BI 695501 Compared to Adalimumab in Patients With Active Rheumatoid Arthritis

NCT ID: NCT02137226

Last Updated: 2018-01-19

Study Results

Results available

Outcome measurements, participant flow, baseline characteristics, and adverse events have been published for this study.

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

645 participants

Study Classification

INTERVENTIONAL

Study Start Date

2015-01-26

Study Completion Date

2016-10-18

Brief Summary

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Primary Objective:

The primary objective of this trial is to establish an equivalence in efficacy between BI 695501 and US-licensed Humira® in patients with active Rheumatoid arthritis based on a statistical comparison of the proportion of patients meeting American College of Rheumatology 20% (ACR20) response rate at Week 12 and ACR20 response rate at Week 24 between BI 695501 and US-licensed Humira®.

Secondary Objectives:

The secondary objectives of this trial are to compare the efficacy, safety and immunogenicity of BI 695501 and US-licensed Humira® in patients with active RA including those undergoing the transition from US-licensed Humira® to BI 695501 after 24 weeks.

Detailed Description

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Conditions

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Arthritis, Rheumatoid

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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BI 695501

one injection every 2 weeks for 48 weeks (25 injections in total)

Group Type EXPERIMENTAL

BI 695501

Intervention Type DRUG

BI 695501, every two weeks for 48 weeks (25 injections in total)

US-licensed Humira®

one injection every 2 weeks for 48 weeks (25 injections in total)

Group Type ACTIVE_COMPARATOR

US-licensed Humira®

Intervention Type DRUG

one injection every 2 weeks for 48 weeks (25 injections in total)

Interventions

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BI 695501

BI 695501, every two weeks for 48 weeks (25 injections in total)

Intervention Type DRUG

US-licensed Humira®

one injection every 2 weeks for 48 weeks (25 injections in total)

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* All patients must sign and date an Informed Consent Form consistent with International Conference on Harmonisation Good Clinical Practice (ICH GCP) guidelines and local legislation prior to participation in the trial (i.e. prior to any trial procedures, which include medication washout and restrictions) and be willing to follow the protocol.
* Male or female participants, between 18 and 80 years of age, who have a diagnosis of moderately to severely active Rheumatoid arthritis for at least 6 months as defined by at least six swollen joints (66 joint count) and at least six tender joints (68 joint count) at Screening and Baseline (Day 1), and either an Erythrocyte sedimentation rate of \>28 mm/hour OR a C-reactive protein (CRP) level \>1.0 mg/dL (normal: \<0.4 mg/dL) at Screening. Patients must currently be receiving methotrexate (MTX) therapy.
* Current treatment for Rheumatoid arthritis on an outpatient basis:

1. Must be receiving and tolerating oral or parenteral MTX therapy at a dose of 15 to 25 mg per week (dose may be as low as 10 mg per week if the patient is unable to tolerate a higher dose) for at least 12 weeks immediately prior to Day 1. The dose and administration route should remain stable for at least 4 weeks prior to Day 1 until Week 24. After Week 24 the administration route can be changed at the investigator's discretion. Patients receiving a lower dose of MTX (10 to 14 mg/week) should be doing so as a result of a documented history of intolerance to higher doses of MTX.
2. Patients must be willing to receive oral folic acid (at least 5 mg/week or as per local practice) or folinic acid (at least 1 mg/week or as per local practice) or equivalent during the entire trial (mandatory comedication for MTX treatment).
3. Disease modifying antirheumatic drug (DMARD) use will be restricted according to guidelines listed in the trial protocol.
4. If receiving current treatment with oral corticosteroids (other than intra-articular or parenteral), the dose must not exceed 10 mg/day prednisolone or equivalent. During the 4 weeks prior to Baseline (Day 1) the dose must remain stable.
5. Any concomitant non-steroidal anti-inflammatory drugs (NSAIDs) must be stable for at least 2 weeks prior to Day 1.
6. Patients may be taking oral hydroxychloroquine provided that the dose is not greater than 400 mg/day or chloroquine provided that the dose is not greater than 250 mg/day. These doses must have been stable for a minimum of 12 weeks prior to Day 1. The hydroxychloroquine or chloroquine treatment will need to be continued at a stable dose with the same formulation until the end of the trial.
* For participants of reproductive potential (males and females), a reliable means of contraception has to be used throughout trial participation(acceptable methods of birth control include for example birth control pills, intrauterine devices \[IUDs\], surgical sterilization, vasectomized partner and double barrier method.. All patients (males and females of child-bearing potential) must also agree to use an acceptable method of contraception for 6 months following completion or discontinuation from the trial medication.

