Long-term Follow-up Study of GLPG0634 in Active Rheumatoid Arthritis Participants

NCT ID: NCT02065700

Last Updated: 2024-06-04

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

739 participants

Study Classification

INTERVENTIONAL

Study Start Date

2014-02-25

Study Completion Date

2023-01-19

Brief Summary

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The primary objective of the study was to evaluate the long-term safety and tolerability of filgotinib (formerly GLPG0634) for the treatment of rheumatoid arthritis.

Participants were enrolled in this open-label long-term follow-up study after they had completed one of the two core studies, GLPG0634-CL-203 (DARWIN1) (NCT01888874) or GLPG0634-CL-204 (DARWIN2) (NCT01894516), and were evaluated for any side effects that might have occured (long-term safety and tolerability) when taking filgotinib. During the course of the study, participants were also examined for long-term effects of filgotinib administration on disease activity (efficacy), participant's disability, fatigue, and quality of life.

Detailed Description

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Conditions

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Rheumatoid Arthritis

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Filgotinib Darwin 1

Participants in Study GLPG0634-CL-203 (NCT01888874) were rolled-over to receive an oral dose of filgotinib at a daily dose of 200 milligrams (mg) in this extension study, with the exception of male participants in the United States (US) who were limited to a daily dose of 100 mg due to a Food and Drug Administration (FDA) requirement based on a non-clinical finding. Treatment was administered until marketing, local (if applicable) regulatory and/or pertinent local reimbursement approval.

In case of intolerance or for safety reasons, and as per investigator's discretion, a daily dose of filgotinib 200 mg could be decreased to 100 mg per day, and later returned to 200 mg per day after the reasons for decreasing the dose were resolved.

Group Type EXPERIMENTAL

Filgotinib

Intervention Type DRUG

Administered as Oral Tablets

Filgotinib Darwin 2

Participants from Study GLPG0634-CL-204 (NCT01894516) were rolled-over to receive oral dose of filgotinib tablet at 200 mg once daily (q.d) in this extension study. Treatment was administered until marketing, local (if applicable) regulatory and/or pertinent local reimbursement approval.

Participants started the study with the same dose level (filgotinib 200 mg per day) and in case of intolerance or safety reasons and as per investigator's discretion, the daily dose of filgotinib was decreased to 100 mg q.d and was returned to 200 mg per day after the reasons for decreasing the dose had resolved and at the investigator's discretion.

Group Type EXPERIMENTAL

Filgotinib

Intervention Type DRUG

Administered as Oral Tablets

Interventions

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Filgotinib

Administered as Oral Tablets

Intervention Type DRUG

Other Intervention Names

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GS-6034 GLPG0634

Eligibility Criteria

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Inclusion Criteria

* Participants who completed one of the qualifying core studies GLPG0634-CL-203 or GLPG0634-CL-204 and may benefit from filgotinib long-term treatment according to the Investigator's judgment
* Females of childbearing potential and sexually active men must agree to use highly effective method of birth control as specified in the protocol, during the study and for at least 12 weeks after the last dose of filgotinib

Exclusion Criteria

* Participants who prematurely withdrew from one of the 2 core studies (GLPG0634-CL-203 or GLPG0634-CL-204), for any reason
* Persistent abnormal lab values during one of the 2 core studies (GLPG0634-CL-203 or GLPG0634-CL-204), according to the Investigator's judgment
* Diagnosis of rheumatic autoimmune disease or inflammatory joint disease other than rheumatoid arthritis, except for secondary Sjogren's syndrome
* Any condition or circumstances which, in the opinion of the Investigator, may make a participant unlikely or unable to complete the study or comply with study procedures and requirements
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Gilead Sciences

INDUSTRY

Sponsor Role collaborator

Galapagos NV

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Galapagos Study Director

Role: STUDY_DIRECTOR

Galapagos NV

Locations

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Arthro, Arthritis Care & Research

Gilbert, Arizona, United States

Site Status

Arizona Arthritis & Rheumatology Research PLLC

Mesa, Arizona, United States

Site Status

C.V. Mehta MD Medical Corp.

