL

5 (Ezetrol®)

Intervention Type DRUG

ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

5 (Lipitor®)

Intervention Type DRUG

After 11day withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

5 (Lipitor®, Ezetrol®)

Intervention Type DRUG

After 11days withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

6(Lipitor®, Ezetrol®>Ezetrol®>Lipitor®)

1. atorvastatin calcium 40mg and ezetimibe 10mg will be administered to healthy volunteers during 7days
2. after 11days withdrawal period, ezetimibe 10mg will be administered to healthy volunteers during 7days
3. after 11days withdrawal period, atorvastatin calcium 40mg will be administered to healthy volunteers during 7days

Group Type EXPERIMENTAL

6(Lipitor®, Ezetrol®)

Intervention Type DRUG

atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

6 (Ezetrol®)

Intervention Type DRUG

After 11days withdrawal period, ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

6 (Lipitor®)

Intervention Type DRUG

After 11day withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

1 (Lipitor®)

atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

1 (Ezetrol®)

After 11days withdrawal period, ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

1 (Lipitor®, Ezetrol®)

After 11days withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

2 (Ezetrol®)

ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

2(Lipitor®, Ezetrol®)

After 11days withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

2 (Lipitor®)

After 11day withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

3(Lipitor®, Ezetrol®)

atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

3 (Lipitor®)

After 11day withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

3 (Ezetrol®)

After 11day withdrawal period, ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

4 (Lipitor®)

atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

4(Lipitor®, Ezetrol®)

After 11days withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

4 (Ezetrol®)

After 11day withdrawal period, ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

5 (Ezetrol®)

ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

5 (Lipitor®)

After 11day withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

5 (Lipitor®, Ezetrol®)

After 11days withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

6(Lipitor®, Ezetrol®)

atorvastatin calcium 40mg, Lipitor® 40mg and ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

6 (Ezetrol®)

After 11days withdrawal period, ezetimibe 10mg, Ezetrol® 10mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

6 (Lipitor®)

After 11day withdrawal period, atorvastatin calcium 40mg, Lipitor® 40mg will be administered to healthy volunteers during 7days

Intervention Type DRUG

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

Lipitor® 40mg Ezetrol® 10mg Lipitor® 40mg, Ezetrol® 10mg Ezetrol® 10mg Lipitor® 40mg, Ezetrol® 10mg Lipitor® 40mg Lipitor® 40mg, Ezetrol® 10mg Lipitor® 40mg Ezetrol® 10mg Lipitor® 40mg Lipitor® 40mg, Ezetrol® 10mg Ezetrol® 10mg Ezetrol® 10mg Lipitor® 40mg Lipitor® 40mg, Ezetrol® 10mg Lipitor® 40mg, Ezetrol® 10mg Ezetrol® 10mg Lipitor® 40mg

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

1. Age Eligible for Study : 19 Years to 45 Years
2. If males, Body weight ≥ 55kg, If females, Body weight ≥ 50kg
3. BSA ≥ 18.5, \<25
4. Accepts healthy volunteers
5. If female, Negative for pregnancy test at the screening and pre dose of Day 1
6. The subjects who agree with performing contraception during the study
7. The subjects who agreed with written informed consent

Exclusion Criteria

1. The subjects with impaired hepatic function, renal function, nervous system etc.
2. The subjects have a gastrointestinal disease or surgery which can be effected in absorption of Investigational product
3. The subjects with high blood pressure or low blood pressure (Systolic blood pressure\>150mmHg or \<90mmHg, Diastolic blood pressure\>100mmHg or \<50mmHg
4. The subjects with abnormal Laboratory test (AST, ALT\>1.25 fold of upper normal limit, Total bilirubin\>1.5 fold of upper normal limit, CPK\>2 fold of upper normal limit, Estimated Glomerular filtration rate\<60mL/min/1.73m2 by Modification of Diet in Renal disease formula
5. The subjects have drug abuse history within 1year or Positive for urine drug test at screening
6. The subjects who took prescription only medicine whch can be effected in metabolism of Investigational product within 14days
7. The subjects who took over the counter drug whch can be effected in metabolism of Investigational product within 7days
Minimum Eligible Age

19 Years

Maximum Eligible Age

45 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Chong Kun Dang Pharmaceutical

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Min Soo Park, Ph.D. M.D

Role: PRINCIPAL_INVESTIGATOR

Severance Hospital

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

ChongKunDang

Seoul, , South Korea

Site Status

Countries

Review the countries where the study has at least one active or historical site.

South Korea

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

152DDI14016

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.

CKD-337(2) Drug-drug Interaction Study
NCT02422030 COMPLETED PHASE1
CKD-337 Drug Interaction Study
NCT02066207 COMPLETED PHASE1
Multiple Ascending Dose and DDI Study
NCT03031119 COMPLETED PHASE1
Teneligliptin and Atorvastatin DDI Study
NCT03769870 COMPLETED PHASE1