Exclusion Criteria

* ACR functional Class IV or wheelchair/bed bound.
* Primary or secondary immunodeficiency, including known history of HIV infection, or a positive test at Screening.
* History of Tuberculosis, latent Tuberculosis, or positive purified protein derivative test or interferon gamma-releasing assay .
* Known clinically significant coronary artery disease or significant cardiac arrhythmias or severe congestive heart failure, or interstitial lung disease.
* Previous treatment with \>=2 biologic agents.
* Previous treatment with adalimumab or adalimumab biosimilar.
* Current treatment or previous treatment with leflunomide within 8 weeks.
* History of a severe allergic reaction or anaphylactic reaction to a biological agent or history of hypersensitivity to adalimumab or any component of the trial drug.
* History of cancer including solid tumors, hematologic malignancies, and carcinoma in situ.
* Has evidence of positive serology for Hepatitis B virus or Hepatitis C virus
* Receipt of a live/attenuated vaccine within 12 weeks prior to the Screening Visit. Patients who are expecting to receive any live virus or bacterial vaccinations during the trial, or up to 3 months after the last dose of trial drug.
* Any treatment that, in the opinion of the investigator, may place the patient at unacceptable risk during the trial.
* Patients with a significant disease other than Rheumatoid arthritis and/or a significant uncontrolled disease (such as, but not limited to, nervous system, renal, hepatic, endocrine, or gastrointestinal disorders). A significant disease is defined as a disease which, in the opinion of the investigator, may (i) put the patient at risk because of participation in the trial, or (ii) influence the results of the trial, or (iii) cause concern regarding the patient's ability to participate in the trial.
* Premenopausal, sexually active women who are pregnant or nursing, or are of child-bearing potential and not practicing an acceptable method of birth control, or do not plan to continue practicing an acceptable method of birth control throughout the trial.
* History of, or current, inflammatory joint disease other than Rheumatoid arthritis or other systemic autoimmune disorder.
* Diagnosis of juvenile idiopathic arthritis, and/or Rheumatoid arthritis before age 16.
* Any planned surgical procedure within 12 weeks prior to the Screening Visit or for the duration of the trial.
* Known active infection of any kind (excluding fungal infections of nail beds), or any major episode of infection requiring hospitalization or treatment with intravenous anti infectives within 4 weeks of the Screening Visit or completion of oral anti-infectives within 2 weeks of the Screening Visit.
* History of deep space/tissue infection within 52 weeks of the Screening Visit.
* History of serious infection or opportunistic infection in the last 2 years.
* Any neurological, vascular or systemic disorder that might affect any of the efficacy assessments.
* Currently active alcohol or drug abuse or history of alcohol or drug abuse within 2 years of the Screening Visit.
* Treatment with intravenous Gamma Globulin or the Prosorba® Column within 6 months of the Screening Visit.
* Treatment with intravenous, intramuscular, intra-articular and parenteral corticosteroids within 6 weeks prior to Day 1 or throughout the trial.
* Aspartate aminotransferase (AST) or alanine aminotransferase (ALT) \>1.5 times upper limit of normal.
* Hemoglobin \<8.0 g/dL.
* Platelets \<100,000/µL.
* Leukocyte count \<4000/µL.
* Creatinine clearance \<60 mL/min.
* Patients who are currently participating in another clinical trial or who have been participating in another clinical trial with another investigational drug within a minimum of 12 weeks or five half-lives (whichever is longer) of the drug prior to Day 1.
* Patients with a history of any clinically significant adverse reaction to murine or chimeric proteins.
Minimum Eligible Age

