A 16 Week Study to Evaluate the Efficacy and Safety of PF-06882961 in Adults With Type 2 Diabetes Mellitus

NCT ID: NCT03985293

Last Updated: 2022-06-30

Study Results

Results available

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Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

412 participants

Study Classification

INTERVENTIONAL

Study Start Date

2019-10-15

Study Completion Date

2021-07-07

Brief Summary

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This multicenter, randomized, double-blind, placebo controlled, parallel group study is being conducted to provide data on efficacy, safety, tolerability and pharmacokinetics (PK) of multiple dose levels of PF-06882961 in adults with type 2 diabetes mellitus (T2DM) inadequately controlled on metformin and/or diet and exercise. In addition, the study is intended to enable selection of efficacious doses for future clinical development of PF-06882961.

Detailed Description

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Conditions

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Diabetes Mellitus, Type 2

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Study Groups

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Placebo

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

4 matching placebo tablets taken twice a day (BID)

PF-06882961 2.5 milligrams (mg)

Group Type EXPERIMENTAL

PF-06882961

Intervention Type DRUG

Participants will be randomized to one of 5 active doses (2.5, 10, 40, 80, or 120 mg), taking 4 tablets twice daily for 16 weeks.

PF-06882961 10 mg

Group Type EXPERIMENTAL

PF-06882961

Intervention Type DRUG

Participants will be randomized to one of 5 active doses (2.5, 10, 40, 80, or 120 mg), taking 4 tablets twice daily for 16 weeks.

PF-06882961 40 mg

Participants will be titrated up to 2 weeks to reach desired dose level

Group Type EXPERIMENTAL

PF-06882961

Intervention Type DRUG

Participants will be randomized to one of 5 active doses (2.5, 10, 40, 80, or 120 mg), taking 4 tablets twice daily for 16 weeks.

PF-06882961 80 mg

Participants will be titrated up to 4 weeks to reach desired dose level

Group Type EXPERIMENTAL

PF-06882961

Intervention Type DRUG

Participants will be randomized to one of 5 active doses (2.5, 10, 40, 80, or 120 mg), taking 4 tablets twice daily for 16 weeks.

PF-06882961 120 mg

Participants will be titrated up to 6 weeks to reach desired dose level

Group Type EXPERIMENTAL

PF-06882961

Intervention Type DRUG

Participants will be randomized to one of 5 active doses (2.5, 10, 40, 80, or 120 mg), taking 4 tablets twice daily for 16 weeks.

Interventions

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Placebo

4 matching placebo tablets taken twice a day (BID)

Intervention Type DRUG

PF-06882961

Participants will be randomized to one of 5 active doses (2.5, 10, 40, 80, or 120 mg), taking 4 tablets twice daily for 16 weeks.

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* Patients with T2DM who are treated with metformin and/or diet and exercise
* HbA1c greater than or equal to 7% and less than or equal to 10.5%
* Total body weight \>50 kg (110 lb) with BMI 24.5 to 45.4 kg/m\^2

Exclusion Criteria

* Any condition possibly affecting drug absorption
* Diagnosis of Type 1 diabetes
* History of myocardial infarction, unstable angina, arterial revascularization, stroke, heart failure, or transient ischemic attack within 6 months of screening
* Any malignancy not considered cured
* Personal or family history of MTC or MEN2, or participants with suspected MTC
* Acute pancreatitis or history of chronic pancreatitis
* Symptomatic gallbladder disease
* Known medical history of active proliferative retinopathy and/or macular edema
* Known medical history of active liver disease, including chronic active hepatitis B or C, or primary biliary cirrhosis
* Known history of HIV
* Supine blood pressure greater than or equal to 160 mmHg (systolic) or greater than or equal to 100 mmHg (diastolic)
* Clinically relevant ECG abnormalities
* Positive urine drug test
Minimum Eligible Age

18 Years

Maximum Eligible Age

75 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Pfizer

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Pfizer CT.gov Call Center

Role: STUDY_DIRECTOR

Pfizer

Locations

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Holy Trinity Medical Clinic

Harbor City, California, United States

Site Status

Innovative Clinical Research, Inc.

