Study To Evaluate The Efficacy And Safety Of PH-797804 For 12 Weeks In Adults With Moderate To Severe Chronic Obstructive Pulmonary Disease (COPD) On A Background Of Tiotropium Bromide

NCT ID: NCT01543919

Last Updated: 2014-10-27

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

730 participants

Study Classification

INTERVENTIONAL

Study Start Date

2012-04-30

Study Completion Date

2013-09-30

Brief Summary

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PH-797804 is an oral anti-inflammatory drug that may reduce the inflammation that is associated with Chronic Obstructive Pulmonary Disease (COPD). PH-797804 will be dosed to patients with Chronic Obstructive Pulmonary Disease (COPD) to evaluate its potential safety and efficacy profile in Chronic Obstructive Pulmonary Disease (COPD)

Detailed Description

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Conditions

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Pulmonary Disease, Chronic Obstructive

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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PH-787904 (arm1)

Group Type EXPERIMENTAL

PH-797804

Intervention Type DRUG

0.25 mg oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

PH-787904 (arm2)

Group Type EXPERIMENTAL

PH-797804

Intervention Type DRUG

1 mg oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

PH-787904 (arm3)

Group Type EXPERIMENTAL

PH-797804

Intervention Type DRUG

3 mg oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

PH-787904 (arm4)

Group Type EXPERIMENTAL

PH-797804

Intervention Type DRUG

6 mg oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

PH-787904 (arm5)

Group Type EXPERIMENTAL

PH-797804

Intervention Type DRUG

10 mg oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

Placebo

Group Type EXPERIMENTAL

Placebo

Intervention Type DRUG

Placebo oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

Interventions

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PH-797804

0.25 mg oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

Intervention Type DRUG

PH-797804

1 mg oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

Intervention Type DRUG

PH-797804

3 mg oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

Intervention Type DRUG

PH-797804

6 mg oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

Intervention Type DRUG

PH-797804

10 mg oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

Intervention Type DRUG

Placebo

Placebo oral tablet plus tiotropium bromide 18 microgram once daily for 12 weeks

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Male or female subjects between, and including, the ages of 40 and 80 years.
* Subjects with a diagnosis, for at least 6 months, of moderate to severe COPD (GOLD) and who meet the criteria for Stage II-III disease: Subjects must have a post-bronchodilator FEV1/FVC ratio \<0.7 and a post-bronchodilator FEV1 of 30 - 80% (inclusive) of the predicted value for age, height, race and sex using European Community for Coal and Steel ECCS standards or NHANES III standards.
* Subjects must have a smoking history of at least 10 pack-years\* and meet one of the following criteria: They are current smokers, or they are ex-smokers who have abstained from smoking for at least 6 months.
* Subjects treated with tiotropium bromide (SPIRIVA HandiHaler) 18 microgram daily for at least 1 month prior to screening.
* Subjects must have had stable disease for at least 1 month prior to screening. During the screening and run-in phase subjects must be able to manage disease symptoms adequately with tiotropium bromide +/- salbutamol (albuterol) rescue medication (subjects should not use \>10 actuations \[100 microgram/actuations\] daily for more than 2 consecutive days), without reliance on other therapies including oral or inhaled corticosteroids, other long-acting bronchodilators, nebulizer therapy, theophylline, roflumilast or regular oxygen.

Exclusion Criteria

* A COPD exacerbation requiring treatment with oral steroids or hospitalization for the treatment of COPD within 3 months of screening.
* History of a lower respiratory tract infection or significant disease instability during the month preceding screening or during the time between screening and randomization.
* History or presence of respiratory failure, cor pulmonale or right ventricular failure.
* Subjects with home oxygen therapy (either PRN or long-term oxygen therapy).
* Any clearly documented history of adult asthma or other chronic respiratory disorders (eg, bronchiectasis, pulmonary fibrosis, pneumoconiosis).
* Known previous diagnosis of Hepatitis B or C or HIV infection (specific screening is not required).
* History of cancer (other than cutaneous basal cell) in the previous 5 years.
* Active or past history of GI hemorrhage of any etiology, peptic ulceration, erosive esophagitis, gastric outlet obstruction or inflammatory bowel disease.
* Regular use of aspirin at a dose greater than 325 mg/day.
* History within the previous 6 months of: myocardial infarction, cardiac arrhythmia (eg, atrial fibrillation, paroxysmal atrial fibrillation, atrial flutter, supraventricular tachycardia, ventricular tachycardia), left ventricular failure, unstable angina, coronary angioplasty, coronary artery bypass grafting (CABG) or cerebrovascular accident (including transient ischemic attacks).
* A family history of long QT syndrome.
* Presenting with: Any condition possibly affecting oral drug absorption (eg, gastrectomy or clinically significant diabetic gastroenteropathy).
* Any clinically significant skin lesions as described in Common Terminology Criteria for Adverse Events for Dermatology (CTCAE) Version 3.0.
* Any clinically significant active systemic or cutaneous infection including herpetic lesions.
* Congestive heart failure requiring treatment New York Heart Association (NYHA) Class III-IV.
* ECG abnormalities at screening or randomization, including those listed below: Subjects with pre-randomization evidence of QTcF prolongation (defined as \>450 ms) at screening or baseline (Week 0) are not eligible for randomization. This assessment is based on a confirmed mean of the triplicate ECG recordings and is made by the investigator at the time of ECG collection.
* Predominant heart rhythm other than normal sinus rhythm eg, atrial fibrillation, atrial flutter, supraventricular tachycardia.
* Atrioventricular (AV) block greater than first degree.
* Resting heart rate \>100 or \<40 bpm.
* Evidence of previous myocardial infarction in the absence of clinical history consistent with these findings.
* Evidence of acute ischemia.
Minimum Eligible Age