18 Years

Maximum Eligible Age

80 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Boehringer Ingelheim

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Boehringer Ingelheim

Role: STUDY_CHAIR

Boehringer Ingelheim

Locations

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Pinnacle Research Group, LLC

Anniston, Alabama, United States

Site Status

Rheumatology Associates

Birmingham, Alabama, United States

Site Status

Achieve Clinical Research, LLC

Birmingham, Alabama, United States

Site Status

Arizona Arthritis and Rheumatology Research, PLLC

Glendale, Arizona, United States

Site Status

Arizona Arthritis and Rheumatology Research, PLLC

Mesa, Arizona, United States

Site Status

Arizona Arthritis and Rheumatology Research, PLLC

Phoenix, Arizona, United States

Site Status

Arizona Arthritis and Rheumatology Research, PLLC

Phoenix, Arizona, United States

Site Status

TriWest Research Associates, LLC

El Cajon, California, United States

Site Status

Advanced Medical Research, LLC

La Palma, California, United States

Site Status

ProHealth Partners

Long Beach, California, United States

Site Status

The Permanente Medical Group

Santa Clara, California, United States

Site Status

Inland Rheumatology Clinical Trials, Inc.

Upland, California, United States

Site Status

Medvin Clinical Research

Whittier, California, United States

Site Status

Alpine Clinical Research Center

Boulder, Colorado, United States

Site Status

Orthopedic Research Institute

Boynton Beach, Florida, United States

Site Status

Clinical Research of West Florida, Inc.

Clearwater, Florida, United States

Site Status

Universal Clinical Research

Coral Gables, Florida, United States

Site Status

Science and Research Institute, Inc.

Jupiter, Florida, United States

Site Status

San Marcus Research Clinic, Inc.

Miami, Florida, United States

Site Status

L&amp;amp;C Professional Medical Research Institute

Miami, Florida, United States

Site Status

Family Clinical Trials, Incorporated

Pembroke Pines, Florida, United States

Site Status

Physician Research Collaboration

South Miami, Florida, United States

Site Status

West Broward Rheumatology Associates, Incorporated

Tamarac, Florida, United States

Site Status

Clinical Research of West Florida, Inc.

Tampa, Florida, United States

Site Status

McIlwain Medical Group, PA

Tampa, Florida, United States

Site Status

Lovelace Scientific Resources, Incorporated

Venice, Florida, United States

Site Status

Institute of Arthritis Research

Idaho Falls, Idaho, United States

Site Status

Goldpoint Clinical Research, LLC

Indianapolis, Indiana, United States

Site Status

Heartland Research Associates, LLC

Wichita, Kansas, United States

Site Status

The Arthritis &amp;amp; Diabetes Clinic, Incorporated

Monroe, Louisiana, United States

Site Status

Klein and Associates, M.D., P.A.

Cumberland, Maryland, United States

Site Status

Clinical Pharmacology Study Group

Worcester, Massachusetts, United States

Site Status

Henry Ford Health System

Detroit, Michigan, United States

Site Status

Arthritis Education and Treatment Center

Grand Rapids, Michigan, United States

Site Status

North MS Medical Clinics, Incorporated

Tupelo, Mississippi, United States

Site Status

Glacier View Research Institute

Kalispell, Montana, United States

Site Status

Accurate Clinical Research, Inc.

Lincoln, Nebraska, United States

Site Status

NJP Clinical Research

Clifton, New Jersey, United States

Site Status

Albuquerque Center For Rheumatology

Albuquerque, New Mexico, United States

Site Status

Anna Imperato, MD PLLC

Manhasset, New York, United States

Site Status

Box Arthritis &amp;amp; Rheumatology of the Carolinas

Charlotte, North Carolina, United States

Site Status

Medication Management, LLC

Greensboro, North Carolina, United States

Site Status

PMG Research of Salisbury, LLC

Salisbury, North Carolina, United States

Site Status

Wake Forest University School of Medicine

Winston-Salem, North Carolina, United States

Site Status

STAT Research, Incorporated

Dayton, Ohio, United States

Site Status

Clinical Research Source, Inc.