Harbor City, California, United States

Site Status

Long Beach Clinical Trials Services, Inc.

Long Beach, California, United States

Site Status

National Research Institute

Los Angeles, California, United States

Site Status

Catalina Research Institute, LLC

Montclair, California, United States

Site Status

Empire Clinical Research

Pomona, California, United States

Site Status

Rancho Cucamonga Clinical Research

Rancho Cucamonga, California, United States

Site Status

Encompass Clinical Research

Spring Valley, California, United States

Site Status

University Clinical Investigators, Incorporated

Tustin, California, United States

Site Status

San Fernando Valley Health Institute, LLC

Van Nuys, California, United States

Site Status

Diablo Clinical Research Incorporated

Walnut Creek, California, United States

Site Status

Accel Research Sites - DeLand Clinical Research Unit

DeLand, Florida, United States

Site Status

East Coast Institute for Research, LLC

Jacksonville, Florida, United States

Site Status

East Coast Institute for Research, LLC

Jacksonville, Florida, United States

Site Status

New Horizon Research Center

Miami, Florida, United States

Site Status

NewPhase Clinical Trials, Corp.

Miami Beach, Florida, United States

Site Status

Sunshine Research Center, Inc

Opa-locka, Florida, United States

Site Status

Andres Patron D.O. P.A.

Pembroke Pines, Florida, United States

Site Status

Ellipsis Group

Alpharetta, Georgia, United States

Site Status

East Coast Institute for Research, LLC

Macon, Georgia, United States

Site Status

Cedar Crosse Research Center

Chicago, Illinois, United States

Site Status

Buynak Clinical Research

Valparaiso, Indiana, United States

Site Status

Viable Research Management LLC

Henderson, Nevada, United States

Site Status

Premier Research

Trenton, New Jersey, United States

Site Status

PharmQuest

Greensboro, North Carolina, United States

Site Status

Lillestol Research LLC

Fargo, North Dakota, United States

Site Status

Velocity Clinical Research

Cincinnati, Ohio, United States

Site Status

Conrad Clinical Research

Edmond, Oklahoma, United States

Site Status

Family Medical Associates

Levittown, Pennsylvania, United States

Site Status

Preferred Primary Care Physicians, Inc.

Pittsburgh, Pennsylvania, United States

Site Status

Spartanburg Medical Research

Spartanburg, South Carolina, United States

Site Status

Palmetto Clinical Research

Summerville, South Carolina, United States

Site Status

Palmetto Primary Care Physicians (physicals only)

Summerville, South Carolina, United States

Site Status

Dallas Diabetes Research Center

Dallas, Texas, United States

Site Status

Endocrine Associates

Houston, Texas, United States

Site Status

PrimeCare Medical Group

Houston, Texas, United States

Site Status

Juno Research, LLC

Houston, Texas, United States

Site Status

Northeast Clinical Research of San Antonio

Live Oak, Texas, United States

Site Status

Sun Research Institute

San Antonio, Texas, United States

Site Status

DM Clinical Research

Tomball, Texas, United States

Site Status

Martin Diagnostic Clinic

Tomball, Texas, United States

Site Status

Rainier Clinical Research Center, Inc.

Renton, Washington, United States

Site Status

MHAT Dobrich AD

Dobrich, , Bulgaria

Site Status

Medical Center ASKLEPII OOD

Dupnitsa, , Bulgaria

Site Status

UMHAT Pulmed

Plovdiv, , Bulgaria

Site Status

Fourth MHAT - Sofia EAD

Sofia, , Bulgaria

Site Status

MHAT "Doverie" AD

Sofia, , Bulgaria

Site Status

MC "New rehabilitation center" EOOD

Stara Zagora, , Bulgaria

Site Status

GA Research Associates Ltd.

Moncton, New Brunswick, Canada

Site Status

Aggarwal and Associates Limited

Brampton, Ontario, Canada

Site Status

Manna Research (Toronto)

Toronto, Ontario, Canada

Site Status

Manna Research (Quebec)

Lévis, Quebec, Canada

Site Status

Manna Research (Mirabel)

Mirabel, Quebec, Canada

Site Status

Diex Recherche Quebec Inc.

