A Study of Avoralstat In Participants With Diabetic Macular Edema

NCT ID: NCT07228559

Last Updated: 2026-02-04

Study Results

Results pending

The study team has not published outcome measurements, participant flow, or safety data for this trial yet. Check back later for updates.

Basic Information

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Recruitment Status

RECRUITING

Clinical Phase

PHASE1

Total Enrollment

9 participants

Study Classification

INTERVENTIONAL

Study Start Date

2025-10-02

Study Completion Date

2026-09-30

Brief Summary

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The goal of this study is to assess the safety and therapeutic potential of a single dose of avoralstat in adult participants with DME.

Detailed Description

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Study BCX4161-111 is an open-label, single ascending dose study with 24 weeks follow-up in participants with DME. Three cohorts with a minimum of 3 participants enrolled in each cohort with 3 dose levels of avoralstat (low, medium, high) are planned.

Conditions

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Diabetic Macular Edema (DME)

Study Design

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Allocation Method

NA

Intervention Model

SINGLE_GROUP

Primary Study Purpose

TREATMENT

Blinding Strategy

NONE

Study Groups

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Single dose suprachoroidal injection of avoralstat

Group Type EXPERIMENTAL

avoralstat

Intervention Type DRUG

BCX4161 for suprachoroidal injection

Interventions

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avoralstat

BCX4161 for suprachoroidal injection

Intervention Type DRUG

Eligibility Criteria

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Inclusion Criteria

1. Male or female aged 18 years or older
2. Glycated hemoglobin A (HbA1c) \< 10% at screening
3. Diagnosis of DME with center involvement requiring medical treatment within 6 months of screening and decreased visual acuity attributable to DME
4. Mild-to-severe non-proliferative diabetic retinopathy (NPDR) with DRSS \< 61 in the study eye at screening
5. BCVA between 35 and 80 ETDRS letters (20/25 to 20/200 Snellen equivalent), inclusive, in the study eye at screening
6. CST measured by Heidelberg OCT between 325 and 600 μm in the study eye at screening

Exclusion Criteria

1. Participants who have previously received more than 3 anti-VEGF injections
2. Any history of retinal surgery or other surgical intervention for diabetic ocular complications or anticipated need for use of laser photocoagulation course of any of the procedures listed in the criteria in the study eye during the study period
3. Current medically untreated diabetes mellitus or previous medically untreated diabetes mellitus with initiation of oral or injectable anti-diabetic medication ≤ 3 months prior to screening
4. Active intraocular or periocular infection or active intraocular inflammation in the study eye
5. Intraocular surgery ≤ 3 months prior to screening or anticipated need for ocular surgery in the study eye during the study period
Minimum Eligible Age

18 Years

Eligible Sex

ALL

Accepts Healthy Volunteers

No

Sponsors

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BioCryst Pharmaceuticals

INDUSTRY

Sponsor Role lead

Responsible Party

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Responsibility Role SPONSOR

Locations

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Investigative Site 6

Sacramento, California, United States

Site Status RECRUITING

Investigative Site 7

Katy, Texas, United States

Site Status RECRUITING

Investigative Site 8

The Woodlands, Texas, United States

Site Status RECRUITING

Investigative Site 1

Sydney, New South Wales, Australia

Site Status RECRUITING

Investigative Site 2

Sydney, New South Wales, Australia

Site Status RECRUITING

Investigative Site 3

Sydney, New South Wales, Australia

Site Status RECRUITING

Investigative Site 4

Adelaide, South Australia, Australia

Site Status RECRUITING

Investigative Site 5

Melbourne, Victoria, Australia

Site Status RECRUITING

Countries

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United States Australia

Central Contacts

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BioCryst Pharmaceuticals, Inc.

Role: CONTACT

+1 919 859 1302

Other Identifiers

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BCX4161-111

Identifier Type: -

Identifier Source: org_study_id

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