Perrysburg, Ohio, United States

Site Status

Altoona Center for Clinical Research, P.C.

Duncansville, Pennsylvania, United States

Site Status

Mountain View Clinical Research

Greer, South Carolina, United States

Site Status

Center for Inflammatory Disease

Nashville, Tennessee, United States

Site Status

Austin Regional Clinic

Austin, Texas, United States

Site Status

Adriana Pop Moody Clinic PA

Corpus Christi, Texas, United States

Site Status

Metroplex Clinical Research Center

Dallas, Texas, United States

Site Status

Accurate Clinical Management LLC

Houston, Texas, United States

Site Status

Pioneer Research Solutions, Inc.

Houston, Texas, United States

Site Status

Accurate Clinical Research, Incorporated

Houston, Texas, United States

Site Status

Rheumatology Clinic Of Houston, P.A.

Houston, Texas, United States

Site Status

Accurate Clinical Research, Incorporated

Houston, Texas, United States

Site Status

Houston Rheumatology Consultants, PLLC

Houston, Texas, United States

Site Status

Arthritis &amp;amp; Osteoporosis Associates LLP

Lubbock, Texas, United States

Site Status

Accurate Clinical Research, Incorporated

Nassau Bay, Texas, United States

Site Status

Heartland Research Associates, LLC

San Antonio, Texas, United States

Site Status

Danville Orthopedic Clinic, Incorporated

Danville, Virginia, United States

Site Status

Arthritis Northwest, PLLC

Spokane, Washington, United States

Site Status

MHAT &quot;Trimontium&quot;, OOD, Plovdiv

Plovdiv, , Bulgaria

Site Status

MHAT &quot;Eurohospital&quot; - Plovdiv, OOD

Plovdiv, , Bulgaria

Site Status

MHAT - Kaspela, EOOD

Plovdiv, , Bulgaria

Site Status

Medical Center &quot;Teodora&quot;, EOOD, Ruse

Rousse, , Bulgaria

Site Status

MHAT,Fourth Dept. of Therapeutics & Cardiology, Ruse

Rousse, , Bulgaria

Site Status

MHAT Shumen AD, Shumen

Shumen, , Bulgaria

Site Status

MHAT Lyulin

Sofia, , Bulgaria

Site Status

DCC 17 - Sofia EOOD

Sofia, , Bulgaria

Site Status

MMA HAT Sofia, Bulgaria

Sofia, , Bulgaria

Site Status

UMHAT Sv. Ivan Rilski EAD

Sofia, , Bulgaria

Site Status

DCC 'Chaika', EOOD, Varna

Varna, , Bulgaria

Site Status

MDHAT 'Dr. Stefan Cherkezov', AD

Veliko Tarnovo, , Bulgaria

Site Status

Corporacion de Beneficencia Osorno

Osorno, , Chile

Site Status

Quantum Research Santiago, Puerto Varas

Puerto Varas, , Chile

Site Status

BIOMEDICA, Santiago

Santiago, , Chile

Site Status

Centro de Estudios Reumatológicos

Santiago, , Chile

Site Status