Québec, Quebec, Canada

Site Status

Alpha Recherche Clinique

Québec, Quebec, Canada

Site Status

Diex Recherche Sherbrooke Inc.

Sherbrooke, Quebec, Canada

Site Status

Diex Recherche Victoriaville Inc.

Victoriaville, Quebec, Canada

Site Status

Centre de Recherche Saint-Louis

Québec, , Canada

Site Status

Belinus Orvosi es Szamitastechnikai Bt

Debrecen, , Hungary

Site Status

Debreceni Egyetem Klinikai Kozpont

Debrecen, , Hungary

Site Status

CRU Hungary Kft.

Miskolc, , Hungary

Site Status

Borbanya Praxis Egeszsegugyi KFT

Nyíregyháza, , Hungary

Site Status

Clinfan Kft.

Szekszárd, , Hungary

Site Status

Zdrowie Osteo-Medic s.c. Lidia i Artur Racewicz, Agnieszka i Jerzy Supronik

Bialystok, , Poland

Site Status

Medyczne Centrum Diabetologiczno-Endokrynologiczno-Metaboliczne DIAB-ENDO-MET Sp. z o. o.

Krakow, , Poland

Site Status

Prywatny Gabinet Lekarski i Wizyty Lekarskie Jan Ruxer

Lodz, , Poland

Site Status

MEDICOME Sp. z o.o.

Oświęcim, , Poland

Site Status

KO-MED CENTRA KLINICZNE Sp. z o.o. Ośrodek Badań Klinicznych w Puławach

Puławy, , Poland

Site Status

Centralny Szpital Kliniczny MSWiA

Warsaw, , Poland

Site Status

Metabol KLINIK s.r.o.

Bratislava, , Slovakia

Site Status

Medispektrum, s.r.o

Bratislava, , Slovakia

Site Status

HUMAN-CARE, s.r.o.

Košice, , Slovakia

Site Status

SchronerMED s.r.o.

Moldava nad Bodvou, , Slovakia

Site Status

Funkystuff, s.r.o.

Nové Zámky, , Slovakia

Site Status

DIAB s.r.o.

Rožňava, , Slovakia

Site Status

MUDr. Jana Rociakova, s.r.o.

Žilina, , Slovakia

Site Status

Yonsei University-Wonju Severance Christian Hospital

Wŏnju, Gangwon-do, South Korea

Site Status

Hanyang University Guri Hospital

Guri-si, Gyeonggi-do, South Korea

Site Status

Ajou University Hospital

Suwon, Gyeonggi-do, South Korea

Site Status

Samsung Medical Center

Gangnam-Gu, Seoul, South Korea

Site Status

Far Eastern Memorial Hospital

New Taipei City, , Taiwan

Site Status

Taichung Veterans General Hospital

Taichung, , Taiwan

Site Status

National Cheng Kung University Hospital

Tainan City, , Taiwan

Site Status

Countries

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United States Bulgaria Canada Hungary Poland Slovakia South Korea Taiwan

References

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Saxena AR, Frias JP, Brown LS, Gorman DN, Vasas S, Tsamandouras N, Birnbaum MJ. Efficacy and Safety of Oral Small Molecule Glucagon-Like Peptide 1 Receptor Agonist Danuglipron for Glycemic Control Among Patients With Type 2 Diabetes: A Randomized Clinical Trial. JAMA Netw Open. 2023 May 1;6(5):e2314493. doi: 10.1001/jamanetworkopen.2023.14493.

Reference Type DERIVED
PMID: 37213102 (View on PubMed)

Provided Documents

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Document Type: Study Protocol

View Document

Document Type: Statistical Analysis Plan

View Document

Related Links

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https://pmiform.com/clinical-trial-info-request?StudyID=C3421005

To obtain contact information for a study center near you, click here.

Other Identifiers

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2019-000218-12

Identifier Type: EUDRACT_NUMBER

Identifier Source: secondary_id

C3421005

Identifier Type: -

Identifier Source: org_study_id

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