Hemet, California, United States

Site Status

Desert Medical Advances

Palm Desert, California, United States

Site Status

RASF Clinical Research Center

Boca Raton, Florida, United States

Site Status

Millenium Research

Ormond Beach, Florida, United States

Site Status

Lovelace Scientific Resources

Venice, Florida, United States

Site Status

Springfield Clinic

Springfield, Illinois, United States

Site Status

Klein and Associates MD, PA

Hagerstown, Maryland, United States

Site Status

Physicians East

Greenville, North Carolina, United States

Site Status

Health Research of Oklahoma

Oklahoma City, Oklahoma, United States

Site Status

Low County Rheumatology PA

Charleston, South Carolina, United States

Site Status

West Tennessee Research Institute

Jackson, Tennessee, United States

Site Status

Austin Rheumatology Research PA

Austin, Texas, United States

Site Status

Pioneer Research Solutions Inc

Houston, Texas, United States

Site Status

Atencion Integral en Reumatologa

Buenos Aires, , Argentina

Site Status

CER Intituto Medico

Buenos Aires, , Argentina

Site Status

Organizacion Medica de Investigaciones (OMI)

Buenos Aires, , Argentina

Site Status

Instituto Reumatologico Strusberg

Córdoba, , Argentina

Site Status

CIMeL Centro dee Investigacion Medico Lanus

Lanús, , Argentina

Site Status

Instituto CAICI

Rosario, , Argentina

Site Status

Instituto de Asistencia Reumatologia Integral - IARI

San Fernando, , Argentina

Site Status

Centro Médico Privado de Reumatologia

San Miguel de Tucumán, , Argentina

Site Status

Flinders Medical Centre

Bedford Park, Flinders Drive, South Australia, Australia

Site Status

Monash Medical Centre

Clayton, Victoria, Australia

Site Status

Princess Alexandra Hospital

Woolloongabba, , Australia

Site Status

Cliniques Universitaires St-Luc

Brussels, , Belgium

Site Status

UZ Leuven

Leuven, , Belgium

Site Status

University "Multiprofile Hospital for Active Treatment - Kaspela" LTD

Plovdiv, , Bulgaria

Site Status

Multiprofile Hospital for Active Treatment - Ruse

Rousse, , Bulgaria

Site Status

Diagnostic Consultative Center "Sveta Anna" LTD

Sofia, , Bulgaria

Site Status

National Multiprofile Transport Hospital "Tsar Boris III," Sofia, Clinical of Internal Diseases

Sofia, , Bulgaria

Site Status

University Multiprofile Hospital for Active Treatment "SV. Ivan Rilski" EAD, Sofia, Rheumatology Clinic

Sofia, , Bulgaria

Site Status

Hospital Regional "Guillermo Grant Benavente"

Santiago, , Chile

Site Status

Prosalud

Santiago, , Chile

Site Status

Someal SA

Santiago, , Chile

Site Status

Centro de Investigacion Clinica del Sur

Temuco, , Chile

Site Status

Consulta Privada Dra. Ponce

Temuco, , Chile

Site Status

Medicity S.A.S.

Bucaramanga, Santander Department, Colombia

Site Status

Circaribe S.A.S

Barranquilla, , Colombia

Site Status

Centro de Investigacion en Reumatologia y Especialidades Medicas (CIREEM)

Bogotá, , Colombia

Site Status

Riesgo De Fractura Cayre Ips7

Bogotá, , Colombia

Site Status

Idearg Sas

Bogotá, , Colombia

Site Status

Preventive Care SAS

Cundinamarca, , Colombia

Site Status

Hospital Pablo Tobon Uribe

Medellín, , Colombia

Site Status

Revmatologie S.R.O

Brno, , Czechia

Site Status

Revmatologicka a interni ambulance

Kladno, , Czechia

Site Status

Revmatologicka ambulance

Praha-Nusle, , Czechia

Site Status

PV-Medical S.R.O.

Zlín, , Czechia

Site Status

Hospitaux de Hautepierre

Strasbourg, , France

Site Status

Schlossparkklinik - Akad. Lehrkrankenhaus Charite

Berlin, , Germany

Site Status

MVZ Rheumatologie and Autoimmun Medizin HH GmbH

Hamburg, , Germany

Site Status

Centro Clinico

Guatemala City, , Guatemala

Site Status

Clinica de Especialidades Medicas

Guatemala City, , Guatemala

Site Status

Clinica Medica Especializada en Reumatologia

Guatemala City, , Guatemala

Site Status

Clinica Medica

Guatemala City, , Guatemala

Site Status

Reuma S.A.