40 Years

Maximum Eligible Age

80 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Pfizer Investigational Site

Birmingham, Alabama, United States

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Birmingham, Alabama, United States

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Birmingham, Alabama, United States

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Jasper, Alabama, United States

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Phoenix, Arizona, United States

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Montclair, California, United States

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San Diego, California, United States

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Waterbury, Connecticut, United States

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Newark, Delaware, United States

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Brandon, Florida, United States

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Chiefland, Florida, United States

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Chiefland, Florida, United States

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Clearwater, Florida, United States

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Clearwater, Florida, United States

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New Port Richey, Florida, United States

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Pensacola, Florida, United States

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Tampa, Florida, United States

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Williston, Florida, United States

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Duluth, Georgia, United States

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Fort Mitchell, Kentucky, United States

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Lexington, Kentucky, United States

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Baltimore, Maryland, United States

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Edina, Minnesota, United States

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Fridley, Minnesota, United States

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Minneapolis, Minnesota, United States

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Rochester, Minnesota, United States

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St Louis, Missouri, United States

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Albuquerque, New Mexico, United States

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Albuquerque, New Mexico, United States

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Albuquerque, New Mexico, United States

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Rochester, New York, United States

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Charlotte, North Carolina, United States

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Cincinnati, Ohio, United States

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Cincinnati, Ohio, United States

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Cincinnati, Ohio, United States

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Oklahoma City, Oklahoma, United States

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Philadelphia, Pennsylvania, United States

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Pawtucket, Rhode Island, United States

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Warwick, Rhode Island, United States

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Charleston, South Carolina, United States

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Charleston, South Carolina, United States

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Kingsport, Tennessee, United States

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Houston, Texas, United States

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San Antonio, Texas, United States

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Midvale, Utah, United States

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Buenos Aires, , Argentina

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Rousse, , Bulgaria

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Sevlievo, , Bulgaria

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Sofia, , Bulgaria

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Sofia, , Bulgaria

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Stara Zagora, , Bulgaria

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Troyan Municipality, , Bulgaria

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Veliko Tarnovo, , Bulgaria

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Winnipeg, Manitoba, Canada

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Toronto, Ontario, Canada

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Toronto, Ontario, Canada

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Montreal, Quebec, Canada

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Québec, Quebec, Canada

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Saint Romuald, Quebec, Canada

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Sherbrooke, Quebec, Canada

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Karlovy Vary, , Czechia

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Liberec, , Czechia

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Mělník, , Czechia

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Prague, , Czechia

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Prague, , Czechia

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Rokycany, , Czechia

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Teplice, , Czechia

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Berlin, , Germany

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Berlin, , Germany

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Dresden, , Germany

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Gelnhausen, , Germany

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Großhansdorf, , Germany

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Hamburg, , Germany

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Hamburg, , Germany

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Hanover, , Germany

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Kassel, , Germany

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Lübeck, , Germany

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Schwerin, , Germany

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Balassagyarmat, , Hungary

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Budaörs, , Hungary

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Budapest, , Hungary

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Debrecen, , Hungary

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Szeged, , Hungary

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Szombathely, , Hungary

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Törökbálint, , Hungary

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Nagoya, Aichi-ken, Japan

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Seto-shi, Aichi-ken, Japan

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Toyota, Aichi-ken, Japan

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Noda, Chiba, Japan

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Fukuoka, Fukuoka, Japan

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Yanagawa, Fukuoka, Japan

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Kanazawa, Ishikawa-ken, Japan

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Takamatsu, Kagawa-ken, Japan

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Kawasaki-shi, Kanagawa, Japan

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Zama, Kanagawa, Japan

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Kumamoto, Kumamoto, Japan

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Saiki, Oita Prefecture, Japan

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Osaka, Osaka, Japan

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Meguro-ku, Tokyo, Japan

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Setagaya City, Tokyo, Japan

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Warsaw, , Poland

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Wroclaw, , Poland

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Wroclaw, , Poland

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Bardejov, , Slovakia

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Bojnice, , Slovakia

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Bratislava, , Slovakia

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Bratislava, , Slovakia

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Humenné, , Slovakia

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Košice, , Slovakia

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Liptovský Hrádok, , Slovakia

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Námestovo, , Slovakia

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Poprad, , Slovakia

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Spišská Nová Ves, , Slovakia

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Štúrovo, , Slovakia

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Bloemfontein, Free State, South Africa

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Gatesville, Western Cape, South Africa

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Parow, Western Cape, South Africa

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Cape Town, , South Africa

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Cape Town, , South Africa

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Durban, , South Africa

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Durban, , South Africa

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Pretoria, , South Africa

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Petrel, Alicante, Spain

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Mérida, Badajoz, Spain

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Salt, Girona, Spain

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Pozuelo de Alarcón, Madrid, Spain

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Gothenburg, , Sweden

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Linköping, , Sweden

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Lund, , Sweden

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Malmo, , Sweden

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Skene, , Sweden

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Taipei, , Taiwan

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Countries

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United States Argentina Bulgaria Canada Czechia Germany Hungary Japan Poland Slovakia South Africa Spain Sweden Taiwan

Related Links

Other Identifiers

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A6631033

Identifier Type: -

Identifier Source: org_study_id

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