Combination of Baricitinib and Anti-TNF in Rheumatoid Arthritis

NCT ID: NCT04870203

Last Updated: 2025-12-19

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE3

Total Enrollment

178 participants

Study Classification

INTERVENTIONAL

Study Start Date

2021-07-15

Study Completion Date

2027-03-31

Brief Summary

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As stated by the European League Against Rheumatism (EULAR) and the Société Française de Rhumatologie (SFR), treatment of patients with rheumatoid arthritis (RA) should target sustained remission or at least low disease activity. However, despite significant advances based on various combinations of conventional synthetic disease-modifying antirheumatic drugs (DMARDs) and biologic DMARDs, RA therapies meet treatment goals only in some patients:

* 40 to 50% of patients with early RA, treated with methotrexate (MTX) monotherapy as first-line therapy,
* 20 to 30% of patients treated with a combination of MTX and biologic as second-line therapy.
* Less than 10% of patients treated with a combination of MTX and another targeted DMARD, such as baricitinib, as third-line therapy.

Therefore, new strategies targeted at achieving a higher percentage of remission are needed, that do not require waiting for multiple failed therapies. Combinations of biologics have shown synergistic improvement of symptoms in murine models of RA relative to the improvement observed with either agent alone. However, in RA patients, only five randomised clinical trials (RCTs) have explored the efficacy and safety of combining tumour necrosis factor (TNF) inhibitor with another biologic (anakinra, abatacept, rituximab or bimekizumab).

Baricitinib is a selective, reversible and competitive inhibitor of Janus kinases (Jaki). This treatment is efficient in a number of therapeutic scenarios in RA and showed a clinical superiority over adalimumab in one RCT (RA-BEAM study in MTX inadequate responders). Of note, baricitinib inhibits many of the pro-inflammatory cytokines involved in the pathogenesis of RA but does not block signalling downstream of TNF. Owing to the interest in combining different mechanisms of action, the investigators plan to assess the efficacy and safety of combination therapy with baricitinib and a TNF inhibitor. The investigators are aware that combining targeted therapies is not recommended due to a potential increase in the frequency of serious adverse events. However, several case series on patients treated with a combination of targeted therapies have been published, suggesting a certain efficacy in patients with refractory RA. The first ones focused on inflammatory bowel diseases and psoriasis, but more recently, combination of tofacitinib (which belongs to the same Jaki family as baricitinib) with various biologics has been reported in a sample of RA patients. No serious adverse effects were reported over a mean of approximately 11 months of therapy. The clinical improvement was mild but noticeable in these refractory RA cases.

Recently, data of interest from the RA-BEAM study have been reported. Patients who switched from adalimumab to baricitinib showed improvements in disease control. Because the switch from adalimumab to baricitinib occurred without a washout period, and because adalimumab has a mean circulating half-life of approximately 14 days, patients would have received several weeks of dual TNF and Jak1/Jak2 inhibition in the course of the change of treatment. The observation of increased efficacy, with no apparent acute safety issues during the weeks when patients were exposed to both adalimumab and baricitinib, is of interest, and supports our strategy to combine the two treatments for patients with refractory RA.

The investigators consider that there is a need for investigation into the addition of anti-TNF to baricitinib in patients suffering of refractory RA (inadequate response to TNF inhibitors). The investigators hypothesize that in this population, based on ACR50 score, this combination therapy will decrease disease activity more efficiently than a switch to another targeted DMARD, such as baricitinib.

Detailed Description

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Intensive combination therapies have revolutionised the management of solid neoplasms, hematologic malignancies, and acquired-immune-deficiency syndrome. These intensive strategies are based on the need to obtain rapid control of disease activity to afford the chance of stable full remission and avoid irreversible complications. The same goal applies to management of RA. Because current therapeutic strategies may fall short of these target goals and fail to improve quality of life in some patients, novel approaches are needed to improve outcomes. RA is a complex disease involving numerous cell types and inflammatory mediators of innate and adaptive immune systems. The investigators are aware that most of combination bDMARD strategies have been associated with little or no incremental benefit in efficacy compared to single-biologic therapy. However, our study will target mechanisms that differ from those in previous studies. Strategies that simultaneously target different pathways involved in the pathogenesis of RA may enhance treatment responses in patients with RA. Of note, baricitinib does not directly block signalling downstream of TNF, even if an indirect effect on TNF production is likely to occur. Targeting multiple inflammatory cytokines in combination may lead to more effective treatment and enhanced clinical responses in patients with RA compared to the current second-line strategies. The different mechanisms of action of baricitinib and anti-TNF, should ensure the efficacy of the combination. No concurrent trial evaluating similar strategies is registered at ClinicalTrial.gov.

