Comparison Study of the Glycemic Effects, Safety, and Tolerability of Exenatide Once Weekly Suspension to Sitagliptin and Placebo in Subjects With Type 2 Diabetes Mellitus

NCT ID: NCT01652729

Last Updated: 2015-08-20

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE3

Total Enrollment

365 participants

Study Classification

INTERVENTIONAL

Study Start Date

2013-02-28

Study Completion Date

2014-04-30

Brief Summary

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To compare the effect on glycemic control (HbA1c) of exenatide suspension administered once weekly to that achieved by sitagliptin or placebo administered once daily for 28 weeks in subjects with type 2 diabetes mellitus.

Detailed Description

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Conditions

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Diabetes Type 2

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Exenatide once weekly suspension

Exenatide once weekly suspension 2mg subcutaneous injection

Group Type EXPERIMENTAL

Exenatide once weekly suspension

Intervention Type DRUG

Sitagliptin 100mg

Overencapsulated Sitagliptin 100mg oral tablet once daily

Group Type ACTIVE_COMPARATOR

Sitagliptin

Intervention Type DRUG

Placebo

Placebo oral capsule once daily

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

Placebo oral capsule once daily

Interventions

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Exenatide once weekly suspension

Intervention Type DRUG

Sitagliptin

Intervention Type DRUG

Placebo

Placebo oral capsule once daily

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* At least 18 years old
* Diagnosed with type 2 diabetes mellitus
* HbA1c of 7.1% to 11.0%, inclusive, at screening
* Has stable body weight, i.e., not varying by \>3% for at least 3 months prior to screening
* Fasting plasma glucose concentration \<280 mg/dL (15.5 mmol/L) at screening
* Body mass index of \<45 kg/m2 at screening
* Has been treated with a stable regimen of ≥1500 mg/day metformin for a minimum of 2 months prior to Visit 1 (Screening)

Exclusion Criteria

* History of pancreatitis or triglycerides \>=500 mg/dL
* Medullary carcinoma or multiple endocrine neoplasia (MEN2) or a family history of either
* History of renal transplantation, or is currently receiving renal dialysis, or has an estimated creatinine clearance \<50 mL/min
* Active cardiovascular disease
* Presence or history of severe congestive heart failure
* Central nervous system disease, including epilepsy
* Liver disease
* History of severe gastrointestinal diseases
* Clinically significant malignant disease
* Repeated severe hypoglycemia within the last 6 months
* Any exposure to exenatide (BYETTA® or BYDUREON™) or any GLP-1 analog
* Any DPP-4 inhibitor within 3 months prior screening
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Peter Ohman

Role: STUDY_CHAIR

AstraZeneca

Locations

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Research Site

Birmingham, Alabama, United States

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Huntsville, Alabama, United States

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Phoenix, Arizona, United States

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Phoenix, Arizona, United States

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Beverly Hills, California, United States

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Buena Park, California, United States

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Chino, California, United States

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Chula Vista, California, United States

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Encinitas, California, United States

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Greenbrae, California, United States

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Los Angeles, California, United States

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Los Angeles, California, United States

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North Hollywood, California, United States

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Walnut Creek, California, United States

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West Hills, California, United States

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Boca Raton, Florida, United States

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Hialeah, Florida, United States

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Miami, Florida, United States

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Miami, Florida, United States

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Miami, Florida, United States

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Port Orange, Florida, United States

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St. Petersburg, Florida, United States

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Chicago, Illinois, United States

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Evanston, Illinois, United States

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Indianapolis, Indiana, United States

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Oxon Hill, Maryland, United States

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Omaha, Nebraska, United States

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Henderson, Nevada, United States

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Las Vegas, Nevada, United States

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Las Vegas, Nevada, United States

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Albuquerque, New Mexico, United States

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Buffalo, New York, United States

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Hartsdale, New York, United States

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Charlotte, North Carolina, United States

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Clayton, North Carolina, United States

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Durham, North Carolina, United States

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Greensboro, North Carolina, United States

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Mooresville, North Carolina, United States

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Salisbury, North Carolina, United States

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Cincinnati, Ohio, United States

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Franklin, Ohio, United States

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Marion, Ohio, United States

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Yukon, Oklahoma, United States

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Eugene, Oregon, United States

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Portland, Oregon, United States

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Greer, South Carolina, United States

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Simpsonville, South Carolina, United States

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Rapid City, South Dakota, United States

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Chattanooga, Tennessee, United States

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Carrolton, Texas, United States

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Corpus Christi, Texas, United States

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Dallas, Texas, United States

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Houston, Texas, United States

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Houston, Texas, United States

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Katy, Texas, United States

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San Antonio, Texas, United States

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Salt Lake City, Utah, United States

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Salt Lake City, Utah, United States

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Burke, Virginia, United States

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Spokane, Washington, United States

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Countries

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United States

References

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Guja C, Frias JP, Suchower L, Hardy E, Marr G, Sjostrom CD, Jabbour SA. Safety and Efficacy of Exenatide Once Weekly in Participants with Type 2 Diabetes and Stage 2/3 Chronic Kidney Disease. Diabetes Ther. 2020 Jul;11(7):1467-1480. doi: 10.1007/s13300-020-00815-z. Epub 2020 Apr 18.

Reference Type DERIVED
PMID: 32306296 (View on PubMed)

Gadde KM, Vetter ML, Iqbal N, Hardy E, Ohman P; DURATION-NEO-2 study investigators. Efficacy and safety of autoinjected exenatide once-weekly suspension versus sitagliptin or placebo with metformin in patients with type 2 diabetes: The DURATION-NEO-2 randomized clinical study. Diabetes Obes Metab. 2017 Jul;19(7):979-988. doi: 10.1111/dom.12908. Epub 2017 Mar 17.

Reference Type DERIVED
PMID: 28205322 (View on PubMed)

Related Links

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Other Identifiers

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MB001-004

Identifier Type: OTHER

Identifier Source: secondary_id

BCB120

Identifier Type: -

Identifier Source: org_study_id

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