Study in Healthy Recreational Polydrug Users to Measure the Abuse Potential of TC-5214

NCT ID: NCT01500018

Last Updated: 2012-03-22

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

WITHDRAWN

Clinical Phase

PHASE1

Study Classification

INTERVENTIONAL

Study Start Date

2012-01-31

Study Completion Date

2012-04-30

Brief Summary

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This is a single dose, crossover study to assess the abuse potential of TC-5214 compared to placebo, ketamine, and phentermine in healthy recreational polydrug users.

Detailed Description

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A Single-center, Single-dose, Double-blind, Randomized, Placebo- and Active-controlled Crossover Study to Evaluate the Abuse Potential of TC-5214 in Healthy Recreational Polydrug Users.

Conditions

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Drug Abuse Healthy

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

TRIPLE

Participants Caregivers Investigators

Study Groups

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Crossover Treatment Sequence 1

Period 1: Placebo, Period 2: Phentermine 45 mg, Period 3: Phentermine 90 mg, Period 4: Ketamine 100 mg, Period 5: TC-5214 2 mg, Period 6: TC-5214 8 mg, Period 7: TC-5214 16 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 2

Period 1: Phentermine 45 mg, Period 2: Ketamine 100 mg , Period 3: Placebo, Period 4: TC-5214 8 mg , Period 5: Phentermine 90 mg, Period 6: TC-5214 16 mg, Period 7: TC-5214 2 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 3

Period 1: Ketamine 100 mg, Period 2: TC-5214 8 mg, Period 3: Phentermine 45 mg, Period 4: TC-5214 16 mg, Period 5: Placebo, Period 6: TC-5214 2 mg, Period 7: Phentermine 90 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 4

Period 1: TC-5214 8 mg, Period 2: TC-5214 16 mg, Period 3: Ketamine 100 mg, Period 4: TC-5214 2 mg, Period 5: Phentermine 45 mg , Period 6: Phentermine 90 mg, Period 7: Placebo

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 5

Period 1: TC-5214 16 mg, Period 2: TC-5214 2 mg, Period 3: TC-5214 8 mg, Period 4: Phentermine 90 mg, Period 5: Ketamine 100 mg, Period 6: Placebo , Period 7: Phentermine 45 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 6

Period 1: TC-5214 2 mg, Period 2: Phentermine 90 mg, Period 3: TC-5214 16 mg, Period 4: Placebo, Period 5: TC-5214 8 mg, Period 6:Phentermine 45 mg , Period 7: Ketamine 100 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 7

Period 1: Phentermine 90 mg, Period 2: Placebo, Period 3: TC-5214 2 mg, Period 4: Phentermine 45 mg, Period 5: TC-5214 16 mg, Period 6: Ketamine 100 mg, Period 7: TC-5214 8 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 8

Period 1: TC-5214 16 mg, Period 2: TC-5214 8 mg, Period 3: TC-5214 2 mg, Period 4: Ketamine 100 mg, Period 5: Phentermine 90 mg, Period 6: Phentermine 45 mg, Period 7: Placebo

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 9

Period 1: TC-5214 2 mg, Period 2: TC-5214 16 mg, Period 3: Phentermine 90 mg, Period 4: TC-5214 8 mg, Period 5: Placebo, Period 6: Ketamine 100 mg, Period 7:

Phentermine 45 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 10

Period 1: Phentermine 90 mg, Period 2: TC-5214 2 mg, Period 3: Placebo, Period 4: TC-5214 16 mg Ketamine 100 mg, Period 5: Phentermine 45 mg, Period 6: TC-5214 8 mg, Period 7: TC-5214 2 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 11

Period 1: Placebo, Period 2: Phentermine 90 mg, Period 3:Phentermine 45 mg, Period 4: TC-5214 2 mg, Period 5: Ketamine 100 mg, Period 6: TC-5214 16 mg, Period 7: TC-5214 8 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 12

Period 1: Phentermine 45 mg, Period 2: Placebo, Period 3: Ketamine 100 mg, Period 4:Phentermine 90 mg, Period 5: TC-5214 8 mg, Period 6: TC-5214 2 mg, Period 7: TC-5214 16 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 13