Centro Medico Prosalud

Santiago, , Chile

Site Status

CINVEC - Centro de Investigacion Clinica V Reg.,Vina del Mar

Viña del Mar, , Chile

Site Status

Pärnu Hospital, Pärnu

Pärnu, , Estonia

Site Status

Medita Kliinik OÜ, Tartu

Tartu, , Estonia

Site Status

Rheumazentrum Prof. Dr. G. Neeck, Bad Doberan

Bad Doberan, , Germany

Site Status

ACURA Kliniken Rheinland-Pfalz AG, Bad Kreuznach

Bad Kreuznach, , Germany

Site Status

Kerckhoff-Klinik, Bad Nauheim

Bad Nauheim, , Germany

Site Status

SMO.MD GmbH, Magdeburg

Magdeburg, , Germany

Site Status

Szegedi Tudomanyegyetem Szent-Gyorgyi Albert Klin. Kozpont

Szeged, , Hungary

Site Status

Csolnoky Ferenc Korhaz, Veszprem

Veszprém, , Hungary

Site Status

Hospital Tengku Ampuan Afzan

Kuantan, , Malaysia

Site Status

Hospital Pulau Pinang

Pulau Pinang, , Malaysia

Site Status

CGM Research Trust, The Princess Margaret Hospital Cantebury

Cantebury, , New Zealand

Site Status

Gabinet Internistyczno-Reumatologiczny Piotr Adrian Klimiuk

Bialystok, , Poland

Site Status

Szpital Uniwersytecki nr 2 im.dr J. Biziela

Bydgoszcz, , Poland

Site Status

Wojewodzki Szpital Zespolony w Elblagu

Elblag, , Poland

Site Status

Medica Pro Familia Spolka Akcyjna, Oddzial w Gdyni

Gdynia, , Poland

Site Status

MCBK Iwona Czajkowska Anna Podrazka- Szczepaniak S.C.

Grodzisk Mazowiecki, , Poland

Site Status

Medical Centre Pratia Katowice I

Katowice, , Poland

Site Status

Medical Centre Pratia Krakow

Krakow, , Poland

Site Status

Specialist Center ALL-MED, Krakow

Krakow, , Poland

Site Status

Niepubliczny ZOZ, &quot;Nasz Lekarz&quot;, Lekarzy Rodzinnych z

Torun, , Poland

Site Status

Medical Centre Pratia Warszawa

Warsaw, , Poland

Site Status

Reumatika, Rheumatology Center, non-public outpatient clinic

Warsaw, , Poland

Site Status

Wojewodzki Szpital Specjalistyczny we Wroclawiu

Wroclaw, , Poland

Site Status

Kemerovo SMA b/o War Veterans Regional Clinical Hospital

Kemerovo, , Russia

Site Status

Practicheskaya Meditsina Ltd

Moscow, , Russia

Site Status

Republic Kareliya Republican Hosp. named after V.A. Baranov

Petrozavodsk, , Russia

Site Status

Samara Regional Clinical Hospital n.a MI Kalinin, Samara

Samara, , Russia

Site Status

Reg. Hospital for war veterans

Saratov, , Russia

Site Status

Stavropol State Medical Academy

Stavropol, , Russia

Site Status

Emergency Clinical Hospital n. a. N. V. Soloviev, Yaroslavl

Yaroslavl, , Russia

Site Status

SBHI of Yaroslavl Area &quot;Clinical Hospital #3&quot;

