Effects of Once and Twice Daily Dosing Regimen of Ertugliflozin (PF-04971729, MK-8835) In Participants With Type 2 Diabetes (MK-8835-040)

NCT ID: NCT01054300

Last Updated: 2019-11-21

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

52 participants

Study Classification

INTERVENTIONAL

Study Start Date

2010-02-17

Study Completion Date

2010-04-07

Brief Summary

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This is a Phase 1 randomized, double-blind, sponsor open, 4 arm, 2 way cross-over study using 2 cohorts. The objective of the study is to evaluate the pharmacodynamics (PD) effects and the pharmacokinetic (PK) of single day dosing of 2 mg and 4 mg doses of ertugliflozin (Ertu, PF-04971729/MK-8835) each administered once vs twice daily (morning \[AM\] and evening \[PM\]) in adults with type 2 diabetes.

Detailed Description

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Conditions

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Diabetes Mellitus, Type 2 Adult

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

CROSSOVER

Primary Study Purpose

OTHER

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

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Cohort 1: Ertu 2 mg/Placebo (Pbo)→Ertu 1 mg/Ertu 1 mg

Period 1: Ertu 2 mg in the AM and Pbo in the PM for 1 day. Period 2: Ertu 1 mg in the AM and Ertu 1 mg in the PM for 1 day. There was a \>= 7 day washout period between Period 1 and Period 2.

Group Type EXPERIMENTAL

Ertugliflozin 2 mg single dose

Intervention Type DRUG

Ertugliflozin 2 mg dose (two 1 mg strength tablets), administered as a single dose

Ertugliflozin 2 mg split into twice daily

Intervention Type DRUG

Ertugliflozin 1 mg dose (1 mg strength tablet) administered twice daily x 1 day

Placebo

Intervention Type DRUG

Placebo to ertugliflozin administered as a single dose

Cohort 1: Ertu 1 mg/Ertu 1 mg→Ertu 2 mg/Pbo

Period 1: Ertu 1 mg in the AM and Ertu 1 mg in the PM for 1 day. Period 2: Ertu 2 mg in the AM and Pbo in the PM for 1 day. There was a \>= 7 day washout period between Period 1 and Period 2.

Group Type EXPERIMENTAL

Ertugliflozin 2 mg single dose

Intervention Type DRUG

Ertugliflozin 2 mg dose (two 1 mg strength tablets), administered as a single dose

Ertugliflozin 2 mg split into twice daily

Intervention Type DRUG

Ertugliflozin 1 mg dose (1 mg strength tablet) administered twice daily x 1 day

Placebo

Intervention Type DRUG

Placebo to ertugliflozin administered as a single dose

Cohort 2: Ertu 4 mg/Pbo→Ertu 2 mg/Ertu 2 mg

Period 1: Ertu 4 mg in the AM and Pbo in the PM for 1 day. Period 2: Ertu 2 mg in the AM and Ertu 2 mg in the PM for 1 day. There was a \>= 7 day washout period between Period 1 and Period 2.

Group Type EXPERIMENTAL

Ertugliflozin 4 mg single dose

Intervention Type DRUG

Ertugliflozin 4 mg dose (four 1 mg strength tablets), administered as a single dose

Ertugliflozin 4 mg split into twice daily

Intervention Type DRUG

Ertugliflozin 2 mg dose (two 1 mg strength tablets) administered twice daily x 1 day

Placebo

Intervention Type DRUG

Placebo to ertugliflozin administered as a single dose

Cohort 2: Ertu 2 mg/Ertu 2 mg→Ertu 4 mg/Pbo

Period 1: Ertu 2 mg in the AM and Ertu 2 mg in the PM for 1 day. Period 2: Ertu 4 mg in the AM and Pbo in the PM for 1 day. There was a \>= 7 day washout period between Period 1 and Period 2.

Group Type EXPERIMENTAL

Ertugliflozin 4 mg single dose

Intervention Type DRUG

Ertugliflozin 4 mg dose (four 1 mg strength tablets), administered as a single dose

Ertugliflozin 4 mg split into twice daily

Intervention Type DRUG

Ertugliflozin 2 mg dose (two 1 mg strength tablets) administered twice daily x 1 day

Placebo

Intervention Type DRUG

Placebo to ertugliflozin administered as a single dose

Interventions

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Ertugliflozin 2 mg single dose

Ertugliflozin 2 mg dose (two 1 mg strength tablets), administered as a single dose

Intervention Type DRUG

Ertugliflozin 2 mg split into twice daily

Ertugliflozin 1 mg dose (1 mg strength tablet) administered twice daily x 1 day

Intervention Type DRUG

Ertugliflozin 4 mg single dose

Ertugliflozin 4 mg dose (four 1 mg strength tablets), administered as a single dose

Intervention Type DRUG

Ertugliflozin 4 mg split into twice daily

Ertugliflozin 2 mg dose (two 1 mg strength tablets) administered twice daily x 1 day

Intervention Type DRUG

Placebo

Placebo to ertugliflozin administered as a single dose

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Participants with type 2 diabetes mellitus, either treatment-naïve or on up to 2 acceptable oral anti-diabetes drugs for at least 8-weeks prior to study.

Exclusion Criteria

* Participants with type 1 diabetes mellitus, participants with stroke, unstable angina, heart attack in last 6-months, uncontrolled blood pressure.
Minimum Eligible Age

18 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role collaborator

Merck Sharp & Dohme LLC

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Medical Director

Role: STUDY_DIRECTOR

Merck Sharp & Dohme LLC

References

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Dawra VK, Liang Y, Shi H, Bass A, Hickman A, Terra SG, Zhou S, Cutler D, Sahasrabudhe V. A PK/PD study comparing twice-daily to once-daily dosing regimens of ertugliflozin in healthy subjects . Int J Clin Pharmacol Ther. 2019 Apr;57(4):207-216. doi: 10.5414/CP203343.

Reference Type RESULT
PMID: 30802200 (View on PubMed)

Fediuk DJ, Sahasrabudhe V, Dawra VK, Zhou S, Sweeney K. Population Pharmacokinetic Analyses of Ertugliflozin in Select Ethnic Populations. Clin Pharmacol Drug Dev. 2021 Nov;10(11):1297-1306. doi: 10.1002/cpdd.970. Epub 2021 Jul 2.

Reference Type DERIVED
PMID: 34213819 (View on PubMed)

Other Identifiers

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B1521007

Identifier Type: OTHER

Identifier Source: secondary_id

MK-8835-040

Identifier Type: OTHER

Identifier Source: secondary_id

8835-040

Identifier Type: -

Identifier Source: org_study_id

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