Safety and Efficacy Study of LB80380 in the Treatment-naive Patients of Chronic Hepatitis B

NCT ID: NCT01026610

Last Updated: 2012-10-05

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

115 participants

Study Classification

INTERVENTIONAL

Study Start Date

2009-08-31

Study Completion Date

2011-05-31

Brief Summary

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The purpose of the study is to investigate the safety and the antiviral activity of two doses of LB80380 for 48 weeks in treatment-naive patients with chronic hepatitis B infection compared to entecavir 0.5 mg.

Detailed Description

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LB80380, an oral prodrug, is a promising candidate nucleotide analogue with antiviral activity against wild-type HBV. LB80380 is undergoing clinical development by LG Life Sciences for use in the treatment of chronic HBV infection.

In this study, the treatment period is 48-week with 24-week of follow-up period.

Conditions

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Chronic Hepatitis B

Keywords

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Chronic hepatitis B LB80380 treatment-naive entecavir

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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LB80380 90 mg

LB80380 90 mg (90 mg + placebo), once daily oral dose

Group Type EXPERIMENTAL

LB80380 90 mg

Intervention Type DRUG

LB80380 90 mg + placebo tablets, once daily, for 48 weeks

LB80380 150 mg

LB80380 150 mg (60 mg + 90 mg), once daily oral dose

Group Type EXPERIMENTAL

LB80380 150 mg

Intervention Type DRUG

LB80380 60 mg + 90 mg tablets, once daily, for 48 weeks

entecavir 0.5 mg

entecavir 0.5 mg, once daily oral dose

Group Type ACTIVE_COMPARATOR

entecavir 0.5 mg

Intervention Type DRUG

entecavir 0.5 mg tablet, once daily, for 48 weeks

Interventions

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LB80380 90 mg

LB80380 90 mg + placebo tablets, once daily, for 48 weeks

Intervention Type DRUG

LB80380 150 mg

LB80380 60 mg + 90 mg tablets, once daily, for 48 weeks

Intervention Type DRUG

entecavir 0.5 mg

entecavir 0.5 mg tablet, once daily, for 48 weeks

Intervention Type DRUG

Other Intervention Names

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LB80380 LB80380 Baraclude

Eligibility Criteria

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Inclusion Criteria

* Female or male, 18 to 65 years of age, inclusive
* Chronic hepatitis B
* Not treated with anti-viral therapeutics including interferon or pegylated interferons for more than 12 weeks before Screening
* Not treated with anti-viral therapeutics including interferon or pegylated interferons 6 months within Screening
* Compensated chronic hepatitis B
* HBeAg positive or HBeAg negative
* Elevated serum ALT level (1.2-10 X ULN, inclusive)

Exclusion Criteria

* Co-infection with hepatitis C or D virus (HCV or HDV) or HIV
* Decompensated liver disease
* Creatinine clearance (calculated by Cockroft-Gault formula) less than 50 ml/min
* Screening alpha-fetoprotein (AFP) value greater than or equal to 50 ng/mL, and a follow-up ultrasonography performed prior to baseline shows findings indicative of HCC
* Treatment with immunomodulatory agent or corticosteroids within 6 months prior to study entry.
* Pregnancy or breast-feeding
* Patient is currently abusing alcohol or illicit drugs
* Significant systemic illnesses other than liver diseases
* Presence of other causes of liver disease
* A history of organ transplantation

Presence of anti-HBs at screening
Minimum Eligible Age

18 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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LG Life Sciences

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Queen Mary Hospital

Hong Kong, , China

Site Status

Hanyang University Guri Hospital

Guri-si, Gyeonggi-do, South Korea

Site Status

Inha University Hospital

Incheon, Inchen, South Korea

Site Status

Kyungpook National University Hospital

Daegu, , South Korea

Site Status

Pusan National University Yangsan Hospital

Pusan, , South Korea

Site Status

Kangnam Severance Hospital, Yonsei University

Seoul, , South Korea

Site Status

Korea University Medical Center

Seoul, , South Korea

Site Status

Severance Hospital of Yonsei University

Seoul, , South Korea

Site Status

The Catholic University of Korea, Seoul St. Mary's Hospital

Seoul, , South Korea

Site Status

Ulsan University Hospital

Ulsan, , South Korea

Site Status

Countries

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China South Korea

References

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Fung J, Lai CL, Yuen MF. LB80380: a promising new drug for the treatment of chronic hepatitis B. Expert Opin Investig Drugs. 2008 Oct;17(10):1581-8. doi: 10.1517/13543784.17.10.1581.

Reference Type BACKGROUND
PMID: 18808318 (View on PubMed)

Yuen MF, Lee SH, Kang HM, Kim CR, Kim J, Ngai V, Lai CL. Pharmacokinetics of LB80331 and LB80317 following oral administration of LB80380, a new antiviral agent for chronic hepatitis B (CHB), in healthy adult subjects, CHB patients, and mice. Antimicrob Agents Chemother. 2009 May;53(5):1779-85. doi: 10.1128/AAC.01290-08. Epub 2009 Feb 17.

Reference Type BACKGROUND
PMID: 19223649 (View on PubMed)

Other Identifiers

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BVCL007

Identifier Type: -

Identifier Source: org_study_id