Safety/Tolerability and Pharmacokinetics/Pharmacodynamics of YH4808 After Oral Administration in Healthy Male Subjects

NCT ID: NCT01007019

Last Updated: 2014-07-10

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

Get a concise snapshot of the trial, including recruitment status, study phase, enrollment targets, and key timeline milestones.

Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

134 participants

Study Classification

INTERVENTIONAL

Study Start Date

2009-11-30

Study Completion Date

2012-03-31

Brief Summary

Review the sponsor-provided synopsis that highlights what the study is about and why it is being conducted.

First in human study

Detailed Description

Dive into the extended narrative that explains the scientific background, objectives, and procedures in greater depth.

Study to evaluate the safety and tolerability, pharmacokinetics/pharmacodynamics (PK/PD) parameters of an escalating, single dose/repeat doses of YH4808 in healthy subjects.

Conditions

See the medical conditions and disease areas that this research is targeting or investigating.

Healthy

Study Design

Understand how the trial is structured, including allocation methods, masking strategies, primary purpose, and other design elements.

Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

BASIC_SCIENCE

Blinding Strategy

DOUBLE

Participants Investigators

Study Groups

Review each arm or cohort in the study, along with the interventions and objectives associated with them.

YH4808 30mg

1.Single dose

2.12 volunteers were administered YH4808 30mg or active/placebo comparators.(YH4808:active:placebo=8:2:2)

Group Type EXPERIMENTAL

YH4808 30mg

Intervention Type DRUG

YH4808 30mg (single dose)

YH4808 50mg

1.Single dose

2.12 volunteers were administered YH4808 50mg or active/placebo comparators.(YH4808:active:placebo=8:2:2)

Group Type EXPERIMENTAL

YH4808 50mg

Intervention Type DRUG

YH4808 50mg (single dose)

YH4808 100mg

1.Single dose

2.12 volunteers were administered YH4808 100mg or active/placebo comparators.(YH4808:active:placebo=8:2:2)

Group Type EXPERIMENTAL

YH4808 100mg

Intervention Type DRUG

YH4808 100mg (single dose)

YH4808 200mg

1.Single dose

2.12 volunteers were administered YH4808 200mg or active/placebo comparators.(YH4808:active:placebo=8:2:2)

Group Type EXPERIMENTAL

YH4808 200mg

Intervention Type DRUG

YH4808 200mg (single dose)

YH4808 400mg

1.Single dose

2.12 volunteers were administered YH4808 400mg or active/placebo comparators.(YH4808:active:placebo=8:2:2)

Group Type EXPERIMENTAL

YH4808

Intervention Type DRUG

YH4808 400mg (single dose)

YH4808 100mg(repeat doses)

1.Repeat doses

2.12 volunteers were administered YH4808 100mg or active/placebo comparators.(YH4808:active:placebo=8:2:2)

Group Type EXPERIMENTAL

YH4808 100mg (repeat dose)

Intervention Type DRUG

YH4808 100mg (repeat dose)

YH4808 200mg(repeat doses)

1.Repeat doses

2.16 volunteers were administered YH4808 200mg or active/placebo comparators.(YH4808:active:placebo=8:6:2)

Group Type EXPERIMENTAL

YH4808 200mg (repeat dose)

Intervention Type DRUG

YH4808 200mg (repeat dose)

YH4808 400mg(repeat doses)

1.Repeat dose

2.12 volunteers were administered YH4808 400mg or active/placebo comparators.(YH4808:active:placebo=8:2:2)

Group Type EXPERIMENTAL

YH4808 400 mg (repeat doses)

Intervention Type DRUG

YH4808 400 mg (repeat doses)

YH4808 600mg

1.Single dose

2.12 volunteers were administered YH4808 600mg or active/placebo comparators.(YH4808:active:placebo=8:2:2)

Group Type EXPERIMENTAL

YH4808 600mg

Intervention Type DRUG

YH4808 600mg

YH4808 800mg

1.Single dose

2.12 volunteers were administered YH4808 800mg or active/placebo comparators.(YH4808:active:placebo=8:2:2)

Group Type EXPERIMENTAL

YH4808 800mg (single dose)

Intervention Type DRUG

YH4808 800mg (single dose)

Placebo

Group Type PLACEBO_COMPARATOR

Placebo

Intervention Type DRUG

10 volunteers will be administered matched placebo.

Esomeprazole 40mg

Group Type ACTIVE_COMPARATOR

Esomeprazole 40mg

Intervention Type DRUG

24 volunteers will be administered Esomeprazole 40mg

Interventions

Learn about the drugs, procedures, or behavioral strategies being tested and how they are applied within this trial.