Yaroslavl, , Russia

Site Status

Institute of Rheumatology, Belgrade

Belgrade, , Serbia

Site Status

Institute for Treatment and Rehabilitation, Niska Banja

Niška Banja, , Serbia

Site Status

Clinical Center of Vojvodina

Novi Sad, , Serbia

Site Status

General Hospital &quot;Dr Laza K. Lazarevic&quot; Sabac, Sabac

Šabac, , Serbia

Site Status

Daegu Catholic University Medical Center

Daegu, , South Korea

Site Status

Chungnam National University Hospital

Daejeon, , South Korea

Site Status

Seoul National University Hospital

Seoul, , South Korea

Site Status

Konkuk University Medical Center

Seoul, , South Korea

Site Status

Hospital A Coruña

A Coruña, , Spain

Site Status

Hospital Universitario de Cruces

Barakaldo, , Spain

Site Status

Fundación Jiménez Díaz

Madrid, , Spain

Site Status

Hosp. Nuestra Señora de la Esperanza, Santiago de Compostela

Santiago de Compostela, , Spain

Site Status

Hospital Clínico de Santiago

Santiago de Compostela, , Spain

Site Status

Siriraj Hospital

Bangkoknoi, , Thailand

Site Status

Songklanagarind Hospital

Hat Yai, , Thailand

Site Status

Pramongkutklao Hospital

Rajathevee, , Thailand

Site Status

Ivano-Frankivsk Nat. Medical University, Dept. Endocrinology

Ivano-Frankivsk, , Ukraine

Site Status

L.T. Malaya Institute of Therapy AMS of Ukraine

Kharkiv, , Ukraine

Site Status

CI of Healthcare Kharkiv CCH #8, Kharkiv

Kharkiv, , Ukraine

Site Status

SI NSC M.D. Strazhesko Institute Cardiology of NAMSU, Kyiv

Kyiv, , Ukraine

Site Status

SI D.F.Chebotariov Institute of Gerontology of NAMSU, Kyiv

Kyiv, , Ukraine

Site Status

Oleksandrivska Clinical Hospital

Kyiv, , Ukraine

Site Status

M.V. Sklifosovskyi Poltava RCH, Poltava

Poltava, , Ukraine

Site Status

M.I. Pyrogov VRCH, Vinnytsia

Vinnytsia, , Ukraine

Site Status

MCIC MC LLC Health Clinic, Vinnytsia

Vinnytsia, , Ukraine

Site Status

Zaporizhzhia Regional Clinical Hospital, Zaporizhzhia

Zaporizhzhia, , Ukraine

Site Status

Countries

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United States Bulgaria Chile Estonia Germany Hungary Malaysia New Zealand Poland Russia Serbia South Korea Spain Thailand Ukraine

References

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Strand V, McCabe D, Bender S. Immunogenicity of adalimumab reference product and adalimumab-adbm in patients with rheumatoid arthritis, Crohn's disease and chronic plaque psoriasis: a pooled analysis of the VOLTAIRE trials. BMJ Open. 2024 Nov 17;14(11):e081687. doi: 10.1136/bmjopen-2023-081687.

Reference Type DERIVED
PMID: 39551590 (View on PubMed)

Strand V, Bender S, McCabe D. Effects of Adalimumab-adbm Versus Adalimumab Reference Product on Patient-Reported Outcomes in Rheumatoid Arthritis: Results from VOLTAIRE-RA. Rheumatol Ther. 2024 Oct;11(5):1291-1302. doi: 10.1007/s40744-024-00687-w. Epub 2024 Aug 9.

Reference Type DERIVED
PMID: 39120847 (View on PubMed)

Cohen SB, Lee EC. Plain language summary of the VOLTAIRE-RA in patients with moderate-to-severe rheumatoid arthritis. Immunotherapy. 2022 Oct;14(15):1183-1190. doi: 10.2217/imt-2022-0106. Epub 2022 Sep 6.

Reference Type DERIVED
PMID: 36065786 (View on PubMed)

Huizinga TWJ, Torii Y, Muniz R. Adalimumab Biosimilars in the Treatment of Rheumatoid Arthritis: A Systematic Review of the Evidence for Biosimilarity. Rheumatol Ther. 2021 Mar;8(1):41-61. doi: 10.1007/s40744-020-00259-8. Epub 2020 Dec 1.

Reference Type DERIVED
PMID: 33263165 (View on PubMed)

Kang J, Eudy-Byrne RJ, Mondick J, Knebel W, Jayadeva G, Liesenfeld KH. Population pharmacokinetics of adalimumab biosimilar adalimumab-adbm and reference product in healthy subjects and patients with rheumatoid arthritis to assess pharmacokinetic similarity. Br J Clin Pharmacol. 2020 Nov;86(11):2274-2285. doi: 10.1111/bcp.14330. Epub 2020 Jun 11.

Reference Type DERIVED
PMID: 32363771 (View on PubMed)

Cohen SB, Alonso-Ruiz A, Klimiuk PA, Lee EC, Peter N, Sonderegger I, Assudani D. Similar efficacy, safety and immunogenicity of adalimumab biosimilar BI 695501 and Humira reference product in patients with moderately to severely active rheumatoid arthritis: results from the phase III randomised VOLTAIRE-RA equivalence study. Ann Rheum Dis. 2018 Jun;77(6):914-921. doi: 10.1136/annrheumdis-2017-212245. Epub 2018 Mar 7.

Reference Type DERIVED
PMID: 29514803 (View on PubMed)

Other Identifiers

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2012-002945-40

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

1297.2

Identifier Type: -

Identifier Source: org_study_id

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