Ritonavir-Boosted GS-9137 vs. Ritonavir-Boosted Protease Inhibitor(s) in Combination With Background ART.

NCT ID: NCT00298350

Last Updated: 2008-07-29

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

COMPLETED

Clinical Phase

PHASE2

Total Enrollment

278 participants

Study Classification

INTERVENTIONAL

Study Start Date

2006-02-28

Study Completion Date

2007-07-31

Brief Summary

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The purpose of this study is to evaluate the non-inferiority of ritonavir-boosted GS-9137 relative to a ritonavir-boosted Comparator Protease Inhibitor when used as part of combination antiretroviral regimens in subjects who have failed, or are failing, protease inhibitor therapy.

Detailed Description

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Conditions

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HIV HIV-1 Human Immunodeficiency Virus

Study Design

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Allocation Method

RANDOMIZED

Intervention Model

PARALLEL

Primary Study Purpose

TREATMENT

Blinding Strategy

QUADRUPLE

Participants Caregivers Investigators Outcome Assessors

Interventions

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GS-9137 - A Novel HIV-1 Integrase Inhibitor

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

* HIV RNA greater than or equal to 1000 c/mL.
* Failed/Failing protease inhibitor based antiretroviral therapy.
* Stable antiretroviral therapy for greater than or equal to 30 days prior to screening.
* Negative Serum Pregnancy Test.
* GFR by Cockcroft Gault greater than or equal to 80 mL/min.
* AST \& ALT less than or equal to 2.5x ULN.
* Total Bilirubin less than or equal to 1.5 mg/dL.
* Albumin greater than 3.5 mg/dL.
* Prothrombin Time INR 1.0-1.4
* Platelets greater than or equal to 50,000.
* Hemoglobin greater than or equal to 8.0 mg/dL.
* Absolute Neutrophil Count greater than or equal to 1000.

Exclusion Criteria

* New AIDS defining condition within 30 days of baseline.
* Prior treatment with HIV-1 integrase inhibitor (except patients from 183-101).
* Ascites or encephalopathy.
* Breast Feeding.
* Cancer Diagnosis (besides Kaposi Sarcoma or Basal Cell Carcinoma).
Minimum Eligible Age

18 Years

Maximum Eligible Age

65 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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Gilead Sciences

INDUSTRY

Sponsor Role lead

Responsible Party

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Gilead Sciences INC

Locations

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Phoenix, Arizona, United States

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Little Rock, Arkansas, United States

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Beverly Hills, California, United States

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Fountain Valley, California, United States

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Long Beach, California, United States

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Los Angeles, California, United States

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Newport Beach, California, United States

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Oakland, California, United States

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San Diego, California, United States

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San Francisco, California, United States

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Stanford, California, United States

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Sunnyvale, California, United States

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Torrance, California, United States

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Denver, Colorado, United States

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Norwalk, Connecticut, United States

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Washington D.C., District of Columbia, United States

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Atlantis, Florida, United States

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Fort Lauderdale, Florida, United States

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Miami, Florida, United States

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North Miami Beach, Florida, United States

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North Palm Beach, Florida, United States

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Orlando, Florida, United States

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Sarasota, Florida, United States

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Tampa, Florida, United States

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Vero Beach, Florida, United States

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Decatur, Georgia, United States

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Macon, Georgia, United States

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Chicago, Illinois, United States

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Baltimore, Maryland, United States

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Boston, Massachusetts, United States

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Springfield, Massachusetts, United States

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Detroit, Michigan, United States

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St Louis, Missouri, United States

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Henderson, Nevada, United States

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Hillsborough, New Jersey, United States

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Santa Fe, New Mexico, United States

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Albany, New York, United States

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Manhasset, New York, United States

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New York, New York, United States

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Huntersville, North Carolina, United States

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Winston-Salem, North Carolina, United States

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Cleveland, Ohio, United States

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Hershey, Pennsylvania, United States

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Philadelphia, Pennsylvania, United States

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Columbia, South Carolina, United States

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Dallas, Texas, United States

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Houston, Texas, United States

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Annandale, Virginia, United States

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Hampton, Virginia, United States

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Seattle, Washington, United States

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Tacoma, Washington, United States

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Milwaukee, Wisconsin, United States

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San Juan, , Puerto Rico

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Santurce, , Puerto Rico

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Countries

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United States Puerto Rico

References

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Zolopa AR, Berger DS, Lampiris H, Zhong L, Chuck SL, Enejosa JV, Kearney BP, Cheng AK. Activity of elvitegravir, a once-daily integrase inhibitor, against resistant HIV Type 1: results of a phase 2, randomized, controlled, dose-ranging clinical trial. J Infect Dis. 2010 Mar 15;201(6):814-22. doi: 10.1086/650698.

Reference Type DERIVED
PMID: 20146631 (View on PubMed)

Related Links

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Other Identifiers

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GS-US-183-0105

Identifier Type: -

Identifier Source: org_study_id

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