YH4808 100mg

YH4808 100mg (single dose)

Intervention Type DRUG

YH4808 200mg

YH4808 200mg (single dose)

Intervention Type DRUG

YH4808

YH4808 400mg (single dose)

Intervention Type DRUG

YH4808 100mg (repeat dose)

YH4808 100mg (repeat dose)

Intervention Type DRUG

YH4808 200mg (repeat dose)

YH4808 200mg (repeat dose)

Intervention Type DRUG

YH4808 600mg

YH4808 600mg

Intervention Type DRUG

YH4808 800mg (single dose)

YH4808 800mg (single dose)

Intervention Type DRUG

YH4808 400 mg (repeat doses)

YH4808 400 mg (repeat doses)

Intervention Type DRUG

Placebo

10 volunteers will be administered matched placebo.

Intervention Type DRUG

Esomeprazole 40mg

24 volunteers will be administered Esomeprazole 40mg

Intervention Type DRUG

YH4808 30mg

YH4808 30mg (single dose)

Intervention Type DRUG

YH4808 50mg

YH4808 50mg (single dose)

Intervention Type DRUG

Other Intervention Names

Discover alternative or legacy names that may be used to describe the listed interventions across different sources.

YH4808 30mg (single dose) YH4808 50mg (single dose) YH4808 100mg (single dose) YH4808 200mg (single dose) YH4808 400mg (single dose) 10 volunteers will be administered matched placebo. 24 volunteers will be administered Esomeprazole 40mg

Eligibility Criteria

Check the participation requirements, including inclusion and exclusion rules, age limits, and whether healthy volunteers are accepted.

Inclusion Criteria

* Healthy male volunteers in the age between 20 to 45 years old
* Subjects who were determined to be appropriate through screening
* Weight: over 50kg, within ±20% of ideal body weight
* Subjects who signed written consent after receiving thorough explanation on trial purpose, content, and characteristics of investigational drug

Exclusion Criteria

* Clinically significant disorder in liver, kidney, cardiovascular, respiratory system, endocrine system and CNS in the physical examination and clinical laboratory tests or a medical history of malignant tumor or psychological disease
* Medical history of gastrointestinal disease or acid restraining surgery, gastric/esophagus surgery (excluding appendectomy, hernia surgery)
* A history of hypersensitivity to drugs or clinically significant allergic disease
* Clinically significant abnormal values in blood chemistry(≥ 1.5 fold of normal upper limit in the levels of SGOT, SGPT)
* Subjects who were unable to be applicable for pH meter catheter
* Subjects who had a history of drug abuse or who had a positive results on urine drug screening
* Subjects who had taken usual dose of any prescription drugs within 14 days before the treatment or who had used usual dose of OTC drugs within 7 days before the treatment(cf, be able to be enrolled in this study according to an investigatory consideration)
* Subjects who participated in another clinical trial within 3 months before enrolling in this study
* Subjects who donated whole blood within 2 months or component blood within 1 month or who are donated within 1 month before the treatment
* Subjects who drank Over 21 units/week of alcohol or subjects who weren't able to stop drinking alcohol during the hospitalization
* Subjects who stopped smoking within 3 months before the treatment
* Subjects who had a beverage containing grapefruits within 24hrs before the hospitalization or who had a beverage containing grapefruits during the hospitalization
* Subjects who had a beverage containing caffeine during the hospitalization
* H.pylori positive results on the Urease breath test(Only repeat doses)
* Subjects with clinically significant observations considered as unsuitable based on medical judgment by investigators
Minimum Eligible Age

20 Years

Maximum Eligible Age

45 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

Meet the organizations funding or collaborating on the study and learn about their roles.

Yuhan Corporation

INDUSTRY

Sponsor Role lead

Responsible Party

Identify the individual or organization who holds primary responsibility for the study information submitted to regulators.

Responsibility Role SPONSOR

Principal Investigators

Learn about the lead researchers overseeing the trial and their institutional affiliations.

Kyung-Sang Yu, MD, PhD

Role: PRINCIPAL_INVESTIGATOR

Seoul National University Hospital

Locations

Explore where the study is taking place and check the recruitment status at each participating site.

Clinical trials center, Seoul national university hospital

Seoul, , South Korea

Site Status

Countries

Review the countries where the study has at least one active or historical site.

South Korea

Other Identifiers

Review additional registry numbers or institutional identifiers associated with this trial.

YCD142 (YH4808-101)

Identifier Type: -

Identifier Source: org_study_id

More Related Trials

Additional clinical trials that may be relevant based on similarity analysis.