Duration of P-glycoprotein Inhibition After Oral Administration of HM30181AK Tablet

NCT ID: NCT00954304

Last Updated: 2010-09-13

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE1

Total Enrollment

30 participants

Study Classification

INTERVENTIONAL

Study Start Date

2009-06-30

Study Completion Date

2009-09-30

Brief Summary

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The purposes of this study are to investigate the duration of P-glycoprotein inhibition after oral administration of HM30181AK tablet in healthy male subject and proper dose of HM30181AK tablet.

Detailed Description

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Conditions

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Healthy

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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1mg group

Administration of HM30181AK 1mg on day 4 and Loperamide 16mg (Loperamide 2mg x 8cap) on day 1,4,8,11,15

Group Type EXPERIMENTAL

HM30181AK 1mg

Intervention Type DRUG

HM30181AK 1mg tablet

Loperamide 2mg

Intervention Type DRUG

Loperamide 2mg capsule

5mg group

Administration of HM30181AK 5mg on day 4 and Loperamide 16mg(Loperamide 2mg x 8cap) on day 1,4,8,11,15

Group Type EXPERIMENTAL

HM30181AK 5mg

Intervention Type DRUG

HM30181AK 5mg tablet

Loperamide 2mg

Intervention Type DRUG

Loperamide 2mg capsule

10mg group

Administration of HM30181AK 10mg(HM30181AK 5mg x 2tab)on day 4 and Loperamide 16mg (Loperamide 2mg x 8cap) on day 1,4,8,11,15

Group Type EXPERIMENTAL

HM30181AK 5mg

Intervention Type DRUG

HM30181AK 5mg tablet

Loperamide 2mg

Intervention Type DRUG

Loperamide 2mg capsule

15mg group

Administration of HM30181AK 15mg on day 4 and Loperamide 16mg (Loperamide 2mg x 8cap) on day 1,4,8,11,15

Group Type EXPERIMENTAL

HM30181AK 15mg

Intervention Type DRUG

HM30181AK 15mg tablet

Loperamide 2mg

Intervention Type DRUG

Loperamide 2mg capsule

60mg group

Administration of HM30181AK 60mg on day 4 and Loperamide 16mg (Loperamide 2mg x 8cap) on day 1,4,8,11,15

Group Type EXPERIMENTAL

HM30181AK 60mg

Intervention Type DRUG

HM30181AK 60mg tablet

Loperamide 2mg

Intervention Type DRUG

Loperamide 2mg capsule

Interventions

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HM30181AK 1mg

HM30181AK 1mg tablet

Intervention Type DRUG

HM30181AK 5mg

HM30181AK 5mg tablet

Intervention Type DRUG

HM30181AK 15mg

HM30181AK 15mg tablet

Intervention Type DRUG

HM30181AK 60mg

HM30181AK 60mg tablet

Intervention Type DRUG

Loperamide 2mg

Loperamide 2mg capsule

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Healthy male volunteers aged 20 to 50 years at screening
2. Subjects whose weights are heavier than or equal to 50 kg and ±20% of ideal body weight

* Ideal body weight = (height cm - 100) x 0.9
3. Subjects who provided written, voluntary informed consent to participate in this clinical trial and to comply the directions including contraception after being fully informed of and understand this trial

Exclusion Criteria

1. Subjects who have the clinically significant diseases or history in liver, kidney, nervous system, respiratory system, endocrine system, blood tumor and cardiovascular system.
2. History of the gastrointestinal diseases which may affect the absorption of oral drugs (e.g., Crohn's disease) or gastrointestinal operations (excluding simple typhlotomy and hernia repair).
3. The following results in laboratory test

* AST, ALT \> 1.25 x upper limits of normal
4. Systolic blood pressure below 100 mmHg or above 150 mmHg or diastolic blood pressure below 65 mmHg or above 95 mmHg in vital signs
5. History of drug allergy or other allergies which are clinically significant
6. History of drug abuse or positive reaction for drug abuse in urine screening test
7. Subjects who took prescription drugs or herbal medicines within 2 weeks prior to the first day of drug administration or OTC or vitamin preparations within 1 week prior to the first day of drug administration If the subjects meet other criteria, they could participate in the trial in the judgement of investigator.)
8. Subjects who have participated in other clinical trial within 2 months prior to the first day of drug administration
9. Whole blood donation within 2 months prior to the first day of drug administration or apheresis donation within 2 weeks prior to the first day of drug administration
10. Subject who are continuously drinking alcohol (over 21 units/week) or who cannot quit drinking during clinical trial period
11. Subject who are smoking over 10 cigar/day
12. Subjects who eat food containing caffeine or grapefruit or drink alcohol in prohibited period
13. Subjects who are inappropriate in the judgement of the investigator due to the reasons including clinical laboratory test results
Minimum Eligible Age

20 Years

Maximum Eligible Age

50 Years

Eligible Sex

MALE

Accepts Healthy Volunteers

Yes

Sponsors

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Hanmi Pharmaceutical Company Limited

INDUSTRY

Sponsor Role lead

Responsible Party

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Hanmi Pharmaceutical Company Limited

Principal Investigators

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Kyung-Sang Yu, MD., Ph.D

Role: PRINCIPAL_INVESTIGATOR

Seoul National University Hospital

Locations

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Seoul National University Hospital

Seoul, , South Korea

Site Status

Countries

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South Korea

Other Identifiers

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HM-OXL-104

Identifier Type: -

Identifier Source: org_study_id