Guatemala City, , Guatemala

Site Status

Reuma-Centro

Guatemala City, , Guatemala

Site Status

Gyogyszervizs galo Kozpont Kft

Balatonfüred, , Hungary

Site Status

QualiClinic Kft.

Budapest, , Hungary

Site Status

Reumatologiai Kft.

Budapest, , Hungary

Site Status

Markhot Ferenc Hospital, Rheumatology

Eger, , Hungary

Site Status

Csolnoky Ferenc Hospital, Rheumatology

Veszprém, , Hungary

Site Status

Carmel Medical Center

Haifa, , Israel

Site Status

Rambam Medical Center

Haifa, , Israel

Site Status

Ltd M&M Centr

Ādaži, , Latvia

Site Status

SIA Arijas Ancane's Family Doctor

Baldone, , Latvia

Site Status

Daugavpils Regional Hospital

Daugavpils, , Latvia

Site Status

L. Atikes doktorats

Liepāja, , Latvia

Site Status

'Bruninieku' polyclinic

Riga, , Latvia

Site Status

Centro de Estudios de Investigacion Basica y Clinica, SC

Guadalajara, , Mexico

Site Status

Centro Medico Dalinde

Mexico City, , Mexico

Site Status

Arke Estudios Clinicos S.A. de C.V.

México, , Mexico

Site Status

Clinstile, S.A. de C.V.

México, , Mexico

Site Status

Hospital General de México

México, , Mexico

Site Status

Hospital Universitario José E. Gonzalez

Monterrey, , Mexico

Site Status

OSMO

Oaxaca City, , Mexico

Site Status

IMSP Institutul de Cardiologie

Chisinau, , Moldova

Site Status

Waikato Hospital

Hamilton, , New Zealand

Site Status

Timaru Rheumatology Studies

Timaru, , New Zealand

Site Status

NZOZ Osteo-Medic s.c.

Bialystok, , Poland

Site Status

Centrum Medyczne Silesiana Sp. Z.o.o.

Bytom, , Poland

Site Status

Centrum Medyczne Pratia Katowice

Katowice, , Poland

Site Status

Centrum Medyczne Plejady

Krakow, , Poland

Site Status

NZOZ "DOBRY LEKARZ" Specjalistyczne Poradnie Lekarskie

Krakow, , Poland

Site Status

Specjalistyczne Centrum Medyczne Nowomed

Krakow, , Poland

Site Status

NZOZ Przychodnia Lekarska "Eskulap"

Skierniewice, , Poland

Site Status

Powiatowy Zaklad Opieki Zdrowotnej w Starachowicach

Starachowice, , Poland

Site Status

NZOZ "Nasz Lekarz" Pratyka Grupowa Lekarzy Rodzinnychz

Torun, , Poland

Site Status

AMED Medical Center

Warsaw, , Poland

Site Status

Rheumatica Sp. Z.o.o.

Warsaw, , Poland

Site Status

Spitalul Clinic Sfanta Maria

Bucharest, , Romania

Site Status

Spitalul Clinic Judetean de Urgenta Sf. Apostol Andrei Galati

Galati, , Romania

Site Status

First Moscow State Medical University n.a. I.M. Sechenova of the Ministry of Health

Moscow, , Russia

Site Status

Scientific Research Institute of Rheumatology

Moscow, , Russia

Site Status

City Clinical Hospital #5

Nizhny Novgorod, , Russia

Site Status

GBOU VPO Orenburg State Medical University

Orenburg, , Russia

Site Status

Ryazan State Medical University

Ryazan, , Russia

Site Status

City Hospital #26

Saint Petersburg, , Russia

Site Status

Regional Clinical Hospital

Saratov, , Russia

Site Status

Vladimir Regional State Instituion of Healthcare

Vladimir, , Russia

Site Status

Complejo Hospitalario Universitario A Coruña (CHUAC)

A Coruña, , Spain

Site Status

Sanatorio Nuestra Señora de la Esperanza

A Coruña, , Spain

Site Status

Hospital Parc Tauli

Sabadell, , Spain

Site Status

Communal Institution of Healthcare - Kharkiv City Clinical Hospital #13

Kharkiv, , Ukraine

Site Status

Kharkiv Medical Academy of Postgraduate Education, Department of Cardiology

Kharkiv, , Ukraine

Site Status

L.T. Malaya Therapy Institute of National Academy of Medical Sciences of Ukraine

Kharkiv, , Ukraine

Site Status

Kherson City Clinical Hospital N. A. Afanasii and Olga Tropin

Kherson, , Ukraine

Site Status

Municipal Non-Profit Institution Consultative and Diagnostic Centre of Desnyasky District of Kyiv