Conditions

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Rheumatoid Arthritis

Keywords

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baricitinib adalimumab etanercept placebo

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Period A : placebo-controlled trial \*\*\* Period B : controlled trial - study switch to an open-label design from the 17th August 2024
Primary Study Purpose

TREATMENT

Blinding Strategy

TRIPLE

Participants Caregivers Investigators
Period A : Participant / Care provider / Investigator \*\*\* Period B : An independent efficacy assessor will perform the joint evaluation, whereas the investigator will evaluate safety.

Study Groups

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Period B : baricitinib + anti-TNF

Group Type EXPERIMENTAL

baricitinib treatment

Intervention Type DRUG

4 mg daily during 12 months

anti-TNF therapy

Intervention Type DRUG

adalimumab at 40 mg every 2 weeks or etanercept 50 mg per week according to treatments history

Period B : baricitinib

Group Type ACTIVE_COMPARATOR

baricitinib treatment

Intervention Type DRUG

4 mg daily during 12 months

Period A : baricitinib + anti-TNF

Group Type EXPERIMENTAL

baricitinib treatment

Intervention Type DRUG

4 mg daily during 12 months

anti-TNF therapy

Intervention Type DRUG

adalimumab at 40 mg every 2 weeks or etanercept 50 mg per week according to treatments history

Period A : baricitinib + placebo

Group Type PLACEBO_COMPARATOR

baricitinib treatment

Intervention Type DRUG

4 mg daily during 12 months

Placebo

Intervention Type DRUG

40 mg every 2 weeks during 6 months only during Period A

Interventions

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baricitinib treatment

4 mg daily during 12 months

Intervention Type DRUG

anti-TNF therapy

adalimumab at 40 mg every 2 weeks or etanercept 50 mg per week according to treatments history

Intervention Type DRUG

Placebo

40 mg every 2 weeks during 6 months only during Period A

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Male or female;
* Age between 18 and 65 years-old;
* Adult patient with a diagnosis of RA as defined by the ACR/EULAR 2010 criteria for the classification of RA;
* Patient who presents an inadequate response to at least one bDMARD or tsDMARD for at least 12 weeks prior to study entry at a dose that is considered acceptable to assess clinical response adequately;
* Patient affected by active RA (DAS28-ESR \> 3.2 or sDAI \> 11 or cDAI \> 10) eligible to receive a bDMARD or tsDMARD according to the French Society of Rheumatology guidelines;
* Patient treated by prednisone dosage ≤ 10mg per day. The corticosteroids dosage will be decreased to 7,5 mg/day at the beginning of the study (W0);
* Person affiliated with or beneficiary of the French social security scheme;
* Free, informed and written consent signed by the participant and the investigator (on the day of inclusion at the latest and before any examination required by the research project).