Period 1: Ketamine 100 mg, Period 2: Phentermine 45 mg, Period 3: TC-5214 8 mg, Period 4: Placebo, Period 5: TC-5214 16 mg, Period 6: Phentermine 90 mg, Period 7: TC-5214 2 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Crossover Treatment Sequence 14

Period 1: TC-5214 8 mg, Period 2: Ketamine 100 mg, Period 3: TC-5214 16 mg, Period 4: Phentermine 45 mg, Period 5: TC-5214 2 mg, Period 6: Placebo, Period 7: Phentermine 90 mg

Group Type EXPERIMENTAL

TC-5214

Intervention Type DRUG

Single oral dose of 2 mg

TC-5214 Placebo

Intervention Type DRUG

Single oral dose

Ketamine

Intervention Type DRUG

Single oral dose of 100 mg

Phentermine

Intervention Type DRUG

Single oral dose of 45 mg

TC-5214

Intervention Type DRUG

Single oral dose of 8 mg

TC-5214

Intervention Type DRUG

Single oral dose of 16 mg

Phentermine

Intervention Type DRUG

Single oral dose of 90 mg

Interventions

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TC-5214

Single oral dose of 2 mg

Intervention Type DRUG

TC-5214 Placebo

Single oral dose

Intervention Type DRUG

Ketamine

Single oral dose of 100 mg

Intervention Type DRUG

Phentermine

Single oral dose of 45 mg

Intervention Type DRUG

TC-5214

Single oral dose of 8 mg

Intervention Type DRUG

TC-5214

Single oral dose of 16 mg

Intervention Type DRUG

Phentermine

Single oral dose of 90 mg

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Current recreational polydrug users with experience with at least 2 drug classes of abuse.
* At least 10 lifetime uses of stimulants drugs (eg, amphetamine, cocaine, methamphetamine) and 10 lifetime occasions of recreational use of psychedelic drugs (eg, cannabis, ketamine, dextromethorphan, PCP, MDMA \[ecstasy\], LSD, mesacline, or psilocybin).
* Recreational use of other classes of drugs is permitted, including opioids (eg, codeine, morphine, or heroin), minor tranquilizers, or sedatives (eg, benzodiazepines or barbiturates).
* Male or female volunteers aged 18 to 55, inclusive with a body mass index (BMI) within the range of 19.0 to 33.0 kg/m2, inclusive, and a minimum weight of 50.0 kg at screening.
* Must pass qualification phase eligibility criteria.

Exclusion Criteria

* Self-reported history of drug or alcohol dependence (except caffeine) in the past 12 months, including subjects who have ever been in a drug rehabilitation program (other than treatment for smoking cessation).
* Unwillingness or inability to abstain from recreational drug use for the duration of the study from screening until follow-up.
* Positive for hepatitis B, hepatitis C, or human immunodeficiency virus (HIV) at screening.
* Any significant unstable hepatic, renal, pulmonary, cardiovascular, ophthalmologic, neurologic, or any other medical conditions that might confound the study or put the volunteer at greater risk during study participation.
* Currently smoking more than 20 cigarettes (or 2 cigars) per day, and/or unwillingness to abstain from smoking for durations of at least 12 hours.
* Use of tobacco cessation product within 1 month (eg, nicotine substitution products, bupropion, etc).
Minimum Eligible Age

18 Years

Maximum Eligible Age

55 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

Yes

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Hans A Eriksson, MD

Role: STUDY_DIRECTOR

AstraZeneca Kvzmbergagatan 12, 15185,Sodertalje, Sweden

Pierre Geoffroy, MDCM, MSC, FCFP

Role: PRINCIPAL_INVESTIGATOR

Syneos Health

Brendan Smyth, MD

Role: STUDY_DIRECTOR

AstraZeneca 180 Concord Pike, Wilmington,DE 19850-5437

Other Identifiers

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D4130C00022

Identifier Type: -

Identifier Source: org_study_id

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