Kiev, , Ukraine

Site Status

Municipal Non-profit Enterprise Consultative and Diagnostic Center of Pechersk District of Kiev city

Kyiv, , Ukraine

Site Status

Vinnitsya Regional Clinical Hospital Named after M.I.Pirogov, Rheumatology Department

Vinnytsia, , Ukraine

Site Status

Countries

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United States Argentina Australia Belgium Bulgaria Chile Colombia Czechia France Germany Guatemala Hungary Israel Latvia Mexico Moldova New Zealand Poland Romania Russia Spain Ukraine

References

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Genovese MC, Kavanaugh A, Winthrop K, et al. Long Term Safety of Filgotinib in the Treatment of Rheumatoid Arthritis: Week 84 Data from a Phase 2b Open-Label Extension Study [abstract]. Arthritis Rheumatol. 2017; 69 (suppl 10).

Reference Type RESULT

Kavanaugh A, Westhovens R, Winthrop K, et al. Rheumatoid Arthritis Treatment with Filgotinib: Week 156 Safety and Efficacy Data from a Phase 2b Open-Label Extension Study [abstract]. Arthritis Rheumatol. 2019; 71 (suppl 10).

Reference Type RESULT

R. Westhovens, R. Alten, K. Winthrop, et al. Long term safety of filgotinib in the treatment of rheumatoid arthritis: week 108 data from a phase 2b open-label extension study. [abstract]. Ann Rheum Dis. 2018;77 (suppl 2)

Reference Type RESULT

Kavanaugh A, Genovese MC, Winthrop K, et al. Rheumatoid Arthritis Treatment with Filgotinib: Week 132 Safety Data from a Phase 2b Open-Label Extension Study [abstract]. Arthritis Rheumatol. 2018; 70 (suppl 9).

Reference Type RESULT

Kavanaugh A, Westhovens RR, Winthrop KL, Lee SJ, Tan Y, An D, Ye L, Sundy JS, Besuyen R, Meuleners L, Stanislavchuk M, Spindler AJ, Greenwald M, Alten R, Genovese MC. Safety and Efficacy of Filgotinib: Up to 4-year Results From an Open-label Extension Study of Phase II Rheumatoid Arthritis Programs. J Rheumatol. 2021 Aug;48(8):1230-1238. doi: 10.3899/jrheum.201183. Epub 2021 Feb 1.

Reference Type RESULT
PMID: 33526618 (View on PubMed)

Westhovens R, Winthrop KL, Kavanaugh A, Greenwald M, Dagna L, Cseuz R, Besuyen R, de Vries D, Modgill V, Le LH, Genovese MC, Emery P, Verschueren P, Alten R. Safety and efficacy of filgotinib in patients with rheumatoid arthritis: final results of the DARWIN 3 long-term extension study. RMD Open. 2025 Jan 30;11(1):e004857. doi: 10.1136/rmdopen-2024-004857.

Reference Type DERIVED
PMID: 39884731 (View on PubMed)

Balsa A, Wassenberg S, Tanaka Y, Tournadre A, Orzechowski HD, Rajendran V, Lendl U, Stiers PJ, Watson C, Caporali R, Galloway J, Verschueren P. Effect of Filgotinib on Body Mass Index (BMI) and Effect of Baseline BMI on the Efficacy and Safety of Filgotinib in Rheumatoid Arthritis. Rheumatol Ther. 2023 Dec;10(6):1555-1574. doi: 10.1007/s40744-023-00599-1. Epub 2023 Sep 25.

Reference Type DERIVED
PMID: 37747626 (View on PubMed)

Combe B, Besuyen R, Gomez-Centeno A, Matsubara T, Sancho Jimenez JJ, Yin Z, Buch MH. Geographic Analysis of the Safety and Efficacy of Filgotinib in Rheumatoid Arthritis. Rheumatol Ther. 2023 Feb;10(1):35-51. doi: 10.1007/s40744-022-00494-1. Epub 2022 Oct 7.

Reference Type DERIVED
PMID: 36205910 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Other Identifiers

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2012-003655-11

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

GLPG0634-CL-205

Identifier Type: -

Identifier Source: org_study_id

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