Exclusion Criteria

* Patient previously treated with baricitinib;
* Patient previously treated by both adalimumab and etanercept. If the patient received previously only one of these two treatments, he/she can be included in the study with the treatment he/she has not yet received (if he/she is randomized in the experimental COMBI group);
* Patient affected by another form of inflammatory arthritis with the exception of secondary Sjögren syndrome;
* Patient who presents contraindications to the study treatments;
* Patients who is an active smoker or former smokers with a maximum exposure of 10 years;
* Patient who is currently receiving glucocorticosteroids at doses \>10 mg of prednisone per day (or equivalent) or has been receiving an unstable dosing regimen of corticosteroids within 4 weeks of study entry;
* Patient who is currently receiving more than 1 concomitant csDMARD (MTX, leflunomide, hydroxychloroquine or sulfasalazine) at the time of study entry;
* Patient who is currently receiving or has received csDMARDs (eg, gold salts, cyclosporine, azathioprine, or any other immunosuppressives) other than MTX (up to 25 mg/week), leflunomide (up to 20 mg/day), hydroxychloroquine (up to 400 mg/day), or sulfasalazine (up to 3000 mg/day) within 4 weeks prior to study entry.
* Doses of hydroxychloroquine or sulfasalazine should be stable for at least 4 weeks prior to study entry; if either has been recently discontinued, the patient must not have taken any dose within 4 weeks prior to study entry.
* Immunosuppression related to organ transplantation is not permitted;
* Patient who has received any parenteral corticosteroid administered by intramuscular or intravenous injection within 4 weeks prior to study entry, or is anticipated to require parenteral injection of corticosteroids during the study;
* Patient who had 3 or more joints injected with intraarticular corticosteroids or hyaluronic acid within 4 weeks prior to study entry. Joints injected with intraarticular corticosteroids or hyaluronic acid within 2 weeks prior to study entry or within 6 weeks prior to planned randomization cannot be counted in the TJC and SJC for entry or enrollment purposes;
* Patient with haemoglobin less than 80 g/L, absolute lymphocyte count lower than 0.5×109/L, absolute neutrophil count less than 1×109/L, or platelet count less than 100×109/L; clearance creatinine less than 60 mL/min; total bilirubin more than 1.5 times the upper limit of normal (ULN) at screening, aspartate aminotransferase, or alanine amino-transferase more than 2 times the upper limit of normal (ULN) at screening.
* Patient with co-administration with OAT3 inhibitors (such as probenecid);
* Patient who has a history or presence of cardiovascular, respiratory, hepatic, gastrointestinal, endocrine, hematological, neurological, or neuropsychiatric diseases or any other serious and/or unstable illness that, in the opinion of the investigator, could constitute a risk when taking investigational product or could interfere with the interpretation of data;
* Patient with an history of Moderate to severe heart failure (NYHA classes III/IV);
* Patient with an history of Major Adverse Cardiovascular Events (non-fatal myocardial infarction or non-fatal stroke);
* Patient who has a history of Venous Thromboembolic Event (VTE) (DVT/PE) within 12 weeks prior to randomization or have a history of recurrent (\>1) VTE (DVT/PE). Prior DVT with PE where events overlapped in time (i.e., with PE considered resulting from DVT) is not considered recurrent DVT/PE for the purpose of this criterion.
* Patient who has been exposed to a live vaccine within 12 weeks prior to planned randomization or are expected to need/receive a live vaccine during the course of the study (with the exception of herpes zoster vaccination). Investigators should review the vaccination status of their patients and follow the local guidelines for adult vaccination with nonlive vaccines intended to prevent infectious disease prior to entering patients into the study;
* Patient with an active cancer;
* Patient with malignancy or history of malignancy;
* Patient who has a current or recent (\<30 days prior to study entry) clinically serious viral, bacterial, fungal, or parasitic infection;
* Patient who is immunocompromised and, in the opinion of the investigator, is at an unacceptable risk for participating in the study;
* Patient with a history of active hepatitis B virus (HBV), hepatitis C virus (HCV), or human immunodeficiency virus (HIV);
* Patient who had household contact with a person with active tuberculosis (TB) and did not receive appropriate and documented prophylaxis for TB;
* Patient who has evidence of active TB or has previously had evidence of active TB and did not receive appropriate and documented treatment;
* Patient who has evidence of latent TB (as documented by a positive Purified Protein Derivative (PPD), no clinical symptoms consistent with active TB, and a normal chest x-ray at screening) unless patient completes at least 3 weeks of appropriate treatment prior to study entry and agrees to complete the remainder of treatment while in the trial
* Patient who had any major surgery within 8 weeks prior to study entry or will require major surgery during the study that, in the opinion of the investigator, would pose an unacceptable risk to the patient;
* Pregnant or breastfeeding woman, or woman who refuses to use an effective contraception during the study course;
* Patient governed by articles L 1121-5 to L 1121-8 (persons deprived of their liberty by a judicial or administrative decision, minors, persons of legal age who are the object of a legal protection measure or unable to express their consent).
Minimum Eligible Age

18 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Eli Lilly and Company

INDUSTRY

Sponsor Role collaborator

Biogen

INDUSTRY

Sponsor Role collaborator

Ministry for Health and Solidarity, France

OTHER_GOV

Sponsor Role collaborator

University Hospital, Bordeaux

OTHER

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Christophe RICHEZ, Prof

Role: PRINCIPAL_INVESTIGATOR

University Hospital, Bordeaux

Edouard LHOMME, MD

Role: STUDY_CHAIR

University Hospital, Bordeaux

Locations

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Polyclinique de Limoges - service de rhumatologie

Limoges, , France

Site Status RECRUITING

Groupement des Hôpitaux de l'Institut Catholique de Lille - service de rhumatologie

