A Phase I, Open-Label, Multi-center Study to Assess the Safety, Tolerability and Pharmacokinetics of AZD6244 (ARRY-142886)

NCT ID: NCT00600496

Last Updated: 2025-11-13

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

ACTIVE_NOT_RECRUITING

Clinical Phase

PHASE1

Total Enrollment

140 participants

Study Classification

INTERVENTIONAL

Study Start Date

2007-12-14

Study Completion Date

2025-12-31

Brief Summary

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This study is being conducted to determine if a combination of AZD6244 given orally twice a day with standard doses of selected chemotherapies will be safe and tolerable for cancer patients with advanced solid tumors. The highest tolerated dose of AZD6244 in combination with selected chemotherapies will be evaluated. The study will also investigate how AZD6244 in combination with standard chemotherapies are absorbed, distributed and excreted by the body as well as the length of time that the drugs remain in the body. Initial and periodic assessments will establish patient response to the combination therapies

Detailed Description

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Conditions

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Breast Cancer Breast Neoplasms Colon Cancer Colonic Cancer Colon Neoplasms Lung Cancer Melanoma Kidney Cancer

Keywords

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ARRY-142886 AZD6244 Cancer Colon Cancer Breast Cancer Lung Cancer Melanoma Kidney Cancer

Study Design

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Allocation Method

NON_RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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1

AZD6244 + docetaxel

Group Type EXPERIMENTAL

AZD6244

Intervention Type DRUG

twice daily oral dose

Docetaxel

Intervention Type DRUG

intravenous infusion

2

AZD6244 + Dacarbazine

Group Type EXPERIMENTAL

AZD6244

Intervention Type DRUG

twice daily oral dose

Dacarbazine

Intervention Type DRUG

intravenous infusion

3

AZD6244 + Erlotinib

Group Type EXPERIMENTAL

AZD6244

Intervention Type DRUG

twice daily oral dose

Erlotinib

Intervention Type DRUG

daily oral dose

4

AZD6244 + Temsirolimus

Group Type EXPERIMENTAL

AZD6244

Intervention Type DRUG

twice daily oral dose

Temsirolimus

Intervention Type DRUG

intravenous infusion

Interventions

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AZD6244

twice daily oral dose

Intervention Type DRUG

Dacarbazine

intravenous infusion

Intervention Type DRUG

Erlotinib

daily oral dose

Intervention Type DRUG

Docetaxel

intravenous infusion

Intervention Type DRUG

Temsirolimus

intravenous infusion

Intervention Type DRUG

Other Intervention Names

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ARRY-142886 Taxotere®

Eligibility Criteria

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Inclusion Criteria

* Patients will have measurable and/or non-measurable disease, lacking curative options for whom the selected chemotherapy agents represent the standard of care
* WHO performance status 0-1
* Patients must be able to swallow AZD6244 capsules

Exclusion Criteria

* Prior treatment with a MEK inhibitor
* Participation in a clinical study during the last 30 days or have not recovered from side effects of an investigational study drug
* Brain metastases or spinal cord compression unless treated and stable (for at least 1 month) off steroids
Minimum Eligible Age

18 Years

Maximum Eligible Age

130 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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AstraZeneca

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Principal Investigators

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Patricia LoRusso, DO

Role: PRINCIPAL_INVESTIGATOR

Barbara Ann Karmanos Cancer Institute

Roger Cohen, MD

Role: PRINCIPAL_INVESTIGATOR

Fox Chase Cancer Center

Jeffrey Infante, MD

Role: PRINCIPAL_INVESTIGATOR

SCRI Development Innovations, LLC

Kevin Kim, MD

Role: PRINCIPAL_INVESTIGATOR

M.D. Anderson Cancer Center

Locations

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Research Site

Detroit, Michigan, United States

Site Status

Research Site

Philadelphia, Pennsylvania, United States

Site Status

Research Site

Nashville, Tennessee, United States

Site Status

Research Site

Houston, Texas, United States

Site Status

Countries

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United States

References

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Patel SP, Lazar AJ, Papadopoulos NE, Liu P, Infante JR, Glass MR, Vaughn CS, LoRusso PM, Cohen RB, Davies MA, Kim KB. Clinical responses to selumetinib (AZD6244; ARRY-142886)-based combination therapy stratified by gene mutations in patients with metastatic melanoma. Cancer. 2013 Feb 15;119(4):799-805. doi: 10.1002/cncr.27790. Epub 2012 Sep 12.

Reference Type DERIVED
PMID: 22972589 (View on PubMed)

Infante JR, Cohen RB, Kim KB, Burris HA 3rd, Curt G, Emeribe U, Clemett D, Tomkinson HK, LoRusso PM. A phase I dose-escalation study of Selumetinib in combination with Erlotinib or Temsirolimus in patients with advanced solid tumors. Invest New Drugs. 2017 Oct;35(5):576-588. doi: 10.1007/s10637-017-0459-7. Epub 2017 Apr 19.

Reference Type DERIVED
PMID: 28424891 (View on PubMed)

LoRusso PM, Infante JR, Kim KB, Burris HA 3rd, Curt G, Emeribe U, Clemett D, Tomkinson HK, Cohen RB. A phase I dose-escalation study of selumetinib in combination with docetaxel or dacarbazine in patients with advanced solid tumors. BMC Cancer. 2017 Mar 6;17(1):173. doi: 10.1186/s12885-017-3143-6.

Reference Type DERIVED
PMID: 28264648 (View on PubMed)

Related Links

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Other Identifiers

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D1532C00004

Identifier Type: -

Identifier Source: org_study_id