Lomme, , France

Site Status RECRUITING

AP-HM - service de rhumatologie

Marseille, , France

Site Status RECRUITING

Hôpital Saint-Joseph - service de rhumatologie

Marseille, , France

Site Status RECRUITING

CHU de Montpellier - service de rhumatologie

Montpellier, , France

Site Status RECRUITING

CHU de Nice - service de rhumatologie

Nice, , France

Site Status RECRUITING

CH de Niort - service de rhumatologie

Niort, , France

Site Status RECRUITING

CHU de Nîmes - service de rhumatologie

Nîmes, , France

Site Status NOT_YET_RECRUITING

Nouvel Hôpital Orléans La Source - service de rhumatologie

Orléans, , France

Site Status RECRUITING

AP-HP - Hôpital Bichat - service de rhumatologie

Paris, , France

Site Status RECRUITING

AP-HP - Hôpital Cochin - service de rhumatologie

Paris, , France

Site Status RECRUITING

AP-HP - Hôpital La Pitié-Salpetrière - service de rhumatologie

Paris, , France

Site Status RECRUITING

AP-HP - Hôpital Saint-Antoine - service de rhumatologie

Paris, , France

Site Status NOT_YET_RECRUITING

CH de Pau - service de rhumatologie

Pau, , France

Site Status RECRUITING

Hospices Civils de Lyon - service de rhumatologie

Pierre-Bénite, , France

Site Status RECRUITING

Hopital NOVO - service de rhumatologie

Pontoise, , France

Site Status RECRUITING

CH de Reims - service de rhumatologie

Reims, , France

Site Status RECRUITING

CHU de Saint-Etienne- service de rhumatologie

Saint-Etienne, , France

Site Status RECRUITING

CH de la Côte Basque - service de rhumatologie

Bayonne, , France

Site Status RECRUITING

CH de Belfort - service de rhumatologie

Belfort, , France

Site Status RECRUITING

AP-HP - Hopital Avicenne - service de rhumatologie

Bobigny, , France

Site Status NOT_YET_RECRUITING

CHU de Bordeaux - service de rhumatologie

Bordeaux, , France

Site Status RECRUITING

CHU de Brest - Service de rhumatologie

Brest, , France

Site Status RECRUITING

Clinique de l'Infirmerie - service de rhumatologie

Caluire-et-Cuire, , France

Site Status RECRUITING

CHU de Clermont-Ferrand - service de rhumatologie

Clermont-Ferrand, , France

Site Status RECRUITING

CH de Dax - service de rhumatologie

Dax, , France

Site Status RECRUITING

CHD VENDEE - service de rhumatologie

La Roche-sur-Yon, , France

Site Status RECRUITING

CH de Saint-Malo - service de rhumatologie

St-Malo, , France

Site Status NOT_YET_RECRUITING

CHRU de Strasbourg - service de rhumatologie

Strasbourg, , France

Site Status RECRUITING

CHU de Toulouse - service de rhumatologie

Toulouse, , France

Site Status RECRUITING

CHRU du Tours - service de rhumtologie

Tours, , France

Site Status RECRUITING

CHRU de Nancy - service de rhumatologie

Vandœuvre-lès-Nancy, , France

Site Status NOT_YET_RECRUITING

AP-HP - Hôpital Kremlin-Bicêtre - service de rhumatologie

Le Kremlin-Bicêtre, , France

Site Status RECRUITING

CH du Mans - service de rhumatologie

Le Mans, , France

Site Status RECRUITING

CH Emile Roux - service rhumatologie

Le Puy-en-Velay, , France

Site Status RECRUITING

service de Rhumatologie - CH Princesse Grace

Monaco, , Monaco

Site Status RECRUITING

Countries

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France Monaco

Central Contacts

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Christophe RICHEZ, Prof

Role: CONTACT

Phone: 05.56.79.55.56

Email: [email protected]

Thomas BARNETCHE, PhD

Role: CONTACT

Email: [email protected]

Facility Contacts

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Alexia HOURDILLE, MD

Role: primary

Anne LOHSE, MD

Role: primary

Luca SEMERANO, Prof

Role: primary

Christophe RICHEZ, Prof

Role: primary

Thomas BARNETCHE, PhD

Role: backup

Divi CORNEC, Prof

Role: primary

André BASCH, MD

Role: primary

Anne TOURNADRE, Prof

Role: primary

Emilie SHIPLEY, MD

Role: primary

Grégoire CORMIER, MD

Role: primary

Raphaele SEROR, Prof

Role: primary

Guillaume DIREZ, MD

Role: primary

Benjamin CASTAGNE, MD

Role: primary

Damien COYRAL, MD

Role: primary

Tristan PASCART, Prof

Role: primary

Thao PHAM, Prof

Role: primary

Damien ROCHE, MD

Role: primary

Jacques MOREL, Prof

Role: primary

Christian ROUX, Prof

Role: primary

Christian LORMEAU, MD

Role: primary

Cécile GAUJOUX-VIALA, Prof

Role: primary

Carine SAILLOT, MD

Role: primary

Philippe DIEUDE, Prof

Role: primary

Jérôme AVOUAC, MD

Role: primary

Bruno FAUTREL, Prof

Role: primary

Jéremie SELLAM, Prof

Role: primary

Vincent GERMAIN, MD

Role: primary

Cyrille CONFAVREUX, Prof

Role: primary

Omar AL TABAA, MD

Role: primary

Jean-Hugues SALMON, Prof

Role: primary

Hubert MAROTTE, Prof

Role: primary

Guillaume COIFFIER, MD

Role: primary

Jacques-Eric GOTTENBERG, Prof

Role: primary

Adeline RUYSSEN-WITRAND, Prof

Role: primary

Denis MULLEMAN, MD

Role: primary

Damien LOEUILLE, Prof

Role: primary

Olivier BROCQ, MD

Role: primary

Role: backup

Other Identifiers

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CHUBX 2019/56

Identifier Type: -

Identifier Source: org_study_id